ketanserin and sb 269970

ketanserin has been researched along with sb 269970 in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's8 (66.67)29.6817
2010's4 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA1
Berardi, F; Colabufo, NA; Contino, M; Lacivita, E; Leopoldo, M; Perrone, R1
Berardi, F; Caroli, A; Colabufo, NA; Contino, M; De Giorgio, P; Di Pilato, P; Hedlund, PB; Lacivita, E; Leopoldo, M; Niso, M; Patarnello, D; Perrone, R; Stroth, N; Svenningsson, P1
Bienkowski, P; Bucki, A; Jaśkowska, J; Kazek, G; Kowalski, P; Kołaczkowski, M; Marcinkowska, M; Mierzejewski, P; Mitka, K; Pawłowski, M; Siwek, A; Wasik, A; Wesołowska, A1
Lepailleur, A; Rochais, C; Thirumaran, SL1
Ge, L; Naylor, RJ; Tuladhar, BR1
Ben Mabrouk, F; Pearlstein, E; Pflieger, JF; Vinay, L1
Pericić, D; Strac, DS; Vlainić, J1
Dogrul, A; Seyrek, M1
Komada, T; Yano, S1
Cao, J; Iwamoto, T; Kadota, K; Kitazawa, T; Nakamura, T; Taneike, T; Teraoka, H1
Castor, MG; Diniz, DA; Duarte, ID; Navarro, LC; Perez, AC; Petrocchi, JA; Romero, TR; Souza, TC1

Reviews

2 review(s) available for ketanserin and sb 269970

ArticleYear
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003
Structure-activity relationships of serotonin 5-HT
    European journal of medicinal chemistry, 2019, Dec-01, Volume: 183

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

2019

Other Studies

10 other study(ies) available for ketanserin and sb 269970

ArticleYear
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides, a class of 5-HT7 receptor agents. 2.
    Journal of medicinal chemistry, 2007, Aug-23, Volume: 50, Issue:17

    Topics: Amides; Animals; Cell Line; Guinea Pigs; Humans; Ileum; Male; Muscle Contraction; Muscle, Smooth; Piperazines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship; Tetrahydronaphthalenes

2007
Investigations on the 1-(2-biphenyl)piperazine motif: identification of new potent and selective ligands for the serotonin(7) (5-HT(7)) receptor with agonist or antagonist action in vitro or ex vivo.
    Journal of medicinal chemistry, 2012, Jul-26, Volume: 55, Issue:14

    Topics: Animals; Guinea Pigs; HeLa Cells; Humans; Ileum; Ligands; Models, Molecular; Molecular Weight; Piperazine; Piperazines; Protein Conformation; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Substrate Specificity

2012
Novel arylsulfonamide derivatives with 5-HT₆/5-HT₇ receptor antagonism targeting behavioral and psychological symptoms of dementia.
    Journal of medicinal chemistry, 2014, Jun-12, Volume: 57, Issue:11

    Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Avoidance Learning; Benzoxazoles; Catalepsy; CHO Cells; Cricetulus; Dementia; Dopamine D2 Receptor Antagonists; HEK293 Cells; Humans; Male; Models, Molecular; Motor Activity; Radioligand Assay; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Sulfonamides

2014
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides

2003
Serotonin refines the locomotor-related alternations in the in vitro neonatal rat spinal cord.
    The European journal of neuroscience, 2005, Volume: 21, Issue:5

    Topics: Animals; Animals, Newborn; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fenclonine; Functional Laterality; In Vitro Techniques; Ketanserin; Motor Activity; N-Methylaspartate; Phenols; Rats; Serotonin; Serotonin Antagonists; Spinal Cord; Statistics as Topic; Sulfonamides

2005
Zimelidine decreases seizure susceptibility in stressed mice.
    Journal of neural transmission (Vienna, Austria : 1996), 2006, Volume: 113, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anticonvulsants; Behavior, Animal; Convulsants; Ketanserin; Male; Mianserin; Mice; Mice, Inbred CBA; Phenols; Picrotoxin; Piperazines; Pyridines; Seizures; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Stress, Psychological; Sulfonamides; Swimming; Zimeldine

2006
Systemic morphine produce antinociception mediated by spinal 5-HT7, but not 5-HT1A and 5-HT2 receptors in the spinal cord.
    British journal of pharmacology, 2006, Volume: 149, Issue:5

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Injections, Spinal; Ketanserin; Male; Metergoline; Mice; Mice, Inbred BALB C; Morphine; Pain; Pain Measurement; Phenols; Piperazines; Pyridines; Reaction Time; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin; Receptors, Serotonin, 5-HT2; Serotonin Antagonists; Spinal Cord; Sulfonamides

2006
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
    Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:3

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin

2007
Excitatory and inhibitory 5-hydroxytryptamine (5-HT) receptors expressed in the isolated porcine uterine muscles.
    European journal of pharmacology, 2008, Dec-14, Volume: 600, Issue:1-3

    Topics: Animals; Dose-Response Relationship, Drug; Female; Gene Expression; Immunohistochemistry; Ketanserin; Phenols; Polymerase Chain Reaction; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Sulfonamides; Swine; Uterine Contraction

2008
Serotonin induces peripheral mechanical antihyperalgesic effects in mice.
    European journal of pharmacology, 2015, Nov-15, Volume: 767

    Topics: Animals; Biphenyl Compounds; Dinoprostone; Dose-Response Relationship, Drug; Hyperalgesia; Ketanserin; Male; Mice; Ondansetron; Pain Measurement; Phenols; Piperazines; Propanolamines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides

2015