ketoconazole and anastrozole

ketoconazole has been researched along with anastrozole in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (27.27)29.6817
2010's8 (72.73)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berk, B; Biltekin, SN; Demirayak, S; Ertas, M; Sahin, Z; Yurttas, L1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Muftuoglu, Y; Mustata, G1
Agard, H; Amato, E; Bankemper, T; Bonfield, K; Keeler, JM; Ma, L; McCallum, A; Paula, S; Roy, D; Steller, J1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Boepple, PA; Crowley, WF; DeCruz, S; Hayes, FJ; Seminara, SB1
Bray, MJ; Schnorr, JA; Veldhuis, JD1
Büyükünal, C; Ceylaner, S; Ercan, O; Evliyaoğlu, O; Özcabı, B; Özcan, R; Tahmiscioğlu Bucak, F; Tüysüz, B1
Baj, F; Baravalle, R; Ciaramella, A; Di Nardo, G; Gilardi, G1

Reviews

1 review(s) available for ketoconazole and anastrozole

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for ketoconazole and anastrozole

ArticleYear
Aromatization mediates testosterone's short-term feedback restraint of 24-hour endogenously driven and acute exogenous gonadotropin-releasing hormone-stimulated luteinizing hormone and follicle-stimulating hormone secretion in young men.
    The Journal of clinical endocrinology and metabolism, 2001, Volume: 86, Issue:6

    Topics: Administration, Cutaneous; Adult; Anastrozole; Aromatase Inhibitors; Circadian Rhythm; Dose-Response Relationship, Drug; Double-Blind Method; Enzyme Inhibitors; Estradiol; Feedback; Follicle Stimulating Hormone; Gonadotropin-Releasing Hormone; Humans; Ketoconazole; Luteinizing Hormone; Male; Nitriles; Prospective Studies; Testosterone; Triazoles

2001

Other Studies

9 other study(ies) available for ketoconazole and anastrozole

ArticleYear
Studies on non-steroidal inhibitors of aromatase enzyme; 4-(aryl/heteroaryl)-2-(pyrimidin-2-yl)thiazole derivatives.
    Bioorganic & medicinal chemistry, 2018, 05-01, Volume: 26, Issue:8

    Topics: Aromatase; Binding Sites; Catalytic Domain; Cell Proliferation; Cell Survival; Drug Design; Enzyme Inhibitors; HEK293 Cells; Humans; MCF-7 Cells; Molecular Docking Simulation; Pyrimidines; Structure-Activity Relationship; Thiazoles

2018
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Pharmacophore modeling strategies for the development of novel nonsteroidal inhibitors of human aromatase (CYP19).
    Bioorganic & medicinal chemistry letters, 2010, May-15, Volume: 20, Issue:10

    Topics: Antineoplastic Agents; Aromatase; Aromatase Inhibitors; Binding Sites; Breast Neoplasms; Computer Simulation; Drug Design; Female; Humans; Models, Chemical; Models, Molecular; Structure-Activity Relationship

2010
Development of a new class of aromatase inhibitors: design, synthesis and inhibitory activity of 3-phenylchroman-4-one (isoflavanone) derivatives.
    Bioorganic & medicinal chemistry, 2012, Apr-15, Volume: 20, Issue:8

    Topics: Aromatase; Aromatase Inhibitors; Dose-Response Relationship, Drug; Drug Design; Humans; Isoflavones; Molecular Structure; Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Differential regulation of gonadotropin secretion by testosterone in the human male: absence of a negative feedback effect of testosterone on follicle-stimulating hormone secretion.
    The Journal of clinical endocrinology and metabolism, 2001, Volume: 86, Issue:1

    Topics: Adult; Anastrozole; Aromatase Inhibitors; Dexamethasone; Enzyme Inhibitors; Estrogen Antagonists; Feedback; Follicle Stimulating Hormone; Glucocorticoids; Gonadal Steroid Hormones; Gonadotropins; Humans; Ketoconazole; Luteinizing Hormone; Male; Nitriles; Testosterone; Triazoles

2001
Testotoxicosis: Report of Two Cases, One with a Novel Mutation in LHCGR Gene.
    Journal of clinical research in pediatric endocrinology, 2015, Volume: 7, Issue:3

    Topics: Anastrozole; Androgen Antagonists; Anilides; Aromatase Inhibitors; Cytochrome P-450 CYP3A Inhibitors; Genetic Predisposition to Disease; Humans; Infant; Ketoconazole; Male; Mutation; Nitriles; Puberty, Precocious; Receptors, LH; Sequence Analysis, DNA; Testosterone; Tosyl Compounds; Triazoles

2015
Identification of endocrine disrupting chemicals acting on human aromatase.
    Biochimica et biophysica acta. Proteins and proteomics, 2018, Volume: 1866, Issue:1

    Topics: Anastrozole; Aromatase; Aromatase Inhibitors; Benzhydryl Compounds; Biological Assay; Endocrine Disruptors; Enzyme-Linked Immunosorbent Assay; Estrone; Gene Expression; Humans; Ketoconazole; Ligands; NADP; Nicotine; Nitriles; Phenols; Protein Binding; Recombinant Proteins; Resveratrol; Sildenafil Citrate; Small Molecule Libraries; Stilbenes; Triazoles

2018