ketanserin has been researched along with tryptamine in 18 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (44.44) | 18.7374 |
1990's | 7 (38.89) | 18.2507 |
2000's | 1 (5.56) | 29.6817 |
2010's | 2 (11.11) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Glennon, RA | 2 |
Andrews, PR; Craik, DJ; Martin, JL | 1 |
Buckingham, J; Glen, RC; Hill, AP; Hyde, RM; Martin, GR; Robertson, AD; Salmon, JA; Woollard, PM | 1 |
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J | 1 |
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR | 1 |
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R | 1 |
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Lepailleur, A; Rochais, C; Thirumaran, SL | 1 |
Horisaka, K; Sugimoto, Y; Yamada, J | 1 |
Aghajanian, GK; Lakoski, JM | 1 |
Bradley, PB; Humphrey, PP; Williams, RH | 1 |
Clancy, BM; Maayani, S; Osman, R | 1 |
de Chaffoy de Courcelles, D; Leysen, JE; Niemegeers, CJ; Van Gompel, P | 1 |
Eyre, P; Ogunbiyi, PO | 1 |
Horisaka, K; Kimura, I; Sugimoto, Y; Watanabe, Y; Yamada, J | 1 |
Baez, M; Johnson, MP; Lucaites, VL; Nelson, DL; Wainscott, DB | 1 |
2 review(s) available for ketanserin and tryptamine
Article | Year |
---|---|
Central serotonin receptors as targets for drug research.
Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin | 1987 |
Structure-activity relationships of serotonin 5-HT
Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship | 2019 |
16 other study(ies) available for ketanserin and tryptamine
Article | Year |
---|---|
Functional group contributions to drug-receptor interactions.
Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship | 1984 |
Computer-aided design and synthesis of 5-substituted tryptamines and their pharmacology at the 5-HT1D receptor: discovery of compounds with potential anti-migraine properties.
Topics: Animals; Aorta; Computer-Aided Design; Drug Design; Haplorhini; In Vitro Techniques; Migraine Disorders; Models, Chemical; Rabbits; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Saphenous Vein; Serotonin Receptor Agonists; Structure-Activity Relationship; Tryptamines | 1995 |
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.
Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction | 1993 |
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection | 1993 |
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents | 1996 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
The 2014 Philip S. Portoghese Medicinal Chemistry Lectureship: The "Phenylalkylaminome" with a Focus on Selected Drugs of Abuse.
Topics: Animals; Central Nervous System Stimulants; Chemistry, Pharmaceutical; Dopamine; Drug Discovery; Hallucinogens; Humans; Illicit Drugs; Norepinephrine; Phenethylamines; Psychotropic Drugs; Receptors, Serotonin; Serotonin | 2017 |
The evidence for the involvement of the 5-HT1A receptor in 5-HT syndrome induced in mice by tryptamine.
Topics: Animals; Behavior, Animal; Haloperidol; Ketanserin; Male; Methysergide; Mice; Mice, Inbred DBA; Propranolol; Receptors, Serotonin; Serotonin; Spiperone; Tryptamines | 1989 |
Effects of ketanserin on neuronal responses to serotonin in the prefrontal cortex, lateral geniculate and dorsal raphe nucleus.
Topics: Animals; Decerebrate State; Electrophysiology; Frontal Lobe; gamma-Aminobutyric Acid; Geniculate Bodies; Ketanserin; Male; Norepinephrine; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Tryptamines | 1985 |
Tryptamine-induced vasoconstrictor responses in rat caudal arteries are mediated predominantly via 5-hydroxytryptamine receptors.
Topics: Animals; Arteries; In Vitro Techniques; Ketanserin; Male; Methysergide; Monoamine Oxidase Inhibitors; Phentolamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tryptamines; Vasoconstriction | 1985 |
Kinetics of competitive drug action at 5-hydroxytryptamine2 receptors in isolated rabbit aorta.
Topics: Animals; Aorta; Binding, Competitive; Diffusion; Indoles; Ketanserin; Kinetics; Male; Methysergide; Muscle, Smooth, Vascular; Rabbits; Receptors, Serotonin; Serotonin; Spiperone; Tryptamines | 1987 |
Opposite regulation of serotonin-S2 and dopamine-D2 receptors in rat brain following chronic receptor blockade.
Topics: Animals; Apomorphine; Behavior, Animal; Corpus Striatum; Diazepam; Dopamine Antagonists; Frontal Lobe; Gene Expression Regulation; Ketanserin; Male; Models, Biological; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin Antagonists; Tryptamines | 1987 |
Effects of tryptamine antagonists on the anaphylactic contractions of the bovine pulmonary smooth muscles.
Topics: Anaphylaxis; Animals; Cattle; Horses; In Vitro Techniques; Ketanserin; Lung; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Pulmonary Artery; Pulmonary Veins; Serotonin Antagonists; Trachea; Tryptamines | 1984 |
Inhibitory effects of tryptamine on tolbutamide-induced hypoglycemia in mice: mediation by 5-HT receptors.
Topics: Animals; Blood Glucose; Hypoglycemia; Indoles; Ketanserin; Male; Methysergide; Mice; Mice, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Time Factors; Tolbutamide; Tropisetron; Tryptamines | 1994 |
Mutations of transmembrane IV and V serines indicate that all tryptamines do not bind to the rat 5-HT2A receptor in the same manner.
Topics: Amino Acid Sequence; Amino Acid Substitution; Amphetamines; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Ergolines; Ketanserin; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Protein Structure, Secondary; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Recombinant Proteins; Serine; Serotonin; Serotonin Antagonists; Tryptamines | 1997 |