ketanserin and piperidines

ketanserin has been researched along with piperidines in 564 studies

Research

Studies (564)

TimeframeStudies, this research(%)All Research%
pre-1990468 (82.98)18.7374
1990's49 (8.69)18.2507
2000's36 (6.38)29.6817
2010's11 (1.95)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berardi, F; Daniele, E; Govoni, S; Leopoldo, M; Lograno, MD; Perrone, R; Tortorella, V1
Bowden, CR; De Coster, R; Heykants, J; Voina, SJ; Woestenborghs, R1
Emilsson, K; Hardebo, JE; Nystedt, S; Owman, C; Szabò, C1
Karnovsky, ML; Polanski, M1
Brazell, C; Campbell, IC; Mitchell, S; Stahl, SM; Twist, EC1
Arora, RC; Meltzer, HY; Nash, JF; Schreiber, MA1
Appell, KC; Barrett, RJ; Kilpatrick, BF; Nolan, JC; Proakis, AG; Walsh, DA1
DeNoble, KF; DeNoble, VJ; Reigel, AL; Schrack, LM1
Gorzalka, BB; Watson, NV1
Beczkowska, IW; Bodnar, RJ1
Beubler, E; Coupar, IM; Hardcastle, J; Hardcastle, PT1
Bird, ED; Crino, PB; Plager, MD; Vogt, BA1
Nakamura, H; Suzukawa, M1
Bennett, DA; Glaeser, BS; Hutchison, AJ; Liebman, JM; Lovell, RA; Sills, MA; Williams, M; Wood, PL1
Broekkamp, CL; Jenck, F; Van Delft, AM1
Dewar, KM; Lima, L; Reader, TA1
Glowinski, J; Godbout, R; Mantz, J; Tassin, JP; Thierry, AM1
Cohen, ML; Mann, JJ; McBride, PA; Nimchinsky, E1
Geyer, MA; Tapson, GS; Wing, LL1
Backus, LI; Grahame-Smith, DG; Sharp, T1
Demetrikopoulos, MK; Flaherty, CF; Grigson, PS; Krauss, KL; Rowan, GA; Weaver, MS1
Bertocci, B; Cesura, AM; Da Prada, M1
Jackson, DA; White, SR1
Cowen, PJ; Gartside, SE1
Campbell, AM; Glatfelter, A; Kunkel, RG; Ulevitch, RJ; Wiggins, RC1
Ahlman, H; Dahlström, A; Lidberg, P2
Delius, W; Dominiak, P; Gessler, I; Grobecker, H; Kees, F1
Vanhoutte, PM1
Gradin, K; Hedner, T; Persson, B; Pettersson, A4
Gradin, K; Hedner, T; Henning, M; Persson, B; Pettersson, A1
Markus, JK; Mylecharane, EJ; Phillips, CA; Shaw, J2
Coghlan, JP; Denton, DA; Mills, EH; Nelson, MA; Scoggins, BA; Spence, CD; Whitworth, JA1
Baudouin-Legros, M; Guicheney, P; Kamal, LA; Le Quan-Bui, KH; Meyer, P1
Ball, SG; Robertson, JI1
Ball, SG; Robertson, JI; Zabludowski, JR2
De Crée, J; De Ryck, M; Hoing, M; Symoens, J1
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; Staessen, J1
Boomsma, F; Man in't Veld, AJ; Schalekamp, MA; Wenting, GJ; Woittiez, AJ1
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; Rorive, G; Staessen, J1
Berglund, G; Hedner, T; Persson, B4
Brown, SA; Simpson, FO; Spears, GF; Waal-Manning, HJ1
Fasano, ML; Ferrara, LA; Mancini, M; Marotta, G; Rubba, P; Soro, S1
Hedner, T; Persson, B3
Ayres, B; Bune, AJ; Chalmers, JP; Graham, JR; West, MJ; Wing, LM2
Kincaid-Smith, P; Murphy, BF; Whitworth, JA1
Armanini, D; Boscaro, M; D'Agostino, D; Mantero, F; Opocher, G; Rocco, S2
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; Staessen, J; Vanhees, L1
Amery, A; Arnout, J; Deckmyn, H; Fiocchi, R; Lijnen, P; Van Russelt, M; Vermylen, J1
De Clerck, F; Xhonneux, B2
De Cree, J; Demoen, B; Leempoels, J; Roels, V; Verhaegen, H2
Brimichová, G; Dzúrik, R; Fetkovská, N; Tison, P2
Freitag, B; Pointel, JP; Schmitt, C; Stoltz, JF; Voisin, P; Zannad, F1
Bogar, L; Dormandy, JA; Matrai, A; Walker, RT1
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; M'Buyamba-Kabangu, JR; Staessen, J1
De Cree, J; Demoen, B; Leempoels, J; Verhaegen, H1
Van Nueten, JM2
Arnold, G; Breuer, J; Meschig, R1
Ahlman, H; Boström, S; Dahlström, A; Vällfors, B1
Arnold, G; Breuer, HW; Breuer, J; Meschig, R1
Marwood, JF; Stokes, GS1
Opie, LH; Saman, S; Thandroyen, F1
Kaumann, AJ2
Ahlman, H; Dahlström, A; Grönstad, K; Jaffe, BM; Nilsson, O; Oberg, K1
Hollenberg, NK1
De Cree, J; Geukens, H; Leempoels, J; Verhaegen, H2
Gush, R; Jayson, MI; Longstaff, J; Williams, EH1
Amery, A; Fagard, R; Laermans, M; Lijnen, P; Lommelen, L; M'Buyamba-Kabangu, JR; Piccart, Y; Staessen, J1
Hirokami, M; Minami, M; Saito, H; Sano, M; Tochihara, M; Togashi, H; Yoshioka, M1
Marsden, CA; Martin, KF1
Altar, CA; Boyar, WC; Marien, MR1
Casthely, PA; Ergin, MA; Goodman, K; Griepp, RB; Jablons, M1
Kienast, J; Verstraete, M1
Coker, SJ; Ellis, AM1
Ball, SG; Robertson, JI; Stott, DJ1
Ball, SG; Hosie, J; Robertson, JI; Stott, DJ1
Cohen, ML; Kurz, KD; Schenck, KW1
Ramage, AG2
Reneman, RS; van der Starre, PJ1
Brunello, N; Galimberti, R; Racagni, G; Riva, M; Rovescalli, AC1
Blauw, GJ; Chang, PC; van Brummelen, P; van Zwieten, PA; Vermeij, P1
Lund, N; Thorborg, P1
Bloomquist, WL; Cohen, ML; Fuller, RW; Snoddy, HD1
Arnt, J; Hyttel, J1
Koshikawa, N; Maruyama, Y; Stephenson, JD1
Chau, NP; Levenson, J; Pithois-Merli, I; Simon, AC1
Ahlman, H; Dahlström, A; Grönstad, K; Jaffe, BM; Oberg, K; Tisell, LE; Zinner, MJ1
Altar, CA; Marshall, JF; O'Neil, S; Walter, RJ1
Frimodt-Møller, C; Hørby-Petersen, J; Mathiesen, FR; Meyhoff, HH; Schmidt, PF1
Bodnar, RJ; Kiefel, JM; Paul, D1
Alling, C; Hansson, E; Simonsson, P1
Gommeren, W; Janssen, PF; Laduron, PM; Leysen, JE; Van Gompel, P; Wynants, J1
Berglund, G; Hedner, T; Persson, B; Pettersson, A1
Andersen, D; Bech, K; Ladegaard, L1
Buchman, O; Grigoriadis, DE; Niznik, HB; Pri-Bar, I; Seeman, P1
Arroyo, JL; Carrasco, MS; De Castro, J; Esteban, J; Sanchez, G1
Aono, J; Ishizuka, N; Nabata, H; Sakai, K1
Andree, TH; Koenig, JI; Meltzer, HY; Mikuni, M; Tong, CY1
Berent, A; Bounameaux, H; Hellemans, H; Holditch, T; Verhaeghe, R1
Assogna, G; Di Lorenzo, M; Feo, B; Pompa, D1
Ramsay, LE1
Ogren, SO1
Greiner, HE; Haase, A; Klockow, M; Schmitges, CJ; Seyfried, C1
Breckenridge, A1
Man in 't Veld, AJ; Schalekamp, MA; van den Meiracker, AH; Wenting, GJ; Woittiez, AJ1
Fisher, R; Gruebel, B; Koehle, W; Rosenthal, J1
Batink, HD; Boddeke, E; Doods, HN; Hugtenburg, JG; Korstanje, C; Sprenkels, R; Thoolen, MJ; Van Zwieten, PA1
Altar, CA; Neale, RF; Stone, GA; Wasley, AM1
Cameron, CM; Cameron, HA; Ramsay, LE1
Di Chiara, G; Longoni, R; Spina, L1
Hedner, T; Persson, B; Pettersson, A2
Hewson, G; Hill, RG; Hughes, J; Leighton, GE1
Knuppel, RA; Montenegro, R; O'Brien, WF; Shah, D1
Appel, JB; Cunningham, KA; Ginn, SR; Nielsen, EB1
Arnt, J1
Mylecharane, EJ; Phillips, CA; Shaw, J1
Laduron, PM; Leysen, JE; Van Dun, J; Wouters, W4
Heiligers, J; Mylecharane, EJ; Saxena, PR1
Janssens, WJ; Van Nueten, JM; Vanhoutte, PM1
Parag, KB; Seedat, YK1
Houvenaghel, A; Schrauwen, E1
Beck, SG; Clarke, WP; Goldfarb, J1
Auer, LM; Leber, K; Sayama, I1
Grekin, RJ; Gross, MD; Shenker, Y1
Apelian, A; Jageneau, AH; Khachadurian, AK; Schneider, SH; Tendler, M1
Barrett, JE; Brady, LS1
Lawang, A; Saxena, PR1
Skolnick, P; Weissman, BA; Youdim, MB1
Feniuk, W; Humphrey, PP; Perren, MJ; Watts, AD1
Gomar, C; Luis, M; Nalda, MA1
Demling, RH; Fox, R; Hechtman, H; Huval, W; Wong, C1
Jähnchen, E; Lühr, A; Radkow, N; Trenk, D1
De Roe, C; Laduron, PM; Luabeya, MK; Maloteaux, JM; Trouet, A1
Battaglia, G; Creese, I; Newton, PL; Norman, AB1
Clineschmidt, BV; Pettibone, DJ; Reiss, DR; Robinson, JL1
Gorzalka, BB; Mendelson, SD4
Ei-Fawal, HA; Eyre, P; Gordon, V; Ogunbiyi, PO1
Hoffmann, D; Wesemann, W2
Allegra, C; Assogna, G; Bonifacio, M; Mari, A; Tonelli, V1
Assogna, G; Attilia, ML; Cavalieri, G; Ceccanti, M; De Lorenzo, A; Romeo, M1
Colli, R; Di Giovanni, V1
Forler, C; Fozard, JR; Middlemiss, DN; Tricklebank, MD1
Engel, G; Hoyer, D; Kalkman, HO2
Man in't Veld, AJ; Ritsema van Eck, HJ; Schalekamp, MA; van den Meiracker, AH; Wenting, GJ; Woittiez, AJ; Zantvoort, FA1
Porter, JM; Taylor, LM1
Kellar, KJ; Stockmeier, CA2
Agid, Y; Baron, JC; Comar, D; Crouzel, C; Deniker, P; Samson, Y1
De Clerck, F; Janssen, PA; Tollenaere, JP; Xhonneux, B1
Biegon, A; Kargman, S; McEwen, BS; Snyder, L1
Ashton, JH; Benedict, CR; Buja, LM; Campbell, WB; Fitzgerald, C; Raheja, S; Taylor, A; Willerson, JT1
Cernohorský, D; Hamet, A; Král, B1
Engel, G; Göthert, M; Hillenbrand, K; Hoyer, D; Schlicker, E1
Hibert, M; Middlemiss, DN1
Barrett, JE; Mansbach, RS1
Pranzatelli, MR; Snodgrass, SR1
Dusting, GJ; Li, DM1
Connor, HE; Feniuk, W; Humphrey, PP; Perren, MJ1
Attilia, ML; Berbellini, A; Cavaleri, G; Ceccanti, M; De Lorenzo, A; Di Giovanni, MG; Pisculli, M; Santini, P1
Assogna, G; Ceccanti, M; De Lorenzo, A; Di Giovanni, MG; Lais, A; Pisculli, M; Romeo, M; Valgiusti, FC1
Ganey, PE; Hadley, KB; Roth, RA; Sprugel, KH1
Hald, A; Ording, H; Sjøntoft, E1
Eberlein, HJ; Schulte-Sasse, U1
Murrin, LC; Zeng, W1
Abrignani, MG; Alaimo, G; Cutietta, A; Novo, S; Raineri, A; Strano, A1
Harinck-de Weerd, JE; Reneman, RS; van der Starre, PJ1
Armstrong, ML; Heistad, DD; Marcus, ML; Mark, AL; Piegors, DJ1
Lüscher, TF; Vanhoutte, PM1
Zanchetti, A1
Janssens, WJ; Van Nueten, JM1
Gordin, A; Saraste, K; Sundberg, S; Turanlahti, M1
Gould, SE; Kane, JA; Sibbald, B; Tooley, M1
Kirch, W; Ohnhaus, EE1
Mauersberger, H1
Bernardiner, E; Lemus, J; Milei, J1
Assogna, G; Costantini, C; del Rosso, G; Libretti, A; Mara, G; Palermo, A; Pizza, N1
Dona, G; Ribeiro, A; Tammaro, AE1
de Jong, PE; de Zeeuw, D; Navis, G; van der Hem, GK1
Andersson, O; Berglund, G; Hedner, T; Persson, B; Petterson, A1
Cohen, RA1
Göthert, M; Kollecker, P; Schlicker, E1
Bergstrom, DA; Carlson, JH; Walters, JR1
Hösli, E; Hösli, L1
Conn, PJ; Hartig, PR; Hoffman, BJ; Sanders-Bush, E1
Arnout, J; De Clerck, F; Deckmyn, H; Vermylen, J; Xhonneux, B1
Boas, RA1
Berges, LC; Cruz, J; Feltkamp, H; Finkielman, S; Geyer, G; Milei, J; Moscovici, H; Silva, AN; Stumpe, KO1
Hoyer, D; Palacios, JM; Pazos, A; Probst, A1
Marwood, JF; Mennie, BA; Stokes, GS1
Bjertnaes, L; Helgesen, KG1
Seibold, JR; Terregino, CA1
Iida, H; Ikeda, K; Mikawa, M; Mizumura, Y; Sugimoto, T; Takata, M; Tomoda, F; Zhang, X1
Ahlman, H; Dahlström, A; Grönstad, KO; Jaffe, BM1
Bennett, A; Cashman, JN; Thompson, MA1
Carter, JA; Houghton, K1
Hoekman, TB; Howlett, SE; Triggle, CR1
Bottaro, D; Hechtman, HB; Peterson, S; Shepro, D2
Engisch, KL; Wenk, GL1
Ferrara, A; Jaffe, BM; Sherlock, DJ1
Skotnicki, SH; van de Wal, HJ; van Lier, HJ; Wijn, PF1
Arvidsson, S; Bergqvist, D; Haglund, U; Hedner, U; Lindblad, B1
Lagerkvist, BE; Linderholm, H1
Hall, H; Wedel, I1
Hulme, VA; Odendaal, HJ1
Jarvis, LG; Setchell, BP; Sowerbutts, SF1
Leff, P; Martin, GR1
Abrignani, MG; Adamo, L; Alaimo, G; Avellone, G; Cutietta, A; Giordano, U; Indovina, A; Novo, S; Pinto, A; Strano, A1
Kaumann, AJ; Lemoine, H1
Creba, JA; Doyle, VM; Hoyer, D; Rüegg, UT1
Banay-Schwartz, M; Lajtha, A; Manigault, I; Wajda, IJ1
Lin, MT; Tsai, ML1
Foray, J; Hagege, A; Housset, E; Priollet, P; Vayssairat, M1
Glennon, RA1
Hladovec, J2
Delbro, D; Nordström, O1
Griffiths, HB; Whitwam, JG2
Gudelsky, GA; Koenig, JI; Meltzer, HY1
Laruelle, M; Maloteaux, JM; Vanisberg, MA1
Altar, CA; Marien, MR1
Kobayashi, M; Koshikawa, N; Maruyama, Y; Mori, E; Nomura, H; Oka, K; Stephenson, JD1
Barbaccia, ML; Costa, E; Gandolfi, O2
Gordin, A; Mustajoki, P; Pelkonen, R1
Kendall, DA; Nahorski, SR1
Goto, A; Ishii, M; Matsuoka, H; Sugimoto, T1
Godfrey, PP; McClue, SJ; Minchin, MC; Schächter, M; Young, MM1
Bockaert, J; Kemp, DE; Sebben, M; Weiss, S1
Kawasaki, H; Takasaki, K1
Linthicum, DS; Simmons, RD1
Candeletti, S; Ferri, S; Romualdi, P; Spadaro, C; Spampinato, S1
Gommeren, W; Janssen, PA; Leysen, JE; Van Gompel, P; Woestenborghs, R1
Byrne, JH; Ocorr, KA1
Jandhyala, BS; Kivlighn, SD1
Laguzzi, R; Shvaloff, A1
Coghlan, JP; Denton, DA; Nelson, M; Scoggins, BA; Tresham, JJ; Whitworth, JA1
Furukawa, H; Ishikawa, K; Kameyama, T; Nabeshima, T; Yamaguchi, K1
Smits, J; Struyker Boudier, H; van Dorsten, F1
Geyer, MA; Tapson, GS1
Arneklo-Nobin, B; Owman, C1
Hole, DR; Hunter, AJ; Wilson, CA1
Houston, DS; Shepherd, JT; Vanhoutte, PM1
Bieger, D; Triggle, C1
Erne, P; Pletscher, A1
Jennewein, HM; Mierau, J; Saxena, PR; Verdouw, PD1
Affolter, H; Burkard, WP; Pletscher, A1
Appel, JB; Callahan, PM; Cunningham, KA1
Frenken, M; Kaumann, AJ3
Kayaba, K; Kimura, M; Kiyono, S; Koyama, S; Nishizawa, M1
Hayashi, T; Ichida, S; Kita, T; Murakami, T1
Grigoriadis, D; Seeman, P1
Olesen, SP1
Anwyl, R; Rowan, MJ1
Fasano, ML; Ferrara, LA; Iannuzzi, A; Rubba, P; Soro, S1
Karasawa, A; Kubo, K; Nakamizo, N; Shuto, K1
Aghajanian, GK; Lakoski, JM1
de Aguiar, JC; Graeff, FG; Schütz, MT1
Bevan, J; Heptinstall, S2
Bradley, PB; Humphrey, PP; Williams, RH1
Comar, D; Maziere, M; Turner, JH1
Klotz, U; Ratge, D; Reimann, IW; Wisser, H1
Koshikawa, N; Smokcum, RW; Stephenson, JD1
Buczko, W1
Beetens, J; De Clerck, F; Reneman, RS; Van Gorp, L1
Burns, EC; Dillon, MJ; Dunger, DB1
Heiligers, J; Mylecharane, EJ; Saxena, PR; Tio, R1
Kurowski, M2
Frost, JJ; Hartig, PR; Scheffel, U; Wagner, HN1
Hechtman, DH; Jageneau, A1
Glaser, T; Traber, J1
Clarke, KA; Parker, AJ; Stirk, GC1
Cameron, HA; Ramsay, LE1
Doğan, N; Ilhan, M; Kayaalp, SO; Tuncer, M1
Reneman, S; van de Water, A; Wouters, L; Xhonneux, R1
Cowen, KJ; McGourty, JC; Silas, JH1
Kilbinger, H; Pfeuffer-Friederich, I1
Brimichová, E; Dzúrik, R; Gerová, Z1
Kwan, S; Lam, WK; So, SY1
De Meirleir, K; Hollmann, W; L'Hermite, M; L'Hermite-Balériaux, M; Rost, R1
Burvenich, C; Peeters, G; Vandeputte-Van Messon, G1
Demenge, P; Feuerstein, C; Guerin, B; Mouchet, P; Silice, C1
Nishino, N; Tanaka, C1
Mana, MJ; Paul, D; Pfaus, JG; Pinel, JP1
de Chaffoy de Courcelles, D; Leysen, JE; Niemegeers, CJ; Van Gompel, P1
Altman, HJ; Normile, HJ1
Janssen, CG; Laduron, PM; Thijssen, JB; Van Dun, J; Wouters, W1
Neal, BS; Sparber, SB1
Marcelle, R1
Bounameaux, HM; Hellemans, H; Verhaeghe, R1
Brimichová, G; Dzúrik, R; Petkovská, N; Tison, P1
Cooper, SJ; Cross, AJ; Crow, TJ; Deakin, JF; Ferrier, IN; Johnson, JA; Joseph, MH; Lofthouse, R; Owen, F; Poulter, M1
Laduron, PM; Luabeya, MK; Maloteaux, JM1
Prescott, RW; Ratcliffe, WA; Taylor, PK1
Beubler, E; Bukhave, K; Rask-Madsen, J1
Amery, A; Groeseneken, D; Laermans, M; Lijnen, P; Lommelen, L; Piccart, Y1
Battaglia, G; Borgundvaag, B; Shannon, M; Titeler, M2
Van Nueten, JM; Vanhoutte, PM2
Edwards, CR; Shaikh, S; Williams, BC1
De Cree, J; Symoens, J; Verhaegen, H1
Bertholet, M; David, JL; Demoulin, JC; Kulbertus, HE; Soumagne, D1
Janssen, PA; Van Beek, J; Van Nueten, JM; Vanhoutte, PM; Verbeuren, TJ; Xhonneux, R1
Ilien, B; Laduron, PM; Schotte, A1
de Roose, J; Symoens, J1
Hedner, T; Henning, M; Persson, B1
Feniuk, W; Humphrey, PP; Watts, AD1
Facoory, BD; Laverty, R; Millar, JA1
Leysen, JE; Schuurkes, JA; Van Nueten, JM; Vanhoutte, PM1
Frölich, JC; Reimann, IW1
Iversen, LL; Reynolds, GP; Rossor, MN1
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; Staessen, J; Vermylen, J1
Helmeste, DM; Tang, SW2
Anger, C; Lawin, P; Puchstein, C; Thijs, J; Van Aken, H1
Timmermans, PB; van Zwieten, PA1
McGoon, MD; Vlietstra, RE1
Timmermans, PB; Van Brummelen, P; Van Zwieten, PA1
Barradas, MA; Dandona, P; Fonseca, V; Jeremy, JY; Mikhailidis, DP; Ramage, AG1
Arnold, R; Koop, H1
Humphrey, PP1
Adams, CB; Boullin, DJ; Kaye, AH; Schachter, M; Tagari, PC; Teddy, PJ1
Lagneaux, D; Lecomte, J2
Cheney, DL; Costa, E; Gandolfi, O; Hong, JS1
Bloom, SR; Corsellis, JA; Cross, AJ; Crow, TJ; Ferrier, IN; Johnson, JA1
David, JL; de Clerck, F; Janssen, PA1
de Chaffoy de Courcelles, D; Roevens, P; van Belle, H1
Barnett, DB; Cook, N; Jennings, PE; O'Malley, BP; Rosenthal, FD1
Buczko, W; De Gaetano, G; Gambino, MC1
Awouters, F; Janssen, PA; Kennis, L; Laduron, PM; Leysen, JE; Vandenberk, J1
Kalkman, HO; Timmermans, PB; Van Zwieten, PA1
Janssen, PA; Symoens, J; Van Nueten, JM; Vanhoutte, PM1
Opie, LH1
Battaglia, G; Shannon, M; Titeler, M3
Schalekamp, MA; Wenting, GJ1
McCall, RB; Schuette, MR1
Kendall-Taylor, P; Prescott, RW; Ratcliffe, WA; Watson, MJ; Weightman, DR1
Vincent, JL1
Eyre, P; Ogunbiyi, PO2
Köhler, C2
Bianconi, M; Degli Uberti, EC; Margutti, AR; Pansini, P; Rotola, CA; Trasforini, G1
Andrén, L; Dahlöf, B; Eggertsen, R; Hansson, L; Svensson, A1
Leysen, JE; Niemegeers, CJ; Van Gompel, P; Verwimp, M1
Arvidsson, S; Falk, A; Haglind, E; Haglund, U1
Ball, HA; Parratt, JR; Rodger, IW1
Amery, A; de Schaepdryver, A; Fagard, R; Fiocchi, R; Lijnen, P; Moerman, E; Staessen, J1
Jageneau, AH; Seibold, JR1
Socol, ML; Vaisrub, N; Weiner, CP1
Arvidsson, S; Bergqvist, D; Esquivel, C; Fält, K; Haglund, U; Lindblad, B; Lindström, C1
Hechtman, HB; Shepro, D; Valeri, CR1
Feniuk, W1
de Chaffoy de Courcelles, D; De Clerck, F; Leysen, JE; Niemegeers, CJ; Van Nueten, JM1
De Clerck, F; Reneman, RS; van Nueten, JM1
Anthony, M1
Bosin, TR; Mais, DE1
Roald, OK; Seem, E1
Cox, NH; Dufton, PA1
Ernst, E; Matrai, A1
McGoon, MD; Vanhoutte, PM1
Battaglia, G; Glennon, RA; Shannon, M; Titeler, M1
Glennon, RA; McKenney, JD; Young, R1
Conn, PJ; Sanders-Bush, E1
De Clerck, F; De Gryse, A; Loots, W; Nevelsteen, A1
Lauwers, F; Van Den Broeck, C; Verheyen, A; Vlaminckx, E; Wouters, L1
Kirby, GC; McQueen, DS1
Finch, CE; Marcusson, JO; Morgan, DG; Winblad, B1
Apprill, P; Ashton, J; Buja, LM; Bush, LR; Campbell, WB; Kern, K; Schmitz, J; Tilton, GD; Willerson, JT1
Hedner, T; Henning, M; Persson, B; Pettersson, A1
McLennan, PL; Taylor, DA1
Offord, SJ; Warwick, RO1
Fuller, RW; Snoddy, HD1
Barvais, L; Capouet, V; d'Hollander, A1
Hoyer, D; Palacios, JM; Pazos, A1
Chuang, DM; Costa, E; Nakaki, T; Roth, BL1
Freedman, M; Hamel, L; Luttinger, D; Perrone, M; Ward, SJ1
Engel, G; Hoyer, D; Kalkman, HO; Wick, MB1
Su, C; Uruno, T1
Hechtman, HB; Huval, WV; Lelcuk, S; Shepro, D1
Duncker, DJ; Heiligers, J; Jennewein, HM; Saxena, PR; Verdouw, PD1
Kolling, JB; Reneman, RS; Scheijgrond, HW; van der Starre, PJ1
Taylor, DA; Yap, CY1
De Wet, JI; Diedericks, BJ; Roelofse, JA1
Frey, HH; Reiche, R1
Dentan, M; Fischler, M; Freitag, B; Vourc'h, G; Westerman, MN1
Klotz, U; Okonkwo, PO; Reimann, IW1
Glennon, RA; Rosecrans, JA; Young, R1
Ball, SG; Fraser, R; Inglis, GC; Isles, CG; Murray, GD; Robertson, JI; Zabludowski, JR; Zoccali, C2
Laduron, PM; Maloteaux, JM; Schotte, A2
Gudelsky, GA; Meltzer, HY; Simonovic, M1
Patel, S; Slater, P1
Holliman, CJ; Larsen, KR; Meuleman, TR; Pace, NL; Port, JD; Stanley, TH; Warden, GD1
Lindelauf, F1
Biegon, A; Mann, JJ; McBride, PA; McEwen, B1
Janssen, PA; Van Beek, J; Van Nueten, JM1
Affolter, H; Pletscher, A1
Cohen, RA; Shepherd, JT; Vanhoutte, PM1
Hayashi, T; Ichida, S; Terao, M1
Engel, G; Müller-Schweinitzer, E1
Angus, JA; Wright, CE1
Lund-Johansen, P; Omvik, P1
Bagge, U; Ivarsson, L; Skolnik, G1
Amery, A; Cattaert, A; Fagard, R; Lijnen, P; Moerman, E; Staessen, J; Vanhees, L1
Frazer, A; Lucki, I; Nobler, MS1
Iwanov, V; Medcalf, RL; Moulds, RF1
Carpeggiani, C; De Caterina, R; L'Abbate, A1
Berre, J; Degaute, JP; Domb, M; Simon, P; Vandesteene, A; Vincent, JL1
De Clerck, F; Janssen, PA; Leysen, J; Xhonneux, B1
Creese, I; Hamblin, MW; Leff, SE1
Coltart, DJ; Juul, SM; Walker, JM; Wilmshurst, PT1
Arnold, L; Iversen, LL; Mountjoy, CQ; Reynolds, GP; Rossor, MN; Roth, M1
Bugiardini, R; Chierchia, S; Freedman, SB; Maseri, A; Rodriguez-Plaza, L; Smith, G1
De Ridder, W; Van Nueten, JM; Vanhoutte, PM1
Gelfan, R; Socol, ML; Weiner, CP1
Barbieri, C; Bevilacqua, M; Bigatti, G; Diena, A; Guffanti, A; Norbiato, G; Rauhe, WG; Sala, M; Scorza, D1
Heym, J; Jacobs, BL; Rasmussen, K1
Hölzenspies, AJ; Kalenda, Z1
Boomsma, F; Man in 't Veld, AJ; Schalekamp, MA; Wenting, GJ; Woittiez, AJ1
Krohg, K; Roald, OK; Stranden, E1
De Clerck, F; Van Nueten, JM1
Makabali, GL; Mandal, AK; Morris, JA1
Dunham, BM; Hechtman, HB; Huval, WV; Jones, AG; Mathieson, MA; Shepro, D; Stemp, LI1
Bagge, U; Ericson, LE; Skolnik, G1
Klotz, U; Okonkwo, PO; Reimann, IW; Woestenborghs, R1
Bury, RW; Kacprowicz, AT; Moulds, RF; Shaw, PG1
Cantalamessa, F; de Caro, G; Massi, M; Micossi, LG1
Barbaccia, ML; Chuang, DM; Costa, E; Gandolfi, O1
de Smet, HL; Gerritsen, HA; Kotora, OV; Perquin, JW; Troost, FA1
De Clerck, F; Gommeren, W; Leysen, JE2
Hill, DC; Meuleman, TR; Mohammad, SF; Pace, NL; Port, JD; Stanley, TH1
Garrett, NJ; Jenner, P; Marsden, CD; Reynolds, GP; Rupniak, N1
Davies, CL1
Arvidsson, S; Bergqvist, D; Esquivel, CO; Haglund, U; Lindblad, B1
Hong, E; Mena, MA; Rión, R1
Brenken, U; Homan van der Heide, JN; Karliczek, GF; Schokkenbroek, R; van den Broeke, JJ1
De Cock, W; De Cree, J; Geukens, H; Leempoels, J; Verhaegen, H2
De Ridder, A; Janssen, PA; Van Nueten, JM; Vanhoutte, PM1
Alexander, JP; Miranda, DR; Stoutenbeek, CP; Zandstra, D1
Laduron, PM; Leysen, JE; Niemegeers, CJ; Van Nueten, JM1
Geerts, R; Gommeren, W; Leysen, JE; Van Gompel, P; Verwimp, M1
Janssen, PF; Laduron, PM; Leysen, JE1
De Clerck, F; Dom, J; Jageneau, A1
de Gaetano, G; Lampugnani, MG1
Simon, V; Somani, P1
Bueno, L; Fioramonti, J; Ooms, L; Ruckebusch, Y1
Janssen, PA; Van Nueten, JM; Vanhoutte, PM; Xhonneux, R1
Hörig, C; Jageneau, AH; Loots, W; Symoens, J1
Barrett, RJ; Sanders-Bush, E; Smith, RL1
Kido, H; Mori, H; Sakamoto, H; Shiba, K; Sumiyoshi, T; Suzuki, K; Urasaki, K; Yamaguchi, N; Yokogawa, K1
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI1
Arruda, K; Glennon, RA; Ismaiel, AM; Teitler, M1
Dykstra, LA; Lin, YP; Powell, KR1
Hansen, MB; Jaffe, BM1
Holtzman, SG; Steinfels, GF1
Cadavid, I; Castro, E; Ferreiro, TG; Fontenla, JA; Loza, MI; Lozoya, E; Manaut, F; Rodriguez, J; Sanz, F; Verde, I1
Colpaert, FC; John, GW; Le Grand, B; Patoiseau, JF; Rieu, JP; Talmant, JM1
Frölich, D; Göthert, M; Likungu, J; Molderings, GJ1
Carr, AA; Johnson, MP; Siegel, BW1
Berardi, F; Giudice, G; Govoni, S; Lucchi, L; Perrone, R; Tortorella, V1
Abi-Dargham, A; al-Tikriti, M; Baldwin, RM; Charney, D; Hoffer, P; Innis, RB; Laruelle, M; Leysen, JE; Mertens, J; Terriere, D; Zea-Ponce, Y1
Assié, MB; Kleven, MS; Koek, W1
López-Giménez, JF; Mengod, G; Palacios, JM; Vilaró, MT4
Buczko, W; Chabielska, E; Małyszko, J; Myśliwiec, M; Pawlak, D; Pawlak, K; Takada, A1
Adamkiewicz, M; Buczko, W; Malyszko, J; Mysliwiec, M; Pawlak, D; Takada, A1
Kulkarni, SK; Ninan, I1
Aloyo, VJ; Harvey, JA; Hoffman, ME; Salt, GL1
Harvey, JA; Hood, H; Romano, AG; Welsh, SE1
Kaibara, M; Mameya, S; Takada, K; Takemura, K; Taniyama, K1
Caldarola-Pastuszka, M; DeLashaw, M; Uphouse, L; Wolf, A1
Chen, K; De Maeyer, E; Kung, MP; Meehan, WP; Ridd, MJ; Seif, I; Shih, JC1
Asai, F; Fujimoto, K; Goto, R; Hayakawa, M; Ito, R; Ogawa, T; Sugidachi, A; Tanaka, N1
Adlersberg, M; Arango, V; Hsiung, S; Kassir, SA; Liu, K; Mann, JJ; Ruggiero, DA; Tamir, H; Underwood, MD1
Naylor, RJ; Tuladhar, BR; Womack, MD1
Cunningham, KA; McMahon, LR1
Hattori, K; Nagatom, T; Nakamura, T; Nakazawa, M; Rashid, M; Watanabe, M1
De los Angeles, J; Dukat, M; Glennon, RA; Herndon, J; Ismaiel, AM; Khorana, N; Metwally, K; Teitler, M1
Baker, GB; Fletcher, PJ; Korth, KM; Robinson, SR1
Audenaert, K; De Vos, F; Dierckx, R; Dumont, F; Jacobs, F; Mertens, J; Peremans, K; Slegers, G; Van Bree, H; Van De Wiele, C; Vandecapelle, M; Verschooten, F1
Fantegrossi, WE; Godlewski, T; Karabenick, RL; Rice, KC; Stephens, JM; Ullrich, T; Woods, JH1
Cunningham, KA; Filip, M; McCreary, AC1
Ge, L; Naylor, RJ; Tuladhar, BR1
Zhang, ZW1
Cao, C; Cho, KW; Han, JH; Kim, SH; Kim, SZ1
Grasby, P; Hirani, E; Hume, S; Sharp, T; Sprakes, M1
Jähnichen, S; Pertz, HH; Radtke, OA1
Gorzalka, BB; Hill, MN; Sun, JC1
Hayslett, RL; Tizabi, Y1
Elfving, B; Gillings, N; Knudsen, GM; Kristiansen, H; Pinborg, LH; Plenge, P1
Asgari, K; Bak, VK; Body, S; Bradshaw, CM; Fone, KC; Glennon, JC; Rickard, JF; Szabadi, E; Zhang, ZQ1
Bindslev, N; Engelmann, BE; Hansen, MB; Larsen, R; Poulsen, SS1
Peña, F; Ramirez, JM; Tryba, AK1
Kajos, M; Kankaanpää, A; Meririnne, E; Seppälä, T1
Abanades, S; Bullich, S; Catafau, AM; Cunningham, VJ; Danus, M; Eersels, JL; Farre, M; Llop, J; Nucci, G; Pavia, J1
Bernard, JF; Comet, MA; Hamon, M; Laguzzi, R; Sévoz-Couche, C1
Komada, T; Yano, S1
Fletcher, PJ; Higgins, GA; Sinyard, J; Tampakeras, M1
Debus, F; Herth, MM; Knudsen, GM; Lüddens, H; Palner, M; Piel, M; Rösch, F1
Harmar, AJ; Jennings, KA; Sharp, T; Sheward, WJ1
Abe, M; Egashira, N; Fujiwara, M; Iwasaki, K; Matsushita, M; Mishima, K; Nishimura, R; Oishi, R; Okuno, R1
Blanckaert, P; Burvenich, I; De Bruyne, S; De Vos, F; Moerman, L; Staelens, S; Wyffels, L1
France, CP; Li, JX; Rice, KC1
Bianchi, P; Calise, D; Escourrou, G; Galinier, M; Guilbeau-Frugier, C; Lairez, O; Mialet-Perez, J; Ordener, C; Parini, A; Pizzinat, N; Roncalli, J; Seif, I; Spreux-Varoquaux, O1
Anju, TR; George, AK; Paulose, CS1
Lefever, TW; Rawls, SM; Walker, EA; Ward, SJ; Whiteside, GT1
France, CP; Javors, MA; Koek, W; Li, JX; Rice, KC; Unzeitig, A1
Doi, A; Ramirez, JM1
Herth, MM; Knudsen, GM; Kramer, V; Palner, M; Rösch, F; Santini, MA1
Estrada-González, V; Márquez-Diosdado, MI; Montes-Rodríguez, CJ; Prospéro-García, O; Soria-Gómez, E1
Cohen, MS; Fantegrossi, WE; Henson, CM; Rice, KC; Simoneau, J; Woods, JH; Zimmerman, SM1
Creed-Carson, M; Nobrega, JN; Oraha, A1
Arai, Y; Kikuchi, T; Mitazaki, S; Nakagawasai, O; Nakaya, K; Niijima-Yaoita, F; Onogi, H; Sato, A; Tadano, T; Tan-No, K; Watanabe, K1
Elizalde, DI; Gallitano, AL; González-Maeso, J; Ingram, WM; Janowski, SA; Kamel, CM; Kozlenkov, A; Levine, S; Lish, JR; Resnik, J; Shoker, J; Williams, AA1
Dyssegaard, A; Ettrup, A; Gillings, N; Hansen, HD; Herth, MM; Knudsen, GM; Ratner, C1
Bailey, JM; Fantegrossi, WE; Gray, BW; Hansen, M; Kristensen, JL; Smith, DA1
Gencer, A; Gunduz, O; Ulugol, A1
Anastasio, NC; Cunningham, KA; Fink, LH; Fox, RG; Moeller, FG; Rice, KC1

Reviews

24 review(s) available for ketanserin and piperidines

ArticleYear
Can peripheral serotonergic blockade explain the hypotensive effect of ketanserin?
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Ketanserin; Methoxamine; Phenylephrine; Piperidines; Receptors, Adrenergic, alpha; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation

1985
Ketanserin: a new hypotensive drug?
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Antihypertensive Agents; Costs and Cost Analysis; Dose-Response Relationship, Drug; Humans; Ketanserin; Kinetics; Patient Compliance; Piperidines; Species Specificity

1985
Serotonin and the heart: effects of ketanserin on myocardial function, heart rate, and arrhythmias.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Coronary Circulation; Coronary Disease; Heart; Heart Rate; Humans; In Vitro Techniques; Ketanserin; Myocardial Contraction; Piperidines; Serotonin; Serotonin Antagonists; Sinoatrial Node

1985
Pharmacology of the interaction between platelets and vessel wall.
    Clinics in haematology, 1986, Volume: 15, Issue:2

    Topics: Animals; Aspirin; Blood Platelets; Blood Vessels; Dextrans; Diltiazem; Dipyridamole; Epoprostenol; Humans; Imidazoles; Ketanserin; Piperidines; Pyrazoles; Pyrazolones; Sulfinpyrazone; Sulfonamides; Thiophenes; Ticlopidine

1986
Antihypertensive mode of action of ketanserin.
    Journal of cardiovascular pharmacology, 1987, Volume: 10 Suppl 3

    Topics: Adrenergic alpha-Antagonists; Aldosterone; Animals; Antihypertensive Agents; Blood Pressure; Carcinoid Heart Disease; Humans; Ketanserin; Piperidines; Prazosin; Ritanserin

1987
Serotonin and vascular reactivity.
    Pharmacological research communications, 1985, Volume: 17, Issue:7

    Topics: Animals; Blood Platelets; Calcium; Cold Temperature; Electric Stimulation; Hypoxia; Ketanserin; Lidoflazine; Methiothepin; Methysergide; Microcirculation; Models, Biological; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation

1985
[New findings and experiences in the field of malignant hyperthermia].
    Der Anaesthesist, 1986, Volume: 35, Issue:1

    Topics: Anesthesia; Animals; Calcium Channel Blockers; Catatonia; Dantrolene; Diagnosis, Differential; Humans; Ketanserin; Malignant Hyperthermia; Neuroleptic Malignant Syndrome; Piperidines; Serotonin Antagonists; Swine

1986
Neurophysiological evidence that D-1 dopamine receptor blockade attenuates postsynaptic but not autoreceptor-mediated effects of dopamine agonists.
    European journal of pharmacology, 1986, Apr-16, Volume: 123, Issue:2

    Topics: Animals; Apomorphine; Basal Ganglia; Benzazepines; Dextroamphetamine; Dopamine Antagonists; Electrophysiology; Ergolines; Globus Pallidus; Haloperidol; Ketanserin; Neurons; Pergolide; Piperidines; Quinpirole; Rats; Receptors, Dopamine; Substantia Nigra

1986
Effects of electroconvulsive shock and serotonin axon lesions on beta-adrenergic and serotonin-2 receptors in rat brain.
    Annals of the New York Academy of Sciences, 1986, Volume: 462

    Topics: Anesthetics; Animals; Axons; Brain; Cerebral Cortex; Cyclic AMP; Dihydroalprenolol; Electroconvulsive Therapy; Frontal Lobe; Hippocampus; Ketanserin; Norepinephrine; Piperidines; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Muscarinic; Receptors, Serotonin; Serotonin; Spiperone; Stress, Physiological; Time Factors; Tritium

1986
[Role of serotonin in the regulation of the circulatory system].
    Polski tygodnik lekarski (Warsaw, Poland : 1960), 1985, Apr-22, Volume: 40, Issue:16

    Topics: Animals; Humans; Hypertension; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Resistance

1985
Cardiovascular pharmacology of ketanserin.
    Bibliotheca cardiologica, 1984, Issue:38

    Topics: Animals; Blood Platelets; Blood Pressure; Drug Interactions; Histamine; Ketanserin; Piperidines; Platelet Aggregation; Receptors, Adrenergic, alpha; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vasoconstriction

1984
Cardiovascular alpha 2-receptors.
    Journal of molecular and cellular cardiology, 1983, Volume: 15, Issue:11

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Affinity Labels; Animals; Blood Pressure; Brain; Calcium Channel Blockers; Cardiovascular Physiological Phenomena; Guanosine Triphosphate; Heart Rate; Humans; Ketanserin; Kidney; Muscle, Smooth, Vascular; Piperazines; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Synaptic Membranes; Tritium; Vasoconstriction

1983
Vasodilator therapy for primary pulmonary hypertension.
    Mayo Clinic proceedings, 1984, Volume: 59, Issue:10

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Blood Pressure; Calcium Channel Blockers; Captopril; Epoprostenol; Hemodynamics; Humans; Hypertension, Pulmonary; Ketanserin; Piperidines; Serotonin Antagonists; Vascular Resistance; Vasodilator Agents

1984
Role of alpha adrenoceptors in hypertension and in antihypertensive drug treatment.
    The American journal of medicine, 1984, Oct-05, Volume: 77, Issue:4A

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Calcium Channel Blockers; Clonidine; Guanfacine; Guanidines; Humans; Hypertension; Ketanserin; Methyldopa; Muscle, Smooth, Vascular; Phenylacetates; Piperazines; Piperidines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Vascular Resistance

1984
Peripheral 5-hydroxytryptamine receptors and their classification.
    Neuropharmacology, 1984, Volume: 23, Issue:12B

    Topics: Animals; Dogs; Guinea Pigs; In Vitro Techniques; Ketanserin; Methysergide; Muscle Relaxation; Muscle, Smooth; Neurotransmitter Agents; Piperidines; Rabbits; Rats; Receptors, Serotonin

1984
Antihypertensive properties of ketanserin (R 41 468).
    Federation proceedings, 1983, Volume: 42, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Dose-Response Relationship, Drug; Humans; Ketanserin; Muscle, Smooth, Vascular; Norepinephrine; Piperidines; Platelet Aggregation; Receptors, Adrenergic, alpha; Serotonin Antagonists

1983
5-hydroxytryptamine and precapillary vessels.
    Federation proceedings, 1983, Volume: 42, Issue:2

    Topics: Angiotensin II; Animals; Dinoprost; Drug Interactions; Histamine; Ketanserin; Methysergide; Norepinephrine; Piperidines; Prostaglandins F; Receptors, Adrenergic, alpha; Serotonin; Vasoconstriction

1983
Place of vasoactive agents in the treatment of acute circulatory failure.
    Resuscitation, 1984, Volume: 11, Issue:3-4

    Topics: Cardiac Output; Depression, Chemical; Dobutamine; Dopamine; Fluid Therapy; Humans; Ketanserin; Nitroglycerin; Nitroprusside; Phentolamine; Piperidines; Shock; Stimulation, Chemical; Sympathomimetics; Vasodilator Agents

1984
Role of humoral mediators in adult respiratory distress syndrome.
    Chest, 1984, Volume: 86, Issue:4

    Topics: Animals; Arachidonic Acids; Chemotaxis, Leukocyte; Chromones; Dogs; Guinea Pigs; Humans; Hypertension, Pulmonary; Inflammation; Ketanserin; Leukocyte Count; Leukocytes; Lung; Piperidines; Platelet Activating Factor; Pulmonary Embolism; Respiratory Distress Syndrome; Serotonin; Serotonin Antagonists; SRS-A; Thromboxane A2

1984
An analysis of 5-hydroxytryptamine receptors mediating contraction of isolated smooth muscle.
    Neuropharmacology, 1984, Volume: 23, Issue:12B

    Topics: Animals; Binding, Competitive; Cats; Cyproheptadine; Dogs; In Vitro Techniques; Ketanserin; Methoxamine; Methysergide; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Piperidines; Rabbits; Rats; Receptors, Serotonin

1984
Serotonin-S2 receptor binding sites and functional correlates.
    Neuropharmacology, 1984, Volume: 23, Issue:12B

    Topics: Animals; Binding Sites; Blood Platelets; Cats; Cerebral Cortex; Humans; In Vitro Techniques; Ketanserin; Kinetics; Models, Biological; Muscle, Smooth, Vascular; Piperidines; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin

1984
Platelet-vessel wall interactions: implication of 5-hydroxytryptamine. A review.
    Agents and actions, 1984, Volume: 15, Issue:5-6

    Topics: Animals; Blood Platelets; Blood Vessels; Capillary Permeability; Endothelium; Humans; In Vitro Techniques; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Receptors, Serotonin; Serotonin; Vasoconstriction

1984
Serotonin antagonists.
    Australian and New Zealand journal of medicine, 1984, Volume: 14, Issue:6

    Topics: Cyproheptadine; Depression; Ergotamine; Humans; Hypertension; Ketanserin; Lisuride; Methysergide; Mianserin; Migraine Disorders; Piperidines; Pizotyline; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Diseases

1984
Ketanserin and spiperone as templates for novel serotonin 5-HT(2A) antagonists.
    Current topics in medicinal chemistry, 2002, Volume: 2, Issue:6

    Topics: Animals; Drug Design; Isoquinolines; Ketanserin; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Structure-Activity Relationship

2002

Trials

78 trial(s) available for ketanserin and piperidines

ArticleYear
Ketanserin and alpha 1-adrenergic antagonism in humans.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Double-Blind Method; Heart Rate; Humans; Ketanserin; Male; Middle Aged; Phenylephrine; Piperidines; Serotonin Antagonists; Valsalva Maneuver

1985
Hemodynamic response to chronic ketanserin treatment in essential hypertension.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Cardiac Output; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Hemodynamics; Humans; Hypertension; Ketanserin; Male; Methoxamine; Phenylephrine; Physical Exertion; Piperidines; Random Allocation; Serotonin Antagonists; Stroke Volume; Vascular Resistance

1985
Double-blind comparison of ketanserin with propranolol in hypertensive patients: interim report.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Aged; Antihypertensive Agents; Body Weight; Clinical Trials as Topic; Double-Blind Method; Female; Follow-Up Studies; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Patient Compliance; Piperidines; Propranolol; Random Allocation

1985
Clinical studies with ketanserin in hypertension.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Aged; Blood Pressure; Clinical Trials as Topic; Diuretics; Erythrocyte Deformability; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Physical Exertion; Piperidines; Pulse; Random Allocation; Serotonin Antagonists; Time Factors

1985
Study with the competitive 5-HT2-serotonergic antagonist ketanserin.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Heart Rate; Humans; Hypertension; Ketanserin; Leg; Metoprolol; Physical Exertion; Piperidines; Random Allocation; Regional Blood Flow; Serotonin Antagonists

1985
Antihypertensive properties of ketanserin in combination with beta-adrenergic blocking agents.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adrenergic beta-Antagonists; Antihypertensive Agents; Blood Pressure; Drug Therapy, Combination; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Serotonin Antagonists; Time Factors

1985
Effect of ketanserin on blood pressure and biochemical parameters in patients with essential hypertension.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Antihypertensive Agents; Blood Pressure; Body Weight; Clinical Trials as Topic; Diuretics; Double-Blind Method; Drug Therapy, Combination; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation

1985
Effect of ketanserin in primary aldosteronism.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Aldosterone; Blood Pressure; Humans; Hydrocortisone; Hyperaldosteronism; Hypertension; Ketanserin; Piperidines; Potassium; Renin; Serotonin Antagonists; Time Factors

1985
Effect of ketanserin on the hyperreactivity of platelets to 5-hydroxytryptamine in patients with cardiovascular diseases.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Aged; beta-Thromboglobulin; Blood Platelets; Cardiovascular Diseases; Double-Blind Method; Humans; Ketanserin; Middle Aged; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists

1985
Serotonin and the flow properties of blood.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Blood Flow Velocity; Blood Viscosity; Hemoglobins; Humans; Ischemia; Ketanserin; Leg; Piperidines; Rheology; Serotonin; Serotonin Antagonists

1985
Ketanserin and red blood cell sodium content in hypertension.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Aged; Erythrocyte Deformability; Erythrocytes; Humans; Hypertension; Ketanserin; Middle Aged; Myocardial Infarction; Ouabain; Piperidines; Serotonin; Serotonin Antagonists; Sodium

1985
Comparison of blood pressure ratio by Doppler velocimetry and by plethysmography during treatment with ketanserin, a 5-HT2 receptor antagonist: a measure of improved collateral and microcirculatory flow.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Aged; Arm; Blood Pressure; Collateral Circulation; Female; Humans; Ketanserin; Male; Microcirculation; Middle Aged; Piperidines; Plethysmography; Regional Blood Flow; Rheology; Serotonin Antagonists; Thigh

1985
Effects of ketanserin on peripheral blood flow, haemorheology, and platelet function in patients with Raynaud's phenomenon.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Aged; Blood Platelets; Blood Viscosity; Female; Fingers; Humans; Ketanserin; Male; Middle Aged; Piperidines; Raynaud Disease; Regional Blood Flow; Rheology; Serotonin Antagonists

1985
Does acute serotonergic type-2 antagonism reduce blood pressure? Comparative effects of single doses of ritanserin and ketanserin in essential hypertension.
    Journal of cardiovascular pharmacology, 1987, Volume: 10 Suppl 3

    Topics: Adult; Affect; Aged; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin; Ritanserin

1987
Experience with ketanserin and ritanserin in hypertensive patients.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Ritanserin

1988
The alpha-adrenergic receptor blocking effect of ketanserin and the interaction between alpha-adrenergic and S2-serotonergic receptor blockade.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Blood Pressure; Droperidol; Female; Humans; Ketanserin; Male; Middle Aged; Phentolamine; Phenylephrine; Piperidines; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin

1988
Comparative haemodynamic effects of ketanserin and ritanserin in the proximal and distal upper limb circulations of hypertensive patients.
    European journal of clinical pharmacology, 1989, Volume: 37, Issue:3

    Topics: Arm; Blood Pressure; Brachial Artery; Double-Blind Method; Hand; Humans; Hypertension; Ketanserin; Middle Aged; Piperidines; Regional Blood Flow; Rheology; Ritanserin; Serotonin Antagonists; Vascular Resistance

1989
Placebo-controlled, double-blind, two-centre trial of ketanserin in intermittent claudication.
    Lancet (London, England), 1985, Dec-07, Volume: 2, Issue:8467

    Topics: Adult; Aged; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Extremities; Female; Humans; Intermittent Claudication; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Regional Blood Flow; Serotonin Antagonists

1985
Ketanserin--a new antihypertensive agent.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adrenergic beta-Antagonists; Clinical Trials as Topic; Diuretics; Dose-Response Relationship, Drug; Humans; Hypertension; Ketanserin; Piperidines; Placebos

1986
Ketanserin: haemodynamic effects and mechanism of action.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adrenergic beta-Antagonists; Clinical Trials as Topic; Double-Blind Method; Heart Rate; Humans; Hypertension; Ketanserin; Piperidines; Placebos; Pressoreceptors; Random Allocation; Receptors, Serotonin; Reflex

1986
Moderate essential hypertension control: a double-blind crossover study between a serotonin antagonist and a post-synaptic alpha-blocker.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Prazosin; Serotonin Antagonists

1986
Comparison of single doses of ketanserin and placebo in chronic stable angina.
    British journal of clinical pharmacology, 1986, Volume: 22, Issue:1

    Topics: Adrenergic beta-Antagonists; Adult; Angina Pectoris; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Drug Therapy, Combination; Electrocardiography; Exercise Test; Female; Heart Rate; Humans; Ketanserin; Male; Middle Aged; Piperidines

1986
Chronic 5-HT2-receptor blockade by ritanserin does not reduce blood pressure in patients with essential hypertension.
    Acta medica Scandinavica, 1987, Volume: 222, Issue:4

    Topics: Aged; Clinical Trials as Topic; Double-Blind Method; Female; Histamine H2 Antagonists; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Ritanserin; Time Factors

1987
The effect of serotonergic blockade in postpartum preeclamptic patients.
    American journal of obstetrics and gynecology, 1985, Sep-15, Volume: 153, Issue:2

    Topics: Adult; Blood Pressure; Double-Blind Method; Female; Humans; Ketanserin; Piperidines; Pre-Eclampsia; Pregnancy; Puerperal Disorders; Random Allocation; Serotonin Antagonists; Time Factors

1985
A comparative study of ketanserin and metoprolol in essential hypertension.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1985, Oct-12, Volume: 68, Issue:8

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Metoprolol; Middle Aged; Piperidines; Random Allocation; Time Factors

1985
The effect of ketanserin, a 5-HT2-receptor antagonist, on 5-hydroxytryptamine-induced irreversible platelet aggregation in patients with cardiovascular diseases.
    Agents and actions, 1985, Volume: 16, Issue:5

    Topics: Aged; Arterial Occlusive Diseases; beta-Thromboglobulin; Cardiovascular Diseases; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Myocardial Infarction; Piperidines; Placebos; Platelet Aggregation; Serotonin

1985
The effect of ketanserin on post-anaesthetic vasoconstriction and shivering.
    European journal of anaesthesiology, 1985, Volume: 2, Issue:3

    Topics: Adult; Anesthesia; Blood Gas Analysis; Blood Pressure; Body Temperature; Female; Heart Rate; Humans; Ketanserin; Middle Aged; Piperidines; Pulse; Serotonin Antagonists; Shivering; Vasoconstriction

1985
Raynaud's disease: a new therapeutic approach with a 5-HT2 receptors blocker.
    Bollettino chimico farmaceutico, 1985, Volume: 124, Issue:10

    Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Raynaud Disease; Serotonin Antagonists

1985
Ketanserin hypertension and chronic alcoholism DB study in 40 patients.
    Bollettino chimico farmaceutico, 1985, Volume: 124, Issue:10

    Topics: Alcoholism; Blood Pressure; Chronic Disease; Female; Humans; Hypertension; Ketanserin; Male; Piperidines

1985
Chronic effect of ketanserin in mild to moderate essential hypertension.
    Hypertension (Dallas, Tex. : 1979), 1986, Volume: 8, Issue:2

    Topics: Adult; Aged; Blood Pressure; Circadian Rhythm; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Posture; Random Allocation

1986
Effects of ketanserin on ambulatory blood pressure monitoring in patients with essential hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adult; Ambulatory Care; Blood Pressure Determination; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Placebos; Propranolol

1986
Comparison of ketanserin and pindolol in hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adult; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Pindolol; Piperidines; Random Allocation

1986
A comparative study of ketanserin and metoprolol in essential hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adult; Aged; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Metoprolol; Middle Aged; Piperidines; Placebos

1986
Double-blind comparison of ketanserin with atenolol: antihypertensive activity and effect on platelet function.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adult; Aged; Atenolol; Blood Platelets; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Ketanserin; Male; Middle Aged; Piperidines; Placebos; Platelet Aggregation

1986
Long-term safety and efficacy of ketanserin in essential hypertension: ketanserin versus or in combination with metoprolol.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypertension; Ketanserin; Male; Metoprolol; Middle Aged; Piperidines; Random Allocation

1986
Ketanserin versus metoprolol in the treatment of essential hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adult; Aged; Female; Follow-Up Studies; Heart Rate; Humans; Hypertension; Ketanserin; Male; Metoprolol; Middle Aged; Piperidines; Placebos

1986
Clinical experience with ketanserin in the treatment of hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Double-Blind Method; Heart Rate; Humans; Hypertension; Ketanserin; Metoprolol; Piperidines

1986
Ketanserin in the treatment of mild hypertension in elderly patients: preliminary results of a controlled double-blind trial.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Piperidines

1986
Blood pressure reduction and pharmacokinetics of ketanserin in hypertensive patients.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Aged; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines

1986
Intra arterial ketanserin in peripheral vascular disease.
    Angiology, 1986, Volume: 37, Issue:4

    Topics: Aged; Clinical Trials as Topic; Female; Humans; Injections, Intra-Arterial; Ischemia; Ketanserin; Leg; Male; Middle Aged; Piperidines; Serotonin Antagonists; Sympathectomy, Chemical

1986
[Multicenter study with 3 different doses of ketanserin in essential arterial hypertension].
    Arquivos brasileiros de cardiologia, 1985, Volume: 45, Issue:4

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Drug Administration Schedule; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Vascular Resistance

1985
Ketanserin and prazosin: a comparison of antihypertensive and biochemical effects.
    Clinical pharmacology and therapeutics, 1986, Volume: 40, Issue:1

    Topics: Adult; Aldosterone; Blood Pressure; Cholesterol; Drug Evaluation; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Physical Exertion; Piperidines; Prazosin; Random Allocation; Renin

1986
Selective antagonism of S2-serotonergic receptors relieves but does not prevent cold induced vasoconstriction in primary Raynaud's phenomenon.
    The Journal of rheumatology, 1986, Volume: 13, Issue:2

    Topics: Adult; Cold Temperature; Female; Humans; Ketanserin; Piperidines; Raynaud Disease; Receptors, Adrenergic; Receptors, Serotonin; Vasoconstriction

1986
Influence of ketanserin pretreatment on the haemodynamic responses to sternotomy.
    Anaesthesia, 1986, Volume: 41, Issue:5

    Topics: Drug Evaluation; Hemodynamics; Humans; Hypertension; Indoles; Intraoperative Complications; Ketanserin; Middle Aged; Myocardial Revascularization; Piperidines; Premedication; Serotonin; Serotonin Antagonists; Sternum

1986
Quantitative study of the effects of Ketanserin in patients with primary Raynaud's phenomenon. A randomized, double blind, placebo controlled investigation and an additional long term open trial.
    Microcirculation, endothelium, and lymphatics, 1985, Volume: 2, Issue:6

    Topics: Adolescent; Adult; Aged; Blood Flow Velocity; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation; Raynaud Disease; Skin Temperature; Vascular Resistance

1985
Effects of ketanserin on blood pressure, peripheral circulation and haemocoagulative parameters in essential hypertensives with or without arteriosclerosis obliterans of the lower limbs.
    International journal of clinical pharmacology research, 1986, Volume: 6, Issue:3

    Topics: Adult; Antihypertensive Agents; Arteriosclerosis Obliterans; Blood Coagulation; Blood Pressure; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Leg; Male; Middle Aged; Piperidines; Propranolol; Random Allocation; Regional Blood Flow

1986
Ketanserin and the cardiovascular system. 2. A study of its effects in patients undergoing myocardial revascularisation.
    Anaesthesia, 1986, Volume: 41, Issue:7

    Topics: Antihypertensive Agents; Cardiopulmonary Bypass; Drug Evaluation; Female; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Myocardial Revascularization; Piperidines

1986
Cardiovascular effects of ketanserin, a new antiserotonergic agent in the treatment of arterial hypertension.
    Journal of clinical pharmacology, 1985, Volume: 25, Issue:3

    Topics: Adult; Blood Pressure; Body Weight; Exercise Test; Heart Rate; Hemodynamics; Humans; Hypertension; Ketanserin; Metoprolol; Middle Aged; Piperidines; Regional Blood Flow; Serotonin Antagonists; Vascular Resistance

1985
Effect of intravenous ketanserin on plasma catecholamines and renin activity in normal volunteers.
    European journal of clinical pharmacology, 1985, Volume: 28, Issue:3

    Topics: Adult; Catecholamines; Female; Humans; Injections, Intravenous; Ketanserin; Male; Piperidines; Renin; Serotonin Antagonists

1985
Inhibition of cold-induced vasoconstriction with ketanserin.
    Microvascular research, 1985, Volume: 30, Issue:1

    Topics: Adult; Cold Temperature; Hand; Humans; Ibuprofen; Ketanserin; Ketoconazole; Male; Middle Aged; Piperidines; Regional Blood Flow; Serotonin; Skin Temperature; Thromboxane B2; Vasoconstriction

1985
Ketanserin in essential hypertension: a double-blind, placebo-controlled study.
    Postgraduate medical journal, 1985, Volume: 61, Issue:717

    Topics: Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines

1985
Controlled trial of ketanserin in hypertension.
    British journal of clinical pharmacology, 1985, Volume: 20, Issue:1

    Topics: Adult; Aged; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin

1985
Ketanserin in chronic sympathetic dystrophy. An acute controlled trial.
    Clinical rheumatology, 1984, Volume: 3, Issue:4

    Topics: Adult; Clinical Trials as Topic; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Reflex Sympathetic Dystrophy; Serotonin Antagonists

1984
Effect of an oral serotonin antagonist, ketanserin, on plasma ACTH concentrations in Nelson's syndrome.
    British medical journal (Clinical research ed.), 1984, Sep-29, Volume: 289, Issue:6448

    Topics: Adrenocorticotropic Hormone; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Nelson Syndrome; Piperidines; Pituitary Neoplasms; Serotonin Antagonists

1984
Ketanserin in acute superficial thrombophlebitis.
    Lancet (London, England), 1982, Aug-21, Volume: 2, Issue:8295

    Topics: Acute Disease; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Pain; Piperidines; Random Allocation; Serotonin Antagonists; Thrombophlebitis

1982
Is ketanserin a D receptor antagonist?
    Lancet (London, England), 1983, Mar-26, Volume: 1, Issue:8326 Pt 1

    Topics: Adult; Animals; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Piperidines; Random Allocation; Rats; Receptors, Serotonin; Serotonin Antagonists

1983
Mechanism of antihypertensive action of ketanserin in man.
    British medical journal (Clinical research ed.), 1983, Aug-06, Volume: 287, Issue:6389

    Topics: Adrenergic alpha-Antagonists; Adult; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Ketanserin; Male; Methoxamine; Piperidines

1983
Alpha 1 antagonistic and antiserotoninergic action during administration of ketanserin.
    British medical journal (Clinical research ed.), 1983, Nov-19, Volume: 287, Issue:6404

    Topics: Adrenergic alpha-Antagonists; Humans; Hypertension; Ketanserin; Piperidines; Serotonin Antagonists

1983
The effect of ketanserin on blood pressure and biochemical parameters in treated patients with essential hypertension.
    Clinical and experimental hypertension. Part A, Theory and practice, 1984, Volume: 6, Issue:6

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Diuretics; Double-Blind Method; Drug Therapy, Combination; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation; Serotonin Antagonists

1984
Placebo-controlled double-blind trial of ketanserin in treatment of intermittent claudication.
    Lancet (London, England), 1984, Oct-06, Volume: 2, Issue:8406

    Topics: Aged; Blood Flow Velocity; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Erythrocyte Deformability; Exercise Test; Humans; Intermittent Claudication; Ketanserin; Leg; Middle Aged; Piperidines; Plethysmography; Regional Blood Flow; Serotonin Antagonists

1984
Ketanserin in combination with beta-adrenergic receptor blocking agents in the treatment of essential hypertension.
    British journal of clinical pharmacology, 1984, Volume: 18, Issue:5

    Topics: Adrenergic beta-Antagonists; Aged; Antihypertensive Agents; Blood Pressure; Drug Therapy, Combination; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines

1984
The effect of ketanserin, a specific serotonin antagonist on the PRL, GH, ACTH and cortisol responses to hypoglycaemia in normal subjects.
    Clinical endocrinology, 1984, Volume: 20, Issue:2

    Topics: Adrenocorticotropic Hormone; Adult; Growth Hormone; Humans; Hydrocortisone; Hypoglycemia; Ketanserin; Male; Piperidines; Pituitary Hormones, Anterior; Prolactin; Serotonin Antagonists

1984
Ketanserin in hypertension. Early clinical evaluation and dose finding study of a new 5-HT2 receptor antagonist.
    Acta medica Scandinavica, 1983, Volume: 214, Issue:2

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation; Serotonin Antagonists

1983
Haemodynamic and humoral responses to chronic ketanserin treatment in essential hypertension.
    British heart journal, 1984, Volume: 51, Issue:2

    Topics: Adult; Antihypertensive Agents; Clinical Trials as Topic; Double-Blind Method; Female; Hemodynamics; Humans; Hypertension; Ketanserin; Male; Methoxamine; Physical Exertion; Piperidines; Pressoreceptors; Renin-Angiotensin System

1984
Treatment of Raynaud's phenomenon with ketanserin, a selective antagonist of the serotonin2 (5-HT2) receptor.
    Arthritis and rheumatism, 1984, Volume: 27, Issue:2

    Topics: Adult; Aged; Clinical Trials as Topic; Female; Fingers; Humans; Ketanserin; Male; Middle Aged; Pilot Projects; Piperidines; Plethysmography; Raynaud Disease; Receptors, Serotonin; Regional Blood Flow; Scleroderma, Systemic; Serotonin Antagonists

1984
[Serotonin antagonists in the treatment of hypertension].
    Casopis lekaru ceskych, 1984, Mar-16, Volume: 123, Issue:11

    Topics: Administration, Oral; Clinical Trials as Topic; Female; Humans; Hypertension; Infusions, Parenteral; Ketanserin; Male; Piperidines; Serotonin Antagonists

1984
Experience with ketanserin, a serotonin (S2) antagonist, in longterm treatment of essential hypertension.
    Clinical and experimental hypertension. Part A, Theory and practice, 1984, Volume: 6, Issue:3

    Topics: Adult; Aged; Chronic Disease; Clinical Trials as Topic; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Placebos; Serotonin Antagonists

1984
Control of preeclamptic hypertension by ketanserin, a new serotonin receptor antagonist.
    American journal of obstetrics and gynecology, 1984, Jul-01, Volume: 149, Issue:5

    Topics: Adult; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Infusions, Parenteral; Ketanserin; Piperidines; Pre-Eclampsia; Pregnancy; Random Allocation; Serotonin Antagonists

1984
Mechanism of antihypertensive action of ketanserin in man.
    British medical journal (Clinical research ed.), 1983, Oct-08, Volume: 287, Issue:6398

    Topics: Antihypertensive Agents; Blood Pressure; Humans; Ketanserin; Piperidines

1983
Treatment of Raynaud's phenomenon with ketanserin in patients with connective tissue disorders.
    British medical journal (Clinical research ed.), 1984, Sep-08, Volume: 289, Issue:6445

    Topics: Adult; Clinical Trials as Topic; Connective Tissue Diseases; Double-Blind Method; Female; Fingers; Humans; Ketanserin; Microcirculation; Middle Aged; Piperidines; Raynaud Disease; Scleroderma, Systemic; Serotonin Antagonists; Ultrasonography

1984
Ketanserin in essential hypertension: effects during rest and exercise.
    European journal of clinical pharmacology, 1983, Volume: 25, Issue:3

    Topics: Antihypertensive Agents; Blood Pressure; Catecholamines; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Physical Exertion; Piperidines; Rest

1983
Responses of the systemic circulation and of the renin-angiotensin-aldosterone system to ketanserin at rest and exercise in normal man.
    Clinical science (London, England : 1979), 1984, Volume: 66, Issue:1

    Topics: Adult; Blood Pressure; Cardiac Output; Catecholamines; Heart Rate; Hemodynamics; Humans; Ketanserin; Lactates; Male; Physical Exertion; Piperidines; Posture; Renin-Angiotensin System; Respiration; Rest; Serotonin Antagonists

1984
A double-blind, placebo-controlled study of ketanserin in patients with Prinzmetal's angina. Evidence against a role for serotonin in the genesis of coronary vasospasm.
    Circulation, 1984, Volume: 69, Issue:5

    Topics: Aged; Angina Pectoris, Variant; Coronary Disease; Coronary Vasospasm; Double-Blind Method; Drug Evaluation; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Piperidines; Placebos; Platelet Aggregation; Serotonin; Serotonin Antagonists

1984
Effect of the 5-hydroxytryptamine type 2 receptor antagonist, ketanserin, on blood pressure, the renin-angiotensin system and sympatho-adrenal function in patients with essential hypertension.
    British journal of clinical pharmacology, 1984, Volume: 17, Issue:3

    Topics: Adrenal Glands; Adult; Aged; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Norepinephrine; Phenylephrine; Piperidines; Posture; Renin-Angiotensin System; Serotonin Antagonists; Sympathetic Nervous System

1984
Treatment of Raynaud's phenomenon with the 5-HT2-receptor antagonist ketanserin.
    British medical journal (Clinical research ed.), 1982, Oct-16, Volume: 285, Issue:6348

    Topics: Adult; Aged; Female; Fingers; Humans; Ketanserin; Male; Middle Aged; Piperidines; Raynaud Disease; Regional Blood Flow; Serotonin Antagonists; Skin Temperature

1982
The antihypertensive effects of a pure and selective serotonin-receptor blocking agent (R 41 468) in elderly patients.
    Angiology, 1981, Volume: 32, Issue:2

    Topics: Age Factors; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Depression, Chemical; Female; Heart Rate; Humans; Hypertension; Injections, Intravenous; Ketanserin; Male; Middle Aged; Myocardial Contraction; Piperidines; Placebos; Receptors, Serotonin; Research Design; Serotonin Antagonists

1981
The antihypertensive effects of ketanserin (R 41468), a novel 5-hydroxytryptamine-blocking agent, in patients with essential hypertension.
    Clinical science (London, England : 1979), 1981, Volume: 61 Suppl 7

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines

1981
Characterization of the SPECT 5-HT2A receptor ligand 123I-R91150 in healthy volunteers: part 2--ketanserin displacement.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2006, Volume: 47, Issue:6

    Topics: Adult; Brain; Humans; Image Interpretation, Computer-Assisted; Iodine Radioisotopes; Ketanserin; Ligands; Male; Metabolic Clearance Rate; Piperidines; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Reference Values; Tissue Distribution; Tomography, Emission-Computed, Single-Photon

2006

Other Studies

462 other study(ies) available for ketanserin and piperidines

ArticleYear
Oxygen isosteric derivatives of 3-(3-hydroxyphenyl)-N-n-propylpiperidine.
    Journal of medicinal chemistry, 1992, Aug-07, Volume: 35, Issue:16

    Topics: Animals; Brain; Dopamine Agents; In Vitro Techniques; Ketanserin; Mice; Oxygen; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1992
Stimulation by risperidone of rat prolactin secretion in vivo and in cultured pituitary cells in vitro.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Animals; Antipsychotic Agents; Cells, Cultured; Haloperidol; Isoxazoles; Ketanserin; Male; Piperidines; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Risperidone; Spiro Compounds; Stimulation, Chemical

1992
Uptake and release of serotonin in rat cerebrovascular nerves after subarachnoid hemorrhage.
    Stroke, 1992, Volume: 23, Issue:1

    Topics: Animals; Basilar Artery; Electric Stimulation; Ischemic Attack, Transient; Ketanserin; Male; Oxidopamine; Paroxetine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Subarachnoid Hemorrhage; Sympathetic Nervous System; Tetrodotoxin; Vasoconstriction

1992
Serotonergic aspects of the response of human platelets to immune-adjuvant muramyl dipeptide.
    Journal of neuroimmunology, 1992, Volume: 37, Issue:1-2

    Topics: Acetylmuramyl-Alanyl-Isoglutamine; Adenosine Diphosphate; Adjuvants, Immunologic; Blood Platelets; Carrier Proteins; Humans; Imipramine; Ketanserin; Lysergic Acid Diethylamide; Paroxetine; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1992
5HT2 receptor changes in rat cortex and platelets following chronic ritanserin and clorgyline administration.
    Biochemical pharmacology, 1990, Jan-01, Volume: 39, Issue:1

    Topics: Animals; Blood Platelets; Cerebral Cortex; Clorgyline; Homovanillic Acid; Hydroxyindoleacetic Acid; Ketanserin; Lysergic Acid Diethylamide; Male; Norepinephrine; Piperidines; Propylamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin

1990
Effect of 3,4-methylenedioxymethamphetamine on [3H]paroxetine binding in the frontal cortex and blood platelets of rats.
    Biochemical pharmacology, 1991, Jan-01, Volume: 41, Issue:1

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Blood Platelets; Frontal Lobe; Hydroxyindoleacetic Acid; Ketanserin; Kinetics; Male; N-Methyl-3,4-methylenedioxyamphetamine; Paroxetine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Time Factors; Tritium

1991
AHR-16303B, a novel antagonist of 5-HT2 receptors and voltage-sensitive calcium channels.
    Journal of cardiovascular pharmacology, 1991, Volume: 17, Issue:1

    Topics: Animals; Atrial Function; Blood Pressure; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Chloride; Diuresis; Dose-Response Relationship, Drug; Edema; Guinea Pigs; Heart Atria; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Nimodipine; Piperidines; Platelet Aggregation; Propiophenones; Rabbits; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Histamine H1; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Tritium; Verapamil

1991
Visual recognition memory in squirrel monkeys: effects of serotonin antagonists on baseline and hypoxia-induced performance deficits.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:4

    Topics: Animals; Avoidance Learning; Cognition; Dose-Response Relationship, Drug; Hypoxia; Ketanserin; Male; Memory; Mianserin; Piperidines; Psychomotor Performance; Reinforcement Schedule; Saimiri; Serotonin Antagonists

1991
DOI-induced inhibition of copulatory behavior in male rats: reversal by 5-HT2 antagonists.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:3

    Topics: Amphetamines; Animals; Copulation; Ejaculation; Female; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Tranquilizing Agents

1991
Naloxone and serotonin receptor subtype antagonists: interactive effects upon deprivation-induced intake.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 38, Issue:3

    Topics: Animals; Drug Interactions; Feeding Behavior; Food Deprivation; Indoles; Ketanserin; Male; Methysergide; Naloxone; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Tropisetron

1991
Stimulatory effects of 5-hydroxytryptamine on fluid secretion and transmural potential difference in rat small intestine are mediated by different receptor subtypes.
    The Journal of pharmacy and pharmacology, 1990, Volume: 42, Issue:1

    Topics: Animals; Blood Pressure; Body Fluids; Cisapride; Dose-Response Relationship, Drug; Female; Intestine, Small; Ketanserin; Male; Membrane Potentials; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1990
Laminar distributions of muscarinic acetylcholine, serotonin, GABA and opioid receptors in human posterior cingulate cortex.
    Neuroscience, 1990, Volume: 36, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aged; Autoradiography; Cerebral Cortex; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Humans; Iodocyanopindolol; Ketanserin; Male; Middle Aged; Oxotremorine; Paroxetine; Pindolol; Piperidines; Pirenzepine; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1990
Effects of ketanserin tartrate on 3-hydroxy, 3-methylglutaryl coenzyme A reductase activity in cultured human skin fibroblasts.
    Cardiovascular drugs and therapy, 1990, Volume: 4 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Cells, Cultured; Fibroblasts; Humans; Hydroxymethylglutaryl CoA Reductases; Ketanserin; Piperidines; Prazosin; Ritanserin; Serotonin Antagonists

1990
CGS 18102A, a benzopyranopyridine anxiolytic with 5-HT1 agonist and 5-HT2 antagonist properties.
    Progress in clinical and biological research, 1990, Volume: 361

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Benzopyrans; Binding, Competitive; Cerebral Cortex; Ketanserin; Kinetics; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1990
5-HT1C receptors in the serotonergic control of periaqueductal gray induced aversion in rats.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: Amphetamines; Animals; Cyproheptadine; Indoles; Ketanserin; Male; Periaqueductal Gray; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reinforcement, Psychology; Ritanserin; Serotonin; Serotonin Antagonists

1990
[3H]ketanserin binds to non-5-HT2 sites in rabbit cerebral cortex and neostriatum.
    Neurochemical research, 1990, Volume: 15, Issue:5

    Topics: Animals; Binding, Competitive; Caudate Nucleus; Cell Membrane; Cerebral Cortex; Corpus Striatum; Frontal Lobe; Ketanserin; Kinetics; Male; Methysergide; Mianserin; Piperidines; Putamen; Rabbits; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1990
Inhibition of spontaneous and evoked unit activity in the rat medial prefrontal cortex by mesencephalic raphe nuclei.
    Brain research, 1990, Jul-30, Volume: 524, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Animals; Brain; Cerebral Cortex; Electric Stimulation; Evoked Potentials; Ketanserin; Male; Membrane Potentials; Neurons; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Ritanserin; Serotonin

1990
Inhibition of serotonin-amplified human platelet aggregation by ketanserin, ritanserin, and the ergoline 5HT2 receptor antagonists-LY53857, sergolexole, and LY237733.
    Life sciences, 1990, Volume: 47, Issue:23

    Topics: Adult; Ergolines; Female; Humans; Ketanserin; Lysergic Acid; Male; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1990
5HT-2 mediation of acute behavioral effects of hallucinogens in rats.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Behavior, Animal; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Hallucinogens; Ketanserin; Male; Mescaline; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Tetrahydronaphthalenes

1990
Behavioural evidence for a functional interaction between central 5-HT2 and 5-HT1A receptors.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Behavior, Animal; Central Nervous System; Dose-Response Relationship, Drug; Haloperidol; Ketanserin; Male; Methoxydimethyltryptamines; Piperidines; Prazosin; Pyrimidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Stereotyped Behavior; Tetrahydronaphthalenes

1990
Effect of serotonergic drugs on negative contrast in consummatory behavior.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Animals; Buspirone; Chlordiazepoxide; Cyproheptadine; Dose-Response Relationship, Drug; Ethanol; Feeding Behavior; Fenclonine; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Male; Midazolam; Nucleus Accumbens; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Serotonin Antagonists

1990
Binding of [3H]dihydrotetrabenazine and [125I]azidoiodoketanserin photoaffinity labeling of the monoamine transporter of platelet 5-HT organelles.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: Affinity Labels; Animals; Azides; Biogenic Monoamines; Blood Platelets; Blood Proteins; Cell Membrane; Guinea Pigs; Humans; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Paroxetine; Photochemistry; Piperidines; Rabbits; Rats; Receptors, Serotonin; Subcellular Fractions; Tetrabenazine

1990
Receptor subtypes mediating facilitation by serotonin of excitability of spinal motoneurons.
    Neuropharmacology, 1990, Volume: 29, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; In Vitro Techniques; Injections, Intravenous; Iontophoresis; Ketanserin; Male; Methysergide; Microelectrodes; Motor Neurons; Piperidines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes

1990
Mediation of ACTH and prolactin responses to 5-HTP by 5-HT2 receptors.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: 5-Hydroxytryptophan; Adrenocorticotropic Hormone; Animals; Dose-Response Relationship, Drug; Ketanserin; Male; Metergoline; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone

1990
Acute hypotension due to platelet serotonin-induced chemoreflexes after intravenous injection of dextran sulfate in the rabbit.
    Circulation research, 1985, Volume: 57, Issue:2

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Autonomic Nervous System; Blood Platelets; Bradycardia; Chemoreceptor Cells; Cimetidine; Complement C3; Dextran Sulfate; Dextrans; Factor XII; Histamine; Histamine Release; Hypotension; Injections, Intravenous; Ketanserin; Leukocyte Count; Lung; Male; Methysergide; Piperidines; Rabbits; Serotonin

1985
On the nature of the contractile motor responses of the rat stomach elicited by serotonin or substance P in vitro.
    Journal of neural transmission, 1985, Volume: 63, Issue:1

    Topics: Animals; Atropine; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Stomach; Substance P; Tachyphylaxis; Tetrodotoxin

1985
Effect of ketanserin on hemodynamics, plasma-catecholamine concentrations, and serotonin uptake by platelets in volunteers and patients with congestive heart failure.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Aged; Blood Platelets; Catecholamines; Dopamine; Female; Heart Failure; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Norepinephrine; Piperidines; Serotonin; Serotonin Antagonists; Stroke Volume; Vascular Resistance

1985
Antihypertensive effects of ketanserin in the spontaneously hypertensive rat: mode of action.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Time Factors

1985
Chronic serotonergic blockade with ketanserin in the spontaneously hypertensive rat.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Blood Pressure; Heart Rate; Ketanserin; Male; Piperidines; Rats; Rats, Inbred SHR; Serotonin Antagonists

1985
Evidence for a central component to the hypotensive action of ketanserin in the dog.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Dogs; Ganglionic Blockers; Hexamethonium Compounds; Ketanserin; Mecamylamine; Nicotine; Norepinephrine; Piperidines; Vasoconstriction

1985
Serotonergic mechanisms and blood pressure in sheep.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adrenergic alpha-Antagonists; Adrenocorticotropic Hormone; Animals; Blood Pressure; Female; Heart Rate; Hypertension; Ketanserin; Phenylephrine; Piperidines; Prazosin; Serotonin; Serotonin Antagonists; Sheep

1985
Platelet serotonin in essential hypertension and in mental depression.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Antidepressive Agents; Blood Platelets; Depressive Disorder; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Serotonin; Serotonin Antagonists; Sex Factors

1985
Is there alpha-adrenergic blockade and/or serotonergic blockade during chronic ketanserin treatment?
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Humans; Ketanserin; Malignant Carcinoid Syndrome; Phenylephrine; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists

1985
The acute antihypertensive effect of ketanserin increases with age.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Aged; Aging; Antihypertensive Agents; Blood Pressure; Female; Humans; Hypertension; Injections, Intravenous; Ketanserin; Male; Middle Aged; Piperidines

1985
Ketanserin: a possible tool for studying the role of serotonin in hypertension.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Aldosterone; Blood Pressure; Female; Hemodynamics; Humans; Hypertension; Ketanserin; Male; Middle Aged; Norepinephrine; Phentolamine; Phenylephrine; Piperidines; Regional Blood Flow; Renal Circulation; Renin; Serotonin; Serotonin Antagonists; Time Factors

1985
A comparative and long-term evaluation of ketanserin in the treatment of essential hypertension.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adrenergic beta-Antagonists; Adult; Blood Pressure; Diuretics; Female; Humans; Hypertension; Ketanserin; Male; Piperidines; Serotonin Antagonists; Time Factors

1985
Ketanserin in the acute management of severe hypertension.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adolescent; Adult; Blood Pressure; Creatinine; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Renin; Serotonin Antagonists; Time Factors

1985
Platelet hypersensitivity to serotonin after prolonged ketanserin intake?
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Blood Platelets; Humans; Ketanserin; Male; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists

1985
Continuous inhibition of platelet S2-serotonergic receptors during chronic administration of ketanserin in humans.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adenosine Diphosphate; Blood Platelets; Collagen; Epinephrine; Female; Humans; Ketanserin; Male; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin Antagonists; Time Factors

1985
Blood pressure, 5-OH indoleacetic acid, and vanilmandelic acid excretion and blood platelet aggregation in hypertensive patients treated with ketanserin.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Blood Pressure; Female; Heart Rate; Humans; Hydroxyindoleacetic Acid; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists; Time Factors; Vanilmandelic Acid

1985
Effects of ketanserin on platelet function and red cell filterability in hypertension and peripheral vascular disease.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adult; Aged; Blood Platelets; Erythrocyte Deformability; Erythrocytes; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Serotonin Antagonists; Vascular Diseases

1985
Effects of ketanserin on the intracellular concentration and transmembrane fluxes of sodium and potassium in erythrocytes of normal male subjects.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Cell Membrane Permeability; Erythrocyte Membrane; Erythrocytes; Furosemide; Humans; Ketanserin; Lithium; Male; Ouabain; Piperidines; Potassium; Serotonin Antagonists; Sodium

1985
Serotonin and the blood vessel wall.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Drug Interactions; In Vitro Techniques; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation

1985
Serotonin-induced vasoconstriction in the perfused canine femoral artery can be blocked in vivo by ketanserin.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Blood Pressure; Dogs; Female; Femoral Artery; Hemodynamics; In Vitro Techniques; Isosorbide Dinitrate; Ketanserin; Male; Piperidines; Prazosin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasoconstriction

1985
Influence of ketanserin on 5-hydroxytryptamine-induced cerebrovascular spasm in the cat.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Cats; Cerebrovascular Circulation; Ischemic Attack, Transient; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Serotonin; Serotonin Antagonists

1985
Effects of serotonin on the cardiopulmonary circulatory system with and without 5-HT2-receptor blockade by ketanserin.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Dogs; Hypertension, Pulmonary; Ketanserin; Piperidines; Pulmonary Artery; Pulmonary Embolism; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Resistance

1985
Bucindolol has serotonin and alpha-adrenoceptor blocking properties.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; In Vitro Techniques; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Regional Blood Flow; Serotonin Antagonists

1985
Two classes of myocardial 5-hydroxytryptamine receptors that are neither 5-HT1 nor 5-HT2.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Animals; Cats; Female; Heart Rate; In Vitro Techniques; Ketanserin; Male; Myocardial Contraction; Myocardium; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1985
The pentagastrin test in the diagnosis of the carcinoid syndrome.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Carcinoid Tumor; Female; Gastrointestinal Neoplasms; Humans; Hydroxyindoleacetic Acid; Ketanserin; Male; Malignant Carcinoid Syndrome; Pentagastrin; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Substance P; Time Factors

1985
Large and small vessel responses to serotonin in the peripheral circulation.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 7

    Topics: Arteriosclerosis; Humans; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasodilation; Vasodilator Agents

1985
Intra-erythrocyte concentration and transmembrane fluxes of sodium and potassium during acute and short-term administration of ketanserin in normal male subjects.
    Methods and findings in experimental and clinical pharmacology, 1985, Volume: 7, Issue:9

    Topics: Adult; Erythrocyte Membrane; Erythrocytes; Humans; Ion Channels; Ketanserin; Male; Piperidines; Potassium; Sodium; Sodium-Potassium-Exchanging ATPase

1985
[Effect of ketanserin on blood pressure in rats].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1985, Volume: 86, Issue:6

    Topics: Adrenal Glands; Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hydroxyindoleacetic Acid; Ketanserin; Male; Norepinephrine; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Serotonin; Sympathetic Nervous System

1985
In vivo voltammetry in the suprachiasmatic nucleus of the rat: effects of RU24969, methiothepin and ketanserin.
    European journal of pharmacology, 1986, Feb-11, Volume: 121, Issue:1

    Topics: Animals; Dibenzothiepins; Electrophysiology; Hydroxyindoleacetic Acid; Ketanserin; Male; Methiothepin; Microelectrodes; Oxidation-Reduction; Phenethylamines; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Suprachiasmatic Nucleus; Time Factors

1986
125I-LSD autoradiography confirms the preferential localization of caudate-putamen S2 receptors to the caudal (peripallidal) region.
    Brain research, 1986, Apr-30, Volume: 372, Issue:1

    Topics: Animals; Autoradiography; Butaclamol; Caudate Nucleus; Frontal Lobe; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Putamen; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin

1986
Ketanserin in the preoperative and intraoperative management of a patient with carcinoid tumor undergoing tricuspid valve replacement.
    Anesthesia and analgesia, 1986, Volume: 65, Issue:7

    Topics: Blood Pressure; Carcinoid Tumor; Cardiopulmonary Bypass; Female; Histamine Release; Humans; Intraoperative Care; Intraoperative Complications; Ketanserin; Middle Aged; Piperidines; Preoperative Care; Serotonin; Tricuspid Valve; Tricuspid Valve Insufficiency

1986
Ketanserin and ritanserin can reduce reperfusion-induced but not ischaemia-induced arrhythmias in anaesthetised rats.
    Journal of cardiovascular pharmacology, 1987, Volume: 10, Issue:4

    Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Coronary Vessels; Female; Guinea Pigs; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists

1987
Antihypertensive effects of ketanserin and ritanserin in the spontaneously hypertensive rat.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin; Sympathetic Nervous System

1988
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Ergolines; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pyrimidinones; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone

1988
Are drugs that act both on serotonin receptors and alpha 1-adrenoceptors more potent hypotensive agents than those that act only on alpha 1-adrenoceptors?
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Cats; Cinanserin; Ergolines; Ketanserin; Male; Metergoline; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes

1988
Age-related changes in rat serotonergic and adrenergic systems and in receptor responsiveness to subchronic desipramine treatment.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:3

    Topics: Aging; Animals; Brain; Clonidine; Desipramine; Dihydroalprenolol; Hydroxyindoleacetic Acid; Imipramine; Ketanserin; Kinetics; Male; Paroxetine; Piperidines; Prazosin; Proteins; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Serotonin; Serotonin; Time Factors

1988
Arterial and venous effects of serotonin in the forearm of healthy subjects are not age-related.
    Journal of cardiovascular pharmacology, 1989, Volume: 14, Issue:1

    Topics: Adult; Aged; Aging; Blood Pressure; Forearm; Heart Rate; Humans; Ketanserin; Male; Methoxamine; Middle Aged; Piperidines; Regional Blood Flow; Ritanserin; Serotonin; Serotonin Antagonists

1989
Serotonin as a modulator of skeletal muscle oxygenation: effects of ketanserin and ritanserin on oxygen pressure distributions.
    International journal of microcirculation, clinical and experimental, 1989, Volume: 8, Issue:2

    Topics: Animals; Ketanserin; Muscles; Oxygen; Oxygen Consumption; Piperidines; Pressure; Rabbits; Ritanserin; Serotonin; Serotonin Antagonists

1989
Lack of a difference between ketanserin and ritanserin in central vs. peripheral serotonin receptor antagonism.
    Life sciences, 1989, Volume: 45, Issue:13

    Topics: Animals; Blood Pressure; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1989
Facilitation of 8-OHDPAT-induced forepaw treading of rats by the 5-HT2 agonist DOI.
    European journal of pharmacology, 1989, Feb-14, Volume: 161, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprenolol; Amphetamines; Animals; Behavior, Animal; Cerebral Cortex; Injections, Subcutaneous; Ketanserin; Male; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Tetrahydronaphthalenes

1989
Production of wet-dog shakes in rats and down-regulation of spinal 5-HT2 receptors.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: Animals; Behavior, Animal; Brain Stem; Ketanserin; Male; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spinal Cord

1989
The pentagastrin test in the diagnosis of the carcinoid syndrome. Blockade of gastrointestinal symptoms by ketanserin.
    Annals of surgery, 1985, Volume: 201, Issue:1

    Topics: Aged; Calcium; Digestive System; Female; Humans; Ketanserin; Liver Neoplasms; Male; Malignant Carcinoid Syndrome; Middle Aged; Pentagastrin; Piperidines; Serotonin; Serotonin Antagonists; Substance P; Vasomotor System

1985
Brain dopamine and serotonin receptor sites revealed by digital subtraction autoradiography.
    Science (New York, N.Y.), 1985, May-03, Volume: 228, Issue:4699

    Topics: Animals; Autoradiography; Brain; Butaclamol; Computers; Ketanserin; Piperidines; Radiographic Image Enhancement; Radionuclide Imaging; Rats; Receptors, Dopamine; Receptors, Serotonin; Spiperone; Sulpiride

1985
The effects of a new serotonin receptor antagonist (ketanserin) on lower urinary tract function in patients with prostatism.
    The Journal of urology, 1985, Volume: 133, Issue:6

    Topics: Aged; Blood Pressure; Humans; Ketanserin; Male; Middle Aged; Piperidines; Pressure; Prostatic Hyperplasia; Serotonin Antagonists; Urethra; Urinary Bladder; Urodynamics

1985
Reduction in opioid and non-opioid forms of swim analgesia by 5-HT2 receptor antagonists.
    Brain research, 1989, Oct-23, Volume: 500, Issue:1-2

    Topics: Analgesia; Endorphins; Ketanserin; Methysergide; Physical Exertion; Piperidines; Receptors, Serotonin; Serotonin Antagonists

1989
5-Hydroxytryptamine stimulates the formation of inositol phosphate in astrocytes from different regions of the brain.
    Neuropharmacology, 1987, Volume: 26, Issue:9

    Topics: Animals; Astrocytes; Brain; Cyclic AMP; Inositol Phosphates; Ketanserin; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Stimulation, Chemical; Sugar Phosphates; Tissue Distribution

1987
Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist.
    Molecular pharmacology, 1985, Volume: 27, Issue:6

    Topics: Animals; Binding, Competitive; Biogenic Amines; Brain; Cerebellum; Cerebral Cortex; Corpus Striatum; Female; Guinea Pigs; Haloperidol; Hippocampus; Histamine H2 Antagonists; In Vitro Techniques; Ketanserin; Kinetics; Male; Organ Specificity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1985
Treatment of arterial hypertension with ketanserin in mono- and combination therapy.
    Clinical pharmacology and therapeutics, 1985, Volume: 38, Issue:2

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Blood Pressure; Drug Therapy, Combination; Female; Follow-Up Studies; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Serotonin Antagonists

1985
Hypotensive actions of ketanserin in dogs: involvement of a centrally mediated inhibition of sympathetic vascular tone.
    European journal of pharmacology, 1985, May-20, Volume: 111, Issue:3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Dogs; Female; Heart Rate; Hexamethonium; Hexamethonium Compounds; Ketanserin; Male; Mecamylamine; Nicotine; Piperidines; Sympathetic Nervous System; Vascular Resistance; Vasomotor System

1985
Effect of somatostatin on bethanechol-stimulated gastric acid secretion and gastric antral motility in dogs with gastric fistula.
    Scandinavian journal of gastroenterology, 1985, Volume: 20, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Bethanechol Compounds; Dogs; Domperidone; Dose-Response Relationship, Drug; Female; Gastric Acid; Gastric Fistula; Gastrointestinal Motility; Ketanserin; Male; Piperidines; Propranolol; Pyloric Antrum; Receptors, Dopamine; Receptors, Serotonin; Somatostatin

1985
Dopamine D2 receptors selectively labeled by a benzamide neuroleptic: [3H]-YM-09151-2.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Corpus Striatum; Dogs; Guanylyl Imidodiphosphate; Ketanserin; Kinetics; Piperidines; Receptors, Dopamine; Sodium; Spiperone; Substrate Specificity; Tetrahydronaphthalenes

1985
[Endocrine and metabolic changes induced in surgery by the combination of ketanserin and alfentanyl].
    Agressologie: revue internationale de physio-biologie et de pharmacologie appliquees aux effets de l'agression, 1985, Volume: 26, Issue:7

    Topics: Abdomen; Adolescent; Adult; Aged; Alfentanil; Analgesics, Opioid; Drug Therapy, Combination; Female; Fentanyl; Humans; Intraoperative Complications; Ketanserin; Male; Middle Aged; Piperidines; Premedication; Serotonin Antagonists; Stress, Physiological

1985
Mechanism of the hypotensive effect of a novel phenylpiperazine derivative, SGB-1534: antagonism at alpha 1-adrenergic and 5-HT2 receptors.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 277, Issue:1

    Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Antihypertensive Agents; Decerebrate State; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Piperidines; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Serotonin Antagonists

1985
Differential effect of subchronic treatment with various neuroleptic agents on serotonin2 receptors in rat cerebral cortex.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Animals; Antipsychotic Agents; Cerebral Cortex; Chlorpromazine; Clozapine; Female; Haloperidol; Imipramine; Ketanserin; Loxapine; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Sulpiride

1986
[Ketanserin in association with a beta blocker and a diuretic in the treatment of essential hypertension].
    Bollettino chimico farmaceutico, 1985, Volume: 124, Issue:10

    Topics: Adrenergic beta-Antagonists; Blood Pressure; Diuretics; Drug Therapy, Combination; Humans; Hypertension; Ketanserin; Piperidines

1985
Ketanserin in intermittent claudication.
    Lancet (London, England), 1986, Mar-15, Volume: 1, Issue:8481

    Topics: Humans; Intermittent Claudication; Ketanserin; Piperidines

1986
Serotonin receptor involvement in the avoidance learning deficit caused by p-chloroamphetamine-induced serotonin release.
    Acta physiologica Scandinavica, 1986, Volume: 126, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Amphetamines; Animals; Avoidance Learning; Brain; Ketanserin; Male; p-Chloroamphetamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Histamine H1; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Serotonin

1986
Studies on the receptor profile of bisoprolol.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Bisoprolol; Cattle; Dihydroalprenolol; Domperidone; Humans; In Vitro Techniques; Ketanserin; Male; Piperidines; Prazosin; Propanolamines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Histamine; Receptors, Muscarinic; Spiperone; Tetrahydronaphthalenes; Yohimbine

1986
Characterization of flufylline, fluprofylline, ritanserin, butanserin and R 56413 with respect to in-vivo alpha 1-,alpha 2- and 5-HT2-receptor antagonism and in-vitro affinity for alpha 1-,alpha 2- and 5-HT2-receptors: comparison with ketanserin.
    The Journal of pharmacy and pharmacology, 1986, Volume: 38, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Decerebrate State; Histamine H2 Antagonists; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Theophylline; Vasoconstriction

1986
Typical and atypical antipsychotic occupancy of D2 and S2 receptors: an autoradiographic analysis in rat brain.
    Brain research bulletin, 1986, Volume: 16, Issue:4

    Topics: Animals; Antipsychotic Agents; Autoradiography; Binding, Competitive; Brain; Caudate Nucleus; Haloperidol; Ketanserin; Kinetics; Male; Nucleus Accumbens; Olfactory Bulb; Piperidines; Putamen; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Spiperone

1986
Permissive role of D-1 receptor stimulation by endogenous dopamine for the expression of postsynaptic D-2-mediated behavioural responses. Yawning in rats.
    European journal of pharmacology, 1987, Feb-10, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Azepines; Benzazepines; Brain Chemistry; Dopamine; Ergolines; Kainic Acid; Ketanserin; Male; Metergoline; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sulpiride; Yawning

1987
Quipazine reduces food intake in the rat by activation of 5-HT2-receptors.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: Animals; Diet; Dose-Response Relationship, Drug; Eating; Histamine H2 Antagonists; Imidazoles; Ketanserin; Methysergide; Ondansetron; Pindolol; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1988
Antagonism of the LSD cue by putative serotonin antagonists: relationship to inhibition of in vivo [3H]spiroperidol binding.
    Behavioural brain research, 1985, Volume: 16, Issue:2-3

    Topics: Animals; Cerebellum; Corpus Striatum; Frontal Lobe; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Pizotyline; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin

1985
Behavioural stimulation is induced by separate dopamine D-1 and D-2 receptor sites in reserpine-pretreated but not in normal rats.
    European journal of pharmacology, 1985, Jul-11, Volume: 113, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Catalepsy; Ergolines; Hydroxydopamines; Ketanserin; Male; Motor Activity; Oxidopamine; Pergolide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Stereotyped Behavior

1985
The effects of ketanserin, methysergide and LY 53857 on sympathetic nerve activity.
    European journal of pharmacology, 1985, Jul-31, Volume: 113, Issue:3

    Topics: Anesthesia; Animals; Blood Pressure; Cats; Ergolines; Heart Rate; Hemodynamics; Ketanserin; Lactates; Lactic Acid; Male; Methysergide; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Sympathetic Nervous System

1985
Mechanisms involved in the vasodilator action of 5-hydroxytryptamine in the dog femoral arterial circulation in vivo.
    European journal of pharmacology, 1985, Jul-31, Volume: 113, Issue:3

    Topics: Animals; Blood Pressure; Carbon Dioxide; Dogs; Dose-Response Relationship, Drug; Female; Femoral Artery; Hindlimb; Ketanserin; Male; Muscle, Smooth, Vascular; Ornipressin; Piperidines; Pizotyline; Regional Blood Flow; Serotonin; Sympathetic Nervous System; Vasodilator Agents

1985
Solubilization of rat brain serotonin-S2 receptors using CHAPS/salt.
    European journal of pharmacology, 1985, Sep-10, Volume: 115, Issue:1

    Topics: Animals; Brain Chemistry; Centrifugation, Density Gradient; Cholic Acids; Filtration; In Vitro Techniques; Ketanserin; Microsomes; Nerve Tissue Proteins; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Sodium Chloride

1985
Analysis of the heart rate effects of 5-hydroxytryptamine in the cat; mediation of tachycardia by 5-HT1-like receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 330, Issue:2

    Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Isoproterenol; Ketanserin; Male; Methysergide; Piperidines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tropanes; Vagus Nerve

1985
Hemodynamic evaluation of endotoxic shock in anesthetized piglets: antagonism of endogenous vasoactive substances.
    Circulatory shock, 1985, Volume: 16, Issue:1

    Topics: Adrenal Cortex Hormones; Anesthesia; Animals; Bacterial Toxins; Blood Pressure; Cardiac Output; Enterotoxins; Escherichia coli Proteins; Flurbiprofen; Heart Rate; Hemodynamics; Ketanserin; Narcotic Antagonists; Piperidines; Prednisone; Pulmonary Circulation; Serotonin Antagonists; Shock, Septic; Swine; Time Factors; Vascular Resistance

1985
Spiperone differentiates multiple 5-hydroxytryptamine responses in rat hippocampal slices in vitro.
    European journal of pharmacology, 1985, Oct-08, Volume: 116, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Butyrophenones; Hippocampus; In Vitro Techniques; Ketanserin; Piperidines; Rats; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes

1985
Effect of serotonin and its antagonist ketanserin on pial vessels.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1985, Volume: 5, Issue:4

    Topics: Administration, Topical; Animals; Arteries; Carbon Dioxide; Cats; Cerebrovascular Circulation; Ketanserin; Oxygen; Pia Mater; Piperidines; Rest; Serotonin; Serotonin Antagonists; Veins

1985
Peripheral serotonin2 receptor blockade does not inhibit 5-hydroxytryptophan-induced aldosterone stimulation.
    The Journal of clinical endocrinology and metabolism, 1985, Volume: 61, Issue:6

    Topics: 5-Hydroxytryptophan; Adult; Aldosterone; Humans; Ketanserin; Male; Methysergide; Piperidines; Potassium; Renin; Serotonin; Serotonin Antagonists

1985
Effects of ketanserin, a 5-HT2-receptor antagonist, on the blood flow response to temperature changes in the diabetic foot.
    Journal of clinical pharmacology, 1985, Volume: 25, Issue:6

    Topics: Adult; Aged; Diabetes Mellitus; Female; Foot; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Piperidines; Plethysmography; Regional Blood Flow; Serotonin Antagonists; Temperature

1985
Effects of serotonin receptor agonists and antagonists on schedule-controlled behavior of squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Cinanserin; Conditioning, Operant; Cyproheptadine; Electroshock; Female; Ketanserin; Male; Metergoline; Methysergide; Piperazines; Piperidines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri

1985
A comparison of cardiovascular and smooth muscle effects of 5-hydroxytryptamine and 5-carboxamidotryptamine, a selective agonist of 5-HT1 receptors.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 277, Issue:2

    Topics: Airway Resistance; Animals; Cyproheptadine; Guinea Pigs; Heart Rate; Hemodynamics; Ileum; In Vitro Techniques; Ketanserin; Male; Mecamylamine; Methysergide; Muscle, Smooth; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Urinary Bladder

1985
Monoaminergic involvement in the pharmacological actions of buspirone.
    British journal of pharmacology, 1985, Volume: 86, Issue:3

    Topics: Animals; Apomorphine; Behavior, Animal; Brain; Buspirone; Dopamine; Ketanserin; Male; Methoxydimethyltryptamines; Monoamine Oxidase; p-Chloroamphetamine; Piperazines; Piperidines; Psychotropic Drugs; Pyrimidines; Rats; Serotonin

1985
A comparison of 5-hydroxytryptamine receptors mediating contraction in rabbit aorta and dog saphenous vein: evidence for different receptor types obtained by use of selective agonists and antagonists.
    British journal of pharmacology, 1985, Volume: 86, Issue:3

    Topics: Animals; Aorta; Dogs; In Vitro Techniques; Ketanserin; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rabbits; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Antagonists; Spiperone

1985
Relationship of increased lung serotonin levels to endotoxin-induced pulmonary hypertension in sheep. Effect of a serotonin antagonist.
    The American review of respiratory disease, 1985, Volume: 132, Issue:6

    Topics: Animals; Blood Pressure; Endotoxins; Escherichia coli; Hypertension, Pulmonary; Hypoxia; Ketanserin; Lung; Lymph; Oxygen; Piperidines; Platelet Count; Pulmonary Artery; Serotonin; Serotonin Antagonists; Sheep

1985
Lack of effect of propranolol on the steady-state plasma levels of ketanserin.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:8

    Topics: Adult; Blood Pressure; Female; Heart Rate; Humans; Ketanserin; Liver; Male; Middle Aged; Piperidines; Propranolol; Time Factors

1985
Chronic 5-HT2 receptor blockade with ritanserin does not reduce blood pressure in the spontaneously hypertensive rat.
    Journal of neural transmission, 1985, Volume: 64, Issue:2

    Topics: Animals; Blood Pressure; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Heart Rate; Hypertension; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Receptors, Serotonin; Ritanserin; Time Factors

1985
Different subcellular localization of muscarinic and serotonin (S2) receptors in human, dog, and rat brain.
    Journal of neurochemistry, 1986, Volume: 46, Issue:2

    Topics: Adult; Aged; Animals; Brain; Brain Chemistry; Centrifugation, Density Gradient; Dexetimide; Dogs; Humans; Ketanserin; Mathematics; Microscopy, Electron; Middle Aged; Piperidines; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Receptors, Serotonin; Species Specificity; Subcellular Fractions

1986
In vitro and in vivo irreversible blockade of cortical S2 serotonin receptors by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline: a technique for investigating S2 serotonin receptor recovery.
    Journal of neurochemistry, 1986, Volume: 46, Issue:2

    Topics: Animals; Cerebral Cortex; Domperidone; Dose-Response Relationship, Drug; Ketanserin; Kinetics; Male; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin

1986
Characterization of 5-hydroxytryptamine receptors in rat stomach fundus.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:3

    Topics: Animals; Binding, Competitive; Brain Chemistry; Gastric Fundus; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Piperazines; Piperidines; Propranolol; Pyrazines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium

1985
Serotonin type 2 antagonists inhibit lordosis behavior in the female rat: reversal with quipazine.
    Life sciences, 1986, Jan-06, Volume: 38, Issue:1

    Topics: Analysis of Variance; Animals; Butyrophenones; Cyproheptadine; Estradiol; Female; Ketanserin; Methiothepin; Piperidines; Pizotyline; Posture; Progesterone; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Sexual Behavior, Animal

1986
Reactivity of the bronchial artery to 5-hydroxytryptamine.
    Research communications in chemical pathology and pharmacology, 1985, Volume: 50, Issue:3

    Topics: Animals; Bronchial Arteries; Cattle; Female; Horses; In Vitro Techniques; Ketanserin; Male; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sheep; Vasoconstriction

1985
Solubilized ketanserin binding sites from pig platelet membranes.
    Thrombosis research, 1985, Sep-15, Volume: 39, Issue:6

    Topics: Animals; Binding Sites; Binding, Competitive; Blood Platelets; Cell Membrane; In Vitro Techniques; Ketanserin; Kinetics; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Solubility; Swine

1985
Peripheral arterial diseases: treatment with ketanserin as i.v. infusion. An open study in 20 patients.
    Bollettino chimico farmaceutico, 1985, Volume: 124, Issue:10

    Topics: Arteriosclerosis; Humans; Infusions, Parenteral; Ketanserin; Piperidines; Regional Blood Flow

1985
Subtypes of the 5-HT receptor mediating the behavioural responses to 5-methoxy-N,N-dimethyltryptamine in the rat.
    European journal of pharmacology, 1985, Oct-29, Volume: 117, Issue:1

    Topics: Animals; Apomorphine; Behavior, Animal; Betaxolol; Haloperidol; Ketanserin; Male; Pindolol; Piperidines; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reserpine; Spiperone

1985
Molecular pharmacology of 5-HT1 and 5-HT2 recognition sites in rat and pig brain membranes: radioligand binding studies with [3H]5-HT, [3H]8-OH-DPAT, (-)[125I]iodocyanopindolol, [3H]mesulergine and [3H]ketanserin.
    European journal of pharmacology, 1985, Nov-26, Volume: 118, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Chemistry; Choroid Plexus; Ergolines; In Vitro Techniques; Iodocyanopindolol; Ketanserin; Male; Membranes; Pindolol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tetrahydronaphthalenes

1985
Drug treatment of claudication: vasodilators, hemorrheologic agents, and antiserotonin drugs.
    Journal of vascular surgery, 1986, Volume: 3, Issue:2

    Topics: Double-Blind Method; Erythrocyte Deformability; Humans; Intermittent Claudication; Ketanserin; Pentoxifylline; Piperidines; Serotonin Antagonists; Theobromine; Vasodilator Agents

1986
In vivo regulation of the serotonin-2 receptor in rat brain.
    Life sciences, 1986, Jan-13, Volume: 38, Issue:2

    Topics: Amitriptyline; Animals; Brain Chemistry; Electroshock; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tritium

1986
[In vivo study of central serotoninergic receptors in man using positron tomography].
    Revue neurologique, 1985, Volume: 141, Issue:8-9

    Topics: Brain; Cerebellum; Chlorpromazine; Frontal Lobe; Humans; Ketanserin; Kinetics; Piperidines; Receptors, Serotonin; Tomography, Emission-Computed

1985
Dependence of the antagonism at human platelet 5-HT2 receptors by ketanserin on the reaction pH.
    Thrombosis research, 1985, Dec-01, Volume: 40, Issue:5

    Topics: Amidines; Blood Platelets; Butyrophenones; Cyproheptadine; Female; Humans; Hydrogen-Ion Concentration; Ketanserin; Kinetics; Male; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1985
Characterization and localization of serotonin receptors in human brain postmortem.
    Brain research, 1986, Jan-15, Volume: 363, Issue:1

    Topics: Adult; Aged; Autoradiography; Binding, Competitive; Diencephalon; Female; Frontal Lobe; Hippocampus; Humans; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin; Spiperone; Telencephalon

1986
Serotonin as a mediator of cyclic flow variations in stenosed canine coronary arteries.
    Circulation, 1986, Volume: 73, Issue:3

    Topics: Animals; Coronary Circulation; Coronary Disease; Coronary Vessels; Dogs; Hemodynamics; Ketanserin; Male; Periodicity; Piperidines; Serotonin

1986
Comparative effects of oxygen, nifedipine and ketanserin in hypoxic pulmonary hypertension.
    Cor et vasa, 1985, Volume: 27, Issue:6

    Topics: Adult; Carbon Dioxide; Cardiac Output; Female; Heart Rate; Humans; Hypertension, Pulmonary; Hypoxia; Ketanserin; Lung Diseases, Obstructive; Lung Volume Measurements; Male; Middle Aged; Nifedipine; Oxygen; Oxygen Inhalation Therapy; Piperidines; Pulmonary Wedge Pressure; Serotonin Antagonists

1985
Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:1

    Topics: Animals; Cerebral Cortex; In Vitro Techniques; Isoproterenol; Ketanserin; Kinetics; Male; Pindolol; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Subcellular Fractions; Swine

1986
Stereoselective blockade at the 5-HT autoreceptor and inhibition of radioligand binding to central 5-HT recognition sites by the optical isomers of methiothepin.
    Neuropharmacology, 1986, Volume: 25, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dibenzothiepins; Frontal Lobe; In Vitro Techniques; Ketanserin; Male; Methiothepin; Piperidines; Rats; Receptors, Serotonin; Serotonin; Stereoisomerism; Tetrahydronaphthalenes

1986
Effects of MK-212 (6-chloro-2[1-piperazinyl]pyrazine) on schedule-controlled behavior and their reversal by 5-HT antagonists in the pigeon.
    Neuropharmacology, 1986, Volume: 25, Issue:1

    Topics: Animals; Columbidae; Conditioning, Operant; Cues; Generalization, Stimulus; Ketanserin; Male; Metergoline; Methysergide; Piperidines; Pyrazines; Receptors, Serotonin; Reinforcement Schedule

1986
Antimyoclonic properties of S2 serotonin receptor antagonists in the rat.
    Neuropharmacology, 1986, Volume: 25, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Brain Chemistry; Butyrophenones; Cinanserin; Ketanserin; Male; Myoclonus; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1986
Catecholamine release and potentiation of thromboxane A2 production by nicotine in the greyhound.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Pressure; Catecholamines; Dioxanes; Dogs; Epinephrine; Female; Heart Rate; Idazoxan; Imidazoles; In Vitro Techniques; Ketanserin; Male; Nicotine; Phenoxybenzamine; Piperidines; Thromboxane A2; Vasoconstriction

1986
5-Carboxamidotryptamine is a selective agonist at 5-hydroxytryptamine receptors mediating vasodilatation and tachycardia in anaesthetized cats.
    British journal of pharmacology, 1986, Volume: 87, Issue:2

    Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Ketanserin; Male; Methiothepin; Methysergide; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasodilation

1986
Ketanserin (S2-receptor blocking agent), platelet activity and chronic alcoholism.
    International journal of clinical pharmacology research, 1986, Volume: 6, Issue:1

    Topics: Adult; Alcoholism; beta-Thromboglobulin; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Serotonin Antagonists

1986
Ketanserin (S2-receptor blocking agents), hypertension and chronic alcoholism.
    International journal of clinical pharmacology research, 1986, Volume: 6, Issue:1

    Topics: Adult; Alcoholism; Antihypertensive Agents; Blood Pressure; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Time Factors

1986
Monocrotaline pyrrole-induced cardiopulmonary toxicity is not altered by metergoline or ketanserin.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:1

    Topics: Angiotensin II; Animals; Blood Platelets; Blood Pressure; Cardiomegaly; Ergolines; Ketanserin; Lung; Male; Metergoline; Monocrotaline; Organ Size; Piperidines; Pyrrolizidine Alkaloids; Rats; Receptors, Serotonin; Serotonin

1986
Ketanserin and malignant hyperthermia in pigs.
    Acta anaesthesiologica Scandinavica, 1986, Volume: 30, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Body Temperature; Carbon Dioxide; Halothane; Heart Rate; Hydrogen-Ion Concentration; Ketanserin; Lactates; Malignant Hyperthermia; Piperidines; Potassium; Serotonin Antagonists; Succinylcholine; Swine

1986
Postnatal ontogeny of dopamine D2 receptors in rat striatum.
    Biochemical pharmacology, 1986, Apr-01, Volume: 35, Issue:7

    Topics: Age Factors; Animals; Animals, Newborn; Corpus Striatum; Ketanserin; Kinetics; Mathematics; Piperidines; Rats; Receptors, Dopamine; Spiperone

1986
Symposium on serotonin and cardiovascular regulation: a new approach to hypertension. Satellite symposium of the Second European Meeting on Hypertension. 9 June 1985, Milan, Italy.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Animals; Humans; Hypertension; Ketanserin; Piperidines; Serotonin; Serotonin Antagonists

1986
Nitroprusside and ketanserin in the treatment of postoperative hypertension following coronary artery bypass grafting: a haemodynamic and ventilatory comparison.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Blood Pressure; Coronary Artery Bypass; Female; Ferricyanides; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Nitroprusside; Piperidines; Postoperative Complications; Pulmonary Artery; Vascular Resistance

1986
Potentiation of vasoconstrictor responses to serotonin in the limb of atherosclerotic monkeys.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Animals; Arteriosclerosis; Hindlimb; Hypercholesterolemia; Ketanserin; Macaca fascicularis; Methysergide; Piperidines; Serotonin; Vasoconstriction

1986
Serotonin and the blood vessel wall.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Animals; Blood Platelets; Heart; Hypertension; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred SHR; Serotonin; Vasoconstriction; Vasodilation

1986
Serotonin and cardiovascular regulation: a new approach to hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Cardiovascular Diseases; Drug Therapy, Combination; Humans; Hypertension; Ketanserin; Piperidines; Serotonin

1986
Augmentation of vasoconstrictor responses to serotonin by acute and chronic factors: inhibition by ketanserin.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Animals; Drug Synergism; Ketanserin; Norepinephrine; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Sheep; Vasoconstriction; Vasodilation

1986
Renal effects of ketanserin in essential hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adult; Angiotensins; Female; Glomerular Filtration Rate; Humans; Hypertension; Ketanserin; Kidney; Male; Middle Aged; Piperidines; Renin

1986
Regional haemodynamics and antihypertensive effects during long-term ketanserin treatment.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Female; Hemodynamics; Humans; Hypertension; Ketanserin; Long-Term Care; Male; Middle Aged; Piperidines

1986
Contractions of isolated canine coronary arteries resistant to S2-serotonergic blockade.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Angiotensin II; Animals; Blood Platelets; Cocaine; Coronary Vessels; Cyproheptadine; Dibenzothiepins; Dinoprost; Dogs; Drug Resistance; Endothelium; Femoral Artery; In Vitro Techniques; Ketanserin; Methiothepin; Piperidines; Potassium; Prostaglandins F; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sympathetic Nervous System; Vasoconstriction

1986
Receptor-mediated effects of serotonin and 5-methoxytryptamine on noradrenaline release in the rat vena cava and in the heart of the pithed rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2

    Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Decerebrate State; Desipramine; Electric Stimulation; Heart; Heart Rate; Ketanserin; Male; Myocardium; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Tryptamines; Vagotomy; Vena Cava, Inferior

1986
Effects of ketanserin, a selective 5-HT2 serotonergic antagonist, on the secondary recruitment of human platelets in vitro.
    Agents and actions, 1986, Volume: 17, Issue:5-6

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Blood Platelets; Collagen; Epinephrine; Humans; Ketanserin; Kinetics; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1986
Binding sites for [3H]dopamine and dopamine-antagonists on cultured astrocytes of rat striatum and spinal cord: an autoradiographic study.
    Neuroscience letters, 1986, Apr-11, Volume: 65, Issue:2

    Topics: Animals; Astrocytes; Autoradiography; Binding Sites; Cells, Cultured; Corpus Striatum; Domperidone; Dopamine; Dopamine Antagonists; Flupenthixol; Ketanserin; Piperidines; Rats; Spinal Cord; Spiperone; Stereoisomerism; Tritium

1986
A unique serotonin receptor in choroid plexus is linked to phosphatidylinositol turnover.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:11

    Topics: Animals; Cerebral Cortex; Choroid Plexus; In Vitro Techniques; Ketanserin; Mianserin; Phosphatidylinositols; Piperidines; Rats; Receptors, Serotonin; Spiperone

1986
Continuous inhibition of the platelet S2-serotonergic receptors during the long term administration of ketanserin.
    Thrombosis research, 1986, Jun-01, Volume: 42, Issue:5

    Topics: Blood Platelets; Humans; Ketanserin; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin

1986
Serotonin receptors in the human brain. II. Characterization and autoradiographic localization of 5-HT1C and 5-HT2 recognition sites.
    Brain research, 1986, Jun-18, Volume: 376, Issue:1

    Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Cerebral Cortex; Choroid Plexus; Ergolines; Female; Humans; Ketanserin; Male; Membranes; Middle Aged; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tissue Distribution; Tritium

1986
The effect of ketanserin on hypoxia-induced vasoconstriction in isolated lungs.
    International journal of microcirculation, clinical and experimental, 1986, Volume: 5, Issue:1

    Topics: Animals; Hypoxia; In Vitro Techniques; Ketanserin; Lung; Perfusion; Piperidines; Pulmonary Circulation; Rats; Rats, Inbred Strains; Vasoconstriction

1986
Cardiovascular effects of ketanserin in conscious rabbits.
    Japanese heart journal, 1986, Volume: 27, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension, Renovascular; Injections, Intravenous; Ketanserin; Male; Norepinephrine; Piperidines; Rabbits; Renin; Serotonin Antagonists

1986
Regional and selective changes in blood flow of the feline small intestine induced by endoluminal serotonin.
    Acta physiologica Scandinavica, 1986, Volume: 127, Issue:2

    Topics: Animals; Atropine; Cats; Intestinal Mucosa; Jejunum; Ketanserin; Male; Microspheres; Perfusion; Piperidines; Receptors, Muscarinic; Receptors, Serotonin; Regional Blood Flow; Serotonin

1986
Peri-operative management of carcinoid syndrome using ketanserin.
    Anaesthesia, 1986, Volume: 41, Issue:6

    Topics: Aged; Antihypertensive Agents; Embolization, Therapeutic; Female; Hepatic Artery; Humans; Hypertension; Intraoperative Period; Ketanserin; Malignant Carcinoid Syndrome; Piperidines

1986
Effects of noradrenaline, serotonin, and selected antagonists on the vascular smooth muscle of normal and dystrophic chickens.
    Canadian journal of physiology and pharmacology, 1986, Volume: 64, Issue:5

    Topics: Animals; Chickens; Dose-Response Relationship, Drug; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Muscular Dystrophy, Animal; Norepinephrine; Organ Size; Piperidines; Prazosin; Reference Values; Serotonin; Serotonin Antagonists; Tetrodotoxin

1986
Serotonin, norepinephrine, and histamine mediation of endothelial cell barrier function in vitro.
    Journal of cellular physiology, 1986, Volume: 128, Issue:2

    Topics: Animals; Aorta; Cattle; Cell Line; Cells, Cultured; Diffusion; Diphenhydramine; Endothelium; Histamine; Ketanserin; Norepinephrine; Phenoxybenzamine; Piperidines; Propranolol; Serotonin; Serum Albumin, Bovine; Trypan Blue

1986
[3H]ketanserin (serotonin type 2) binding increases in rat cortex following basal forebrain lesions with ibotenic acid.
    Journal of neurochemistry, 1986, Volume: 47, Issue:3

    Topics: Animals; Cerebral Cortex; Choline O-Acetyltransferase; Diencephalon; Frontal Lobe; Hippocampus; Ibotenic Acid; Ketanserin; Male; Oxazoles; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Telencephalon

1986
Comparative effects of ketanserin, atropine and methysergide on the gastrointestinal effects of hyperserotoninemia in the awake dog.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:2

    Topics: Animals; Atropine; Digestive System; Dogs; Gastrointestinal Motility; Ketanserin; Methysergide; Piperidines; Receptors, Serotonin; Serotonin; Water-Electrolyte Balance

1986
The influence of ketanserin on hemostasis in vitro.
    Thrombosis research, 1986, Jul-15, Volume: 43, Issue:2

    Topics: Adenosine Diphosphate; Adult; Blood Coagulation; Collagen; Epinephrine; Female; Fibrinolysis; Hemostasis; Humans; In Vitro Techniques; Ketanserin; Male; Piperidines; Platelet Aggregation; Serotonin Antagonists

1986
Cold hands after exposure to arsenic or vibrating tools: effects of ketanserin on finger blood pressure and skin temperature.
    Acta pharmacologica et toxicologica, 1986, Volume: 58, Issue:5

    Topics: Administration, Oral; Adult; Arsenic Poisoning; Blood Pressure; Double-Blind Method; Hand; Humans; Injections, Intravenous; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation; Raynaud Disease; Regional Blood Flow; Skin Temperature; Vibration

1986
Comparisons between the in vitro binding of two substituted benzamides and two butyrophenones to dopamine-D2 receptors in the rat striatum.
    Acta pharmacologica et toxicologica, 1986, Volume: 58, Issue:5

    Topics: Animals; Benzamides; Butyrophenones; Corpus Striatum; Domperidone; In Vitro Techniques; Ketanserin; Kinetics; Male; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride

1986
Intrapartum treatment of preeclamptic hypertension by ketanserin.
    American journal of obstetrics and gynecology, 1986, Volume: 155, Issue:2

    Topics: Blood Pressure; Female; Fetal Heart; Heart Rate; Humans; Hypertension; Ketanserin; Obstetric Labor Complications; Piperidines; Pre-Eclampsia; Pregnancy; Uterine Contraction

1986
The increase in testicular vascular permeability induced by human chorionic gonadotrophin involves 5-hydroxytryptamine and possibly oestrogens, but not testosterone, prostaglandins, histamine or bradykinin.
    The Australian journal of experimental biology and medical science, 1986, Volume: 64 ( Pt 2)

    Topics: Aminoglutethimide; Androstatrienes; Animals; Aromatase Inhibitors; Bradykinin; Capillary Permeability; Chorionic Gonadotropin; Dihydrotestosterone; Estrogens; Histamine; Ketanserin; Kinetics; Male; Piperidines; Prostaglandins; Rats; Rats, Inbred Strains; Serotonin; Testis; Testosterone

1986
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
    British journal of pharmacology, 1986, Volume: 88, Issue:3

    Topics: Animals; Aorta, Thoracic; In Vitro Techniques; Jugular Veins; Ketanserin; Male; Methysergide; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Trazodone

1986
Allosteric properties of 5-HT2 receptors in tracheal smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:2

    Topics: Allosteric Regulation; Animals; Binding, Competitive; Cattle; Female; Guinea Pigs; Ketanserin; Kinetics; Male; Methysergide; Models, Biological; Muscle Relaxation; Muscle, Smooth; Piperidines; Potassium; Receptors, Serotonin; Serotonin; Species Specificity; Trachea

1986
Serotonin increases the production of inositol phosphates and mobilises calcium via the 5-HT2 receptor in A7r5 smooth muscle cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:2

    Topics: Animals; Aorta; Calcium; Cell Line; Cerebral Cortex; Inositol Phosphates; Ketanserin; Kinetics; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sugar Phosphates; Time Factors

1986
Modulation of the serotonin S2-receptor in brain after chronic lithium.
    Neurochemical research, 1986, Volume: 11, Issue:7

    Topics: Animals; Cerebral Cortex; Corpus Striatum; Domperidone; Ketanserin; Kinetics; Lithium; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin

1986
Hypertension and tachycardia produced by inhibition of reuptake of 5-hydroxytryptamine by fluoxetine in the rat.
    Neuropharmacology, 1986, Volume: 25, Issue:7

    Topics: Adrenalectomy; Animals; Blood Pressure; Brain; Female; Fluoxetine; Heart Rate; Injections, Intraventricular; Ketanserin; Piperidines; Propylamines; Rats; Rats, Inbred Strains; Serotonin; Vagotomy

1986
Does ketanserin relieve frostbite?
    The Practitioner, 1986, Volume: 230, Issue:1415

    Topics: Adult; Frostbite; Humans; Ketanserin; Male; Piperidines; Serotonin Antagonists

1986
Harmine reverses the inhibition of lordosis by the 5-HT2 antagonists pirenperone and ketanserin in the female rat.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:1

    Topics: Alkaloids; Animals; Estradiol; Female; Harmine; Ketanserin; Ovariectomy; Piperidines; Posture; Progesterone; Rats; Rats, Inbred Strains; Receptors, Serotonin; Sexual Behavior, Animal

1986
Discriminative stimulus properties of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH DPAT).
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Discrimination Learning; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ketanserin; Male; Naphthalenes; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes

1986
A sensitive model of venous thrombosis in rats.
    Thrombosis research, 1986, Sep-01, Volume: 43, Issue:5

    Topics: Animals; Anticoagulants; Aspirin; Dipyridamole; Disease Models, Animal; Female; Heparin; Ketanserin; Piperidines; Rats; Rats, Inbred Strains; Sulfinpyrazone; Thrombophlebitis; Time Factors

1986
Antithrombotics in view of thrombosis models.
    Thrombosis research, 1986, Sep-01, Volume: 43, Issue:5

    Topics: Animals; Anticoagulants; Arteries; Aspirin; Dipyridamole; Female; Hydroxyethylrutoside; Ketanserin; Piperidines; Pizotyline; Prenylamine; Rats; Rats, Inbred Strains; Sulfinpyrazone; Thrombophlebitis; Thrombosis

1986
Adenosine-induced contractions of the isolated rat trachea are mediated by 5-hydroxytryptamine.
    Acta physiologica Scandinavica, 1986, Volume: 127, Issue:4

    Topics: Adenosine; Animals; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Trachea

1986
Ketanserin and the cardiovascular system. 1. Modification of the effects of pressor amines in patients undergoing myocardial revascularisation.
    Anaesthesia, 1986, Volume: 41, Issue:7

    Topics: Angiotensin II; Antihypertensive Agents; Cardiopulmonary Bypass; Drug Evaluation; Hemodynamics; Humans; Ketanserin; Middle Aged; Myocardial Revascularization; Norepinephrine; Phenylephrine; Piperidines

1986
Thermoregulatory responses to serotonin (5-HT) receptor stimulation in the rat. Evidence for opposing roles of 5-HT2 and 5-HT1A receptors.
    Neuropharmacology, 1986, Volume: 25, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature Regulation; Ketanserin; Male; Methoxydimethyltryptamines; Pindolol; Piperidines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes

1986
Regional and subcellular localization in human brain of [3H]paroxetine binding, a marker of serotonin uptake sites.
    Biological psychiatry, 1988, Volume: 24, Issue:3

    Topics: Adult; Aged; Animals; Binding, Competitive; Brain; Brain Mapping; Cerebral Cortex; Corpus Striatum; Humans; Ketanserin; Male; Middle Aged; Paroxetine; Piperidines; Putamen; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Subcellular Fractions; Synaptosomes

1988
[3H]vesamicol binding in brain: autoradiographic distribution, pharmacology, and effects of cholinergic lesions.
    Synapse (New York, N.Y.), 1988, Volume: 2, Issue:5

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Autoradiography; Brain; Cholinergic Fibers; Frontal Lobe; Haloperidol; Hippocampus; Image Processing, Computer-Assisted; Ketanserin; Male; Neural Pathways; Neurotransmitter Uptake Inhibitors; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains

1988
Changes in cortical 5-HT2 receptors following 5-HTP and paroxetine administration in rats.
    The Journal of Nihon University School of Dentistry, 1988, Volume: 30, Issue:3

    Topics: Animals; Carbidopa; Cerebral Cortex; Ketanserin; Male; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin

1988
Different effects of serotonin antagonists on 3H-mianserin and 3H-ketanserin recognition sites.
    Life sciences, 1985, Feb-25, Volume: 36, Issue:8

    Topics: Animals; Binding Sites; Cerebral Cortex; Cyclic AMP; Dibenzazepines; Ketanserin; Kinetics; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin Antagonists; Time Factors

1985
Serotonin, histamine, and norepinephrine mediation of endothelial and vascular smooth muscle cell movement.
    The American journal of physiology, 1985, Volume: 248, Issue:3 Pt 1

    Topics: Animals; Aorta; Cattle; Cell Movement; Cells, Cultured; Depression, Chemical; Diphenhydramine; Endothelium; Histamine; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Piperidines; Propranolol; Receptors, Adrenergic, beta; Receptors, Histamine H1; Serotonin; Time Factors

1985
Ketanserin without effects on basal anterior pituitary hormone secretion in healthy subjects.
    Journal of endocrinological investigation, 1985, Volume: 8, Issue:1

    Topics: Adrenocorticotropic Hormone; Adult; Blood Glucose; Growth Hormone; Humans; Hydrocortisone; Ketanserin; Luteinizing Hormone; Male; Piperidines; Pituitary Hormones, Anterior; Prolactin; Serotonin Antagonists; Thyroid Hormones; Thyrotropin

1985
5-Hydroxytryptamine-stimulated inositol phospholipid hydrolysis in rat cerebral cortex slices: pharmacological characterization and effects of antidepressants.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 233, Issue:2

    Topics: Affinity Labels; Animals; Antidepressive Agents; Cerebral Cortex; Hydrolysis; Imipramine; Iprindole; Ketanserin; Male; Phenoxybenzamine; Phosphatidylinositols; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin

1985
Role of serotonin type 2 receptors in regulation of aldosterone production.
    The American journal of physiology, 1985, Volume: 249, Issue:2 Pt 1

    Topics: Adrenal Glands; Aldosterone; Angiotensin II; Animals; Cosyntropin; Cyclic AMP; Cyproheptadine; Female; In Vitro Techniques; Ketanserin; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1985
Antihypertensive mechanism of action of ketanserin and some ketanserin analogues in the spontaneously hypertensive rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension; Ketanserin; Phenylephrine; Piperidines; Prazosin; Pyrimidines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Ritanserin; Sympathetic Nervous System

1985
Serotonergic agonists stimulate inositol lipid metabolism in rabbit platelets.
    Life sciences, 1985, Oct-28, Volume: 37, Issue:17

    Topics: Animals; Blood Platelets; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Phosphatidylinositols; Piperidines; Quipazine; Rabbits; Receptors, Serotonin; Serotonin

1985
Serotonin 5-HT1 receptors mediate inhibition of cyclic AMP production in neurons.
    European journal of pharmacology, 1986, Jan-21, Volume: 120, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Brain; Cerebral Cortex; Corpus Striatum; Cyclic AMP; Female; Fetus; Indoles; Ketanserin; Metergoline; Mice; Neurons; Piperidines; Pregnancy; Receptors, Serotonin; Tetrahydronaphthalenes; Vasoactive Intestinal Peptide

1986
Central alpha-2 adrenoceptor-mediated hypertensive response to clonidine in conscious, normotensive rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:3

    Topics: Animals; Azepines; Blood Pressure; Brain; Cimetidine; Clonidine; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Male; Methoxamine; Oxidopamine; Piperidines; Prazosin; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1986
A simple 'free 3H-ligand' assay for rapid screening of hybridoma monoclonal antibodies against neurotransmitter analogs and anti-idiotype antibodies.
    Journal of neuroimmunology, 1986, Volume: 11, Issue:3

    Topics: Animals; Antibodies, Monoclonal; Haloperidol; Hybridomas; Immunoglobulin Idiotypes; Ketanserin; Mice; Pimozide; Piperidines; Receptors, Neurotransmitter

1986
Studies on the antinociceptive effect of intrathecal salmon calcitonin.
    Peptides, 1985, Volume: 6 Suppl 3

    Topics: Analgesics; Animals; Benzomorphans; Calcitonin; Enkephalin, Leucine; Haloperidol; Ketanserin; Male; Methysergide; Nociceptors; Phentolamine; Piperidines; Rats; Receptors, Opioid

1985
Effect of ketanserin on the in vitro regulation of aldosterone.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:1

    Topics: Adrenocorticotropic Hormone; Angiotensin II; Animals; Female; In Vitro Techniques; Ketanserin; Mineralocorticoid Receptor Antagonists; Piperidines; Potassium; Rats; Rats, Inbred Strains

1986
Down regulation of serotonin-S2 receptor sites in rat brain by chronic treatment with the serotonin-S2 antagonists: ritanserin and setoperone.
    Psychopharmacology, 1986, Volume: 88, Issue:4

    Topics: Animals; Brain; Corpus Striatum; Frontal Lobe; Ketanserin; Male; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Neurotransmitter; Receptors, Serotonin; Ritanserin

1986
Evidence for separate receptors that mediate parallel effects of serotonin and small cardioactive peptideB (SCPB) on adenylate cyclase in Aplysia californica.
    Neuroscience letters, 1986, Oct-08, Volume: 70, Issue:2

    Topics: Adenylyl Cyclases; Animals; Aplysia; Enzyme Activation; Ketanserin; Neuropeptides; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1986
Antagonism by methysergide of neurogenic vasoconstriction in the dog forelimb.
    Federation proceedings, 1987, Volume: 46, Issue:2

    Topics: Animals; Dogs; Electric Stimulation; Forelimb; Ketanserin; Median Nerve; Methysergide; Phentolamine; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasoconstriction; Vasodilation

1987
Serotonin receptors in the rat nucleus tractus solitarii and cardiovascular regulation.
    European journal of pharmacology, 1986, Dec-16, Volume: 132, Issue:2-3

    Topics: Animals; Blood Pressure; Body Temperature; Cardiovascular Physiological Phenomena; Heart Rate; Indoles; Ketanserin; Male; Medulla Oblongata; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1986
Ritanserin and serotonergic mechanisms in blood pressure and fluid regulation in sheep.
    Clinical and experimental pharmacology & physiology, 1987, Volume: 14, Issue:7

    Topics: Animals; Blood Pressure; Cardiac Output; Heart Rate; Hypertension; Ketanserin; Phenylephrine; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Sheep; Water-Electrolyte Balance

1987
Protection with phencyclidine against inactivation of 5-HT2 receptors by sulfhydryl-modifying reagents.
    Biochemical pharmacology, 1988, Sep-01, Volume: 37, Issue:17

    Topics: Animals; Behavior, Animal; Ethylmaleimide; Ketanserin; Male; Phencyclidine; Piperidines; Rats; Rats, Inbred F344; Receptors, Serotonin; Ritanserin; Serotonin; Sulfhydryl Reagents

1988
Interference of ketanserin with baroreflex control of the circulation in the conscious spontaneously hypertensive rat.
    Drugs, 1988, Volume: 36 Suppl 1

    Topics: Animals; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Piperidines; Prazosin; Pressoreceptors; Rats; Rats, Inbred SHR; Ritanserin; Serotonin Antagonists

1988
Habituation of tactile startle is altered by drugs acting on serotonin-2 receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1988, Volume: 1, Issue:2

    Topics: Animals; Cinanserin; Cyproheptadine; Habituation, Psychophysiologic; Ketanserin; Male; Piperidines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reference Values; Reflex, Startle; Ritanserin; Serotonin; Serotonin Antagonists; Touch

1988
Adrenergic and serotoninergic mechanisms in human hand arteries and veins studied by fluorescence histochemistry and in vitro pharmacology.
    Blood vessels, 1985, Volume: 22, Issue:1

    Topics: Arteries; Binding, Competitive; Biogenic Amines; Epinephrine; Female; Hand; Humans; Isoproterenol; Ketanserin; Male; Microscopy, Fluorescence; Muscle Contraction; Norepinephrine; Phentolamine; Piperidines; Receptors, Adrenergic; Serotonin; Sympathetic Nervous System; Veins

1985
Studies into the dual effects of serotonergic pharmacological agents on female sexual behaviour in the rat: preliminary evidence that endogenous 5HT is stimulatory.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:1

    Topics: 5-Hydroxytryptophan; Adrenalectomy; Alanine; Animals; Castration; Cinanserin; Female; Ketanserin; Metergoline; Methysergide; Mianserin; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal; Zimeldine

1985
Adenine nucleotides, serotonin, and endothelium-dependent relaxations to platelets.
    The American journal of physiology, 1985, Volume: 248, Issue:3 Pt 2

    Topics: Adenine Nucleotides; Animals; Apyrase; Blood Platelets; Coronary Vessels; Dogs; Endothelium; Female; Ketanserin; Male; Meclofenamic Acid; Methiothepin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists; Vasoconstriction

1985
Pharmacological properties of mechanical responses of the rat oesophageal muscularis mucosae to vagal and field stimulation.
    British journal of pharmacology, 1985, Volume: 84, Issue:1

    Topics: Animals; Dioxolanes; Electric Stimulation; Esophagus; Hexamethonium Compounds; In Vitro Techniques; Ketanserin; Male; Morphine; Muscle Contraction; Muscle, Smooth; N-Methylscopolamine; Naloxone; Piperidines; Rats; Rats, Inbred Strains; Scopolamine Derivatives; Serotonin; Tetrodotoxin; Tubocurarine; Vagus Nerve

1985
Rapid intracellular release of calcium in human platelets by stimulation of 5-HT2-receptors.
    British journal of pharmacology, 1985, Volume: 84, Issue:2

    Topics: Aminoquinolines; Blood Platelets; Calcium; Cytoplasm; Gallic Acid; Humans; In Vitro Techniques; Ketanserin; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1985
N-(3-acetylaminophenyl)piperazine hydrochloride (BEA 1654), a putative 5-HT1 agonist, causes constriction of arteriovenous anastomoses and dilatation of arterioles.
    European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3

    Topics: Animals; Arterioles; Arteriovenous Anastomosis; Carotid Arteries; Hemodynamics; In Vitro Techniques; Ketanserin; Phentolamine; Piperazines; Piperidines; Rats; Receptors, Serotonin; Regional Blood Flow; Swine; Vasoconstriction; Vasodilation

1985
Verapamil, an antagonist at 5-hydroxytryptamine receptors of human blood platelets.
    European journal of pharmacology, 1985, Jan-22, Volume: 108, Issue:2

    Topics: Adenosine Diphosphate; Binding, Competitive; Blood Platelets; Cerebral Cortex; Gallopamil; Humans; In Vitro Techniques; Ketanserin; Membranes; Piperidines; Receptors, Serotonin; Spiperone; Verapamil

1985
Differentiation between the stimulus effects of l-5-hydroxytryptophan and LSD.
    European journal of pharmacology, 1985, Jan-22, Volume: 108, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Benserazide; Cues; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains

1985
A paradox: the 5-HT2-receptor antagonist ketanserin restores the 5-HT-induced contraction depressed by methysergide in large coronary arteries of calf. Allosteric regulation of 5-HT2-receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 328, Issue:3

    Topics: Allosteric Regulation; Animals; Cattle; Coronary Vessels; In Vitro Techniques; Ketanserin; Methysergide; Models, Biological; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vasoconstriction

1985
Ketanserin causes surmountable antagonism of 5-hydroxytryptamine-induced contractions of large coronary arteries of dog.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 328, Issue:3

    Topics: Animals; Coronary Vessels; Dogs; Female; In Vitro Techniques; Ketanserin; Male; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vasoconstriction

1985
Cardiovascular and blood gas responses to ketanserin in canine pulmonary edema induced by oleic acid.
    Anesthesiology, 1985, Volume: 62, Issue:4

    Topics: Animals; Blood Pressure; Carbon Dioxide; Cardiac Output; Dogs; Hemodynamics; Hydrogen-Ion Concentration; Ketanserin; Lung; Oleic Acid; Oleic Acids; Oxygen; Piperidines; Pulmonary Edema; Serotonin; Serotonin Antagonists; Vascular Resistance

1985
Estradiol-induced increase of specific [3H]ketanserin binding sites on rat uterine membranes.
    European journal of pharmacology, 1985, Feb-05, Volume: 108, Issue:3

    Topics: Animals; Binding Sites; Castration; Estradiol; Female; In Vitro Techniques; Ketanserin; Membranes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tritium; Uterus

1985
Characterization of 5-hydroxytryptamine binding sites in the plasma membrane of pig blood platelets.
    Journal of neural transmission, 1985, Volume: 61, Issue:3-4

    Topics: Animals; Binding Sites; Blood Platelets; Brain; Ketanserin; Lysergic Acid Diethylamide; Piperidines; Platelet Aggregation; Serotonin; Sodium; Swine

1985
Complete conversion of brain D2 dopamine receptors from the high- to the low-affinity state for dopamine agonists, using sodium ions and guanine nucleotide.
    Journal of neurochemistry, 1985, Volume: 44, Issue:6

    Topics: Animals; Apomorphine; Brain; Guanine Nucleotides; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Tetrahydronaphthalenes; Tritium

1985
A calcium-dependent reversible permeability increase in microvessels in frog brain, induced by serotonin.
    The Journal of physiology, 1985, Volume: 361

    Topics: Animals; Blood-Brain Barrier; Brain; Calcium; Capillary Permeability; Dose-Response Relationship, Drug; Electric Conductivity; Endothelium; Ketanserin; Piperidines; Rana temporaria; Serotonin; Serotonin Antagonists; Verapamil

1985
The effect of prolonged treatment with tricyclic antidepressants on the actions of 5-hydroxytryptamine in the hippocampal slice of the rat.
    Neuropharmacology, 1985, Volume: 24, Issue:2

    Topics: Animals; Cyproheptadine; Desipramine; Evoked Potentials; Hippocampus; Imipramine; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin

1985
Serotonin antagonist pirenperone inhibits sexual behavior in the male rat: attenuation by quipazine.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Fenclonine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Serotonin Antagonists; Sexual Behavior, Animal; Tranquilizing Agents

1985
Interaction of 5-hydroxytryptamine and ketanserin in rat vas deferens subjected to low frequency field stimulation.
    Japanese journal of pharmacology, 1985, Volume: 37, Issue:3

    Topics: Animals; Drug Interactions; Electric Stimulation; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth; Piperidines; Prazosin; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Vas Deferens

1985
Effects of ketanserin on neuronal responses to serotonin in the prefrontal cortex, lateral geniculate and dorsal raphe nucleus.
    Neuropharmacology, 1985, Volume: 24, Issue:4

    Topics: Animals; Decerebrate State; Electrophysiology; Frontal Lobe; gamma-Aminobutyric Acid; Geniculate Bodies; Ketanserin; Male; Norepinephrine; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Tryptamines

1985
Anti-aversive role of serotonin in the dorsal periaqueductal grey matter.
    Psychopharmacology, 1985, Volume: 85, Issue:3

    Topics: Animals; Avoidance Learning; Electric Stimulation; Electrodes, Implanted; Injections; Ketanserin; Male; Metergoline; Methoxydimethyltryptamines; Periaqueductal Gray; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Zimeldine

1985
Serotonin-induced platelet aggregation in whole blood and the effects of ketanserin and mepyramine.
    Thrombosis research, 1985, Apr-15, Volume: 38, Issue:2

    Topics: Aminopyridines; Dose-Response Relationship, Drug; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Serotonin; Time Factors

1985
Tryptamine-induced vasoconstrictor responses in rat caudal arteries are mediated predominantly via 5-hydroxytryptamine receptors.
    British journal of pharmacology, 1985, Volume: 84, Issue:4

    Topics: Animals; Arteries; In Vitro Techniques; Ketanserin; Male; Methysergide; Monoamine Oxidase Inhibitors; Phentolamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tryptamines; Vasoconstriction

1985
Localization of 11C-radiopharmaceuticals in the Greene melanoma of hamsters.
    European journal of nuclear medicine, 1985, Volume: 10, Issue:9-10

    Topics: Animals; Benzodiazepinones; Carbon Radioisotopes; Chlorpromazine; Cricetinae; Flumazenil; Flunitrazepam; Gallium Radioisotopes; Isotope Labeling; Ketanserin; Melanoma; Mesocricetus; Methionine; Neoplasm Transplantation; Pimozide; Piperidines; Quinuclidinyl Benzilate; Radionuclide Imaging; Tissue Distribution

1985
Is waning of a 5-hydroxytryptamine (5-HT)-mediated syndrome due to 5-HT2 receptor down-regulation?
    Neuroscience letters, 1985, Apr-19, Volume: 55, Issue:3

    Topics: Animals; Cerebral Cortex; Ketanserin; Male; Myoclonus; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Syndrome; Time Factors; Tritium

1985
Platelet-mediated vascular permeability in the rat: a predominant role for 5-hydroxytryptamine.
    Thrombosis research, 1985, May-15, Volume: 38, Issue:4

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Capillary Permeability; Dose-Response Relationship, Drug; Histamine; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Suprofen; Thrombin

1985
Raynaud's disease.
    Archives of disease in childhood, 1985, Volume: 60, Issue:6

    Topics: Antihypertensive Agents; Child; Dinoprostone; Epoprostenol; Female; Humans; Ketanserin; Male; Nifedipine; Nitroprusside; Phenoxybenzamine; Piperidines; Prostaglandins E, Synthetic; Raynaud Disease

1985
Excitatory 5-hydroxytryptamine receptors in the cat urinary bladder are of the M- and 5-HT2-type.
    Journal of autonomic pharmacology, 1985, Volume: 5, Issue:2

    Topics: Animals; Atropine; Cats; Cyproheptadine; Dimethylphenylpiperazinium Iodide; Drug Interactions; Female; Guanethidine; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Urinary Bladder

1985
Simultaneous determination of ketanserin and ketanserinol in biological fluids using ion-pair liquid chromatography and fluorometric detection.
    Journal of chromatography, 1985, May-31, Volume: 341, Issue:1

    Topics: Aged; Antihypertensive Agents; Body Fluids; Chromatography, High Pressure Liquid; Female; Humans; Hydrogen-Ion Concentration; Ketanserin; Kinetics; Piperidines; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet

1985
In vivo binding of 125I-LSD to serotonin 5-HT2 receptors in mouse brain.
    Life sciences, 1985, Aug-19, Volume: 37, Issue:7

    Topics: Animals; Binding, Competitive; Brain; Cinanserin; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Mice; Piperidines; Receptors, Serotonin; Spiperone; Time Factors; Tissue Distribution

1985
Binding of the putative anxiolytic TVX Q 7821 to hippocampal 5-hydroxytryptamine (5-HT) recognition sites.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:3

    Topics: Animals; Binding, Competitive; Cattle; Hippocampus; Ketanserin; Kinetics; Membranes; Piperidines; Pyrimidines; Rats; Receptors, Serotonin

1985
Potentiation of motoneurone excitability by combined administration of 5-HT agonist and TRH analogue.
    Neuropeptides, 1985, Volume: 6, Issue:3

    Topics: Animals; Anterior Horn Cells; Drug Synergism; Female; Fenclonine; Ketanserin; Methoxydimethyltryptamines; Methysergide; Motor Neurons; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Serotonin; Stimulation, Chemical; Thyrotropin-Releasing Hormone

1985
A facilitatory role for serotonin in the sexual behavior of the female rat.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:6

    Topics: Animals; Castration; Estradiol; Female; Ketanserin; Methysergide; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Sexual Behavior, Animal; Spiperone

1985
Serotonin-induced contraction of canine saphenous vein: mediation by 5-HT1 receptors.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 274, Issue:2

    Topics: Animals; Clonidine; Dogs; Drug Interactions; Emetics; In Vitro Techniques; Ketanserin; Mianserin; Muscle Contraction; Naphthols; Piperidines; Receptors, Serotonin; Saphenous Vein; Serotonin; Yohimbine

1985
Cardiovascular effects of ketanserin in closed-chest anesthetized dogs.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 275, Issue:2

    Topics: Anesthesia; Animals; Blood Pressure; Dogs; Electrocardiography; Female; Heart Rate; Hemodynamics; Ketanserin; Male; Piperidines; Respiration; Serotonin; Serotonin Antagonists; Stroke Volume; Vascular Resistance

1985
Two types of receptors for 5-hydroxytryptamine on the cholinergic nerves of the guinea-pig myenteric plexus.
    British journal of pharmacology, 1985, Volume: 85, Issue:2

    Topics: Acetylcholine; Animals; Binding, Competitive; Cocaine; Electric Stimulation; Female; Guinea Pigs; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Myenteric Plexus; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes

1985
[Ketanserin in the treatment of ischemic disease of the lower extremities].
    Casopis lekaru ceskych, 1985, Jul-26, Volume: 124, Issue:30

    Topics: Female; Humans; Ischemia; Ketanserin; Leg; Male; Middle Aged; Piperidines; Regional Blood Flow; Serotonin Antagonists

1985
Selective 5-HT2 receptor blockade in exercise-induced asthma.
    Clinical allergy, 1985, Volume: 15, Issue:4

    Topics: Adolescent; Adult; Asthma; Asthma, Exercise-Induced; Bronchi; Child; Humans; Ketanserin; Piperidines; Receptors, Serotonin; Sleep Stages

1985
Bioavailability and pharmacokinetics of ketanserin in elderly subjects.
    European journal of clinical pharmacology, 1985, Volume: 28, Issue:4

    Topics: Age Factors; Aged; Biological Availability; Female; Half-Life; Humans; Ketanserin; Kinetics; Male; Middle Aged; Piperidines; Serotonin Antagonists

1985
Evidence for serotoninergic control of exercise-induced prolactin secretion.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1985, Volume: 17, Issue:7

    Topics: Adult; Heart Rate; Humans; Ketanserin; Male; Physical Exertion; Piperidines; Prolactin; Serotonin; Time Factors

1985
Effect of serotonin on the motility of smooth muscles in teats of lactating cows.
    The Journal of dairy research, 1985, Volume: 52, Issue:3

    Topics: Animals; Cattle; Female; Ketanserin; Lactation; Mammary Glands, Animal; Methysergide; Mianserin; Milk Ejection; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Piperidines; Pregnancy; Serotonin; Serotonin Antagonists

1985
Changes of the striatal 3H-spiperone binding 3-6 weeks after nigrostriatal denervation and after two years.
    Life sciences, 1985, Sep-09, Volume: 37, Issue:10

    Topics: Animals; Butyrophenones; Corpus Striatum; Denervation; Haloperidol; Hydroxydopamines; Ketanserin; Kinetics; Male; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Spiperone; Substantia Nigra; Time Factors

1985
Target size analysis of serotonin 5-HT1 and 5-HT2 receptors in bovine brain membranes.
    Life sciences, 1985, Sep-23, Volume: 37, Issue:12

    Topics: Animals; Binding, Competitive; Brain Chemistry; Cattle; Caudate Nucleus; Cerebral Cortex; Freeze Drying; Ketanserin; Molecular Weight; Piperidines; Radioligand Assay; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Synaptic Membranes

1985
Attenuation of morphine analgesia by the S2 antagonists, pirenperone and ketanserin.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:3

    Topics: Analgesia; Animals; Dose-Response Relationship, Drug; Ketamine; Ketanserin; Male; Morphine; Piperidines; Rats; Reaction Time; Receptors, Serotonin; Serotonin Antagonists

1988
Opposite regulation of serotonin-S2 and dopamine-D2 receptors in rat brain following chronic receptor blockade.
    Journal of receptor research, 1987, Volume: 7, Issue:1-4

    Topics: Animals; Apomorphine; Behavior, Animal; Corpus Striatum; Diazepam; Dopamine Antagonists; Frontal Lobe; Gene Expression Regulation; Ketanserin; Male; Models, Biological; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin Antagonists; Tryptamines

1987
Different temporal effects of serotonergic antagonists on passive avoidance retention.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:3

    Topics: Animals; Avoidance Learning; Ketanserin; Male; Memory; Mianserin; Mice; Piperidines; Receptors, Serotonin; Retention, Psychology; Serotonin Antagonists; Time Factors

1987
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Frontal Lobe; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1986
Ketanserin and pirenperone attenuate acute morphine withdrawal in rats.
    European journal of pharmacology, 1986, Dec-16, Volume: 132, Issue:2-3

    Topics: Animals; Body Temperature; Conditioning, Operant; Ketanserin; Male; Morphine Dependence; Piperidines; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome

1986
Photoaffinity probes for serotonin and histamine receptors. Synthesis and characterization of two azide analogues of ketanserin.
    The Journal of biological chemistry, 1985, Jul-15, Volume: 260, Issue:14

    Topics: 4-Aminobenzoic Acid; Affinity Labels; Animals; Azides; Binding, Competitive; Cerebellum; Cerebral Cortex; Guinea Pigs; Histamine Antagonists; Ketanserin; Kinetics; Lysergic Acid Diethylamide; Photochemistry; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Receptors, Serotonin; Serotonin Antagonists; Ultraviolet Rays

1985
Photoaffinity labelling of serotonin-S2 receptors with 7-azidoketanserin.
    European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3

    Topics: Affinity Labels; Animals; Azides; Female; Frontal Lobe; In Vitro Techniques; Ketanserin; Light; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1985
Differential photoaffinity labelling of serotonin-S2 receptors and histamine-H1 receptors using 7-azidoketanserin.
    FEBS letters, 1985, Mar-25, Volume: 182, Issue:2

    Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Butyrophenones; Cerebellum; Cerebral Cortex; Female; Guinea Pigs; Ketanserin; Photolysis; Piperidines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Serotonin; Spiperone

1985
[Reciprocal potentiation of the bronchoconstrictor activity of histamine and 5-hydroxytryptamine in the guinea pig].
    Archives internationales de physiologie et de biochimie, 1984, Volume: 92, Issue:3

    Topics: Animals; Bronchi; Drug Synergism; Female; Guinea Pigs; Histamine; Histamine Antagonists; Ketanserin; Male; Piperidines; Serotonin; Serotonin Antagonists

1984
Acute effects of antagonist of S2-receptors.
    Czechoslovak medicine, 1984, Volume: 7, Issue:4

    Topics: Adult; Blood Pressure; Drug Evaluation; Female; Humans; Hydroxyindoleacetic Acid; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Serotonin Antagonists; Vanilmandelic Acid

1984
Neurotransmitter receptors and monoamine metabolites in the brains of patients with Alzheimer-type dementia and depression, and suicides.
    Neuropharmacology, 1984, Volume: 23, Issue:12B

    Topics: Aged; Aging; Alzheimer Disease; Binding, Competitive; Biogenic Amines; Brain; Choline O-Acetyltransferase; Depressive Disorder; Female; Humans; Hydroxyindoleacetic Acid; Ketanserin; Male; Middle Aged; Piperidines; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Serotonin; Serotonin; Sex Factors; Suicide

1984
Regional and cortical laminar distributions of serotonin S2, benzodiazepine, muscarinic, and dopamine D2 receptors in human brain.
    Journal of neurochemistry, 1984, Volume: 43, Issue:4

    Topics: Adult; Aged; Brain; Cerebral Cortex; Diazepam; Humans; Ketanserin; Male; Middle Aged; Piperidines; Quinuclidinyl Benzilate; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Serotonin; Spiperone; Tissue Distribution

1984
Colonic secretion mediated by prostaglandin E2 and 5-hydroxytryptamine may contribute to diarrhea due to morphine withdrawal in the rat.
    Gastroenterology, 1984, Volume: 87, Issue:5

    Topics: Animals; Atropine; Clonidine; Colon; Cyclic AMP; Diarrhea; Dinoprostone; Female; Humans; Indomethacin; Ketanserin; Morphine Dependence; Naloxone; Piperidines; Prostaglandins E; Rats; Rats, Inbred Strains; Serotonin; Substance Withdrawal Syndrome

1984
Assessment of sodium-potassium ATPase activity in human erythrocytes in vitro.
    Methods and findings in experimental and clinical pharmacology, 1984, Volume: 6, Issue:8

    Topics: Erythrocytes; Humans; In Vitro Techniques; Ketanserin; Male; Ouabain; Piperidines; Rubidium; Sodium; Sodium-Potassium-Exchanging ATPase

1984
Alpha 1 adrenergic receptors in the porcine pituitary neurointermediate lobe: detection with [3H]ketanserin.
    Journal of receptor research, 1984, Volume: 4, Issue:7

    Topics: Animals; Binding, Competitive; Brain; Cinanserin; In Vitro Techniques; Ketanserin; Kinetics; Piperidines; Pituitary Gland; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Swine

1984
The specificity of ketanserin in the inhibition of serotonin-induced steroidogenesis in the rat adrenal zona glomerulosa.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1984, Volume: 2, Issue:3

    Topics: Adrenal Cortex; Aldosterone; Animals; Corticosterone; Cyclic AMP; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Methysergide; Piperidines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1984
Acute blood-pressure-lowering effect of ketanserin.
    Lancet (London, England), 1981, May-23, Volume: 1, Issue:8230

    Topics: Aged; Antihypertensive Agents; Blood Pressure; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Serotonin Antagonists

1981
5-HT2-receptor blockade in the treatment of heart failure. A preliminary study.
    Lancet (London, England), 1981, May-30, Volume: 1, Issue:8231

    Topics: Adult; Aged; Blood Pressure; Cardiac Output; Heart Failure; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Pulmonary Wedge Pressure; Serotonin Antagonists; Stroke Volume; Vascular Resistance; Vasoconstriction

1981
Vascular effects of ketanserin (R 41 468), a novel antagonist of 5-HT2 serotonergic receptors.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 218, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Arteries; Blood Pressure; Calcium; Dogs; Guinea Pigs; Hypertension; In Vitro Techniques; Ketanserin; Kidney; Male; Muscle, Smooth, Vascular; Norepinephrine; Organ Specificity; Piperidines; Rats; Serotonin Antagonists; Species Specificity; Stomach; Vasoconstriction; Veins

1981
Solubilized serotonin receptors from rat and dog brain. Selective labelling with [3H]ketanserin.
    FEBS letters, 1982, Feb-22, Volume: 138, Issue:2

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Brain; Butyrophenones; Dogs; Isonipecotic Acids; Ketanserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Solubility; Species Specificity; Spiperone; Time Factors

1982
Cardiovascular effects in the rat of ketanserin, a novel 5-hydroxytryptamine receptor blocking agent.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:7

    Topics: Animals; Blood Pressure; Heart Rate; Hemodynamics; Injections, Intraventricular; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Time Factors

1982
Ketanserin--a novel antihypertensive drug?
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:8

    Topics: Animals; Antihypertensive Agents; In Vitro Techniques; Ketanserin; Muscle, Smooth; Piperidines; Rats; Receptors, Histamine H2

1982
Ketanserin: a selective serotonin antagonist.
    Lancet (London, England), 1982, Oct-16, Volume: 2, Issue:8303

    Topics: Cardiovascular System; Humans; Hypertension; Ketanserin; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1982
Mechanism of action of ketanserin.
    Lancet (London, England), 1982, Nov-20, Volume: 2, Issue:8308

    Topics: Animals; Antihypertensive Agents; Humans; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Spiperone

1982
Ketanserin: a selective antagonist of 5-HT2 serotoninergic receptors.
    Lancet (London, England), 1983, Feb-05, Volume: 1, Issue:8319

    Topics: Animals; Binding Sites; Ketanserin; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists

1983
Preliminary studies of human cortical 5-HT2 receptors and their involvement in schizophrenia and neuroleptic drug action.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Antipsychotic Agents; Cerebral Cortex; Humans; Ketanserin; Piperidines; Receptors, Serotonin; Schizophrenia; Spiperone; Substrate Specificity

1983
Yohimbine and rauwolscine inhibit 5-hydroxytryptamine-induced contraction of large coronary arteries of calf through blockade of 5 HT2 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 323, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Cattle; Coronary Vessels; Drug Combinations; Ketanserin; Muscle Contraction; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Yohimbine

1983
Unusual acute effects of antidepressants and neuroleptics on S2-serotonergic receptors.
    Life sciences, 1983, Dec-19, Volume: 33, Issue:25

    Topics: Amoxapine; Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Fenclonine; Frontal Lobe; Ketanserin; Loxapine; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1983
Influence of ketanserin, an antihypertensive agent with specific 5-HT2-receptor blocking activity, on intracranial pressure.
    Critical care medicine, 1984, Volume: 12, Issue:1

    Topics: Animals; Blood Gas Analysis; Cardiac Output; Cerebral Cortex; Dogs; Female; Hemodynamics; Histamine H2 Antagonists; Intermittent Positive-Pressure Ventilation; Intracranial Pressure; Ketanserin; Male; Piperidines

1984
Ketanserin in intermittent claudication.
    Lancet (London, England), 1984, Nov-24, Volume: 2, Issue:8413

    Topics: Appetite; Blood Pressure; Body Weight; Humans; Intermittent Claudication; Ketanserin; Piperidines

1984
Serotoninergic control of somatostatin and gastrin release from the isolated rat stomach.
    Regulatory peptides, 1984, Volume: 9, Issue:1-2

    Topics: Animals; Gastric Mucosa; Gastrins; In Vitro Techniques; Ketanserin; Male; Methysergide; Perfusion; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Receptors, Serotonin; Serotonin; Somatostatin

1984
The 5-hydroxytryptamine antagonist ketanserin inhibits the vasoconstrictor activity of per-operative CSF, from subarachnoid haemorrhage patients, on isolated tissues.
    Journal of neurology, neurosurgery, and psychiatry, 1983, Volume: 46, Issue:3

    Topics: Adult; Aged; Animals; Female; Humans; Hydroxyindoleacetic Acid; Intracranial Aneurysm; Intraoperative Complications; Ischemic Attack, Transient; Ketanserin; Male; Middle Aged; Piperidines; Postoperative Complications; Rats; Rupture, Spontaneous; Serotonin; Serotonin Antagonists; Subarachnoid Hemorrhage; Vasoconstriction

1983
[Thermogenic shivering in the anesthetized rat].
    Archives internationales de physiologie et de biochimie, 1982, Volume: 90, Issue:5

    Topics: Animals; Body Temperature Regulation; Ketanserin; Pentobarbital; Piperidines; Rats; Shivering

1982
On the neurotoxicity of chlordecone: a role for gamma-aminobutyric acid and serotonin.
    Brain research, 1984, Jun-11, Volume: 303, Issue:1

    Topics: Acetylcholine; Animals; Binding Sites; Brain; Chlordecone; gamma-Aminobutyric Acid; Insecticides; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Spiperone

1984
Serotonin receptor changes in dementia of the Alzheimer type.
    Journal of neurochemistry, 1984, Volume: 43, Issue:6

    Topics: Aged; Alzheimer Disease; Choline O-Acetyltransferase; Female; Humans; Hydroxyindoleacetic Acid; Ketanserin; Male; Piperidines; Postmortem Changes; Receptors, Serotonin; Serotonin; Somatostatin; Tissue Distribution

1984
Inhibition of 5-hydroxytryptamine-induced and -amplified human platelet aggregation by ketanserin (R 41 468), a selective 5-HT2-receptor antagonist.
    Agents and actions, 1982, Volume: 12, Issue:3

    Topics: beta-Thromboglobulin; Blood Platelets; Blood Proteins; Humans; In Vitro Techniques; Ketanserin; Malondialdehyde; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists; Thromboxane B2

1982
[Effect of ketanserin on various properties of pentobarbital in rats].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1983, Volume: 177, Issue:3

    Topics: Animals; Body Temperature; Drug Interactions; Ketanserin; Pentobarbital; Piperidines; Rats; Rats, Inbred Strains; Sleep

1983
Stimulation by serotonin of 40 kDa and 20 kDa protein phosphorylation in human platelets.
    FEBS letters, 1984, Jun-11, Volume: 171, Issue:2

    Topics: Blood Platelets; Blood Proteins; Humans; Ketanserin; Molecular Weight; Myosin-Light-Chain Kinase; Phosphatidic Acids; Phosphorylation; Piperidines; Protein Kinase C; Protein Kinases; Receptors, Serotonin; Serotonin

1984
The role of serotonin (5-HT) in the control of TSH and prolactin release in euthyroid subjects as assessed by the administration of ketanserin (5-HT2 antagonist) and zimelidine (5-HT re-uptake inhibitor).
    Psychoneuroendocrinology, 1984, Volume: 9, Issue:1

    Topics: Female; Humans; Ketanserin; Male; Piperidines; Prolactin; Serotonin; Serotonin Antagonists; Thyrotropin; Thyrotropin-Releasing Hormone; Thyroxine; Zimeldine

1984
Prolongation of rat tail bleeding time by ketanserin: mechanisms of action.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Bleeding Time; Blood Coagulation; Blood Platelets; Blood Pressure; Drug Interactions; Fenclonine; Ketanserin; Male; Metergoline; Piperidines; Platelet Aggregation; Prazosin; Rats; Serotonin; Serotonin Antagonists; Sympatholytics; Tail

1984
Receptor binding profile of R 41 468, a novel antagonist at 5-HT2 receptors.
    Life sciences, 1981, Mar-02, Volume: 28, Issue:9

    Topics: Animals; Brain; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Receptors, Adrenergic, alpha; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Serotonin; Serotonin Antagonists

1981
Characterization of the antihypertensive properties of ketanserin (R 41 468) in rats.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 222, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Ketanserin; Male; Methoxamine; Piperidines; Rats; Receptors, Adrenergic, alpha; Receptors, Serotonin; Vasopressins

1982
Principles of therapy for congestive heart failure.
    European heart journal, 1983, Volume: 4 Suppl A

    Topics: Calcium; Calcium Channel Blockers; Calmodulin; Cardiotonic Agents; Clonidine; Cyclic AMP; Cytosol; Digitalis Glycosides; Diuretics; Heart Failure; Humans; Ketanserin; Models, Cardiovascular; Muscle, Smooth, Vascular; Myocardium; Myosins; Piperidines; Receptors, Adrenergic, alpha; Vasodilator Agents

1983
Modulation of brain S2 serotonin receptors by lithium, sodium and potassium chloride.
    Life sciences, 1983, May-30, Volume: 32, Issue:22

    Topics: Animals; Binding, Competitive; Brain; Chlorides; Dose-Response Relationship, Drug; Female; Ketanserin; Lithium; Lithium Chloride; Piperidines; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium Chloride

1983
Mechanism of antihypertensive action of ketanserin in man.
    British medical journal (Clinical research ed.), 1983, Oct-29, Volume: 287, Issue:6401

    Topics: Antihypertensive Agents; Blood Pressure; Humans; Ketanserin; Piperidines; Receptors, Adrenergic, alpha

1983
Evidence for an alpha-1 receptor-mediated central sympathoinhibitory action of ketanserin.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 228, Issue:3

    Topics: Animals; Blood Pressure; Brain; Cats; Clonidine; Heart Rate; Ketanserin; Piperidines; Receptors, Adrenergic, alpha; Serotonin Antagonists; Sympathetic Nervous System; Sympatholytics

1984
Comparison of iprindole, imipramine and mianserin action on brain serotonergic and beta adrenergic receptors.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 229, Issue:3

    Topics: Animals; Axons; Brain; Cyclic AMP; Dibenzazepines; Imipramine; Indoles; Iprindole; Ketanserin; Male; Mianserin; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin

1984
Tryptaminergic receptors in the bovine pulmonary vasculature: effects of ketanserin.
    Research communications in chemical pathology and pharmacology, 1984, Volume: 44, Issue:1

    Topics: Animals; Cattle; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pulmonary Artery; Pulmonary Veins; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists

1984
Autoradiographic mapping of spirodecanone binding-sites in the hippocampal region of the rat. Evidence for a localization on intrinsic neurons.
    Neuroscience letters, 1984, May-04, Volume: 46, Issue:2

    Topics: Animals; Autoradiography; Binding, Competitive; Brain Mapping; Butyrophenones; Haloperidol; Hippocampus; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Serotonin; Spiperone; Tetrahydronaphthalenes

1984
Effect of ketanserin, an inhibitor of 5-HT2 receptors, on the aldosterone-stimulating action of metoclopramide.
    Hormone research, 1983, Volume: 17, Issue:3

    Topics: Adolescent; Adult; Aldosterone; Humans; Ketanserin; Kinetics; Male; Metoclopramide; Piperidines; Potassium; Prolactin; Receptors, Serotonin; Renin; Serotonin Antagonists

1983
Role and localization of serotonin2 (S2)-receptor-binding sites: effects of neuronal lesions.
    Advances in biochemical psychopharmacology, 1983, Volume: 37

    Topics: Animals; Catecholamines; Cerebral Cortex; Dogs; Female; Guinea Pigs; Kainic Acid; Ketanserin; Kinetics; Male; Nerve Tissue Proteins; Neurons; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Serotonin; Stereotaxic Techniques; Subcellular Fractions

1983
The role of 5-hydroxytryptamine in the feline response to intravenous infusion of live E. coli.
    British journal of pharmacology, 1983, Volume: 79, Issue:3

    Topics: Animals; Blood Pressure; Cats; Escherichia coli Infections; Hemodynamics; Intestines; Ketanserin; Lung; Piperidines; Premedication; Regional Blood Flow; Shock, Septic; Time Factors; Vascular Resistance

1983
The effect of a selective 5-HT2 antagonist, ketanserin, on the pulmonary responses to Escherichia coli endotoxin.
    British journal of pharmacology, 1983, Volume: 80, Issue:2

    Topics: Animals; Blood Gas Analysis; Cats; Endotoxins; Escherichia coli; Female; Hemodynamics; Ketanserin; Lung; Lung Compliance; Male; Piperidines; Serotonin; Serotonin Antagonists

1983
Is 5-HT a mediator in the motor control of the feline pylorus?
    Scandinavian journal of gastroenterology, 1984, Volume: 19, Issue:3

    Topics: Animals; Cats; Dose-Response Relationship, Drug; Electric Stimulation; Female; Fluorescent Antibody Technique; Histocytochemistry; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Pylorus; Serotonin; Serotonin Antagonists

1984
Effects of dihydroergotamine on the feline cardiovascular response to intravenous infusion of live Escherichia coli bacteria.
    European surgical research. Europaische chirurgische Forschung. Recherches chirurgicales europeennes, 1984, Volume: 16, Issue:4

    Topics: Animals; Blood Pressure; Cardiovascular System; Cats; Dihydroergotamine; Escherichia coli Infections; Gastric Mucosa; Intestinal Mucosa; Ketanserin; Piperidines; Regional Blood Flow; Sepsis; Shock, Septic; Vascular Resistance

1984
A role for serotonin in alpha-naphthylthiourea-induced pulmonary edema.
    Toxicology and applied pharmacology, 1984, Jun-30, Volume: 74, Issue:2

    Topics: Animals; Blood Platelets; Clorgyline; Drug Interactions; Fluoxetine; Ketanserin; Lung; Male; Mice; Piperidines; Pulmonary Edema; Reserpine; Serotonin; Serotonin Antagonists; Thiourea; Thrombocytopenia

1984
Treatment of Raynaud's phenomenon with ketanserin.
    British medical journal (Clinical research ed.), 1984, Oct-20, Volume: 289, Issue:6451

    Topics: Adolescent; Humans; Ketanserin; Leg Ulcer; Male; Piperidines; Scleroderma, Systemic

1984
Ketanserin treatment in essential hypertension.
    British heart journal, 1984, Volume: 52, Issue:3

    Topics: Antihypertensive Agents; Humans; Hypertension; Ketanserin; Piperidines

1984
Aggregating platelets contract isolated canine pulmonary arteries by releasing 5-hydroxytryptamine.
    The Journal of clinical investigation, 1984, Volume: 74, Issue:3

    Topics: Animals; Blood Platelets; Dogs; Epinephrine; In Vitro Techniques; Ketanserin; Muscle Contraction; Norepinephrine; Piperidines; Platelet Aggregation; Pulmonary Artery; Serotonin; Serotonin Antagonists; Thromboxane B2

1984
Temperature-sensitive high affinity [3H]serotonin binding: characterization and effects of antidepressant treatment.
    Life sciences, 1984, Aug-13, Volume: 35, Issue:7

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Ketanserin; Kinetics; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Temperature; Tritium

1984
5-HT1 and 5-HT2 binding properties of derivatives of the hallucinogen 1-(2,5-dimethoxyphenyl)-2-aminopropane (2,5-DMA).
    European journal of pharmacology, 1984, Jun-15, Volume: 102, Issue:1

    Topics: Amphetamines; Animals; Binding, Competitive; Cerebral Cortex; Guanylyl Imidodiphosphate; Hallucinogens; In Vitro Techniques; Ketanserin; Male; Membranes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Structure-Activity Relationship

1984
Discriminative stimulus properties of the serotonin agonist 1-(3-trifluoromethylphenyl)piperazine (TFMPP).
    Life sciences, 1984, Oct-01, Volume: 35, Issue:14

    Topics: Animals; Discrimination Learning; DOM 2,5-Dimethoxy-4-Methylamphetamine; Extinction, Psychological; Fenfluramine; Indoles; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin

1984
Interaction of ketanserin and its metabolite ketanserinol with 5HT2 receptors in pulmonary and coronary arteries of calf.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 326, Issue:4

    Topics: Animals; Cattle; Coronary Vessels; In Vitro Techniques; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Pulmonary Artery; Receptors, Serotonin; Yohimbine

1984
Selective 5HT-2 antagonists inhibit serotonin stimulated phosphatidylinositol metabolism in cerebral cortex.
    Neuropharmacology, 1984, Volume: 23, Issue:8

    Topics: Animals; Cerebral Cortex; In Vitro Techniques; Ketanserin; Phosphatidylinositols; Piperidines; Pizotyline; Rats; Serotonin; Serotonin Antagonists

1984
Restoration of post-thrombotic peripheral collateral circulation in the cat by ketanserin, a selective 5-HT2-receptor antagonist.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 270, Issue:2

    Topics: Animals; Blood Platelets; Blood Pressure; Cats; Collateral Circulation; Ketanserin; Piperidines; Prostaglandins; Receptors, Serotonin; Serotonin Antagonists; Thrombosis; Vascular Resistance

1984
Serotonin-induced blood flow changes in the rat hindlegs after unilateral ligation of the femoral artery. Inhibition by the S2 receptor antagonist ketanserin.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 270, Issue:2

    Topics: Angiography; Animals; Body Temperature; Collateral Circulation; Corrosion; Evans Blue; Femoral Artery; Hindlimb; Ketanserin; Ligation; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists

1984
Effects of the antagonists MDL 72222 and ketanserin on responses of cat carotid body chemoreceptors to 5-hydroxytryptamine.
    British journal of pharmacology, 1984, Volume: 83, Issue:1

    Topics: Action Potentials; Animals; Carotid Body; Cats; Chemoreceptor Cells; Domperidone; Dopamine; Electrophysiology; Female; Hypoxia; Ketanserin; Male; Piperidines; Serotonin; Serotonin Antagonists; Tropanes

1984
Serotonin-2 binding sites in human frontal cortex and hippocampus. Selective loss of S-2A sites with age.
    Brain research, 1984, Oct-08, Volume: 311, Issue:1

    Topics: Adolescent; Adult; Aged; Aging; Cerebral Cortex; Hippocampus; Humans; Ketanserin; Kinetics; Methysergide; Middle Aged; Organ Specificity; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1984
The effects of alpha 2-adrenergic and serotonergic receptor antagonists on cyclic blood flow alterations in stenosed canine coronary arteries.
    Circulation research, 1984, Volume: 55, Issue:5

    Topics: Adenosine Diphosphate; Animals; Blood Flow Velocity; Coronary Circulation; Coronary Disease; Dogs; Female; Heart Rate; Hemodynamics; Ketanserin; Male; Piperidines; Platelet Aggregation; Prazosin; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Yohimbine

1984
Guanyl nucleotide and divalent cation regulation of cortical S2 serotonin receptors.
    Journal of neurochemistry, 1984, Volume: 43, Issue:5

    Topics: Animals; Binding, Competitive; Calcium Chloride; Cations, Divalent; Cerebral Cortex; Chlorides; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Ketanserin; Magnesium; Magnesium Chloride; Male; Manganese; Manganese Compounds; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1984
Antihypertensive effects of chronic 5-hydroxytryptamine (5-HT2) receptor blockade with ketanserin in the spontaneously hypertensive rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 327, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Piperidines; Rats; Rats, Inbred SHR; Receptors, Serotonin; Serotonin Antagonists

1984
Antagonism by ketanserin of 5-HT-induced vasoconstriction unmasks a 5-HT-induced vasodilation.
    European journal of pharmacology, 1984, Sep-17, Volume: 104, Issue:3-4

    Topics: Amidines; Animals; Antihypertensive Agents; Blood Pressure; Hypertension; In Vitro Techniques; Ketanserin; Male; Norepinephrine; Piperidines; Rats; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation

1984
Ketanserin alters [3H]serotonin uptake and release in rat hypothalamus.
    European journal of pharmacology, 1984, Sep-17, Volume: 104, Issue:3-4

    Topics: Animals; Calcium; Dose-Response Relationship, Drug; Hypothalamus; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Tritium

1984
Central serotonin antagonist activity of ketanserin.
    Research communications in chemical pathology and pharmacology, 1984, Volume: 46, Issue:1

    Topics: Animals; Brain; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1984
The haemodynamic effects of labetalol, ketanserin and a placebo at the end of a NLA. A double blind study.
    Acta anaesthesiologica Belgica, 1984, Volume: 35 Suppl

    Topics: Adolescent; Adult; Aged; Double-Blind Method; Ethanolamines; Female; Hemodynamics; Humans; Ketanserin; Labetalol; Middle Aged; Piperidines; Placebos; Random Allocation; Serotonin Antagonists; Sympatholytics

1984
Mesulergine, a selective serotonin-2 ligand in the rat cortex, does not label these receptors in porcine and human cortex: evidence for species differences in brain serotonin-2 receptors.
    European journal of pharmacology, 1984, Nov-27, Volume: 106, Issue:3

    Topics: Animals; Brain Chemistry; Cerebral Cortex; Ergolines; Humans; In Vitro Techniques; Ketanserin; Kinetics; Ligands; Male; Piperidines; Rats; Receptors, Serotonin; Species Specificity; Swine; Tritium

1984
Aortic recognition sites for serotonin (5HT) are coupled to phospholipase C and modulate phosphatidylinositol turnover.
    Neuropharmacology, 1984, Volume: 23, Issue:10

    Topics: Animals; Aorta; Hydrolysis; Ketanserin; Male; Phosphatidylinositols; Phospholipases; Piperidines; Rats; Receptors, Serotonin; Serotonin; Type C Phospholipases; Vasoconstriction

1984
The effects of serotonin antagonists in a behavioral despair procedure in mice.
    European journal of pharmacology, 1984, Dec-15, Volume: 107, Issue:1

    Topics: Animals; Behavior, Animal; Cyproheptadine; Guinea Pigs; Ketanserin; Male; Methysergide; Mice; Muscle, Smooth; Piperidines; Pizotyline; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Trazodone; Tritium

1984
Identification of 5HT2-receptors on longitudinal muscle of the guinea pig ileum.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: Animals; Cerebral Cortex; Female; Guinea Pigs; Ileum; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Muscle, Smooth; Piperidines; Rats; Receptors, Serotonin

1984
Guanine nucleotides modulate cortical S2 serotonin receptors.
    Journal of receptor research, 1984, Volume: 4, Issue:7

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone

1984
The distribution of serotonin binding sites in the hippocampal region of the rat brain. An autoradiographic study.
    Neuroscience, 1984, Volume: 13, Issue:3

    Topics: Animals; Autoradiography; Binding Sites; Binding, Competitive; Hippocampus; Ketanserin; Male; Methoxydimethyltryptamines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone

1984
Excitatory and inhibitory effects of 5-hydroxytryptamine in mesenteric arteries of spontaneously hypertensive rats.
    European journal of pharmacology, 1984, Nov-13, Volume: 106, Issue:2

    Topics: Animals; Blood Pressure; Cyproheptadine; Drug Synergism; Hypertension; In Vitro Techniques; Ketanserin; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Norepinephrine; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Serotonin; Synapses

1984
Role of serotonin in patients with acute respiratory failure.
    Annals of surgery, 1984, Volume: 200, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Acute Disease; Adult; Aged; Blood Platelets; Blood Pressure; Cardiac Output; Female; Humans; Intubation, Intratracheal; Ketanserin; Male; Middle Aged; Piperidines; Platelet Count; Pulmonary Wedge Pressure; Respiratory Function Tests; Respiratory Insufficiency; Serotonin; Serotonin Antagonists; Thromboxane B2

1984
Redistribution of carotid artery blood flow by 5-HT: effects of the 5-HT2 receptor antagonists ketanserin and Wal 1307.
    European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4

    Topics: Animals; Carotid Arteries; Dibenzoxazepines; Hemodynamics; Ketanserin; Piperidines; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Swine

1984
Three distinct subtypes of serotonergic receptors mediate the triphasic blood pressure response to serotonin in rats.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1984, Volume: 2, Issue:3

    Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Indoles; Ketanserin; Mice; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Tropisetron

1984
The use of ketanserin, a 5-hydroxytryptamine receptor antagonist, for treatment of postoperative hypertension following coronary artery bypass surgery.
    Anesthesia and analgesia, 1983, Volume: 62, Issue:1

    Topics: Coronary Artery Bypass; Female; Heart Rate; Hemodynamics; Humans; Hypertension; Infusions, Parenteral; Injections, Intravenous; Ketanserin; Male; Middle Aged; Piperidines; Postoperative Complications; Serotonin Antagonists

1983
Involvement of 5-HT2 receptors in the wet-dog shake behaviour induced by 5-hydroxytryptophan in the rat.
    Neuropharmacology, 1983, Volume: 22, Issue:7

    Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Female; Ketanserin; Methysergide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1983
Ketanserin in the treatment of hypertension following coronary artery bypass surgery. A preliminary study.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1983, Oct-01, Volume: 64, Issue:15

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Coronary Artery Bypass; Humans; Hypertension; Ketanserin; Middle Aged; Piperidines; Postoperative Care; Postoperative Complications

1983
Effects of ketanserin and mepyramine on platelet aggregation and on the uptake of 5-hydroxytryptamine into platelets.
    Thrombosis research, 1983, Jun-01, Volume: 30, Issue:5

    Topics: Adenosine Diphosphate; Aminopyridines; Blood Platelets; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1983
Antagonism of the 5-HT-induced bronchoconstriction in the cat.
    Archives internationales de pharmacodynamie et de therapie, 1983, Volume: 263, Issue:1

    Topics: Animals; Bronchi; Carbachol; Cats; Clenbuterol; Cyproheptadine; Female; Hemodynamics; Ketanserin; Male; Piperidines; Pregnancy; Serotonin; Serotonin Antagonists; Theophylline

1983
Prophylactic use of ketanserin in a patient with carcinoid syndrome.
    British journal of anaesthesia, 1983, Volume: 55, Issue:9

    Topics: Female; Humans; Hypertension; Intraoperative Complications; Ketanserin; Malignant Carcinoid Syndrome; Middle Aged; Piperidines; Serotonin Antagonists

1983
Ketanserin, a novel 5-hydroxytryptamine antagonist: monotherapy in essential hypertension.
    British journal of clinical pharmacology, 1983, Volume: 16, Issue:2

    Topics: Adult; Aged; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Ketanserin; Kinetics; Male; Middle Aged; Piperidines; Serotonin Antagonists

1983
Pharmacokinetics of ketanserin in man.
    European journal of clinical pharmacology, 1983, Volume: 25, Issue:1

    Topics: Administration, Oral; Adult; Blood Pressure; Blood Proteins; Female; Half-Life; Heart Rate; Humans; Injections, Intravenous; Ketanserin; Kinetics; Male; Piperidines; Protein Binding

1983
Antagonism of the effects of the hallucinogen DOM and the purported 5-HT agonist quipazine by 5-HT2 antagonists.
    European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

    Topics: Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists

1983
The effect of a 5-HT antagonist, ketanserin, on blood pressure, the renin-angiotensin system and sympathoadrenal function in normal man.
    British journal of clinical pharmacology, 1983, Volume: 16, Issue:3

    Topics: Adrenal Glands; Adult; Blood Pressure; Diet; Heart Rate; Humans; Ketanserin; Male; Phenylephrine; Piperidines; Posture; Renin-Angiotensin System; Serotonin Antagonists; Sympathetic Nervous System; Time Factors

1983
Characterization and regional distribution of serotonin S2-receptors in human brain.
    Brain research, 1983, Oct-16, Volume: 276, Issue:2

    Topics: Brain; Brain Chemistry; Humans; Ketanserin; Kinetics; Piperidines; Receptors, Serotonin

1983
Effects of pirenperone and ketanserin on rat prolactin secretion in vivo and in vitro.
    European journal of pharmacology, 1983, Aug-19, Volume: 92, Issue:1-2

    Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin Antagonists; Tranquilizing Agents

1983
Autoradiographic distribution of serotonin2 receptors in rat brain.
    European journal of pharmacology, 1983, Sep-02, Volume: 92, Issue:3-4

    Topics: Animals; Brain Chemistry; Ketanserin; Male; Piperidines; Rats; Receptors, Serotonin; Tissue Distribution

1983
The effect of ketanserin, a specific serotonin antagonist, on burn shock hemodynamic parameters in a porcine burn model.
    The Journal of trauma, 1983, Volume: 23, Issue:10

    Topics: Animals; Blood Pressure; Body Temperature; Burns; Disease Models, Animal; Heart Rate; Hemodynamics; Ketanserin; Piperidines; Serotonin Antagonists; Shock, Traumatic; Swine

1983
Determination of ketanserin and its major metabolite (reduced ketanserin) in human plasma by high-performance liquid chromatography.
    Journal of chromatography, 1983, Oct-14, Volume: 277

    Topics: Adult; Chromatography, High Pressure Liquid; Female; Humans; Ketanserin; Oxidation-Reduction; Piperidines; Spectrophotometry, Ultraviolet

1983
pH-dependent modulation of agonist interactions with [3H]-ketanserin-labelled S2 serotonin receptors.
    Life sciences, 1983, Nov-14, Volume: 33, Issue:20

    Topics: Animals; Binding, Competitive; Frontal Lobe; Hydrogen-Ion Concentration; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1983
Characterization of serotonin binding sites on human platelets.
    Life sciences, 1983, Nov-14, Volume: 33, Issue:20

    Topics: Adult; Binding, Competitive; Blood Platelets; Frontal Lobe; Humans; Ketanserin; Male; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1983
Inhibitory effect of ketanserin on ergonovine-induced contractions of isolated canine coronary arteries.
    Archives internationales de pharmacodynamie et de therapie, 1983, Volume: 265, Issue:1

    Topics: Animals; Coronary Vessels; Dogs; Ergonovine; In Vitro Techniques; Ketanserin; Methysergide; Piperidines; Serotonin Antagonists; Vasoconstriction

1983
The 5-hydroxytryptamine receptor of blood platelets.
    Journal of neural transmission, 1983, Volume: 57, Issue:4

    Topics: Animals; Binding, Competitive; Blood Platelets; Brain; Calcium; Cell Membrane; Ketanserin; Kinetics; Lysergic Acid Diethylamide; Models, Neurological; Neurons; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1983
5-Hydroxytryptamine can mediate endothelium-dependent relaxation of coronary arteries.
    The American journal of physiology, 1983, Volume: 245, Issue:6

    Topics: Animals; Blood Platelets; Coronary Vessels; Dogs; In Vitro Techniques; Isometric Contraction; Ketanserin; Methysergide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Piperidines; Serotonin; Serotonin Antagonists; Thromboxane B2

1983
Selective inhibition by ketanserin and spiroperidol of 5-HT-induced myometrial contraction.
    European journal of pharmacology, 1983, Dec-09, Volume: 96, Issue:1-2

    Topics: Animals; Butyrophenones; Estradiol; Female; Ketanserin; Ovary; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Spiperone; Uterine Contraction

1983
Evidence for mediation by 5-HT2 receptors of 5-hydroxytryptamine-induced contraction of canine basilar artery.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:4

    Topics: Animals; Basilar Artery; Cerebral Cortex; Dogs; Female; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium

1983
Haemodynamic response to ketanserin in rabbits with Page hypertension: comparison with prazosin.
    Journal of hypertension, 1983, Volume: 1, Issue:2

    Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Hypertension; Ketanserin; Male; Methoxamine; Piperidines; Prazosin; Quinazolines; Rabbits; Receptors, Serotonin; Serotonin Antagonists

1983
Long-term effects on central haemodynamics and body fluid volumes of ketanserin in essential hypertension studies at rest and during dynamic exercise.
    Journal of hypertension, 1983, Volume: 1, Issue:4

    Topics: Adult; Blood Pressure; Body Fluids; Body Weight; Cardiac Output; Female; Heart Rate; Hemodynamics; Humans; Hypertension; Ketanserin; Male; Middle Aged; Oxygen Consumption; Physical Exertion; Piperidines; Rest; Time Factors; Vascular Resistance

1983
The influence of antiserotonin treatment with ketanserin on the pulmonary lodgement of circulating tumour cells in normal and traumatized rats.
    European journal of cancer & clinical oncology, 1983, Volume: 19, Issue:6

    Topics: Animals; Femoral Fractures; Fibrosarcoma; Ketanserin; Lung Neoplasms; Neoplasm Transplantation; Neoplastic Cells, Circulating; Piperidines; Rats; Sarcoma, Experimental; Serotonin Antagonists

1983
Differential actions of serotonin antagonists on two behavioral models of serotonin receptor activation in the rat.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 228, Issue:1

    Topics: Animals; Behavior, Animal; Butyrophenones; Ketanserin; Male; Metergoline; Methysergide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1984
The effects of platelet-derived contractile agents on human digital arteries.
    Clinical science (London, England : 1979), 1984, Volume: 66, Issue:4

    Topics: Arteries; Blood Platelets; Humans; Imidazoles; In Vitro Techniques; Indomethacin; Ketanserin; Muscle Contraction; Piperidines; Platelet Aggregation; Serotonin Antagonists; Thromboxane A2; Time Factors

1984
Ketanserin, a serotonin antagonist. Administration in patients with acute respiratory failure.
    Chest, 1984, Volume: 85, Issue:4

    Topics: Adult; Aged; Blood Proteins; Erythrocyte Indices; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Pulmonary Wedge Pressure; Respiratory Insufficiency; Stroke Volume; Vascular Resistance

1984
The involvement of 5-HT2-receptor sites in the activation of cat platelets.
    Thrombosis research, 1984, Feb-01, Volume: 33, Issue:3

    Topics: Adenosine Diphosphate; Animals; Blood Platelets; Cats; Collagen; Dose-Response Relationship, Drug; Ketanserin; Kinetics; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin

1984
Interactions of agonists with D-2 dopamine receptors: evidence for a single receptor population existing in multiple agonist affinity-states in rat striatal membranes.
    Biochemical pharmacology, 1984, Mar-15, Volume: 33, Issue:6

    Topics: Animals; Binding, Competitive; Butyrophenones; Corpus Striatum; Domperidone; Dopamine Antagonists; Guanine Nucleotides; Ketanserin; Metoclopramide; Piperidines; Radioligand Assay; Rats; Receptors, Dopamine; Sodium; Spiperone; Temperature

1984
Acute effects of ketanserin on left ventricular function, metabolism and coronary blood flow.
    British journal of clinical pharmacology, 1984, Volume: 17, Issue:3

    Topics: Adult; Blood Pressure; Cardiac Catheterization; Coronary Circulation; Female; Heart; Heart Rate; Heart Ventricles; Humans; Ketanserin; Male; Middle Aged; Myocardium; Piperidines; Pulmonary Artery; Vascular Resistance

1984
Reduced binding of [3H]ketanserin to cortical 5-ht2 receptors in senile dementia of the Alzheimer type.
    Neuroscience letters, 1984, Jan-27, Volume: 44, Issue:1

    Topics: Age Factors; Aged; Alzheimer Disease; Cerebral Cortex; Humans; Ketanserin; Piperidines; Receptors, Serotonin; Serotonin Antagonists

1984
Ergonovine-induced myocardial ischemia: no role for serotonergic receptors?
    Circulation, 1984, Volume: 70, Issue:2

    Topics: Aged; Angina Pectoris; Coronary Vasospasm; Coronary Vessels; Ergonovine; Hand; Humans; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Vasoconstriction

1984
Solubilization of serotonin S2-receptors from human brain.
    European journal of pharmacology, 1984, May-04, Volume: 100, Issue:3-4

    Topics: Animals; Brain Chemistry; Dogs; Humans; In Vitro Techniques; Ketanserin; Kinetics; Lysophosphatidylcholines; Membranes; Piperidines; Rats; Receptors, Serotonin; Species Specificity

1984
Ketanserin and vascular contractions in response to cooling.
    European journal of pharmacology, 1984, Apr-06, Volume: 99, Issue:4

    Topics: Animals; Arteries; Cold Temperature; In Vitro Techniques; Ketanserin; Piperidines; Rabbits; Serotonin; Serotonin Antagonists; Vasoconstriction

1984
Intrapartum treatment of preeclamptic hypertension by ketanserin--a serotonin receptor antagonist.
    American journal of obstetrics and gynecology, 1984, Jul-01, Volume: 149, Issue:5

    Topics: Adult; Antihypertensive Agents; Delivery, Obstetric; Female; Humans; Hydralazine; Hypertension; Infant, Newborn; Ketanserin; Piperidines; Pre-Eclampsia; Pregnancy; Serotonin Antagonists; Time Factors; Vascular Resistance

1984
Serotonergic regulation of cortisol secretion in dogs.
    Endocrinology, 1984, Volume: 115, Issue:2

    Topics: Animals; Dogs; Fenfluramine; Hydrocortisone; Ketanserin; Piperidines; Quipazine; Serotonin; Time Factors

1984
Some behavioral effects of hallucinogens are mediated by a postsynaptic serotonergic action: evidence from single unit studies in freely moving cats.
    European journal of pharmacology, 1984, May-18, Volume: 101, Issue:1-2

    Topics: Animals; Apomorphine; Behavior, Animal; Cats; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Female; Hallucinogens; Ketanserin; Lisuride; Lysergic Acid Diethylamide; Metergoline; Mianserin; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Synapses

1984
Effects of tryptamine antagonists on the anaphylactic contractions of the bovine pulmonary smooth muscles.
    Journal of veterinary pharmacology and therapeutics, 1984, Volume: 7, Issue:2

    Topics: Anaphylaxis; Animals; Cattle; Horses; In Vitro Techniques; Ketanserin; Lung; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Pulmonary Artery; Pulmonary Veins; Serotonin Antagonists; Trachea; Tryptamines

1984
Restoration of pulmonary perfusion by a serotonin antagonist.
    Angiology, 1981, Volume: 32, Issue:7

    Topics: Adult; Aged; Blood Pressure; Carbon Dioxide; Embolism, Air; Female; Humans; Infant, Newborn; Intraoperative Complications; Ketanserin; Male; Piperidines; Pulmonary Circulation; Respiration; Respiratory Distress Syndrome; Serotonin Antagonists; Vasodilator Agents

1981
Treatment of hypertension with ketanserin, a new selective 5-HT2 receptor antagonist.
    British medical journal (Clinical research ed.), 1982, Feb-20, Volume: 284, Issue:6315

    Topics: Adult; Aged; Cardiac Output; Female; Heart Rate; Humans; Hypertension; Ketanserin; Kidney; Male; Middle Aged; Norepinephrine; Piperidines; Receptors, Serotonin; Vascular Resistance

1982
Platelet-mediated vascular contractions: inhibition of the serotonergic component by ketanserin.
    Thrombosis research, 1982, Sep-15, Volume: 27, Issue:6

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Depression, Chemical; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Suprofen; Thrombin

1982
An assessment of the participatory role of prostaglandins and serotonin in the pathophysiology of endotoxic shock.
    American journal of obstetrics and gynecology, 1983, Feb-15, Volume: 145, Issue:4

    Topics: Animals; Dogs; Hemodynamics; Indomethacin; Ketanserin; Oxygen; Piperidines; Prostaglandins; Pulmonary Circulation; Serotonin; Serotonin Antagonists; Shock, Septic

1983
Therapeutic benefits of 5-hydroxytryptamine inhibition following pulmonary embolism.
    Annals of surgery, 1983, Volume: 197, Issue:2

    Topics: Animals; Dogs; Female; Ketanserin; Male; Piperidines; Platelet Count; Prostaglandins; Pulmonary Embolism; Pulmonary Wedge Pressure; Receptors, Serotonin; Respiratory Dead Space; Serotonin; Serotonin Antagonists; Vascular Resistance

1983
The effect of thrombocytopenia and antiserotonin treatment on the lodgement of circulating tumor cells. A vital fluorescence microscopic, electron microscopic and isotope study in the rat.
    Journal of cancer research and clinical oncology, 1983, Volume: 105, Issue:1

    Topics: Animals; Female; Fibrosarcoma; Ketanserin; Liver Neoplasms; Male; Microscopy, Electron; Microscopy, Fluorescence; Neoplasm Transplantation; Neoplastic Cells, Circulating; Phagocytosis; Piperidines; Rats; Sarcoma, Experimental; Serotonin Antagonists; Thrombocytopenia

1983
High-performance liquid chromatographic assay with fluorometric detection of ketanserin, a new antihypertensive agent and serotonin S2 antagonist in human plasma, blood and urine.
    Journal of chromatography, 1983, Feb-11, Volume: 272, Issue:2

    Topics: Antihypertensive Agents; Chromatography, High Pressure Liquid; Half-Life; Humans; Ketanserin; Piperidines; Radioimmunoassay; Serotonin Antagonists; Spectrometry, Fluorescence

1983
Determination of ketanserin in human plasma by high-performance liquid chromatography.
    Journal of chromatography, 1983, Feb-11, Volume: 272, Issue:2

    Topics: Chromatography, High Pressure Liquid; Humans; Hypertension; Ketanserin; Piperidines; Time Factors

1983
Ketanserin, a new selective 5-HT2 receptor blocking agent, inhibits the antidiuretic effect of 5-hydroxytryptamine (5-HT) in Wistar rats.
    Archives internationales de pharmacodynamie et de therapie, 1983, Volume: 261, Issue:2

    Topics: Animals; Diuresis; Ketanserin; Kidney; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Time Factors

1983
Differences in the regulatory adaptation of the 5HT recognition sites labelled by 3H-mianserin or 3H-ketanserin.
    Neuropharmacology, 1983, Volume: 22, Issue:1

    Topics: Animals; Axons; Dibenzazepines; Hippocampus; Imipramine; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Synapses; Tritium

1983
Continuous imaging of regional blood flow in peripheral vascular disease using Krypton-81m: effect of Ketanserin, a new selective serotonin antagonist.
    Diagnostic imaging, 1983, Volume: 52, Issue:2-3

    Topics: Animals; Arteriosclerosis Obliterans; Cats; Diabetic Angiopathies; Female; Humans; Hyperemia; Ketanserin; Krypton; Leg; Male; Piperidines; Radioisotopes; Radionuclide Imaging; Regional Blood Flow; Serotonin; Serotonin Antagonists; Thromboangiitis Obliterans; Vascular Diseases

1983
Demonstration of S2-receptor binding sites on cat blood platelets using [3H]ketanserin.
    European journal of pharmacology, 1983, Mar-18, Volume: 88, Issue:1

    Topics: Animals; Binding Sites; Blood Platelets; Cats; Corpus Striatum; Female; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Tritium

1983
Ketanserin prevents platelet aggregation and endotoxin-induced pulmonary vasoconstriction.
    Critical care medicine, 1983, Volume: 11, Issue:8

    Topics: Animals; Dogs; Epinephrine; Hemodynamics; Hypertension, Pulmonary; Ketanserin; Male; Oxygen; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists; Shock, Septic

1983
Chronic clozapine treatment of rats down-regulates cortical 5-HT2 receptors.
    European journal of pharmacology, 1983, May-06, Volume: 89, Issue:3-4

    Topics: Animals; Cerebral Cortex; Clozapine; Dibenzazepines; Ketanserin; Male; Piperidines; Rats; Receptors, Serotonin; Time Factors

1983
Determination of ketanserin in plasma by reversed-phase high-performance liquid chromatography.
    Journal of chromatography, 1983, Jun-10, Volume: 275, Issue:1

    Topics: Chromatography, High Pressure Liquid; Humans; Ketanserin; Piperidines

1983
The effect of serotonin inhibition on initial microvessel hemostasis and platelet aggregation in vivo.
    Thrombosis and haemostasis, 1983, Jun-28, Volume: 49, Issue:3

    Topics: Animals; Bleeding Time; Dihydroergotamine; Female; Hemostasis; Ketanserin; Male; Mesenteric Arteries; Mesenteric Veins; Microcirculation; Piperidines; Platelet Aggregation; Rabbits; Serotonin Antagonists

1983
3H-Ketanserin labels serotonin S2-receptor binding sites on cat blood platelets.
    Archives internationales de pharmacodynamie et de therapie, 1983, Volume: 263, Issue:2

    Topics: Animals; Blood Platelets; Cats; Cell Membrane; In Vitro Techniques; Ketanserin; Kinetics; Piperidines; Receptors, Serotonin

1983
On the mechanism of action of ketanserin, a selective antagonist of the S2 receptors with antihypertensive activity.
    Proceedings of the Western Pharmacology Society, 1983, Volume: 26

    Topics: Animals; Antihypertensive Agents; Dogs; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Norepinephrine; Piperidines; Rats; Serotonin Antagonists; Vasodilation

1983
Is prevention of hypertension after open heart surgery possible by blocking 5HT2-receptors with ketanserin?
    Acta anaesthesiologica Belgica, 1982, Volume: 33, Issue:2

    Topics: Adult; Aged; Anesthesia; Aortic Valve; Coronary Artery Bypass; Heart Valve Prosthesis; Hemodynamics; Humans; Hypertension; Injections, Intravenous; Ketanserin; Middle Aged; Nitrous Oxide; Piperidines; Postoperative Complications; Serotonin Antagonists

1982
Interaction between 5-hydroxytryptamine and other vasoconstrictor substances in the isolated femoral artery of the rabbit; effect of ketanserin (R 41 468).
    European journal of pharmacology, 1982, Feb-05, Volume: 77, Issue:4

    Topics: Animals; Drug Interactions; Evoked Potentials; Femoral Artery; In Vitro Techniques; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rabbits; Serotonin; Vasoconstrictor Agents

1982
The effects of serotonin-receptor blockade after cardiopulmonary by-pass. A pilot study.
    Acta anaesthesiologica Belgica, 1982, Volume: 33, Issue:1

    Topics: Aged; Cardiopulmonary Bypass; Female; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Pilot Projects; Piperidines; Postoperative Complications; Serotonin Antagonists

1982
[3H]Ketanserin (R 41 468), a selective 3H-ligand for serotonin2 receptor binding sites. Binding properties, brain distribution, and functional role.
    Molecular pharmacology, 1982, Volume: 21, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Cerebral Cortex; Female; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Species Specificity

1982
Regional distribution of serotonin-2 receptor binding sites in the brain and effects of neuronal lesions.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 256, Issue:2

    Topics: Animals; Brain; Dogs; Guinea Pigs; Ketanserin; Microsomes; Mitochondria; Neurons; Neurotoxins; Piperidines; Rabbits; Rats; Receptors, Serotonin; Serotonin Antagonists; Species Specificity

1982
In vivo binding of [3H]ketanserin on serotonin S2-receptors in rat brain.
    European journal of pharmacology, 1982, Jun-16, Volume: 81, Issue:1

    Topics: Animals; Brain; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Tritium

1982
Haemorheological effects of ketanserin, a selective 5-HT2 receptor antagonist, in aged, spontaneously hypertensive dogs.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 258, Issue:1

    Topics: Aging; Animals; Blood Cell Count; Blood Pressure; Blood Viscosity; Dogs; Erythrocyte Membrane; Hypertension; Ketanserin; Piperidines; Serotonin Antagonists; Vascular Resistance

1982
Comparative effects of ketanserin, a novel serotonergic receptor antagonist, on 5HT-induced shape change and 5HT uptake in rat and human platelets.
    Biochemical pharmacology, 1982, Sep-15, Volume: 31, Issue:18

    Topics: Adenosine Diphosphate; Animals; Blood Platelets; Clomipramine; Female; Humans; In Vitro Techniques; Ketanserin; Kinetics; Male; Methysergide; Piperidines; Rats; Serotonin; Serotonin Antagonists

1982
Rapid method for determination of ketanserin, a novel antiserotonin drug, by high-performance liquid chromatography.
    Journal of chromatography, 1982, Oct-08, Volume: 232, Issue:1

    Topics: Autoanalysis; Chromatography, High Pressure Liquid; Humans; Ketanserin; Piperidines; Serotonin Antagonists

1982
Effects of Ketanserine on rumino-reticular motility and eructation in sheep: a possible application as an anti-bloating substance.
    Journal of veterinary pharmacology and therapeutics, 1982, Volume: 5, Issue:3

    Topics: Animals; Eructation; Gastrointestinal Motility; Ketanserin; Piperidines; Rumen; Serotonin Antagonists; Sheep

1982
Selectivity of calcium antagonism and serotonin antagonism with respect to venous and arterial tissues.
    Angiology, 1981, Volume: 32, Issue:7

    Topics: Animals; Arteries; Calcium; Cinnarizine; Dogs; Flunarizine; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rabbits; Rats; Serotonin; Serotonin Antagonists; Veins

1981
Vascular activity of ketanserin (R 41 468), a selective 5-HT2 receptor antagonist.
    Archives internationales de pharmacodynamie et de therapie, 1981, Volume: 250, Issue:2

    Topics: Animals; Blood Pressure; Dogs; Guinea Pigs; Humans; In Vitro Techniques; Ketanserin; Piperidines; Rabbits; Rats; Serotonin Antagonists; Vasoconstriction

1981
Plethysmographic registration of volume changes in a hand vein. Effects of serotonin and of a specific antagonist.
    Angiology, 1980, Volume: 31, Issue:12

    Topics: Blood Pressure; Blood Volume; Hand; Heart Rate; Humans; Ketanserin; Piperidines; Plethysmography; Serotonin; Serotonin Antagonists; Veins

1980
Neurochemical and behavioral evidence that quipazine-ketanserin discrimination is mediated by serotonin2A receptor.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: Animals; Brain Mapping; Discrimination Learning; Dose-Response Relationship, Drug; Fluorobenzenes; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
In vivo dopamine-D2 and serotonin-5-HT2 receptor binding study of risperidone and haloperidol.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Cerebellum; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; In Vitro Techniques; Isoxazoles; Ketanserin; Ligands; Male; Neostriatum; Piperidines; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone

1994
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach

1995
Ketanserin analogues: the effect of structural modification on 5-HT2 serotonin receptor binding.
    Journal of medicinal chemistry, 1995, Mar-31, Volume: 38, Issue:7

    Topics: Animals; Binding Sites; Cerebral Cortex; Chemical Phenomena; Chemistry, Physical; In Vitro Techniques; Ketanserin; Magnetic Resonance Spectroscopy; Male; Molecular Structure; Piperazines; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Structure-Activity Relationship

1995
Antinociceptive effects of the kappa opioid, U50,488: lack of modulation by 5-HT2 antagonists.
    Psychopharmacology, 1993, Volume: 112, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Ergolines; Ketanserin; Male; Piperidines; Pyrrolidines; Receptors, Opioid, kappa; Saimiri; Serotonin Antagonists

1993
5-HT receptor subtypes involved in luminal serotonin-induced secretion in rat intestine in vivo.
    The Journal of surgical research, 1994, Volume: 56, Issue:3

    Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Ileum; Indoles; Jejunum; Ketanserin; Male; Methysergide; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Tropisetron; Water-Electrolyte Balance

1994
Monoamine systems in the discriminative effects of spiradoline, a kappa-opioid agonist.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Analgesics; Animals; Avoidance Learning; Biogenic Monoamines; Discrimination, Psychological; Dopamine Antagonists; Fenfluramine; Fluoxetine; Generalization, Stimulus; Ketanserin; Male; Piperidines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Selective Serotonin Reuptake Inhibitors; Serotonin; Synaptic Transmission

1994
Antiserotoninergic activity of 2-aminoethylbenzocyclanones in rat aorta: structure-activity relationships.
    Journal of pharmaceutical sciences, 1993, Volume: 82, Issue:5

    Topics: Animals; Aorta, Thoracic; Butyrophenones; In Vitro Techniques; Ketanserin; Ketones; Molecular Conformation; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1993
Investigation of the mechanism by which ketanserin prolongs the duration of the cardiac action potential.
    Journal of cardiovascular pharmacology, 1995, Volume: 26, Issue:5

    Topics: Action Potentials; Amphetamines; Animals; Guinea Pigs; Heart; Ketanserin; Male; Piperidines; Potassium Channels; Serotonin Antagonists

1995
Inhibition of noradrenaline release via presynaptic 5-HT1D alpha receptors in human atrium.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3

    Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Cisapride; Corticosterone; Desipramine; Heart Atria; Humans; Indoles; Ketanserin; Male; Middle Aged; Norepinephrine; Oxadiazoles; Piperidines; Receptors, Presynaptic; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tritium; Tryptamines

1996
[3H]MDL 100,907: a novel selective 5-HT2A receptor ligand.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:2

    Topics: Animals; Fluorobenzenes; Frontal Lobe; Ketanserin; Ligands; Male; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists

1996
Novel potent sigma 1 ligands: N-[omega-(tetralin-1-yl)alkyl]piperidine derivatives.
    Journal of medicinal chemistry, 1996, Oct-11, Volume: 39, Issue:21

    Topics: Animals; Hippocampus; Ketanserin; Phencyclidine; Piperidines; Rats; Receptors, Phencyclidine; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, sigma; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes

1996
Preclinical evaluation of [123I]R93274 as a SPECT radiotracer for imaging 5-HT2A receptors.
    European journal of pharmacology, 1997, Mar-05, Volume: 321, Issue:3

    Topics: Animals; Benzamides; Brain; Dopamine Antagonists; Female; Iodine Radioisotopes; Ketanserin; Papio; Piperidines; Raclopride; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Salicylamides; Serotonin Antagonists; Tomography, Emission-Computed, Single-Photon

1997
Pharmacological characterization of in vivo properties of putative mixed 5-HT1A agonist/5-HT(2A/2C) antagonist anxiolytics. II. Drug discrimination and behavioral observation studies in rats.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzopyrans; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Nicotinic Acids; Piperazines; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

1997
Selective visualization of rat brain 5-HT2A receptors by autoradiography with [3H]MDL 100,907.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:4

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Fluorobenzenes; Guanylyl Imidodiphosphate; In Situ Hybridization; In Vitro Techniques; Ketanserin; Male; Naphthalenes; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists

1997
A potent 5-hydroxytryptamine receptor (5-HT2A) antagonist, DV-7028, delays arterial thrombosis development in rats.
    Thrombosis research, 1998, Jun-15, Volume: 90, Issue:6

    Topics: Animals; Aorta, Abdominal; Bleeding Time; Ketanserin; Male; Piperidines; Platelet Aggregation; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Thrombophlebitis; Thrombosis; Triazines

1998
Vascular and cardiac effects of DV-7028, a selective, 5-HT2-receptor antagonist in rats.
    Journal of cardiovascular pharmacology, 1998, Volume: 32, Issue:2

    Topics: Animals; Baroreflex; Blood Pressure; Cardiovascular System; Coronary Circulation; Heart; Heart Rate; Hindlimb; Injections, Intravenous; Ketanserin; Male; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Triazines; Vagotomy

1998
5-HT2A receptor antagonists block MK-801-induced stereotypy and hyperlocomotion.
    European journal of pharmacology, 1998, Oct-02, Volume: 358, Issue:2

    Topics: Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Histamine H2 Antagonists; Ketanserin; Locomotion; Male; Mice; Mice, Inbred BALB C; Neuroprotective Agents; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Stereotypic Movement Disorder

1998
[3H]MDL 100,907 labels 5-HT2A serotonin receptors selectively in primate brain.
    Neuropharmacology, 1998, Volume: 37, Issue:9

    Topics: Aged; Aged, 80 and over; Animals; Binding Sites; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Male; Naphthalenes; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Tritium

1998
Agonist and antagonist binding to rabbit cortical 5-HT2A receptors: opposite effects of magnesium.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: Amphetamines; Animals; Cerebral Cortex; Fluorobenzenes; Guanylyl Imidodiphosphate; Ketanserin; Magnesium; Methysergide; Piperidines; Prazosin; Rabbits; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1998
Effect of 5-HT2 receptor antagonists on a cranial nerve reflex in the rabbit: evidence for inverse agonism.
    Psychopharmacology, 1999, Volume: 141, Issue:2

    Topics: Animals; Cranial Nerves; Ergolines; Female; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Piperidines; Rabbits; Receptors, Serotonin; Reflex; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach.
    Japanese journal of pharmacology, 1999, Volume: 79, Issue:1

    Topics: Animals; Atropine; Dioxanes; Enzyme Inhibitors; Female; Gastric Fundus; Granisetron; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscarinic Antagonists; Muscle Relaxation; Muscle Tonus; Nitroarginine; Piperidines; Pyloric Antrum; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Tetrodotoxin

1999
5-HT2C receptor involvement in female rat lordosis behavior.
    Brain research, 1999, Apr-17, Volume: 825, Issue:1-2

    Topics: Animals; Estradiol; Female; Fluorobenzenes; Indoles; Indophenol; Ketanserin; Ovariectomy; Piperidines; Posture; Pyridines; Rats; Rats, Inbred Strains; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sexual Behavior, Animal; Ventromedial Hypothalamic Nucleus

1999
Ketanserin and tetrabenazine abolish aggression in mice lacking monoamine oxidase A.
    Brain research, 1999, Jul-24, Volume: 835, Issue:2

    Topics: Adrenergic Uptake Inhibitors; Aggression; Animals; Brain; Corpus Striatum; Drug Evaluation, Preclinical; Fluorobenzenes; Frontal Lobe; Ketanserin; Male; Mice; Mice, Knockout; Monoamine Oxidase; Neurotransmitter Agents; Piperidines; Radioligand Assay; Serotonin Antagonists; Tetrabenazine

1999
Human striosomes are enriched in 5-HT2A receptors: autoradiographical visualization with [3H]MDL100,907,[125I](+/-)DOI and [3H]ketanserin.
    The European journal of neuroscience, 1999, Volume: 11, Issue:10

    Topics: Adult; Aged; Autoradiography; Female; Fluorobenzenes; Humans; Indophenol; Iodine Radioisotopes; Ketanserin; Male; Middle Aged; Neostriatum; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Tritium

1999
[2-(omega-phenylalkyl)phenoxy]alkylamines.II: Synthesis and selective serotonin-2 receptor binding.
    Chemical & pharmaceutical bulletin, 2000, Volume: 48, Issue:2

    Topics: Animals; Blood Platelets; Blood Vessels; Humans; In Vitro Techniques; Ketanserin; Phenyl Ethers; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Pyrroles; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Structure-Activity Relationship; Succinates; Vasoconstriction

2000
In vitro autoradiography of serotonin 5-HT(2A/2C) receptor-activated G protein: guanosine-5'-(gamma-[(35)S]thio)triphosphate binding in rat brain.
    Journal of neuroscience research, 2000, Sep-15, Volume: 61, Issue:6

    Topics: Amphetamines; Animals; Autoradiography; Brain Chemistry; Dose-Response Relationship, Drug; Fluorobenzenes; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Image Processing, Computer-Assisted; Indoles; Ketanserin; Male; Membrane Proteins; Piperidines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Subcellular Fractions; Sulfur Radioisotopes

2000
Mapping of 5-HT2A receptors and their mRNA in monkey brain: [3H]MDL100,907 autoradiography and in situ hybridization studies.
    The Journal of comparative neurology, 2001, Jan-22, Volume: 429, Issue:4

    Topics: Animals; Autoradiography; Brain; Brain Mapping; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Macaca mulatta; Male; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists

2001
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
Antagonism of 5-hydroxytryptamine(2a) receptors attenuates the behavioral effects of cocaine in rats.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 297, Issue:1

    Topics: Animals; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Discrimination Learning; Dopamine; Fluorobenzenes; Ketanserin; Male; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists

2001
Assessment of affinity and dissociation ability of a newly synthesized 5-HT2 antagonist, AT-1015: comparison with other 5-HT2 antagonists.
    Japanese journal of pharmacology, 2001, Volume: 87, Issue:3

    Topics: Animals; Cerebral Cortex; Isonipecotic Acids; Ketanserin; Male; Piperidines; Rabbits; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists

2001
Multiple 5-HT receptors are involved in the effects of acute MDMA treatment: studies on locomotor activity and responding for conditioned reinforcement.
    Psychopharmacology, 2002, Volume: 162, Issue:3

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Ethylamines; Indoles; Ketanserin; Male; Motor Activity; Oxadiazoles; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors

2002
Biodistribution and displacement studies of the selective 5-HT2A receptor antagonist 123I-5-I-R91150 in the normal dog.
    Nuclear medicine communications, 2002, Volume: 23, Issue:10

    Topics: Animals; Binding, Competitive; Brain; Dogs; Ketanserin; Piperidines; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Tissue Distribution; Tomography, Emission-Computed, Single-Photon; Whole-Body Counting

2002
Pharmacological characterization of the effects of 3,4-methylenedioxymethamphetamine ("ecstasy") and its enantiomers on lethality, core temperature, and locomotor activity in singly housed and crowded mice.
    Psychopharmacology, 2003, Volume: 166, Issue:3

    Topics: Animals; Body Temperature; Cold Temperature; Crowding; Dose-Response Relationship, Drug; Fluorobenzenes; Fluoxetine; Hallucinogens; Ketanserin; Lethal Dose 50; Male; Mice; Motor Activity; N-Methyl-3,4-methylenedioxyamphetamine; Piperidines; Platelet Aggregation Inhibitors; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Social Isolation; Stereoisomerism; Telemetry

2003
Discriminative stimulus properties of (+/-)-fenfluramine: the role of 5-HT2 receptor subtypes.
    Behavioral neuroscience, 2003, Volume: 117, Issue:2

    Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Fenfluramine; Fluorobenzenes; Indoles; Ketanserin; Male; Piperidines; Pyrazines; Pyridines; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Thiophenes

2003
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides

2003
Serotonin induces tonic firing in layer V pyramidal neurons of rat prefrontal cortex during postnatal development.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Apr-15, Volume: 23, Issue:8

    Topics: Age Factors; Animals; Down-Regulation; Female; In Vitro Techniques; Ketanserin; Male; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Signal Transduction

2003
Diverse regulation of atrial natriuretic peptide secretion by serotonin receptor subtypes.
    Cardiovascular research, 2003, Aug-01, Volume: 59, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Alkaloids; Aminobenzoates; Animals; Atrial Natriuretic Factor; Benzophenanthridines; Benzothiazoles; Calcium; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Dose-Response Relationship, Drug; Heart; Heart Atria; Imines; Indoles; Isoquinolines; Ketanserin; Male; Myocytes, Cardiac; Neomycin; para-Aminobenzoates; Perfusion; Phenanthridines; Piperazines; Piperidines; Protein Kinase C; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Staurosporine; Sulfonamides; Thiazoles; Type C Phospholipases

2003
Fenfluramine evokes 5-HT2A receptor-mediated responses but does not displace [11C]MDL 100907: small animal PET and gene expression studies.
    Synapse (New York, N.Y.), 2003, Dec-01, Volume: 50, Issue:3

    Topics: Animals; Carbon Radioisotopes; Cerebellum; Fenfluramine; Fluorobenzenes; Gene Expression; Genes, Immediate-Early; In Situ Hybridization; Ketanserin; Male; Neurons; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Time Factors; Tomography, Emission-Computed

2003
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:1

    Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines

2004
Functional role of the endocannabinoid system and AMPA/kainate receptors in 5-HT2A receptor-mediated wet dog shakes.
    European journal of pharmacology, 2005, May-23, Volume: 516, Issue:1

    Topics: Amphetamines; Animals; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Dose-Response Relationship, Drug; Endocannabinoids; Excitatory Amino Acid Antagonists; Injections, Intraperitoneal; Ketanserin; Male; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, Kainic Acid; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists

2005
Effects of donepezil, nicotine and haloperidol on the central serotonergic system in mice: implications for Tourette's syndrome.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:4

    Topics: Amphetamines; Animals; Behavior, Animal; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Donepezil; Dose-Response Relationship, Drug; Frontal Lobe; Gene Expression; Haloperidol; Humans; Indans; Ketanserin; Male; Mesencephalon; Mice; Mice, Inbred ICR; Nicotine; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin Antagonists; Tourette Syndrome

2005
Binding characteristics of the 5-HT2A receptor antagonists altanserin and MDL 100907.
    Synapse (New York, N.Y.), 2005, Dec-15, Volume: 58, Issue:4

    Topics: Animals; Binding, Competitive; Brain; Carbon Radioisotopes; Fluorine Radioisotopes; Fluorobenzenes; Ketanserin; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2005
Effects of 5-HT2A receptor stimulation on the discrimination of durations by rats.
    Behavioural pharmacology, 2006, Volume: 17, Issue:1

    Topics: Amphetamines; Animals; Association Learning; Brain; Discrimination Learning; Female; Fluorobenzenes; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Piperidines; Psychophysics; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Serotonin Receptor Agonists; Time Perception

2006
Functional characterization of serotonin receptor subtypes in human duodenal secretion.
    Basic & clinical pharmacology & toxicology, 2006, Volume: 98, Issue:2

    Topics: Adult; Aged; Bumetanide; Dioxanes; Duodenum; Female; Helicobacter Infections; Helicobacter pylori; Humans; In Vitro Techniques; Intestinal Secretions; Ion Transport; Ketanserin; Male; Middle Aged; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium Potassium Chloride Symporter Inhibitors

2006
Gasping activity in vitro: a rhythm dependent on 5-HT2A receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Mar-08, Volume: 26, Issue:10

    Topics: Action Potentials; Analysis of Variance; Animals; Animals, Newborn; Biological Clocks; Dose-Response Relationship, Drug; Drug Interactions; Flufenamic Acid; In Vitro Techniques; Ketanserin; Mice; Nerve Net; Neurons; Oxygen; Patch-Clamp Techniques; Piperidines; Receptor, Serotonin, 5-HT2A; Respiratory Burst; Respiratory Center; Respiratory Mechanics; Serotonin Antagonists; Substance P; Synaptic Transmission; Time Factors

2006
Rewarding properties of 1-benzylpiperazine, a new drug of abuse, in rats.
    Basic & clinical pharmacology & toxicology, 2006, Volume: 98, Issue:4

    Topics: Animals; Behavior, Animal; Benzazepines; Conditioning, Psychological; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ketanserin; Male; Piperidines; Psychotropic Drugs; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT3; Reward; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Substance-Related Disorders; Tropanes

2006
Cardiac baroreflex facilitation evoked by hypothalamus and prefrontal cortex stimulation: role of the nucleus tractus solitarius 5-HT2A receptors.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2006, Volume: 291, Issue:4

    Topics: Animals; Atenolol; Atropine Derivatives; Baroreflex; Brain; Electric Stimulation; Fluorobenzenes; Heart; Ketanserin; Male; Microinjections; Neural Inhibition; Neural Pathways; Parasympatholytics; Piperidines; Prefrontal Cortex; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Solitary Nucleus; Stimulation, Chemical; Sympatholytics

2006
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
    Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:3

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin

2007
Opposing effects of 5-HT(2A) and 5-HT(2C) receptor antagonists in the rat and mouse on premature responding in the five-choice serial reaction time test.
    Psychopharmacology, 2007, Volume: 195, Issue:2

    Topics: Aminopyridines; Amphetamines; Animals; Conditioning, Operant; Ethylamines; Fluorobenzenes; Impulsive Behavior; Indoles; Ketanserin; Male; Mice; Mice, Inbred C57BL; Piperidines; Quinolines; Rats; Reaction Time; Serial Learning; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Species Specificity

2007
Total synthesis and evaluation of [18F]MHMZ.
    Bioorganic & medicinal chemistry letters, 2008, Feb-15, Volume: 18, Issue:4

    Topics: Animals; Binding, Competitive; Brain; Fluorine Radioisotopes; Fluorobenzenes; Isotope Labeling; Ketanserin; Kinetics; Piperidines; Radioligand Assay; Radionuclide Imaging; Radiopharmaceuticals; Rats; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2008
Evidence that genetic variation in 5-HT transporter expression is linked to changes in 5-HT2A receptor function.
    Neuropharmacology, 2008, Volume: 54, Issue:5

    Topics: Amphetamines; Analysis of Variance; Animals; Brain; Cytoskeletal Proteins; Dose-Response Relationship, Drug; Fluorobenzenes; Gene Expression; Genetic Variation; Head Movements; Ketanserin; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Nerve Tissue Proteins; Piperidines; Protein Binding; Proto-Oncogene Proteins c-fos; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists

2008
Aripiprazole inhibits marble-burying behavior via 5-hydroxytryptamine (5-HT)1A receptor-independent mechanisms.
    European journal of pharmacology, 2008, Sep-11, Volume: 592, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Anxiety; Aripiprazole; Behavior, Animal; Benzodiazepines; Catalepsy; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Ketanserin; Male; Mice; Mice, Inbred ICR; Olanzapine; Piperazines; Piperidines; Postural Balance; Psychomotor Performance; Pyridines; Quinolones; Quinpirole; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists

2008
Effect of cyclosporin A administration on the biodistribution and multipinhole muSPECT imaging of [123I]R91150 in rodent brain.
    European journal of nuclear medicine and molecular imaging, 2009, Volume: 36, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Brain; Cyclosporine; Iodine Radioisotopes; Ketanserin; Ligands; Male; Mice; Piperidines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tomography, Emission-Computed, Single-Photon

2009
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane in rhesus monkeys: antagonism and apparent pA2 analyses.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 328, Issue:3

    Topics: Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Electroshock; Fluorobenzenes; Hallucinogens; Ketanserin; Macaca mulatta; Phenethylamines; Piperidines; Reaction Time; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Regression Analysis; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

2009
Genetic deletion of MAO-A promotes serotonin-dependent ventricular hypertrophy by pressure overload.
    Journal of molecular and cellular cardiology, 2009, Volume: 46, Issue:4

    Topics: Animals; Aorta; Blood Pressure; Cardiomegaly; Fibrosis; Fluorobenzenes; Gene Deletion; Gene Expression Regulation; Heart Ventricles; Ketanserin; Mice; Mice, Knockout; Monoamine Oxidase; Myocardium; Piperidines; Pressure; Receptors, Serotonin; Serotonin; Stress, Physiological; Ultrasonography

2009
Enhanced 5-HT(2A) receptors in brain stem and ALDH activity in brain stem and liver: 5-HT(2A) regulation on ALDH in primary hepatocytes cultures in vitro.
    Neurochemical research, 2009, Volume: 34, Issue:9

    Topics: Aldehyde Dehydrogenase; Animals; Brain Stem; Ethanol; Fluorobenzenes; Hepatocytes; Ketanserin; Liver; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin

2009
Age-dependent effects of the cannabinoid CB1 antagonist SR141716A on food intake, body weight change, and pruritus in rats.
    Psychopharmacology, 2009, Volume: 206, Issue:1

    Topics: Age Factors; Animals; Brain; Dose-Response Relationship, Drug; Drinking; Eating; Feeding Behavior; Ketanserin; Male; Piperidines; Pruritus; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Serotonin Antagonists; Weight Gain

2009
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM), ketanserin, and (R)-(+)-{alpha}-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-pipidinemethanol (MDL100907) in rats.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:2

    Topics: Analgesics, Opioid; Anesthetics, Dissociative; Animals; Conditioning, Operant; Discrimination, Psychological; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorobenzenes; Ketamine; Ketanserin; Male; Morphine; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

2009
State-dependent interactions between excitatory neuromodulators in the neuronal control of breathing.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Jun-16, Volume: 30, Issue:24

    Topics: Action Potentials; Adrenergic alpha-1 Receptor Antagonists; Animals; Animals, Newborn; Electric Stimulation; Electromyography; Hypoglossal Nerve; In Vitro Techniques; Isoindoles; Ketanserin; Locus Coeruleus; Mice; Microinjections; Neural Inhibition; Neural Pathways; Neurokinin-1 Receptor Antagonists; Neurons; Neurotransmitter Agents; Piperidines; Raphe Nuclei; Receptors, Adrenergic, alpha-1; Receptors, Neurokinin-1; Receptors, Serotonin, 5-HT2; Respiration; Respiratory Center; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2010
Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode.
    Chemical biology & drug design, 2010, Volume: 76, Issue:4

    Topics: Binding, Competitive; Combinatorial Chemistry Techniques; Fluorobenzenes; Hydrophobic and Hydrophilic Interactions; Ketanserin; Ligands; Phenols; Piperidines; Protein Binding; Pyridines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists

2010
Oleamide administered into the nucleus accumbens shell regulates feeding behaviour via CB1 and 5-HT2C receptors.
    The international journal of neuropsychopharmacology, 2010, Volume: 13, Issue:9

    Topics: Aminopyridines; Animals; Eating; Feeding Behavior; Hyperphagia; Hypothalamus; Indoles; Ketanserin; Male; Motor Activity; Nucleus Accumbens; Oleic Acids; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Antagonists

2010
Interaction of 5-HT2A and 5-HT2C receptors in R(-)-2,5-dimethoxy-4-iodoamphetamine-elicited head twitch behavior in mice.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 335, Issue:3

    Topics: Aminopyridines; Amphetamines; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Ethylamines; Fluorobenzenes; Hallucinogens; Head; Indoles; Ketanserin; Male; Mice; Mice, Inbred Strains; Movement; Piperidines; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Spiro Compounds; Sulfonamides

2010
Effects of 5-HT(2A) and 5-HT(2C) receptor antagonists on acute and chronic dyskinetic effects induced by haloperidol in rats.
    Behavioural brain research, 2011, Jun-01, Volume: 219, Issue:2

    Topics: Aminopyridines; Animals; Antipsychotic Agents; Brain Chemistry; Catalepsy; Dyskinesia, Drug-Induced; Fluorobenzenes; Gene Expression Regulation; Haloperidol; Immunohistochemistry; In Situ Hybridization; Indoles; Ketanserin; Male; Mouth; Piperidines; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; RNA, Messenger; Serotonin Antagonists

2011
p-Hydroxyamphetamine causes prepulse inhibition disruption in mice: contribution of serotonin neurotransmission.
    Behavioural brain research, 2011, Oct-10, Volume: 224, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Acoustic Stimulation; Analysis of Variance; Animals; Autoradiography; Brain; Dose-Response Relationship, Drug; Fenclonine; Fluorobenzenes; Inhibition, Psychological; Ketanserin; Male; Mice; p-Hydroxyamphetamine; Piperidines; Reflex, Startle; Serotonin; Serotonin Agents; Serotonin Plasma Membrane Transport Proteins; Time Factors

2011
Reduced levels of serotonin 2A receptors underlie resistance of Egr3-deficient mice to locomotor suppression by clozapine.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2012, Volume: 37, Issue:10

    Topics: Animals; Clozapine; Disease Models, Animal; Early Growth Response Protein 3; Humans; Hypnotics and Sedatives; Ketanserin; Male; Mice; Mice, Transgenic; Motor Activity; Piperidines; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin 5-HT2 Receptor Agonists; Serotonin Antagonists

2012
Direct comparison of [(18) F]MH.MZ and [(18) F] altanserin for 5-HT2A receptor imaging with PET.
    Synapse (New York, N.Y.), 2013, Volume: 67, Issue:6

    Topics: Animals; Brain; Fluorine Radioisotopes; Fluorobenzenes; Ketanserin; Piperidines; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Swine; Tissue Distribution; Tritium

2013
Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT₂A receptors, in mice.
    Psychopharmacology, 2015, Volume: 232, Issue:6

    Topics: Amphetamines; Animals; Dose-Response Relationship, Drug; Fluorobenzenes; Hallucinogens; Head Movements; Ketanserin; Male; Mice; Phenethylamines; Piperidines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2015
Involvement of Descending Serotonergic and Noradrenergic Systems and their Spinal Receptor Subtypes in the Antinociceptive Effect of Dipyrone.
    Drug research, 2015, Volume: 65, Issue:12

    Topics: 5,7-Dihydroxytryptamine; Adrenergic Neurons; Analgesics; Animals; Dipyrone; Dose-Response Relationship, Drug; Injections, Spinal; Ketanserin; Mice; Ondansetron; Oxidopamine; Pain Measurement; Piperidines; Prazosin; Propranolol; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonergic Neurons; Spinal Cord; Sulfonamides; Yohimbine

2015
Individual Differences in Impulsive Action Reflect Variation in the Cortical Serotonin 5-HT2A Receptor System.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2015, Volume: 40, Issue:8

    Topics: Animals; Choice Behavior; Dimethoxyphenylethylamine; Fluorobenzenes; Head Movements; Immunoprecipitation; Impulsive Behavior; Individuality; Ketanserin; Male; Piperidines; Prefrontal Cortex; Protein Binding; Rats; Rats, Sprague-Dawley; Reaction Time; Receptor, Serotonin, 5-HT2A; Serotonin Agents; Tritium

2015