ketanserin and urapidil

ketanserin has been researched along with urapidil in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19905 (25.00)18.7374
1990's9 (45.00)18.2507
2000's2 (10.00)29.6817
2010's4 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Baldanzi, G; Bertoni, A; Capello, D; Fresu, LG; Gesu, A; Graziani, A; Massarotti, A; Ruffo, E; Snow, AL; Talmon, M; Tron, GC; Varma, KSS; Velnati, S1
Blauw, GJ; van Brummelen, P; van Zwieten, PA3
Lauwers, P; Möllhoff, T; Mulier, JP; Müller, E; Van Aken, H1
Kirsten, R; Ochs, JG; Storck, J1
Prichard, BN; Van Zwieten, PA1
van Zwieten, PA1
Doyle, AE1
Timmermans, PB; van Zwieten, PA1
Timmermans, PB; Van Brummelen, P; Van Zwieten, PA1
Baumgärtel, M; Petry, A; Wulf, H1
Innes, PA1
Kal, JE; Kooyman, J; Korsten, HH; Langemeijer, JJ; Porsius, M; van den Ende, R; van der Starre, PJ; van der Stroom, JG; van Wezel, HB; van Zwieten, PA1
Petry, A1
Buñag, RD; Mellick, JR; Thomas, CV1

Reviews

7 review(s) available for ketanserin and urapidil

ArticleYear
Serotonergic receptors and drugs in hypertension.
    Pharmacology & toxicology, 1992, Volume: 70, Issue:6 Pt 2

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Disease Models, Animal; Humans; Hypertension; Ketanserin; Piperazines; Receptors, Serotonin; Vasodilator Agents

1992
Pharmacological profile of antihypertensive drugs with serotonin receptor and alpha-adrenoceptor activity.
    Drugs, 1990, Volume: 40 Suppl 4

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Ketanserin; Piperazines; Receptors, Serotonin; Serotonin Antagonists

1990
Pathophysiological and pharmacotherapeutic aspects of serotonin and serotonergic drugs.
    Clinical physiology and biochemistry, 1990, Volume: 8 Suppl 3

    Topics: Animals; Antihypertensive Agents; Cardiovascular Diseases; Humans; Hypertension; Ketanserin; Piperazines; Receptors, Serotonin; Serotonin

1990
Basic pharmacology of alpha-adrenoceptor antagonists and hybrid drugs.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1988, Volume: 6, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Chemical Phenomena; Chemistry; Humans; Ketanserin; Labetalol; Piperazines

1988
Do hybrid drugs offer an additional benefit over pure alpha 1-blockade for hypertensive patients?
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1988, Volume: 6, Issue:2

    Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Humans; Hypertension; Ketanserin; Labetalol; Piperazines

1988
Cardiovascular alpha 2-receptors.
    Journal of molecular and cellular cardiology, 1983, Volume: 15, Issue:11

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Affinity Labels; Animals; Blood Pressure; Brain; Calcium Channel Blockers; Cardiovascular Physiological Phenomena; Guanosine Triphosphate; Heart Rate; Humans; Ketanserin; Kidney; Muscle, Smooth, Vascular; Piperazines; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Synaptic Membranes; Tritium; Vasoconstriction

1983
Role of alpha adrenoceptors in hypertension and in antihypertensive drug treatment.
    The American journal of medicine, 1984, Oct-05, Volume: 77, Issue:4A

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Calcium Channel Blockers; Clonidine; Guanfacine; Guanidines; Humans; Hypertension; Ketanserin; Methyldopa; Muscle, Smooth, Vascular; Phenylacetates; Piperazines; Piperidines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Vascular Resistance

1984

Trials

4 trial(s) available for ketanserin and urapidil

ArticleYear
Effects of urapidil, ketanserin and sodium nitroprusside on venous admixture and arterial oxygenation following coronary artery bypass grafting.
    British journal of anaesthesia, 1990, Volume: 64, Issue:4

    Topics: Antihypertensive Agents; Coronary Artery Bypass; Heart Rate; Hemodynamics; Humans; Hypertension; Ketanserin; Middle Aged; Nitroprusside; Oxygen; Piperazines; Postoperative Complications; Respiration

1990
The influence of ketanserin or urapidil on haemodynamics, stress response and kidney function during operations for myocardial revascularisation.
    Anaesthesia, 1995, Volume: 50, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Anesthesia, General; Antihypertensive Agents; Double-Blind Method; Epinephrine; Hemodynamics; Humans; Hypertension; Ketanserin; Kidney; Male; Middle Aged; Myocardial Revascularization; Norepinephrine; Piperazines; Prospective Studies

1995
A randomized multicenter double-blind comparison of urapidil and ketanserin in hypertensive patients after coronary artery surgery.
    Journal of cardiothoracic and vascular anesthesia, 1997, Volume: 11, Issue:6

    Topics: Aged; Antihypertensive Agents; Coronary Vessels; Double-Blind Method; Hemodynamics; Humans; Hypertension; Ketanserin; Middle Aged; Piperazines; Postoperative Complications; Respiration

1997
Computer aided monitor-data processing (CAMP). A landmark for unbiased gauging of anaesthetic courses?
    Journal of clinical monitoring and computing, 1998, Volume: 14, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Anesthesia, General; Blood Pressure; Hemodynamics; Humans; Ketanserin; Male; Medical Records Systems, Computerized; Middle Aged; Monitoring, Intraoperative; Myocardial Revascularization; Operating Room Information Systems; Piperazines; Prospective Studies; Serotonin Antagonists

1998

Other Studies

9 other study(ies) available for ketanserin and urapidil

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Identification of a novel DGKα inhibitor for XLP-1 therapy by virtual screening.
    European journal of medicinal chemistry, 2019, Feb-15, Volume: 164

    Topics: Cell Death; Computer Simulation; Diacylglycerol Kinase; Drug Evaluation, Preclinical; Humans; Lymphoproliferative Disorders; Piperidines; Protein Kinase Inhibitors; Pyrimidinones; Quinazolinones; Ritanserin; Thiazoles

2019
Effects of urapidil on 5-hydroxytryptamine induced platelet aggregation and on 14C-5-hydroxytryptamine uptake in platelets.
    International journal of clinical pharmacology, therapy, and toxicology, 1990, Volume: 28, Issue:7

    Topics: Administration, Oral; Adult; Blood Platelets; Carbon Radioisotopes; Epinephrine; Humans; Ketanserin; Nafronyl; Piperazines; Platelet Aggregation Inhibitors; Prazosin; Serotonin; Serotonin Antagonists

1990
An antihypertensive drug with polyfactor mechanism of action: urapidil.
    Annales francaises d'anesthesie et de reanimation, 1989, Volume: 8, Issue:5

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Brain Chemistry; Cats; Humans; Ketanserin; Labetalol; Piperazines; Rats; Receptors, Adrenergic; Receptors, Serotonin

1989
Ketanserin and urapidil during myocardial revascularisation.
    Anaesthesia, 1995, Volume: 50, Issue:12

    Topics: Hemodynamics; Humans; Ketanserin; Myocardial Revascularization; Piperazines; Research Design; Vasodilator Agents

1995
Ketanserin versus urapidil: age-related cardiovascular effects in conscious rats.
    European journal of pharmacology, 2002, Jan-18, Volume: 435, Issue:1

    Topics: Aging; Angiotensins; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Bradycardia; Ketanserin; Male; Piperazines; Rats; Rats, Sprague-Dawley; Reflex

2002