ketanserin and pirenperone

ketanserin has been researched along with pirenperone in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-199016 (69.57)18.7374
1990's6 (26.09)18.2507
2000's1 (4.35)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA1
Janssen, CG; Laduron, PM; Thijssen, JB; Van Dun, J; Wouters, W1
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
DeNoble, KF; DeNoble, VJ; Reigel, AL; Schrack, LM1
Gorzalka, BB; Watson, NV1
Bodnar, RJ; Kiefel, JM; Paul, D1
Appel, JB; Cunningham, KA; Ginn, SR; Nielsen, EB1
Pranzatelli, MR; Snodgrass, SR1
Creba, JA; Doyle, VM; Hoyer, D; Rüegg, UT1
Gorzalka, BB; Mendelson, SD3
Gudelsky, GA; Koenig, JI; Meltzer, HY1
Mana, MJ; Paul, D; Pfaus, JG; Pinel, JP1
Altman, HJ; Normile, HJ1
Neal, BS; Sparber, SB1
Taylor, DA; Yap, CY1
Glennon, RA; Rosecrans, JA; Young, R1
Gudelsky, GA; Meltzer, HY; Simonovic, M1
Dykstra, LA; Lin, YP; Powell, KR1
Holtzman, SG; Steinfels, GF1
Colpaert, FC; John, GW; Le Grand, B; Patoiseau, JF; Rieu, JP; Talmant, JM1

Reviews

1 review(s) available for ketanserin and pirenperone

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987

Other Studies

22 other study(ies) available for ketanserin and pirenperone

ArticleYear
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Frontal Lobe; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1986
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
    British journal of pharmacology, 1997, Volume: 122, Issue:1

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid

1997
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Visual recognition memory in squirrel monkeys: effects of serotonin antagonists on baseline and hypoxia-induced performance deficits.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:4

    Topics: Animals; Avoidance Learning; Cognition; Dose-Response Relationship, Drug; Hypoxia; Ketanserin; Male; Memory; Mianserin; Piperidines; Psychomotor Performance; Reinforcement Schedule; Saimiri; Serotonin Antagonists

1991
DOI-induced inhibition of copulatory behavior in male rats: reversal by 5-HT2 antagonists.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:3

    Topics: Amphetamines; Animals; Copulation; Ejaculation; Female; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Tranquilizing Agents

1991
Reduction in opioid and non-opioid forms of swim analgesia by 5-HT2 receptor antagonists.
    Brain research, 1989, Oct-23, Volume: 500, Issue:1-2

    Topics: Analgesia; Endorphins; Ketanserin; Methysergide; Physical Exertion; Piperidines; Receptors, Serotonin; Serotonin Antagonists

1989
Antagonism of the LSD cue by putative serotonin antagonists: relationship to inhibition of in vivo [3H]spiroperidol binding.
    Behavioural brain research, 1985, Volume: 16, Issue:2-3

    Topics: Animals; Cerebellum; Corpus Striatum; Frontal Lobe; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Pizotyline; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin

1985
Antimyoclonic properties of S2 serotonin receptor antagonists in the rat.
    Neuropharmacology, 1986, Volume: 25, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Brain Chemistry; Butyrophenones; Cinanserin; Ketanserin; Male; Myoclonus; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1986
Serotonin increases the production of inositol phosphates and mobilises calcium via the 5-HT2 receptor in A7r5 smooth muscle cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:2

    Topics: Animals; Aorta; Calcium; Cell Line; Cerebral Cortex; Inositol Phosphates; Ketanserin; Kinetics; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sugar Phosphates; Time Factors

1986
Harmine reverses the inhibition of lordosis by the 5-HT2 antagonists pirenperone and ketanserin in the female rat.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:1

    Topics: Alkaloids; Animals; Estradiol; Female; Harmine; Ketanserin; Ovariectomy; Piperidines; Posture; Progesterone; Rats; Rats, Inbred Strains; Receptors, Serotonin; Sexual Behavior, Animal

1986
Thermoregulatory responses to serotonin (5-HT) receptor stimulation in the rat. Evidence for opposing roles of 5-HT2 and 5-HT1A receptors.
    Neuropharmacology, 1986, Volume: 25, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature Regulation; Ketanserin; Male; Methoxydimethyltryptamines; Pindolol; Piperidines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes

1986
Serotonin antagonist pirenperone inhibits sexual behavior in the male rat: attenuation by quipazine.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Fenclonine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Serotonin Antagonists; Sexual Behavior, Animal; Tranquilizing Agents

1985
A facilitatory role for serotonin in the sexual behavior of the female rat.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:6

    Topics: Animals; Castration; Estradiol; Female; Ketanserin; Methysergide; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Sexual Behavior, Animal; Spiperone

1985
Attenuation of morphine analgesia by the S2 antagonists, pirenperone and ketanserin.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:3

    Topics: Analgesia; Animals; Dose-Response Relationship, Drug; Ketamine; Ketanserin; Male; Morphine; Piperidines; Rats; Reaction Time; Receptors, Serotonin; Serotonin Antagonists

1988
Different temporal effects of serotonergic antagonists on passive avoidance retention.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:3

    Topics: Animals; Avoidance Learning; Ketanserin; Male; Memory; Mianserin; Mice; Piperidines; Receptors, Serotonin; Retention, Psychology; Serotonin Antagonists; Time Factors

1987
Ketanserin and pirenperone attenuate acute morphine withdrawal in rats.
    European journal of pharmacology, 1986, Dec-16, Volume: 132, Issue:2-3

    Topics: Animals; Body Temperature; Conditioning, Operant; Ketanserin; Male; Morphine Dependence; Piperidines; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome

1986
Involvement of 5-HT2 receptors in the wet-dog shake behaviour induced by 5-hydroxytryptophan in the rat.
    Neuropharmacology, 1983, Volume: 22, Issue:7

    Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Female; Ketanserin; Methysergide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1983
Antagonism of the effects of the hallucinogen DOM and the purported 5-HT agonist quipazine by 5-HT2 antagonists.
    European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

    Topics: Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists

1983
Effects of pirenperone and ketanserin on rat prolactin secretion in vivo and in vitro.
    European journal of pharmacology, 1983, Aug-19, Volume: 92, Issue:1-2

    Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin Antagonists; Tranquilizing Agents

1983
Antinociceptive effects of the kappa opioid, U50,488: lack of modulation by 5-HT2 antagonists.
    Psychopharmacology, 1993, Volume: 112, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Ergolines; Ketanserin; Male; Piperidines; Pyrrolidines; Receptors, Opioid, kappa; Saimiri; Serotonin Antagonists

1993
Monoamine systems in the discriminative effects of spiradoline, a kappa-opioid agonist.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Analgesics; Animals; Avoidance Learning; Biogenic Monoamines; Discrimination, Psychological; Dopamine Antagonists; Fenfluramine; Fluoxetine; Generalization, Stimulus; Ketanserin; Male; Piperidines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Selective Serotonin Reuptake Inhibitors; Serotonin; Synaptic Transmission

1994
Investigation of the mechanism by which ketanserin prolongs the duration of the cardiac action potential.
    Journal of cardiovascular pharmacology, 1995, Volume: 26, Issue:5

    Topics: Action Potentials; Amphetamines; Animals; Guinea Pigs; Heart; Ketanserin; Male; Piperidines; Potassium Channels; Serotonin Antagonists

1995