ketanserin has been researched along with piperidines in 564 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 468 (82.98) | 18.7374 |
1990's | 49 (8.69) | 18.2507 |
2000's | 36 (6.38) | 29.6817 |
2010's | 11 (1.95) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Berardi, F; Daniele, E; Govoni, S; Leopoldo, M; Lograno, MD; Perrone, R; Tortorella, V | 1 |
Bowden, CR; De Coster, R; Heykants, J; Voina, SJ; Woestenborghs, R | 1 |
Emilsson, K; Hardebo, JE; Nystedt, S; Owman, C; Szabò, C | 1 |
Karnovsky, ML; Polanski, M | 1 |
Brazell, C; Campbell, IC; Mitchell, S; Stahl, SM; Twist, EC | 1 |
Arora, RC; Meltzer, HY; Nash, JF; Schreiber, MA | 1 |
Appell, KC; Barrett, RJ; Kilpatrick, BF; Nolan, JC; Proakis, AG; Walsh, DA | 1 |
DeNoble, KF; DeNoble, VJ; Reigel, AL; Schrack, LM | 1 |
Gorzalka, BB; Watson, NV | 1 |
Beczkowska, IW; Bodnar, RJ | 1 |
Beubler, E; Coupar, IM; Hardcastle, J; Hardcastle, PT | 1 |
Bird, ED; Crino, PB; Plager, MD; Vogt, BA | 1 |
Nakamura, H; Suzukawa, M | 1 |
Bennett, DA; Glaeser, BS; Hutchison, AJ; Liebman, JM; Lovell, RA; Sills, MA; Williams, M; Wood, PL | 1 |
Broekkamp, CL; Jenck, F; Van Delft, AM | 1 |
Dewar, KM; Lima, L; Reader, TA | 1 |
Glowinski, J; Godbout, R; Mantz, J; Tassin, JP; Thierry, AM | 1 |
Cohen, ML; Mann, JJ; McBride, PA; Nimchinsky, E | 1 |
Geyer, MA; Tapson, GS; Wing, LL | 1 |
Backus, LI; Grahame-Smith, DG; Sharp, T | 1 |
Demetrikopoulos, MK; Flaherty, CF; Grigson, PS; Krauss, KL; Rowan, GA; Weaver, MS | 1 |
Bertocci, B; Cesura, AM; Da Prada, M | 1 |
Jackson, DA; White, SR | 1 |
Cowen, PJ; Gartside, SE | 1 |
Campbell, AM; Glatfelter, A; Kunkel, RG; Ulevitch, RJ; Wiggins, RC | 1 |
Ahlman, H; Dahlström, A; Lidberg, P | 2 |
Delius, W; Dominiak, P; Gessler, I; Grobecker, H; Kees, F | 1 |
Vanhoutte, PM | 1 |
Gradin, K; Hedner, T; Persson, B; Pettersson, A | 4 |
Gradin, K; Hedner, T; Henning, M; Persson, B; Pettersson, A | 1 |
Markus, JK; Mylecharane, EJ; Phillips, CA; Shaw, J | 2 |
Coghlan, JP; Denton, DA; Mills, EH; Nelson, MA; Scoggins, BA; Spence, CD; Whitworth, JA | 1 |
Baudouin-Legros, M; Guicheney, P; Kamal, LA; Le Quan-Bui, KH; Meyer, P | 1 |
Ball, SG; Robertson, JI | 1 |
Ball, SG; Robertson, JI; Zabludowski, JR | 2 |
De Crée, J; De Ryck, M; Hoing, M; Symoens, J | 1 |
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; Staessen, J | 1 |
Boomsma, F; Man in't Veld, AJ; Schalekamp, MA; Wenting, GJ; Woittiez, AJ | 1 |
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; Rorive, G; Staessen, J | 1 |
Berglund, G; Hedner, T; Persson, B | 4 |
Brown, SA; Simpson, FO; Spears, GF; Waal-Manning, HJ | 1 |
Fasano, ML; Ferrara, LA; Mancini, M; Marotta, G; Rubba, P; Soro, S | 1 |
Hedner, T; Persson, B | 3 |
Ayres, B; Bune, AJ; Chalmers, JP; Graham, JR; West, MJ; Wing, LM | 2 |
Kincaid-Smith, P; Murphy, BF; Whitworth, JA | 1 |
Armanini, D; Boscaro, M; D'Agostino, D; Mantero, F; Opocher, G; Rocco, S | 2 |
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; Staessen, J; Vanhees, L | 1 |
Amery, A; Arnout, J; Deckmyn, H; Fiocchi, R; Lijnen, P; Van Russelt, M; Vermylen, J | 1 |
De Clerck, F; Xhonneux, B | 2 |
De Cree, J; Demoen, B; Leempoels, J; Roels, V; Verhaegen, H | 2 |
Brimichová, G; Dzúrik, R; Fetkovská, N; Tison, P | 2 |
Freitag, B; Pointel, JP; Schmitt, C; Stoltz, JF; Voisin, P; Zannad, F | 1 |
Bogar, L; Dormandy, JA; Matrai, A; Walker, RT | 1 |
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; M'Buyamba-Kabangu, JR; Staessen, J | 1 |
De Cree, J; Demoen, B; Leempoels, J; Verhaegen, H | 1 |
Van Nueten, JM | 2 |
Arnold, G; Breuer, J; Meschig, R | 1 |
Ahlman, H; Boström, S; Dahlström, A; Vällfors, B | 1 |
Arnold, G; Breuer, HW; Breuer, J; Meschig, R | 1 |
Marwood, JF; Stokes, GS | 1 |
Opie, LH; Saman, S; Thandroyen, F | 1 |
Kaumann, AJ | 2 |
Ahlman, H; Dahlström, A; Grönstad, K; Jaffe, BM; Nilsson, O; Oberg, K | 1 |
Hollenberg, NK | 1 |
De Cree, J; Geukens, H; Leempoels, J; Verhaegen, H | 2 |
Gush, R; Jayson, MI; Longstaff, J; Williams, EH | 1 |
Amery, A; Fagard, R; Laermans, M; Lijnen, P; Lommelen, L; M'Buyamba-Kabangu, JR; Piccart, Y; Staessen, J | 1 |
Hirokami, M; Minami, M; Saito, H; Sano, M; Tochihara, M; Togashi, H; Yoshioka, M | 1 |
Marsden, CA; Martin, KF | 1 |
Altar, CA; Boyar, WC; Marien, MR | 1 |
Casthely, PA; Ergin, MA; Goodman, K; Griepp, RB; Jablons, M | 1 |
Kienast, J; Verstraete, M | 1 |
Coker, SJ; Ellis, AM | 1 |
Ball, SG; Robertson, JI; Stott, DJ | 1 |
Ball, SG; Hosie, J; Robertson, JI; Stott, DJ | 1 |
Cohen, ML; Kurz, KD; Schenck, KW | 1 |
Ramage, AG | 2 |
Reneman, RS; van der Starre, PJ | 1 |
Brunello, N; Galimberti, R; Racagni, G; Riva, M; Rovescalli, AC | 1 |
Blauw, GJ; Chang, PC; van Brummelen, P; van Zwieten, PA; Vermeij, P | 1 |
Lund, N; Thorborg, P | 1 |
Bloomquist, WL; Cohen, ML; Fuller, RW; Snoddy, HD | 1 |
Arnt, J; Hyttel, J | 1 |
Koshikawa, N; Maruyama, Y; Stephenson, JD | 1 |
Chau, NP; Levenson, J; Pithois-Merli, I; Simon, AC | 1 |
Ahlman, H; Dahlström, A; Grönstad, K; Jaffe, BM; Oberg, K; Tisell, LE; Zinner, MJ | 1 |
Altar, CA; Marshall, JF; O'Neil, S; Walter, RJ | 1 |
Frimodt-Møller, C; Hørby-Petersen, J; Mathiesen, FR; Meyhoff, HH; Schmidt, PF | 1 |
Bodnar, RJ; Kiefel, JM; Paul, D | 1 |
Alling, C; Hansson, E; Simonsson, P | 1 |
Gommeren, W; Janssen, PF; Laduron, PM; Leysen, JE; Van Gompel, P; Wynants, J | 1 |
Berglund, G; Hedner, T; Persson, B; Pettersson, A | 1 |
Andersen, D; Bech, K; Ladegaard, L | 1 |
Buchman, O; Grigoriadis, DE; Niznik, HB; Pri-Bar, I; Seeman, P | 1 |
Arroyo, JL; Carrasco, MS; De Castro, J; Esteban, J; Sanchez, G | 1 |
Aono, J; Ishizuka, N; Nabata, H; Sakai, K | 1 |
Andree, TH; Koenig, JI; Meltzer, HY; Mikuni, M; Tong, CY | 1 |
Berent, A; Bounameaux, H; Hellemans, H; Holditch, T; Verhaeghe, R | 1 |
Assogna, G; Di Lorenzo, M; Feo, B; Pompa, D | 1 |
Ramsay, LE | 1 |
Ogren, SO | 1 |
Greiner, HE; Haase, A; Klockow, M; Schmitges, CJ; Seyfried, C | 1 |
Breckenridge, A | 1 |
Man in 't Veld, AJ; Schalekamp, MA; van den Meiracker, AH; Wenting, GJ; Woittiez, AJ | 1 |
Fisher, R; Gruebel, B; Koehle, W; Rosenthal, J | 1 |
Batink, HD; Boddeke, E; Doods, HN; Hugtenburg, JG; Korstanje, C; Sprenkels, R; Thoolen, MJ; Van Zwieten, PA | 1 |
Altar, CA; Neale, RF; Stone, GA; Wasley, AM | 1 |
Cameron, CM; Cameron, HA; Ramsay, LE | 1 |
Di Chiara, G; Longoni, R; Spina, L | 1 |
Hedner, T; Persson, B; Pettersson, A | 2 |
Hewson, G; Hill, RG; Hughes, J; Leighton, GE | 1 |
Knuppel, RA; Montenegro, R; O'Brien, WF; Shah, D | 1 |
Appel, JB; Cunningham, KA; Ginn, SR; Nielsen, EB | 1 |
Arnt, J | 1 |
Mylecharane, EJ; Phillips, CA; Shaw, J | 1 |
Laduron, PM; Leysen, JE; Van Dun, J; Wouters, W | 4 |
Heiligers, J; Mylecharane, EJ; Saxena, PR | 1 |
Janssens, WJ; Van Nueten, JM; Vanhoutte, PM | 1 |
Parag, KB; Seedat, YK | 1 |
Houvenaghel, A; Schrauwen, E | 1 |
Beck, SG; Clarke, WP; Goldfarb, J | 1 |
Auer, LM; Leber, K; Sayama, I | 1 |
Grekin, RJ; Gross, MD; Shenker, Y | 1 |
Apelian, A; Jageneau, AH; Khachadurian, AK; Schneider, SH; Tendler, M | 1 |
Barrett, JE; Brady, LS | 1 |
Lawang, A; Saxena, PR | 1 |
Skolnick, P; Weissman, BA; Youdim, MB | 1 |
Feniuk, W; Humphrey, PP; Perren, MJ; Watts, AD | 1 |
Gomar, C; Luis, M; Nalda, MA | 1 |
Demling, RH; Fox, R; Hechtman, H; Huval, W; Wong, C | 1 |
Jähnchen, E; Lühr, A; Radkow, N; Trenk, D | 1 |
De Roe, C; Laduron, PM; Luabeya, MK; Maloteaux, JM; Trouet, A | 1 |
Battaglia, G; Creese, I; Newton, PL; Norman, AB | 1 |
Clineschmidt, BV; Pettibone, DJ; Reiss, DR; Robinson, JL | 1 |
Gorzalka, BB; Mendelson, SD | 4 |
Ei-Fawal, HA; Eyre, P; Gordon, V; Ogunbiyi, PO | 1 |
Hoffmann, D; Wesemann, W | 2 |
Allegra, C; Assogna, G; Bonifacio, M; Mari, A; Tonelli, V | 1 |
Assogna, G; Attilia, ML; Cavalieri, G; Ceccanti, M; De Lorenzo, A; Romeo, M | 1 |
Colli, R; Di Giovanni, V | 1 |
Forler, C; Fozard, JR; Middlemiss, DN; Tricklebank, MD | 1 |
Engel, G; Hoyer, D; Kalkman, HO | 2 |
Man in't Veld, AJ; Ritsema van Eck, HJ; Schalekamp, MA; van den Meiracker, AH; Wenting, GJ; Woittiez, AJ; Zantvoort, FA | 1 |
Porter, JM; Taylor, LM | 1 |
Kellar, KJ; Stockmeier, CA | 2 |
Agid, Y; Baron, JC; Comar, D; Crouzel, C; Deniker, P; Samson, Y | 1 |
De Clerck, F; Janssen, PA; Tollenaere, JP; Xhonneux, B | 1 |
Biegon, A; Kargman, S; McEwen, BS; Snyder, L | 1 |
Ashton, JH; Benedict, CR; Buja, LM; Campbell, WB; Fitzgerald, C; Raheja, S; Taylor, A; Willerson, JT | 1 |
Cernohorský, D; Hamet, A; Král, B | 1 |
Engel, G; Göthert, M; Hillenbrand, K; Hoyer, D; Schlicker, E | 1 |
Hibert, M; Middlemiss, DN | 1 |
Barrett, JE; Mansbach, RS | 1 |
Pranzatelli, MR; Snodgrass, SR | 1 |
Dusting, GJ; Li, DM | 1 |
Connor, HE; Feniuk, W; Humphrey, PP; Perren, MJ | 1 |
Attilia, ML; Berbellini, A; Cavaleri, G; Ceccanti, M; De Lorenzo, A; Di Giovanni, MG; Pisculli, M; Santini, P | 1 |
Assogna, G; Ceccanti, M; De Lorenzo, A; Di Giovanni, MG; Lais, A; Pisculli, M; Romeo, M; Valgiusti, FC | 1 |
Ganey, PE; Hadley, KB; Roth, RA; Sprugel, KH | 1 |
Hald, A; Ording, H; Sjøntoft, E | 1 |
Eberlein, HJ; Schulte-Sasse, U | 1 |
Murrin, LC; Zeng, W | 1 |
Abrignani, MG; Alaimo, G; Cutietta, A; Novo, S; Raineri, A; Strano, A | 1 |
Harinck-de Weerd, JE; Reneman, RS; van der Starre, PJ | 1 |
Armstrong, ML; Heistad, DD; Marcus, ML; Mark, AL; Piegors, DJ | 1 |
Lüscher, TF; Vanhoutte, PM | 1 |
Zanchetti, A | 1 |
Janssens, WJ; Van Nueten, JM | 1 |
Gordin, A; Saraste, K; Sundberg, S; Turanlahti, M | 1 |
Gould, SE; Kane, JA; Sibbald, B; Tooley, M | 1 |
Kirch, W; Ohnhaus, EE | 1 |
Mauersberger, H | 1 |
Bernardiner, E; Lemus, J; Milei, J | 1 |
Assogna, G; Costantini, C; del Rosso, G; Libretti, A; Mara, G; Palermo, A; Pizza, N | 1 |
Dona, G; Ribeiro, A; Tammaro, AE | 1 |
de Jong, PE; de Zeeuw, D; Navis, G; van der Hem, GK | 1 |
Andersson, O; Berglund, G; Hedner, T; Persson, B; Petterson, A | 1 |
Cohen, RA | 1 |
Göthert, M; Kollecker, P; Schlicker, E | 1 |
Bergstrom, DA; Carlson, JH; Walters, JR | 1 |
Hösli, E; Hösli, L | 1 |
Conn, PJ; Hartig, PR; Hoffman, BJ; Sanders-Bush, E | 1 |
Arnout, J; De Clerck, F; Deckmyn, H; Vermylen, J; Xhonneux, B | 1 |
Boas, RA | 1 |
Berges, LC; Cruz, J; Feltkamp, H; Finkielman, S; Geyer, G; Milei, J; Moscovici, H; Silva, AN; Stumpe, KO | 1 |
Hoyer, D; Palacios, JM; Pazos, A; Probst, A | 1 |
Marwood, JF; Mennie, BA; Stokes, GS | 1 |
Bjertnaes, L; Helgesen, KG | 1 |
Seibold, JR; Terregino, CA | 1 |
Iida, H; Ikeda, K; Mikawa, M; Mizumura, Y; Sugimoto, T; Takata, M; Tomoda, F; Zhang, X | 1 |
Ahlman, H; Dahlström, A; Grönstad, KO; Jaffe, BM | 1 |
Bennett, A; Cashman, JN; Thompson, MA | 1 |
Carter, JA; Houghton, K | 1 |
Hoekman, TB; Howlett, SE; Triggle, CR | 1 |
Bottaro, D; Hechtman, HB; Peterson, S; Shepro, D | 2 |
Engisch, KL; Wenk, GL | 1 |
Ferrara, A; Jaffe, BM; Sherlock, DJ | 1 |
Skotnicki, SH; van de Wal, HJ; van Lier, HJ; Wijn, PF | 1 |
Arvidsson, S; Bergqvist, D; Haglund, U; Hedner, U; Lindblad, B | 1 |
Lagerkvist, BE; Linderholm, H | 1 |
Hall, H; Wedel, I | 1 |
Hulme, VA; Odendaal, HJ | 1 |
Jarvis, LG; Setchell, BP; Sowerbutts, SF | 1 |
Leff, P; Martin, GR | 1 |
Abrignani, MG; Adamo, L; Alaimo, G; Avellone, G; Cutietta, A; Giordano, U; Indovina, A; Novo, S; Pinto, A; Strano, A | 1 |
Kaumann, AJ; Lemoine, H | 1 |
Creba, JA; Doyle, VM; Hoyer, D; Rüegg, UT | 1 |
Banay-Schwartz, M; Lajtha, A; Manigault, I; Wajda, IJ | 1 |
Lin, MT; Tsai, ML | 1 |
Foray, J; Hagege, A; Housset, E; Priollet, P; Vayssairat, M | 1 |
Glennon, RA | 1 |
Hladovec, J | 2 |
Delbro, D; Nordström, O | 1 |
Griffiths, HB; Whitwam, JG | 2 |
Gudelsky, GA; Koenig, JI; Meltzer, HY | 1 |
Laruelle, M; Maloteaux, JM; Vanisberg, MA | 1 |
Altar, CA; Marien, MR | 1 |
Kobayashi, M; Koshikawa, N; Maruyama, Y; Mori, E; Nomura, H; Oka, K; Stephenson, JD | 1 |
Barbaccia, ML; Costa, E; Gandolfi, O | 2 |
Gordin, A; Mustajoki, P; Pelkonen, R | 1 |
Kendall, DA; Nahorski, SR | 1 |
Goto, A; Ishii, M; Matsuoka, H; Sugimoto, T | 1 |
Godfrey, PP; McClue, SJ; Minchin, MC; Schächter, M; Young, MM | 1 |
Bockaert, J; Kemp, DE; Sebben, M; Weiss, S | 1 |
Kawasaki, H; Takasaki, K | 1 |
Linthicum, DS; Simmons, RD | 1 |
Candeletti, S; Ferri, S; Romualdi, P; Spadaro, C; Spampinato, S | 1 |
Gommeren, W; Janssen, PA; Leysen, JE; Van Gompel, P; Woestenborghs, R | 1 |
Byrne, JH; Ocorr, KA | 1 |
Jandhyala, BS; Kivlighn, SD | 1 |
Laguzzi, R; Shvaloff, A | 1 |
Coghlan, JP; Denton, DA; Nelson, M; Scoggins, BA; Tresham, JJ; Whitworth, JA | 1 |
Furukawa, H; Ishikawa, K; Kameyama, T; Nabeshima, T; Yamaguchi, K | 1 |
Smits, J; Struyker Boudier, H; van Dorsten, F | 1 |
Geyer, MA; Tapson, GS | 1 |
Arneklo-Nobin, B; Owman, C | 1 |
Hole, DR; Hunter, AJ; Wilson, CA | 1 |
Houston, DS; Shepherd, JT; Vanhoutte, PM | 1 |
Bieger, D; Triggle, C | 1 |
Erne, P; Pletscher, A | 1 |
Jennewein, HM; Mierau, J; Saxena, PR; Verdouw, PD | 1 |
Affolter, H; Burkard, WP; Pletscher, A | 1 |
Appel, JB; Callahan, PM; Cunningham, KA | 1 |
Frenken, M; Kaumann, AJ | 3 |
Kayaba, K; Kimura, M; Kiyono, S; Koyama, S; Nishizawa, M | 1 |
Hayashi, T; Ichida, S; Kita, T; Murakami, T | 1 |
Grigoriadis, D; Seeman, P | 1 |
Olesen, SP | 1 |
Anwyl, R; Rowan, MJ | 1 |
Fasano, ML; Ferrara, LA; Iannuzzi, A; Rubba, P; Soro, S | 1 |
Karasawa, A; Kubo, K; Nakamizo, N; Shuto, K | 1 |
Aghajanian, GK; Lakoski, JM | 1 |
de Aguiar, JC; Graeff, FG; Schütz, MT | 1 |
Bevan, J; Heptinstall, S | 2 |
Bradley, PB; Humphrey, PP; Williams, RH | 1 |
Comar, D; Maziere, M; Turner, JH | 1 |
Klotz, U; Ratge, D; Reimann, IW; Wisser, H | 1 |
Koshikawa, N; Smokcum, RW; Stephenson, JD | 1 |
Buczko, W | 1 |
Beetens, J; De Clerck, F; Reneman, RS; Van Gorp, L | 1 |
Burns, EC; Dillon, MJ; Dunger, DB | 1 |
Heiligers, J; Mylecharane, EJ; Saxena, PR; Tio, R | 1 |
Kurowski, M | 2 |
Frost, JJ; Hartig, PR; Scheffel, U; Wagner, HN | 1 |
Hechtman, DH; Jageneau, A | 1 |
Glaser, T; Traber, J | 1 |
Clarke, KA; Parker, AJ; Stirk, GC | 1 |
Cameron, HA; Ramsay, LE | 1 |
Doğan, N; Ilhan, M; Kayaalp, SO; Tuncer, M | 1 |
Reneman, S; van de Water, A; Wouters, L; Xhonneux, R | 1 |
Cowen, KJ; McGourty, JC; Silas, JH | 1 |
Kilbinger, H; Pfeuffer-Friederich, I | 1 |
Brimichová, E; Dzúrik, R; Gerová, Z | 1 |
Kwan, S; Lam, WK; So, SY | 1 |
De Meirleir, K; Hollmann, W; L'Hermite, M; L'Hermite-Balériaux, M; Rost, R | 1 |
Burvenich, C; Peeters, G; Vandeputte-Van Messon, G | 1 |
Demenge, P; Feuerstein, C; Guerin, B; Mouchet, P; Silice, C | 1 |
Nishino, N; Tanaka, C | 1 |
Mana, MJ; Paul, D; Pfaus, JG; Pinel, JP | 1 |
de Chaffoy de Courcelles, D; Leysen, JE; Niemegeers, CJ; Van Gompel, P | 1 |
Altman, HJ; Normile, HJ | 1 |
Janssen, CG; Laduron, PM; Thijssen, JB; Van Dun, J; Wouters, W | 1 |
Neal, BS; Sparber, SB | 1 |
Marcelle, R | 1 |
Bounameaux, HM; Hellemans, H; Verhaeghe, R | 1 |
Brimichová, G; Dzúrik, R; Petkovská, N; Tison, P | 1 |
Cooper, SJ; Cross, AJ; Crow, TJ; Deakin, JF; Ferrier, IN; Johnson, JA; Joseph, MH; Lofthouse, R; Owen, F; Poulter, M | 1 |
Laduron, PM; Luabeya, MK; Maloteaux, JM | 1 |
Prescott, RW; Ratcliffe, WA; Taylor, PK | 1 |
Beubler, E; Bukhave, K; Rask-Madsen, J | 1 |
Amery, A; Groeseneken, D; Laermans, M; Lijnen, P; Lommelen, L; Piccart, Y | 1 |
Battaglia, G; Borgundvaag, B; Shannon, M; Titeler, M | 2 |
Van Nueten, JM; Vanhoutte, PM | 2 |
Edwards, CR; Shaikh, S; Williams, BC | 1 |
De Cree, J; Symoens, J; Verhaegen, H | 1 |
Bertholet, M; David, JL; Demoulin, JC; Kulbertus, HE; Soumagne, D | 1 |
Janssen, PA; Van Beek, J; Van Nueten, JM; Vanhoutte, PM; Verbeuren, TJ; Xhonneux, R | 1 |
Ilien, B; Laduron, PM; Schotte, A | 1 |
de Roose, J; Symoens, J | 1 |
Hedner, T; Henning, M; Persson, B | 1 |
Feniuk, W; Humphrey, PP; Watts, AD | 1 |
Facoory, BD; Laverty, R; Millar, JA | 1 |
Leysen, JE; Schuurkes, JA; Van Nueten, JM; Vanhoutte, PM | 1 |
Frölich, JC; Reimann, IW | 1 |
Iversen, LL; Reynolds, GP; Rossor, MN | 1 |
Amery, A; Fagard, R; Fiocchi, R; Lijnen, P; Staessen, J; Vermylen, J | 1 |
Helmeste, DM; Tang, SW | 2 |
Anger, C; Lawin, P; Puchstein, C; Thijs, J; Van Aken, H | 1 |
Timmermans, PB; van Zwieten, PA | 1 |
McGoon, MD; Vlietstra, RE | 1 |
Timmermans, PB; Van Brummelen, P; Van Zwieten, PA | 1 |
Barradas, MA; Dandona, P; Fonseca, V; Jeremy, JY; Mikhailidis, DP; Ramage, AG | 1 |
Arnold, R; Koop, H | 1 |
Humphrey, PP | 1 |
Adams, CB; Boullin, DJ; Kaye, AH; Schachter, M; Tagari, PC; Teddy, PJ | 1 |
Lagneaux, D; Lecomte, J | 2 |
Cheney, DL; Costa, E; Gandolfi, O; Hong, JS | 1 |
Bloom, SR; Corsellis, JA; Cross, AJ; Crow, TJ; Ferrier, IN; Johnson, JA | 1 |
David, JL; de Clerck, F; Janssen, PA | 1 |
de Chaffoy de Courcelles, D; Roevens, P; van Belle, H | 1 |
Barnett, DB; Cook, N; Jennings, PE; O'Malley, BP; Rosenthal, FD | 1 |
Buczko, W; De Gaetano, G; Gambino, MC | 1 |
Awouters, F; Janssen, PA; Kennis, L; Laduron, PM; Leysen, JE; Vandenberk, J | 1 |
Kalkman, HO; Timmermans, PB; Van Zwieten, PA | 1 |
Janssen, PA; Symoens, J; Van Nueten, JM; Vanhoutte, PM | 1 |
Opie, LH | 1 |
Battaglia, G; Shannon, M; Titeler, M | 3 |
Schalekamp, MA; Wenting, GJ | 1 |
McCall, RB; Schuette, MR | 1 |
Kendall-Taylor, P; Prescott, RW; Ratcliffe, WA; Watson, MJ; Weightman, DR | 1 |
Vincent, JL | 1 |
Eyre, P; Ogunbiyi, PO | 2 |
Köhler, C | 2 |
Bianconi, M; Degli Uberti, EC; Margutti, AR; Pansini, P; Rotola, CA; Trasforini, G | 1 |
Andrén, L; Dahlöf, B; Eggertsen, R; Hansson, L; Svensson, A | 1 |
Leysen, JE; Niemegeers, CJ; Van Gompel, P; Verwimp, M | 1 |
Arvidsson, S; Falk, A; Haglind, E; Haglund, U | 1 |
Ball, HA; Parratt, JR; Rodger, IW | 1 |
Amery, A; de Schaepdryver, A; Fagard, R; Fiocchi, R; Lijnen, P; Moerman, E; Staessen, J | 1 |
Jageneau, AH; Seibold, JR | 1 |
Socol, ML; Vaisrub, N; Weiner, CP | 1 |
Arvidsson, S; Bergqvist, D; Esquivel, C; Fält, K; Haglund, U; Lindblad, B; Lindström, C | 1 |
Hechtman, HB; Shepro, D; Valeri, CR | 1 |
Feniuk, W | 1 |
de Chaffoy de Courcelles, D; De Clerck, F; Leysen, JE; Niemegeers, CJ; Van Nueten, JM | 1 |
De Clerck, F; Reneman, RS; van Nueten, JM | 1 |
Anthony, M | 1 |
Bosin, TR; Mais, DE | 1 |
Roald, OK; Seem, E | 1 |
Cox, NH; Dufton, PA | 1 |
Ernst, E; Matrai, A | 1 |
McGoon, MD; Vanhoutte, PM | 1 |
Battaglia, G; Glennon, RA; Shannon, M; Titeler, M | 1 |
Glennon, RA; McKenney, JD; Young, R | 1 |
Conn, PJ; Sanders-Bush, E | 1 |
De Clerck, F; De Gryse, A; Loots, W; Nevelsteen, A | 1 |
Lauwers, F; Van Den Broeck, C; Verheyen, A; Vlaminckx, E; Wouters, L | 1 |
Kirby, GC; McQueen, DS | 1 |
Finch, CE; Marcusson, JO; Morgan, DG; Winblad, B | 1 |
Apprill, P; Ashton, J; Buja, LM; Bush, LR; Campbell, WB; Kern, K; Schmitz, J; Tilton, GD; Willerson, JT | 1 |
Hedner, T; Henning, M; Persson, B; Pettersson, A | 1 |
McLennan, PL; Taylor, DA | 1 |
Offord, SJ; Warwick, RO | 1 |
Fuller, RW; Snoddy, HD | 1 |
Barvais, L; Capouet, V; d'Hollander, A | 1 |
Hoyer, D; Palacios, JM; Pazos, A | 1 |
Chuang, DM; Costa, E; Nakaki, T; Roth, BL | 1 |
Freedman, M; Hamel, L; Luttinger, D; Perrone, M; Ward, SJ | 1 |
Engel, G; Hoyer, D; Kalkman, HO; Wick, MB | 1 |
Su, C; Uruno, T | 1 |
Hechtman, HB; Huval, WV; Lelcuk, S; Shepro, D | 1 |
Duncker, DJ; Heiligers, J; Jennewein, HM; Saxena, PR; Verdouw, PD | 1 |
Kolling, JB; Reneman, RS; Scheijgrond, HW; van der Starre, PJ | 1 |
Taylor, DA; Yap, CY | 1 |
De Wet, JI; Diedericks, BJ; Roelofse, JA | 1 |
Frey, HH; Reiche, R | 1 |
Dentan, M; Fischler, M; Freitag, B; Vourc'h, G; Westerman, MN | 1 |
Klotz, U; Okonkwo, PO; Reimann, IW | 1 |
Glennon, RA; Rosecrans, JA; Young, R | 1 |
Ball, SG; Fraser, R; Inglis, GC; Isles, CG; Murray, GD; Robertson, JI; Zabludowski, JR; Zoccali, C | 2 |
Laduron, PM; Maloteaux, JM; Schotte, A | 2 |
Gudelsky, GA; Meltzer, HY; Simonovic, M | 1 |
Patel, S; Slater, P | 1 |
Holliman, CJ; Larsen, KR; Meuleman, TR; Pace, NL; Port, JD; Stanley, TH; Warden, GD | 1 |
Lindelauf, F | 1 |
Biegon, A; Mann, JJ; McBride, PA; McEwen, B | 1 |
Janssen, PA; Van Beek, J; Van Nueten, JM | 1 |
Affolter, H; Pletscher, A | 1 |
Cohen, RA; Shepherd, JT; Vanhoutte, PM | 1 |
Hayashi, T; Ichida, S; Terao, M | 1 |
Engel, G; Müller-Schweinitzer, E | 1 |
Angus, JA; Wright, CE | 1 |
Lund-Johansen, P; Omvik, P | 1 |
Bagge, U; Ivarsson, L; Skolnik, G | 1 |
Amery, A; Cattaert, A; Fagard, R; Lijnen, P; Moerman, E; Staessen, J; Vanhees, L | 1 |
Frazer, A; Lucki, I; Nobler, MS | 1 |
Iwanov, V; Medcalf, RL; Moulds, RF | 1 |
Carpeggiani, C; De Caterina, R; L'Abbate, A | 1 |
Berre, J; Degaute, JP; Domb, M; Simon, P; Vandesteene, A; Vincent, JL | 1 |
De Clerck, F; Janssen, PA; Leysen, J; Xhonneux, B | 1 |
Creese, I; Hamblin, MW; Leff, SE | 1 |
Coltart, DJ; Juul, SM; Walker, JM; Wilmshurst, PT | 1 |
Arnold, L; Iversen, LL; Mountjoy, CQ; Reynolds, GP; Rossor, MN; Roth, M | 1 |
Bugiardini, R; Chierchia, S; Freedman, SB; Maseri, A; Rodriguez-Plaza, L; Smith, G | 1 |
De Ridder, W; Van Nueten, JM; Vanhoutte, PM | 1 |
Gelfan, R; Socol, ML; Weiner, CP | 1 |
Barbieri, C; Bevilacqua, M; Bigatti, G; Diena, A; Guffanti, A; Norbiato, G; Rauhe, WG; Sala, M; Scorza, D | 1 |
Heym, J; Jacobs, BL; Rasmussen, K | 1 |
Hölzenspies, AJ; Kalenda, Z | 1 |
Boomsma, F; Man in 't Veld, AJ; Schalekamp, MA; Wenting, GJ; Woittiez, AJ | 1 |
Krohg, K; Roald, OK; Stranden, E | 1 |
De Clerck, F; Van Nueten, JM | 1 |
Makabali, GL; Mandal, AK; Morris, JA | 1 |
Dunham, BM; Hechtman, HB; Huval, WV; Jones, AG; Mathieson, MA; Shepro, D; Stemp, LI | 1 |
Bagge, U; Ericson, LE; Skolnik, G | 1 |
Klotz, U; Okonkwo, PO; Reimann, IW; Woestenborghs, R | 1 |
Bury, RW; Kacprowicz, AT; Moulds, RF; Shaw, PG | 1 |
Cantalamessa, F; de Caro, G; Massi, M; Micossi, LG | 1 |
Barbaccia, ML; Chuang, DM; Costa, E; Gandolfi, O | 1 |
de Smet, HL; Gerritsen, HA; Kotora, OV; Perquin, JW; Troost, FA | 1 |
De Clerck, F; Gommeren, W; Leysen, JE | 2 |
Hill, DC; Meuleman, TR; Mohammad, SF; Pace, NL; Port, JD; Stanley, TH | 1 |
Garrett, NJ; Jenner, P; Marsden, CD; Reynolds, GP; Rupniak, N | 1 |
Davies, CL | 1 |
Arvidsson, S; Bergqvist, D; Esquivel, CO; Haglund, U; Lindblad, B | 1 |
Hong, E; Mena, MA; Rión, R | 1 |
Brenken, U; Homan van der Heide, JN; Karliczek, GF; Schokkenbroek, R; van den Broeke, JJ | 1 |
De Cock, W; De Cree, J; Geukens, H; Leempoels, J; Verhaegen, H | 2 |
De Ridder, A; Janssen, PA; Van Nueten, JM; Vanhoutte, PM | 1 |
Alexander, JP; Miranda, DR; Stoutenbeek, CP; Zandstra, D | 1 |
Laduron, PM; Leysen, JE; Niemegeers, CJ; Van Nueten, JM | 1 |
Geerts, R; Gommeren, W; Leysen, JE; Van Gompel, P; Verwimp, M | 1 |
Janssen, PF; Laduron, PM; Leysen, JE | 1 |
De Clerck, F; Dom, J; Jageneau, A | 1 |
de Gaetano, G; Lampugnani, MG | 1 |
Simon, V; Somani, P | 1 |
Bueno, L; Fioramonti, J; Ooms, L; Ruckebusch, Y | 1 |
Janssen, PA; Van Nueten, JM; Vanhoutte, PM; Xhonneux, R | 1 |
Hörig, C; Jageneau, AH; Loots, W; Symoens, J | 1 |
Barrett, RJ; Sanders-Bush, E; Smith, RL | 1 |
Kido, H; Mori, H; Sakamoto, H; Shiba, K; Sumiyoshi, T; Suzuki, K; Urasaki, K; Yamaguchi, N; Yokogawa, K | 1 |
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI | 1 |
Arruda, K; Glennon, RA; Ismaiel, AM; Teitler, M | 1 |
Dykstra, LA; Lin, YP; Powell, KR | 1 |
Hansen, MB; Jaffe, BM | 1 |
Holtzman, SG; Steinfels, GF | 1 |
Cadavid, I; Castro, E; Ferreiro, TG; Fontenla, JA; Loza, MI; Lozoya, E; Manaut, F; Rodriguez, J; Sanz, F; Verde, I | 1 |
Colpaert, FC; John, GW; Le Grand, B; Patoiseau, JF; Rieu, JP; Talmant, JM | 1 |
Frölich, D; Göthert, M; Likungu, J; Molderings, GJ | 1 |
Carr, AA; Johnson, MP; Siegel, BW | 1 |
Berardi, F; Giudice, G; Govoni, S; Lucchi, L; Perrone, R; Tortorella, V | 1 |
Abi-Dargham, A; al-Tikriti, M; Baldwin, RM; Charney, D; Hoffer, P; Innis, RB; Laruelle, M; Leysen, JE; Mertens, J; Terriere, D; Zea-Ponce, Y | 1 |
Assié, MB; Kleven, MS; Koek, W | 1 |
López-Giménez, JF; Mengod, G; Palacios, JM; Vilaró, MT | 4 |
Buczko, W; Chabielska, E; Małyszko, J; Myśliwiec, M; Pawlak, D; Pawlak, K; Takada, A | 1 |
Adamkiewicz, M; Buczko, W; Malyszko, J; Mysliwiec, M; Pawlak, D; Takada, A | 1 |
Kulkarni, SK; Ninan, I | 1 |
Aloyo, VJ; Harvey, JA; Hoffman, ME; Salt, GL | 1 |
Harvey, JA; Hood, H; Romano, AG; Welsh, SE | 1 |
Kaibara, M; Mameya, S; Takada, K; Takemura, K; Taniyama, K | 1 |
Caldarola-Pastuszka, M; DeLashaw, M; Uphouse, L; Wolf, A | 1 |
Chen, K; De Maeyer, E; Kung, MP; Meehan, WP; Ridd, MJ; Seif, I; Shih, JC | 1 |
Asai, F; Fujimoto, K; Goto, R; Hayakawa, M; Ito, R; Ogawa, T; Sugidachi, A; Tanaka, N | 1 |
Adlersberg, M; Arango, V; Hsiung, S; Kassir, SA; Liu, K; Mann, JJ; Ruggiero, DA; Tamir, H; Underwood, MD | 1 |
Naylor, RJ; Tuladhar, BR; Womack, MD | 1 |
Cunningham, KA; McMahon, LR | 1 |
Hattori, K; Nagatom, T; Nakamura, T; Nakazawa, M; Rashid, M; Watanabe, M | 1 |
De los Angeles, J; Dukat, M; Glennon, RA; Herndon, J; Ismaiel, AM; Khorana, N; Metwally, K; Teitler, M | 1 |
Baker, GB; Fletcher, PJ; Korth, KM; Robinson, SR | 1 |
Audenaert, K; De Vos, F; Dierckx, R; Dumont, F; Jacobs, F; Mertens, J; Peremans, K; Slegers, G; Van Bree, H; Van De Wiele, C; Vandecapelle, M; Verschooten, F | 1 |
Fantegrossi, WE; Godlewski, T; Karabenick, RL; Rice, KC; Stephens, JM; Ullrich, T; Woods, JH | 1 |
Cunningham, KA; Filip, M; McCreary, AC | 1 |
Ge, L; Naylor, RJ; Tuladhar, BR | 1 |
Zhang, ZW | 1 |
Cao, C; Cho, KW; Han, JH; Kim, SH; Kim, SZ | 1 |
Grasby, P; Hirani, E; Hume, S; Sharp, T; Sprakes, M | 1 |
Jähnichen, S; Pertz, HH; Radtke, OA | 1 |
Gorzalka, BB; Hill, MN; Sun, JC | 1 |
Hayslett, RL; Tizabi, Y | 1 |
Elfving, B; Gillings, N; Knudsen, GM; Kristiansen, H; Pinborg, LH; Plenge, P | 1 |
Asgari, K; Bak, VK; Body, S; Bradshaw, CM; Fone, KC; Glennon, JC; Rickard, JF; Szabadi, E; Zhang, ZQ | 1 |
Bindslev, N; Engelmann, BE; Hansen, MB; Larsen, R; Poulsen, SS | 1 |
Peña, F; Ramirez, JM; Tryba, AK | 1 |
Kajos, M; Kankaanpää, A; Meririnne, E; Seppälä, T | 1 |
Abanades, S; Bullich, S; Catafau, AM; Cunningham, VJ; Danus, M; Eersels, JL; Farre, M; Llop, J; Nucci, G; Pavia, J | 1 |
Bernard, JF; Comet, MA; Hamon, M; Laguzzi, R; Sévoz-Couche, C | 1 |
Komada, T; Yano, S | 1 |
Fletcher, PJ; Higgins, GA; Sinyard, J; Tampakeras, M | 1 |
Debus, F; Herth, MM; Knudsen, GM; Lüddens, H; Palner, M; Piel, M; Rösch, F | 1 |
Harmar, AJ; Jennings, KA; Sharp, T; Sheward, WJ | 1 |
Abe, M; Egashira, N; Fujiwara, M; Iwasaki, K; Matsushita, M; Mishima, K; Nishimura, R; Oishi, R; Okuno, R | 1 |
Blanckaert, P; Burvenich, I; De Bruyne, S; De Vos, F; Moerman, L; Staelens, S; Wyffels, L | 1 |
France, CP; Li, JX; Rice, KC | 1 |
Bianchi, P; Calise, D; Escourrou, G; Galinier, M; Guilbeau-Frugier, C; Lairez, O; Mialet-Perez, J; Ordener, C; Parini, A; Pizzinat, N; Roncalli, J; Seif, I; Spreux-Varoquaux, O | 1 |
Anju, TR; George, AK; Paulose, CS | 1 |
Lefever, TW; Rawls, SM; Walker, EA; Ward, SJ; Whiteside, GT | 1 |
France, CP; Javors, MA; Koek, W; Li, JX; Rice, KC; Unzeitig, A | 1 |
Doi, A; Ramirez, JM | 1 |
Herth, MM; Knudsen, GM; Kramer, V; Palner, M; Rösch, F; Santini, MA | 1 |
Estrada-González, V; Márquez-Diosdado, MI; Montes-Rodríguez, CJ; Prospéro-García, O; Soria-Gómez, E | 1 |
Cohen, MS; Fantegrossi, WE; Henson, CM; Rice, KC; Simoneau, J; Woods, JH; Zimmerman, SM | 1 |
Creed-Carson, M; Nobrega, JN; Oraha, A | 1 |
Arai, Y; Kikuchi, T; Mitazaki, S; Nakagawasai, O; Nakaya, K; Niijima-Yaoita, F; Onogi, H; Sato, A; Tadano, T; Tan-No, K; Watanabe, K | 1 |
Elizalde, DI; Gallitano, AL; González-Maeso, J; Ingram, WM; Janowski, SA; Kamel, CM; Kozlenkov, A; Levine, S; Lish, JR; Resnik, J; Shoker, J; Williams, AA | 1 |
Dyssegaard, A; Ettrup, A; Gillings, N; Hansen, HD; Herth, MM; Knudsen, GM; Ratner, C | 1 |
Bailey, JM; Fantegrossi, WE; Gray, BW; Hansen, M; Kristensen, JL; Smith, DA | 1 |
Gencer, A; Gunduz, O; Ulugol, A | 1 |
Anastasio, NC; Cunningham, KA; Fink, LH; Fox, RG; Moeller, FG; Rice, KC | 1 |
24 review(s) available for ketanserin and piperidines
Article | Year |
---|---|
Can peripheral serotonergic blockade explain the hypotensive effect of ketanserin?
Topics: Animals; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Ketanserin; Methoxamine; Phenylephrine; Piperidines; Receptors, Adrenergic, alpha; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation | 1985 |
Ketanserin: a new hypotensive drug?
Topics: Animals; Antihypertensive Agents; Costs and Cost Analysis; Dose-Response Relationship, Drug; Humans; Ketanserin; Kinetics; Patient Compliance; Piperidines; Species Specificity | 1985 |
Serotonin and the heart: effects of ketanserin on myocardial function, heart rate, and arrhythmias.
Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Coronary Circulation; Coronary Disease; Heart; Heart Rate; Humans; In Vitro Techniques; Ketanserin; Myocardial Contraction; Piperidines; Serotonin; Serotonin Antagonists; Sinoatrial Node | 1985 |
Pharmacology of the interaction between platelets and vessel wall.
Topics: Animals; Aspirin; Blood Platelets; Blood Vessels; Dextrans; Diltiazem; Dipyridamole; Epoprostenol; Humans; Imidazoles; Ketanserin; Piperidines; Pyrazoles; Pyrazolones; Sulfinpyrazone; Sulfonamides; Thiophenes; Ticlopidine | 1986 |
Antihypertensive mode of action of ketanserin.
Topics: Adrenergic alpha-Antagonists; Aldosterone; Animals; Antihypertensive Agents; Blood Pressure; Carcinoid Heart Disease; Humans; Ketanserin; Piperidines; Prazosin; Ritanserin | 1987 |
Serotonin and vascular reactivity.
Topics: Animals; Blood Platelets; Calcium; Cold Temperature; Electric Stimulation; Hypoxia; Ketanserin; Lidoflazine; Methiothepin; Methysergide; Microcirculation; Models, Biological; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation | 1985 |
[New findings and experiences in the field of malignant hyperthermia].
Topics: Anesthesia; Animals; Calcium Channel Blockers; Catatonia; Dantrolene; Diagnosis, Differential; Humans; Ketanserin; Malignant Hyperthermia; Neuroleptic Malignant Syndrome; Piperidines; Serotonin Antagonists; Swine | 1986 |
Neurophysiological evidence that D-1 dopamine receptor blockade attenuates postsynaptic but not autoreceptor-mediated effects of dopamine agonists.
Topics: Animals; Apomorphine; Basal Ganglia; Benzazepines; Dextroamphetamine; Dopamine Antagonists; Electrophysiology; Ergolines; Globus Pallidus; Haloperidol; Ketanserin; Neurons; Pergolide; Piperidines; Quinpirole; Rats; Receptors, Dopamine; Substantia Nigra | 1986 |
Effects of electroconvulsive shock and serotonin axon lesions on beta-adrenergic and serotonin-2 receptors in rat brain.
Topics: Anesthetics; Animals; Axons; Brain; Cerebral Cortex; Cyclic AMP; Dihydroalprenolol; Electroconvulsive Therapy; Frontal Lobe; Hippocampus; Ketanserin; Norepinephrine; Piperidines; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Muscarinic; Receptors, Serotonin; Serotonin; Spiperone; Stress, Physiological; Time Factors; Tritium | 1986 |
[Role of serotonin in the regulation of the circulatory system].
Topics: Animals; Humans; Hypertension; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Resistance | 1985 |
Cardiovascular pharmacology of ketanserin.
Topics: Animals; Blood Platelets; Blood Pressure; Drug Interactions; Histamine; Ketanserin; Piperidines; Platelet Aggregation; Receptors, Adrenergic, alpha; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vasoconstriction | 1984 |
Cardiovascular alpha 2-receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Affinity Labels; Animals; Blood Pressure; Brain; Calcium Channel Blockers; Cardiovascular Physiological Phenomena; Guanosine Triphosphate; Heart Rate; Humans; Ketanserin; Kidney; Muscle, Smooth, Vascular; Piperazines; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Synaptic Membranes; Tritium; Vasoconstriction | 1983 |
Vasodilator therapy for primary pulmonary hypertension.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Blood Pressure; Calcium Channel Blockers; Captopril; Epoprostenol; Hemodynamics; Humans; Hypertension, Pulmonary; Ketanserin; Piperidines; Serotonin Antagonists; Vascular Resistance; Vasodilator Agents | 1984 |
Role of alpha adrenoceptors in hypertension and in antihypertensive drug treatment.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Calcium Channel Blockers; Clonidine; Guanfacine; Guanidines; Humans; Hypertension; Ketanserin; Methyldopa; Muscle, Smooth, Vascular; Phenylacetates; Piperazines; Piperidines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Vascular Resistance | 1984 |
Peripheral 5-hydroxytryptamine receptors and their classification.
Topics: Animals; Dogs; Guinea Pigs; In Vitro Techniques; Ketanserin; Methysergide; Muscle Relaxation; Muscle, Smooth; Neurotransmitter Agents; Piperidines; Rabbits; Rats; Receptors, Serotonin | 1984 |
Antihypertensive properties of ketanserin (R 41 468).
Topics: Animals; Antihypertensive Agents; Blood Pressure; Dose-Response Relationship, Drug; Humans; Ketanserin; Muscle, Smooth, Vascular; Norepinephrine; Piperidines; Platelet Aggregation; Receptors, Adrenergic, alpha; Serotonin Antagonists | 1983 |
5-hydroxytryptamine and precapillary vessels.
Topics: Angiotensin II; Animals; Dinoprost; Drug Interactions; Histamine; Ketanserin; Methysergide; Norepinephrine; Piperidines; Prostaglandins F; Receptors, Adrenergic, alpha; Serotonin; Vasoconstriction | 1983 |
Place of vasoactive agents in the treatment of acute circulatory failure.
Topics: Cardiac Output; Depression, Chemical; Dobutamine; Dopamine; Fluid Therapy; Humans; Ketanserin; Nitroglycerin; Nitroprusside; Phentolamine; Piperidines; Shock; Stimulation, Chemical; Sympathomimetics; Vasodilator Agents | 1984 |
Role of humoral mediators in adult respiratory distress syndrome.
Topics: Animals; Arachidonic Acids; Chemotaxis, Leukocyte; Chromones; Dogs; Guinea Pigs; Humans; Hypertension, Pulmonary; Inflammation; Ketanserin; Leukocyte Count; Leukocytes; Lung; Piperidines; Platelet Activating Factor; Pulmonary Embolism; Respiratory Distress Syndrome; Serotonin; Serotonin Antagonists; SRS-A; Thromboxane A2 | 1984 |
An analysis of 5-hydroxytryptamine receptors mediating contraction of isolated smooth muscle.
Topics: Animals; Binding, Competitive; Cats; Cyproheptadine; Dogs; In Vitro Techniques; Ketanserin; Methoxamine; Methysergide; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Piperidines; Rabbits; Rats; Receptors, Serotonin | 1984 |
Serotonin-S2 receptor binding sites and functional correlates.
Topics: Animals; Binding Sites; Blood Platelets; Cats; Cerebral Cortex; Humans; In Vitro Techniques; Ketanserin; Kinetics; Models, Biological; Muscle, Smooth, Vascular; Piperidines; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin | 1984 |
Platelet-vessel wall interactions: implication of 5-hydroxytryptamine. A review.
Topics: Animals; Blood Platelets; Blood Vessels; Capillary Permeability; Endothelium; Humans; In Vitro Techniques; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Receptors, Serotonin; Serotonin; Vasoconstriction | 1984 |
Serotonin antagonists.
Topics: Cyproheptadine; Depression; Ergotamine; Humans; Hypertension; Ketanserin; Lisuride; Methysergide; Mianserin; Migraine Disorders; Piperidines; Pizotyline; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Diseases | 1984 |
Ketanserin and spiperone as templates for novel serotonin 5-HT(2A) antagonists.
Topics: Animals; Drug Design; Isoquinolines; Ketanserin; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Structure-Activity Relationship | 2002 |
78 trial(s) available for ketanserin and piperidines
Article | Year |
---|---|
Ketanserin and alpha 1-adrenergic antagonism in humans.
Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Double-Blind Method; Heart Rate; Humans; Ketanserin; Male; Middle Aged; Phenylephrine; Piperidines; Serotonin Antagonists; Valsalva Maneuver | 1985 |
Hemodynamic response to chronic ketanserin treatment in essential hypertension.
Topics: Adult; Cardiac Output; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Hemodynamics; Humans; Hypertension; Ketanserin; Male; Methoxamine; Phenylephrine; Physical Exertion; Piperidines; Random Allocation; Serotonin Antagonists; Stroke Volume; Vascular Resistance | 1985 |
Double-blind comparison of ketanserin with propranolol in hypertensive patients: interim report.
Topics: Adult; Aged; Antihypertensive Agents; Body Weight; Clinical Trials as Topic; Double-Blind Method; Female; Follow-Up Studies; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Patient Compliance; Piperidines; Propranolol; Random Allocation | 1985 |
Clinical studies with ketanserin in hypertension.
Topics: Aged; Blood Pressure; Clinical Trials as Topic; Diuretics; Erythrocyte Deformability; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Physical Exertion; Piperidines; Pulse; Random Allocation; Serotonin Antagonists; Time Factors | 1985 |
Study with the competitive 5-HT2-serotonergic antagonist ketanserin.
Topics: Adult; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Heart Rate; Humans; Hypertension; Ketanserin; Leg; Metoprolol; Physical Exertion; Piperidines; Random Allocation; Regional Blood Flow; Serotonin Antagonists | 1985 |
Antihypertensive properties of ketanserin in combination with beta-adrenergic blocking agents.
Topics: Adrenergic beta-Antagonists; Antihypertensive Agents; Blood Pressure; Drug Therapy, Combination; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Serotonin Antagonists; Time Factors | 1985 |
Effect of ketanserin on blood pressure and biochemical parameters in patients with essential hypertension.
Topics: Adrenergic beta-Antagonists; Adult; Aged; Antihypertensive Agents; Blood Pressure; Body Weight; Clinical Trials as Topic; Diuretics; Double-Blind Method; Drug Therapy, Combination; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation | 1985 |
Effect of ketanserin in primary aldosteronism.
Topics: Aldosterone; Blood Pressure; Humans; Hydrocortisone; Hyperaldosteronism; Hypertension; Ketanserin; Piperidines; Potassium; Renin; Serotonin Antagonists; Time Factors | 1985 |
Effect of ketanserin on the hyperreactivity of platelets to 5-hydroxytryptamine in patients with cardiovascular diseases.
Topics: Adult; Aged; beta-Thromboglobulin; Blood Platelets; Cardiovascular Diseases; Double-Blind Method; Humans; Ketanserin; Middle Aged; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists | 1985 |
Serotonin and the flow properties of blood.
Topics: Blood Flow Velocity; Blood Viscosity; Hemoglobins; Humans; Ischemia; Ketanserin; Leg; Piperidines; Rheology; Serotonin; Serotonin Antagonists | 1985 |
Ketanserin and red blood cell sodium content in hypertension.
Topics: Adult; Aged; Erythrocyte Deformability; Erythrocytes; Humans; Hypertension; Ketanserin; Middle Aged; Myocardial Infarction; Ouabain; Piperidines; Serotonin; Serotonin Antagonists; Sodium | 1985 |
Comparison of blood pressure ratio by Doppler velocimetry and by plethysmography during treatment with ketanserin, a 5-HT2 receptor antagonist: a measure of improved collateral and microcirculatory flow.
Topics: Aged; Arm; Blood Pressure; Collateral Circulation; Female; Humans; Ketanserin; Male; Microcirculation; Middle Aged; Piperidines; Plethysmography; Regional Blood Flow; Rheology; Serotonin Antagonists; Thigh | 1985 |
Effects of ketanserin on peripheral blood flow, haemorheology, and platelet function in patients with Raynaud's phenomenon.
Topics: Adult; Aged; Blood Platelets; Blood Viscosity; Female; Fingers; Humans; Ketanserin; Male; Middle Aged; Piperidines; Raynaud Disease; Regional Blood Flow; Rheology; Serotonin Antagonists | 1985 |
Does acute serotonergic type-2 antagonism reduce blood pressure? Comparative effects of single doses of ritanserin and ketanserin in essential hypertension.
Topics: Adult; Affect; Aged; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin; Ritanserin | 1987 |
Experience with ketanserin and ritanserin in hypertensive patients.
Topics: Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Ritanserin | 1988 |
The alpha-adrenergic receptor blocking effect of ketanserin and the interaction between alpha-adrenergic and S2-serotonergic receptor blockade.
Topics: Adrenergic alpha-Antagonists; Blood Pressure; Droperidol; Female; Humans; Ketanserin; Male; Middle Aged; Phentolamine; Phenylephrine; Piperidines; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin | 1988 |
Comparative haemodynamic effects of ketanserin and ritanserin in the proximal and distal upper limb circulations of hypertensive patients.
Topics: Arm; Blood Pressure; Brachial Artery; Double-Blind Method; Hand; Humans; Hypertension; Ketanserin; Middle Aged; Piperidines; Regional Blood Flow; Rheology; Ritanserin; Serotonin Antagonists; Vascular Resistance | 1989 |
Placebo-controlled, double-blind, two-centre trial of ketanserin in intermittent claudication.
Topics: Adult; Aged; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Extremities; Female; Humans; Intermittent Claudication; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Regional Blood Flow; Serotonin Antagonists | 1985 |
Ketanserin--a new antihypertensive agent.
Topics: Adrenergic beta-Antagonists; Clinical Trials as Topic; Diuretics; Dose-Response Relationship, Drug; Humans; Hypertension; Ketanserin; Piperidines; Placebos | 1986 |
Ketanserin: haemodynamic effects and mechanism of action.
Topics: Adrenergic beta-Antagonists; Clinical Trials as Topic; Double-Blind Method; Heart Rate; Humans; Hypertension; Ketanserin; Piperidines; Placebos; Pressoreceptors; Random Allocation; Receptors, Serotonin; Reflex | 1986 |
Moderate essential hypertension control: a double-blind crossover study between a serotonin antagonist and a post-synaptic alpha-blocker.
Topics: Adrenergic beta-Antagonists; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Prazosin; Serotonin Antagonists | 1986 |
Comparison of single doses of ketanserin and placebo in chronic stable angina.
Topics: Adrenergic beta-Antagonists; Adult; Angina Pectoris; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Drug Therapy, Combination; Electrocardiography; Exercise Test; Female; Heart Rate; Humans; Ketanserin; Male; Middle Aged; Piperidines | 1986 |
Chronic 5-HT2-receptor blockade by ritanserin does not reduce blood pressure in patients with essential hypertension.
Topics: Aged; Clinical Trials as Topic; Double-Blind Method; Female; Histamine H2 Antagonists; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Ritanserin; Time Factors | 1987 |
The effect of serotonergic blockade in postpartum preeclamptic patients.
Topics: Adult; Blood Pressure; Double-Blind Method; Female; Humans; Ketanserin; Piperidines; Pre-Eclampsia; Pregnancy; Puerperal Disorders; Random Allocation; Serotonin Antagonists; Time Factors | 1985 |
A comparative study of ketanserin and metoprolol in essential hypertension.
Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Metoprolol; Middle Aged; Piperidines; Random Allocation; Time Factors | 1985 |
The effect of ketanserin, a 5-HT2-receptor antagonist, on 5-hydroxytryptamine-induced irreversible platelet aggregation in patients with cardiovascular diseases.
Topics: Aged; Arterial Occlusive Diseases; beta-Thromboglobulin; Cardiovascular Diseases; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Myocardial Infarction; Piperidines; Placebos; Platelet Aggregation; Serotonin | 1985 |
The effect of ketanserin on post-anaesthetic vasoconstriction and shivering.
Topics: Adult; Anesthesia; Blood Gas Analysis; Blood Pressure; Body Temperature; Female; Heart Rate; Humans; Ketanserin; Middle Aged; Piperidines; Pulse; Serotonin Antagonists; Shivering; Vasoconstriction | 1985 |
Raynaud's disease: a new therapeutic approach with a 5-HT2 receptors blocker.
Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Raynaud Disease; Serotonin Antagonists | 1985 |
Ketanserin hypertension and chronic alcoholism DB study in 40 patients.
Topics: Alcoholism; Blood Pressure; Chronic Disease; Female; Humans; Hypertension; Ketanserin; Male; Piperidines | 1985 |
Chronic effect of ketanserin in mild to moderate essential hypertension.
Topics: Adult; Aged; Blood Pressure; Circadian Rhythm; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Posture; Random Allocation | 1986 |
Effects of ketanserin on ambulatory blood pressure monitoring in patients with essential hypertension.
Topics: Adult; Ambulatory Care; Blood Pressure Determination; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Placebos; Propranolol | 1986 |
Comparison of ketanserin and pindolol in hypertension.
Topics: Adult; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Pindolol; Piperidines; Random Allocation | 1986 |
A comparative study of ketanserin and metoprolol in essential hypertension.
Topics: Adult; Aged; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Metoprolol; Middle Aged; Piperidines; Placebos | 1986 |
Double-blind comparison of ketanserin with atenolol: antihypertensive activity and effect on platelet function.
Topics: Adult; Aged; Atenolol; Blood Platelets; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Ketanserin; Male; Middle Aged; Piperidines; Placebos; Platelet Aggregation | 1986 |
Long-term safety and efficacy of ketanserin in essential hypertension: ketanserin versus or in combination with metoprolol.
Topics: Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypertension; Ketanserin; Male; Metoprolol; Middle Aged; Piperidines; Random Allocation | 1986 |
Ketanserin versus metoprolol in the treatment of essential hypertension.
Topics: Adult; Aged; Female; Follow-Up Studies; Heart Rate; Humans; Hypertension; Ketanserin; Male; Metoprolol; Middle Aged; Piperidines; Placebos | 1986 |
Clinical experience with ketanserin in the treatment of hypertension.
Topics: Double-Blind Method; Heart Rate; Humans; Hypertension; Ketanserin; Metoprolol; Piperidines | 1986 |
Ketanserin in the treatment of mild hypertension in elderly patients: preliminary results of a controlled double-blind trial.
Topics: Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Piperidines | 1986 |
Blood pressure reduction and pharmacokinetics of ketanserin in hypertensive patients.
Topics: Aged; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines | 1986 |
Intra arterial ketanserin in peripheral vascular disease.
Topics: Aged; Clinical Trials as Topic; Female; Humans; Injections, Intra-Arterial; Ischemia; Ketanserin; Leg; Male; Middle Aged; Piperidines; Serotonin Antagonists; Sympathectomy, Chemical | 1986 |
[Multicenter study with 3 different doses of ketanserin in essential arterial hypertension].
Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Drug Administration Schedule; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Vascular Resistance | 1985 |
Ketanserin and prazosin: a comparison of antihypertensive and biochemical effects.
Topics: Adult; Aldosterone; Blood Pressure; Cholesterol; Drug Evaluation; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Physical Exertion; Piperidines; Prazosin; Random Allocation; Renin | 1986 |
Selective antagonism of S2-serotonergic receptors relieves but does not prevent cold induced vasoconstriction in primary Raynaud's phenomenon.
Topics: Adult; Cold Temperature; Female; Humans; Ketanserin; Piperidines; Raynaud Disease; Receptors, Adrenergic; Receptors, Serotonin; Vasoconstriction | 1986 |
Influence of ketanserin pretreatment on the haemodynamic responses to sternotomy.
Topics: Drug Evaluation; Hemodynamics; Humans; Hypertension; Indoles; Intraoperative Complications; Ketanserin; Middle Aged; Myocardial Revascularization; Piperidines; Premedication; Serotonin; Serotonin Antagonists; Sternum | 1986 |
Quantitative study of the effects of Ketanserin in patients with primary Raynaud's phenomenon. A randomized, double blind, placebo controlled investigation and an additional long term open trial.
Topics: Adolescent; Adult; Aged; Blood Flow Velocity; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation; Raynaud Disease; Skin Temperature; Vascular Resistance | 1985 |
Effects of ketanserin on blood pressure, peripheral circulation and haemocoagulative parameters in essential hypertensives with or without arteriosclerosis obliterans of the lower limbs.
Topics: Adult; Antihypertensive Agents; Arteriosclerosis Obliterans; Blood Coagulation; Blood Pressure; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Leg; Male; Middle Aged; Piperidines; Propranolol; Random Allocation; Regional Blood Flow | 1986 |
Ketanserin and the cardiovascular system. 2. A study of its effects in patients undergoing myocardial revascularisation.
Topics: Antihypertensive Agents; Cardiopulmonary Bypass; Drug Evaluation; Female; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Myocardial Revascularization; Piperidines | 1986 |
Cardiovascular effects of ketanserin, a new antiserotonergic agent in the treatment of arterial hypertension.
Topics: Adult; Blood Pressure; Body Weight; Exercise Test; Heart Rate; Hemodynamics; Humans; Hypertension; Ketanserin; Metoprolol; Middle Aged; Piperidines; Regional Blood Flow; Serotonin Antagonists; Vascular Resistance | 1985 |
Effect of intravenous ketanserin on plasma catecholamines and renin activity in normal volunteers.
Topics: Adult; Catecholamines; Female; Humans; Injections, Intravenous; Ketanserin; Male; Piperidines; Renin; Serotonin Antagonists | 1985 |
Inhibition of cold-induced vasoconstriction with ketanserin.
Topics: Adult; Cold Temperature; Hand; Humans; Ibuprofen; Ketanserin; Ketoconazole; Male; Middle Aged; Piperidines; Regional Blood Flow; Serotonin; Skin Temperature; Thromboxane B2; Vasoconstriction | 1985 |
Ketanserin in essential hypertension: a double-blind, placebo-controlled study.
Topics: Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines | 1985 |
Controlled trial of ketanserin in hypertension.
Topics: Adult; Aged; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin | 1985 |
Ketanserin in chronic sympathetic dystrophy. An acute controlled trial.
Topics: Adult; Clinical Trials as Topic; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Reflex Sympathetic Dystrophy; Serotonin Antagonists | 1984 |
Effect of an oral serotonin antagonist, ketanserin, on plasma ACTH concentrations in Nelson's syndrome.
Topics: Adrenocorticotropic Hormone; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Nelson Syndrome; Piperidines; Pituitary Neoplasms; Serotonin Antagonists | 1984 |
Ketanserin in acute superficial thrombophlebitis.
Topics: Acute Disease; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Middle Aged; Pain; Piperidines; Random Allocation; Serotonin Antagonists; Thrombophlebitis | 1982 |
Is ketanserin a D receptor antagonist?
Topics: Adult; Animals; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Ketanserin; Male; Piperidines; Random Allocation; Rats; Receptors, Serotonin; Serotonin Antagonists | 1983 |
Mechanism of antihypertensive action of ketanserin in man.
Topics: Adrenergic alpha-Antagonists; Adult; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Ketanserin; Male; Methoxamine; Piperidines | 1983 |
Alpha 1 antagonistic and antiserotoninergic action during administration of ketanserin.
Topics: Adrenergic alpha-Antagonists; Humans; Hypertension; Ketanserin; Piperidines; Serotonin Antagonists | 1983 |
The effect of ketanserin on blood pressure and biochemical parameters in treated patients with essential hypertension.
Topics: Adrenergic beta-Antagonists; Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Diuretics; Double-Blind Method; Drug Therapy, Combination; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation; Serotonin Antagonists | 1984 |
Placebo-controlled double-blind trial of ketanserin in treatment of intermittent claudication.
Topics: Aged; Blood Flow Velocity; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Erythrocyte Deformability; Exercise Test; Humans; Intermittent Claudication; Ketanserin; Leg; Middle Aged; Piperidines; Plethysmography; Regional Blood Flow; Serotonin Antagonists | 1984 |
Ketanserin in combination with beta-adrenergic receptor blocking agents in the treatment of essential hypertension.
Topics: Adrenergic beta-Antagonists; Aged; Antihypertensive Agents; Blood Pressure; Drug Therapy, Combination; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines | 1984 |
The effect of ketanserin, a specific serotonin antagonist on the PRL, GH, ACTH and cortisol responses to hypoglycaemia in normal subjects.
Topics: Adrenocorticotropic Hormone; Adult; Growth Hormone; Humans; Hydrocortisone; Hypoglycemia; Ketanserin; Male; Piperidines; Pituitary Hormones, Anterior; Prolactin; Serotonin Antagonists | 1984 |
Ketanserin in hypertension. Early clinical evaluation and dose finding study of a new 5-HT2 receptor antagonist.
Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation; Serotonin Antagonists | 1983 |
Haemodynamic and humoral responses to chronic ketanserin treatment in essential hypertension.
Topics: Adult; Antihypertensive Agents; Clinical Trials as Topic; Double-Blind Method; Female; Hemodynamics; Humans; Hypertension; Ketanserin; Male; Methoxamine; Physical Exertion; Piperidines; Pressoreceptors; Renin-Angiotensin System | 1984 |
Treatment of Raynaud's phenomenon with ketanserin, a selective antagonist of the serotonin2 (5-HT2) receptor.
Topics: Adult; Aged; Clinical Trials as Topic; Female; Fingers; Humans; Ketanserin; Male; Middle Aged; Pilot Projects; Piperidines; Plethysmography; Raynaud Disease; Receptors, Serotonin; Regional Blood Flow; Scleroderma, Systemic; Serotonin Antagonists | 1984 |
[Serotonin antagonists in the treatment of hypertension].
Topics: Administration, Oral; Clinical Trials as Topic; Female; Humans; Hypertension; Infusions, Parenteral; Ketanserin; Male; Piperidines; Serotonin Antagonists | 1984 |
Experience with ketanserin, a serotonin (S2) antagonist, in longterm treatment of essential hypertension.
Topics: Adult; Aged; Chronic Disease; Clinical Trials as Topic; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Placebos; Serotonin Antagonists | 1984 |
Control of preeclamptic hypertension by ketanserin, a new serotonin receptor antagonist.
Topics: Adult; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Infusions, Parenteral; Ketanserin; Piperidines; Pre-Eclampsia; Pregnancy; Random Allocation; Serotonin Antagonists | 1984 |
Mechanism of antihypertensive action of ketanserin in man.
Topics: Antihypertensive Agents; Blood Pressure; Humans; Ketanserin; Piperidines | 1983 |
Treatment of Raynaud's phenomenon with ketanserin in patients with connective tissue disorders.
Topics: Adult; Clinical Trials as Topic; Connective Tissue Diseases; Double-Blind Method; Female; Fingers; Humans; Ketanserin; Microcirculation; Middle Aged; Piperidines; Raynaud Disease; Scleroderma, Systemic; Serotonin Antagonists; Ultrasonography | 1984 |
Ketanserin in essential hypertension: effects during rest and exercise.
Topics: Antihypertensive Agents; Blood Pressure; Catecholamines; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Physical Exertion; Piperidines; Rest | 1983 |
Responses of the systemic circulation and of the renin-angiotensin-aldosterone system to ketanserin at rest and exercise in normal man.
Topics: Adult; Blood Pressure; Cardiac Output; Catecholamines; Heart Rate; Hemodynamics; Humans; Ketanserin; Lactates; Male; Physical Exertion; Piperidines; Posture; Renin-Angiotensin System; Respiration; Rest; Serotonin Antagonists | 1984 |
A double-blind, placebo-controlled study of ketanserin in patients with Prinzmetal's angina. Evidence against a role for serotonin in the genesis of coronary vasospasm.
Topics: Aged; Angina Pectoris, Variant; Coronary Disease; Coronary Vasospasm; Double-Blind Method; Drug Evaluation; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Piperidines; Placebos; Platelet Aggregation; Serotonin; Serotonin Antagonists | 1984 |
Effect of the 5-hydroxytryptamine type 2 receptor antagonist, ketanserin, on blood pressure, the renin-angiotensin system and sympatho-adrenal function in patients with essential hypertension.
Topics: Adrenal Glands; Adult; Aged; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Norepinephrine; Phenylephrine; Piperidines; Posture; Renin-Angiotensin System; Serotonin Antagonists; Sympathetic Nervous System | 1984 |
Treatment of Raynaud's phenomenon with the 5-HT2-receptor antagonist ketanserin.
Topics: Adult; Aged; Female; Fingers; Humans; Ketanserin; Male; Middle Aged; Piperidines; Raynaud Disease; Regional Blood Flow; Serotonin Antagonists; Skin Temperature | 1982 |
The antihypertensive effects of a pure and selective serotonin-receptor blocking agent (R 41 468) in elderly patients.
Topics: Age Factors; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Depression, Chemical; Female; Heart Rate; Humans; Hypertension; Injections, Intravenous; Ketanserin; Male; Middle Aged; Myocardial Contraction; Piperidines; Placebos; Receptors, Serotonin; Research Design; Serotonin Antagonists | 1981 |
The antihypertensive effects of ketanserin (R 41468), a novel 5-hydroxytryptamine-blocking agent, in patients with essential hypertension.
Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines | 1981 |
Characterization of the SPECT 5-HT2A receptor ligand 123I-R91150 in healthy volunteers: part 2--ketanserin displacement.
Topics: Adult; Brain; Humans; Image Interpretation, Computer-Assisted; Iodine Radioisotopes; Ketanserin; Ligands; Male; Metabolic Clearance Rate; Piperidines; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Reference Values; Tissue Distribution; Tomography, Emission-Computed, Single-Photon | 2006 |
462 other study(ies) available for ketanserin and piperidines
Article | Year |
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Oxygen isosteric derivatives of 3-(3-hydroxyphenyl)-N-n-propylpiperidine.
Topics: Animals; Brain; Dopamine Agents; In Vitro Techniques; Ketanserin; Mice; Oxygen; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone | 1992 |
Stimulation by risperidone of rat prolactin secretion in vivo and in cultured pituitary cells in vitro.
Topics: Animals; Antipsychotic Agents; Cells, Cultured; Haloperidol; Isoxazoles; Ketanserin; Male; Piperidines; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Risperidone; Spiro Compounds; Stimulation, Chemical | 1992 |
Uptake and release of serotonin in rat cerebrovascular nerves after subarachnoid hemorrhage.
Topics: Animals; Basilar Artery; Electric Stimulation; Ischemic Attack, Transient; Ketanserin; Male; Oxidopamine; Paroxetine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Subarachnoid Hemorrhage; Sympathetic Nervous System; Tetrodotoxin; Vasoconstriction | 1992 |
Serotonergic aspects of the response of human platelets to immune-adjuvant muramyl dipeptide.
Topics: Acetylmuramyl-Alanyl-Isoglutamine; Adenosine Diphosphate; Adjuvants, Immunologic; Blood Platelets; Carrier Proteins; Humans; Imipramine; Ketanserin; Lysergic Acid Diethylamide; Paroxetine; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1992 |
5HT2 receptor changes in rat cortex and platelets following chronic ritanserin and clorgyline administration.
Topics: Animals; Blood Platelets; Cerebral Cortex; Clorgyline; Homovanillic Acid; Hydroxyindoleacetic Acid; Ketanserin; Lysergic Acid Diethylamide; Male; Norepinephrine; Piperidines; Propylamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin | 1990 |
Effect of 3,4-methylenedioxymethamphetamine on [3H]paroxetine binding in the frontal cortex and blood platelets of rats.
Topics: 3,4-Methylenedioxyamphetamine; Animals; Blood Platelets; Frontal Lobe; Hydroxyindoleacetic Acid; Ketanserin; Kinetics; Male; N-Methyl-3,4-methylenedioxyamphetamine; Paroxetine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Time Factors; Tritium | 1991 |
AHR-16303B, a novel antagonist of 5-HT2 receptors and voltage-sensitive calcium channels.
Topics: Animals; Atrial Function; Blood Pressure; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Chloride; Diuresis; Dose-Response Relationship, Drug; Edema; Guinea Pigs; Heart Atria; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Nimodipine; Piperidines; Platelet Aggregation; Propiophenones; Rabbits; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Histamine H1; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Tritium; Verapamil | 1991 |
Visual recognition memory in squirrel monkeys: effects of serotonin antagonists on baseline and hypoxia-induced performance deficits.
Topics: Animals; Avoidance Learning; Cognition; Dose-Response Relationship, Drug; Hypoxia; Ketanserin; Male; Memory; Mianserin; Piperidines; Psychomotor Performance; Reinforcement Schedule; Saimiri; Serotonin Antagonists | 1991 |
DOI-induced inhibition of copulatory behavior in male rats: reversal by 5-HT2 antagonists.
Topics: Amphetamines; Animals; Copulation; Ejaculation; Female; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Tranquilizing Agents | 1991 |
Naloxone and serotonin receptor subtype antagonists: interactive effects upon deprivation-induced intake.
Topics: Animals; Drug Interactions; Feeding Behavior; Food Deprivation; Indoles; Ketanserin; Male; Methysergide; Naloxone; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Tropisetron | 1991 |
Stimulatory effects of 5-hydroxytryptamine on fluid secretion and transmural potential difference in rat small intestine are mediated by different receptor subtypes.
Topics: Animals; Blood Pressure; Body Fluids; Cisapride; Dose-Response Relationship, Drug; Female; Intestine, Small; Ketanserin; Male; Membrane Potentials; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1990 |
Laminar distributions of muscarinic acetylcholine, serotonin, GABA and opioid receptors in human posterior cingulate cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aged; Autoradiography; Cerebral Cortex; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Humans; Iodocyanopindolol; Ketanserin; Male; Middle Aged; Oxotremorine; Paroxetine; Pindolol; Piperidines; Pirenzepine; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1990 |
Effects of ketanserin tartrate on 3-hydroxy, 3-methylglutaryl coenzyme A reductase activity in cultured human skin fibroblasts.
Topics: Adrenergic alpha-Antagonists; Cells, Cultured; Fibroblasts; Humans; Hydroxymethylglutaryl CoA Reductases; Ketanserin; Piperidines; Prazosin; Ritanserin; Serotonin Antagonists | 1990 |
CGS 18102A, a benzopyranopyridine anxiolytic with 5-HT1 agonist and 5-HT2 antagonist properties.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Benzopyrans; Binding, Competitive; Cerebral Cortex; Ketanserin; Kinetics; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1990 |
5-HT1C receptors in the serotonergic control of periaqueductal gray induced aversion in rats.
Topics: Amphetamines; Animals; Cyproheptadine; Indoles; Ketanserin; Male; Periaqueductal Gray; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reinforcement, Psychology; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
[3H]ketanserin binds to non-5-HT2 sites in rabbit cerebral cortex and neostriatum.
Topics: Animals; Binding, Competitive; Caudate Nucleus; Cell Membrane; Cerebral Cortex; Corpus Striatum; Frontal Lobe; Ketanserin; Kinetics; Male; Methysergide; Mianserin; Piperidines; Putamen; Rabbits; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Inhibition of spontaneous and evoked unit activity in the rat medial prefrontal cortex by mesencephalic raphe nuclei.
Topics: 5,7-Dihydroxytryptamine; Animals; Brain; Cerebral Cortex; Electric Stimulation; Evoked Potentials; Ketanserin; Male; Membrane Potentials; Neurons; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Ritanserin; Serotonin | 1990 |
Inhibition of serotonin-amplified human platelet aggregation by ketanserin, ritanserin, and the ergoline 5HT2 receptor antagonists-LY53857, sergolexole, and LY237733.
Topics: Adult; Ergolines; Female; Humans; Ketanserin; Lysergic Acid; Male; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
5HT-2 mediation of acute behavioral effects of hallucinogens in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Behavior, Animal; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Hallucinogens; Ketanserin; Male; Mescaline; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Tetrahydronaphthalenes | 1990 |
Behavioural evidence for a functional interaction between central 5-HT2 and 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Behavior, Animal; Central Nervous System; Dose-Response Relationship, Drug; Haloperidol; Ketanserin; Male; Methoxydimethyltryptamines; Piperidines; Prazosin; Pyrimidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Stereotyped Behavior; Tetrahydronaphthalenes | 1990 |
Effect of serotonergic drugs on negative contrast in consummatory behavior.
Topics: Animals; Buspirone; Chlordiazepoxide; Cyproheptadine; Dose-Response Relationship, Drug; Ethanol; Feeding Behavior; Fenclonine; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Male; Midazolam; Nucleus Accumbens; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Binding of [3H]dihydrotetrabenazine and [125I]azidoiodoketanserin photoaffinity labeling of the monoamine transporter of platelet 5-HT organelles.
Topics: Affinity Labels; Animals; Azides; Biogenic Monoamines; Blood Platelets; Blood Proteins; Cell Membrane; Guinea Pigs; Humans; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Paroxetine; Photochemistry; Piperidines; Rabbits; Rats; Receptors, Serotonin; Subcellular Fractions; Tetrabenazine | 1990 |
Receptor subtypes mediating facilitation by serotonin of excitability of spinal motoneurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; In Vitro Techniques; Injections, Intravenous; Iontophoresis; Ketanserin; Male; Methysergide; Microelectrodes; Motor Neurons; Piperidines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes | 1990 |
Mediation of ACTH and prolactin responses to 5-HTP by 5-HT2 receptors.
Topics: 5-Hydroxytryptophan; Adrenocorticotropic Hormone; Animals; Dose-Response Relationship, Drug; Ketanserin; Male; Metergoline; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone | 1990 |
Acute hypotension due to platelet serotonin-induced chemoreflexes after intravenous injection of dextran sulfate in the rabbit.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Autonomic Nervous System; Blood Platelets; Bradycardia; Chemoreceptor Cells; Cimetidine; Complement C3; Dextran Sulfate; Dextrans; Factor XII; Histamine; Histamine Release; Hypotension; Injections, Intravenous; Ketanserin; Leukocyte Count; Lung; Male; Methysergide; Piperidines; Rabbits; Serotonin | 1985 |
On the nature of the contractile motor responses of the rat stomach elicited by serotonin or substance P in vitro.
Topics: Animals; Atropine; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Stomach; Substance P; Tachyphylaxis; Tetrodotoxin | 1985 |
Effect of ketanserin on hemodynamics, plasma-catecholamine concentrations, and serotonin uptake by platelets in volunteers and patients with congestive heart failure.
Topics: Aged; Blood Platelets; Catecholamines; Dopamine; Female; Heart Failure; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Norepinephrine; Piperidines; Serotonin; Serotonin Antagonists; Stroke Volume; Vascular Resistance | 1985 |
Antihypertensive effects of ketanserin in the spontaneously hypertensive rat: mode of action.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Time Factors | 1985 |
Chronic serotonergic blockade with ketanserin in the spontaneously hypertensive rat.
Topics: Animals; Blood Pressure; Heart Rate; Ketanserin; Male; Piperidines; Rats; Rats, Inbred SHR; Serotonin Antagonists | 1985 |
Evidence for a central component to the hypotensive action of ketanserin in the dog.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Dogs; Ganglionic Blockers; Hexamethonium Compounds; Ketanserin; Mecamylamine; Nicotine; Norepinephrine; Piperidines; Vasoconstriction | 1985 |
Serotonergic mechanisms and blood pressure in sheep.
Topics: Adrenergic alpha-Antagonists; Adrenocorticotropic Hormone; Animals; Blood Pressure; Female; Heart Rate; Hypertension; Ketanserin; Phenylephrine; Piperidines; Prazosin; Serotonin; Serotonin Antagonists; Sheep | 1985 |
Platelet serotonin in essential hypertension and in mental depression.
Topics: Adult; Antidepressive Agents; Blood Platelets; Depressive Disorder; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Serotonin; Serotonin Antagonists; Sex Factors | 1985 |
Is there alpha-adrenergic blockade and/or serotonergic blockade during chronic ketanserin treatment?
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Humans; Ketanserin; Malignant Carcinoid Syndrome; Phenylephrine; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists | 1985 |
The acute antihypertensive effect of ketanserin increases with age.
Topics: Adult; Aged; Aging; Antihypertensive Agents; Blood Pressure; Female; Humans; Hypertension; Injections, Intravenous; Ketanserin; Male; Middle Aged; Piperidines | 1985 |
Ketanserin: a possible tool for studying the role of serotonin in hypertension.
Topics: Aldosterone; Blood Pressure; Female; Hemodynamics; Humans; Hypertension; Ketanserin; Male; Middle Aged; Norepinephrine; Phentolamine; Phenylephrine; Piperidines; Regional Blood Flow; Renal Circulation; Renin; Serotonin; Serotonin Antagonists; Time Factors | 1985 |
A comparative and long-term evaluation of ketanserin in the treatment of essential hypertension.
Topics: Adrenergic beta-Antagonists; Adult; Blood Pressure; Diuretics; Female; Humans; Hypertension; Ketanserin; Male; Piperidines; Serotonin Antagonists; Time Factors | 1985 |
Ketanserin in the acute management of severe hypertension.
Topics: Adolescent; Adult; Blood Pressure; Creatinine; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Renin; Serotonin Antagonists; Time Factors | 1985 |
Platelet hypersensitivity to serotonin after prolonged ketanserin intake?
Topics: Adult; Blood Platelets; Humans; Ketanserin; Male; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists | 1985 |
Continuous inhibition of platelet S2-serotonergic receptors during chronic administration of ketanserin in humans.
Topics: Adenosine Diphosphate; Blood Platelets; Collagen; Epinephrine; Female; Humans; Ketanserin; Male; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin Antagonists; Time Factors | 1985 |
Blood pressure, 5-OH indoleacetic acid, and vanilmandelic acid excretion and blood platelet aggregation in hypertensive patients treated with ketanserin.
Topics: Adult; Blood Pressure; Female; Heart Rate; Humans; Hydroxyindoleacetic Acid; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists; Time Factors; Vanilmandelic Acid | 1985 |
Effects of ketanserin on platelet function and red cell filterability in hypertension and peripheral vascular disease.
Topics: Adult; Aged; Blood Platelets; Erythrocyte Deformability; Erythrocytes; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Serotonin Antagonists; Vascular Diseases | 1985 |
Effects of ketanserin on the intracellular concentration and transmembrane fluxes of sodium and potassium in erythrocytes of normal male subjects.
Topics: Cell Membrane Permeability; Erythrocyte Membrane; Erythrocytes; Furosemide; Humans; Ketanserin; Lithium; Male; Ouabain; Piperidines; Potassium; Serotonin Antagonists; Sodium | 1985 |
Serotonin and the blood vessel wall.
Topics: Animals; Drug Interactions; In Vitro Techniques; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation | 1985 |
Serotonin-induced vasoconstriction in the perfused canine femoral artery can be blocked in vivo by ketanserin.
Topics: Animals; Blood Pressure; Dogs; Female; Femoral Artery; Hemodynamics; In Vitro Techniques; Isosorbide Dinitrate; Ketanserin; Male; Piperidines; Prazosin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasoconstriction | 1985 |
Influence of ketanserin on 5-hydroxytryptamine-induced cerebrovascular spasm in the cat.
Topics: Animals; Cats; Cerebrovascular Circulation; Ischemic Attack, Transient; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Serotonin; Serotonin Antagonists | 1985 |
Effects of serotonin on the cardiopulmonary circulatory system with and without 5-HT2-receptor blockade by ketanserin.
Topics: Animals; Dogs; Hypertension, Pulmonary; Ketanserin; Piperidines; Pulmonary Artery; Pulmonary Embolism; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Resistance | 1985 |
Bucindolol has serotonin and alpha-adrenoceptor blocking properties.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; In Vitro Techniques; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Regional Blood Flow; Serotonin Antagonists | 1985 |
Two classes of myocardial 5-hydroxytryptamine receptors that are neither 5-HT1 nor 5-HT2.
Topics: Animals; Cats; Female; Heart Rate; In Vitro Techniques; Ketanserin; Male; Myocardial Contraction; Myocardium; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1985 |
The pentagastrin test in the diagnosis of the carcinoid syndrome.
Topics: Carcinoid Tumor; Female; Gastrointestinal Neoplasms; Humans; Hydroxyindoleacetic Acid; Ketanserin; Male; Malignant Carcinoid Syndrome; Pentagastrin; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Substance P; Time Factors | 1985 |
Large and small vessel responses to serotonin in the peripheral circulation.
Topics: Arteriosclerosis; Humans; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasodilation; Vasodilator Agents | 1985 |
Intra-erythrocyte concentration and transmembrane fluxes of sodium and potassium during acute and short-term administration of ketanserin in normal male subjects.
Topics: Adult; Erythrocyte Membrane; Erythrocytes; Humans; Ion Channels; Ketanserin; Male; Piperidines; Potassium; Sodium; Sodium-Potassium-Exchanging ATPase | 1985 |
[Effect of ketanserin on blood pressure in rats].
Topics: Adrenal Glands; Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hydroxyindoleacetic Acid; Ketanserin; Male; Norepinephrine; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Serotonin; Sympathetic Nervous System | 1985 |
In vivo voltammetry in the suprachiasmatic nucleus of the rat: effects of RU24969, methiothepin and ketanserin.
Topics: Animals; Dibenzothiepins; Electrophysiology; Hydroxyindoleacetic Acid; Ketanserin; Male; Methiothepin; Microelectrodes; Oxidation-Reduction; Phenethylamines; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Suprachiasmatic Nucleus; Time Factors | 1986 |
125I-LSD autoradiography confirms the preferential localization of caudate-putamen S2 receptors to the caudal (peripallidal) region.
Topics: Animals; Autoradiography; Butaclamol; Caudate Nucleus; Frontal Lobe; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Putamen; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin | 1986 |
Ketanserin in the preoperative and intraoperative management of a patient with carcinoid tumor undergoing tricuspid valve replacement.
Topics: Blood Pressure; Carcinoid Tumor; Cardiopulmonary Bypass; Female; Histamine Release; Humans; Intraoperative Care; Intraoperative Complications; Ketanserin; Middle Aged; Piperidines; Preoperative Care; Serotonin; Tricuspid Valve; Tricuspid Valve Insufficiency | 1986 |
Ketanserin and ritanserin can reduce reperfusion-induced but not ischaemia-induced arrhythmias in anaesthetised rats.
Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Coronary Vessels; Female; Guinea Pigs; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists | 1987 |
Antihypertensive effects of ketanserin and ritanserin in the spontaneously hypertensive rat.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin; Sympathetic Nervous System | 1988 |
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Ergolines; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pyrimidinones; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone | 1988 |
Are drugs that act both on serotonin receptors and alpha 1-adrenoceptors more potent hypotensive agents than those that act only on alpha 1-adrenoceptors?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Cats; Cinanserin; Ergolines; Ketanserin; Male; Metergoline; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes | 1988 |
Age-related changes in rat serotonergic and adrenergic systems and in receptor responsiveness to subchronic desipramine treatment.
Topics: Aging; Animals; Brain; Clonidine; Desipramine; Dihydroalprenolol; Hydroxyindoleacetic Acid; Imipramine; Ketanserin; Kinetics; Male; Paroxetine; Piperidines; Prazosin; Proteins; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Serotonin; Serotonin; Time Factors | 1988 |
Arterial and venous effects of serotonin in the forearm of healthy subjects are not age-related.
Topics: Adult; Aged; Aging; Blood Pressure; Forearm; Heart Rate; Humans; Ketanserin; Male; Methoxamine; Middle Aged; Piperidines; Regional Blood Flow; Ritanserin; Serotonin; Serotonin Antagonists | 1989 |
Serotonin as a modulator of skeletal muscle oxygenation: effects of ketanserin and ritanserin on oxygen pressure distributions.
Topics: Animals; Ketanserin; Muscles; Oxygen; Oxygen Consumption; Piperidines; Pressure; Rabbits; Ritanserin; Serotonin; Serotonin Antagonists | 1989 |
Lack of a difference between ketanserin and ritanserin in central vs. peripheral serotonin receptor antagonism.
Topics: Animals; Blood Pressure; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1989 |
Facilitation of 8-OHDPAT-induced forepaw treading of rats by the 5-HT2 agonist DOI.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprenolol; Amphetamines; Animals; Behavior, Animal; Cerebral Cortex; Injections, Subcutaneous; Ketanserin; Male; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Tetrahydronaphthalenes | 1989 |
Production of wet-dog shakes in rats and down-regulation of spinal 5-HT2 receptors.
Topics: Animals; Behavior, Animal; Brain Stem; Ketanserin; Male; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spinal Cord | 1989 |
The pentagastrin test in the diagnosis of the carcinoid syndrome. Blockade of gastrointestinal symptoms by ketanserin.
Topics: Aged; Calcium; Digestive System; Female; Humans; Ketanserin; Liver Neoplasms; Male; Malignant Carcinoid Syndrome; Middle Aged; Pentagastrin; Piperidines; Serotonin; Serotonin Antagonists; Substance P; Vasomotor System | 1985 |
Brain dopamine and serotonin receptor sites revealed by digital subtraction autoradiography.
Topics: Animals; Autoradiography; Brain; Butaclamol; Computers; Ketanserin; Piperidines; Radiographic Image Enhancement; Radionuclide Imaging; Rats; Receptors, Dopamine; Receptors, Serotonin; Spiperone; Sulpiride | 1985 |
The effects of a new serotonin receptor antagonist (ketanserin) on lower urinary tract function in patients with prostatism.
Topics: Aged; Blood Pressure; Humans; Ketanserin; Male; Middle Aged; Piperidines; Pressure; Prostatic Hyperplasia; Serotonin Antagonists; Urethra; Urinary Bladder; Urodynamics | 1985 |
Reduction in opioid and non-opioid forms of swim analgesia by 5-HT2 receptor antagonists.
Topics: Analgesia; Endorphins; Ketanserin; Methysergide; Physical Exertion; Piperidines; Receptors, Serotonin; Serotonin Antagonists | 1989 |
5-Hydroxytryptamine stimulates the formation of inositol phosphate in astrocytes from different regions of the brain.
Topics: Animals; Astrocytes; Brain; Cyclic AMP; Inositol Phosphates; Ketanserin; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Stimulation, Chemical; Sugar Phosphates; Tissue Distribution | 1987 |
Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist.
Topics: Animals; Binding, Competitive; Biogenic Amines; Brain; Cerebellum; Cerebral Cortex; Corpus Striatum; Female; Guinea Pigs; Haloperidol; Hippocampus; Histamine H2 Antagonists; In Vitro Techniques; Ketanserin; Kinetics; Male; Organ Specificity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1985 |
Treatment of arterial hypertension with ketanserin in mono- and combination therapy.
Topics: Adrenergic beta-Antagonists; Adult; Aged; Blood Pressure; Drug Therapy, Combination; Female; Follow-Up Studies; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Serotonin Antagonists | 1985 |
Hypotensive actions of ketanserin in dogs: involvement of a centrally mediated inhibition of sympathetic vascular tone.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Dogs; Female; Heart Rate; Hexamethonium; Hexamethonium Compounds; Ketanserin; Male; Mecamylamine; Nicotine; Piperidines; Sympathetic Nervous System; Vascular Resistance; Vasomotor System | 1985 |
Effect of somatostatin on bethanechol-stimulated gastric acid secretion and gastric antral motility in dogs with gastric fistula.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Bethanechol Compounds; Dogs; Domperidone; Dose-Response Relationship, Drug; Female; Gastric Acid; Gastric Fistula; Gastrointestinal Motility; Ketanserin; Male; Piperidines; Propranolol; Pyloric Antrum; Receptors, Dopamine; Receptors, Serotonin; Somatostatin | 1985 |
Dopamine D2 receptors selectively labeled by a benzamide neuroleptic: [3H]-YM-09151-2.
Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Corpus Striatum; Dogs; Guanylyl Imidodiphosphate; Ketanserin; Kinetics; Piperidines; Receptors, Dopamine; Sodium; Spiperone; Substrate Specificity; Tetrahydronaphthalenes | 1985 |
[Endocrine and metabolic changes induced in surgery by the combination of ketanserin and alfentanyl].
Topics: Abdomen; Adolescent; Adult; Aged; Alfentanil; Analgesics, Opioid; Drug Therapy, Combination; Female; Fentanyl; Humans; Intraoperative Complications; Ketanserin; Male; Middle Aged; Piperidines; Premedication; Serotonin Antagonists; Stress, Physiological | 1985 |
Mechanism of the hypotensive effect of a novel phenylpiperazine derivative, SGB-1534: antagonism at alpha 1-adrenergic and 5-HT2 receptors.
Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Antihypertensive Agents; Decerebrate State; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Piperidines; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Serotonin Antagonists | 1985 |
Differential effect of subchronic treatment with various neuroleptic agents on serotonin2 receptors in rat cerebral cortex.
Topics: 5,7-Dihydroxytryptamine; Animals; Antipsychotic Agents; Cerebral Cortex; Chlorpromazine; Clozapine; Female; Haloperidol; Imipramine; Ketanserin; Loxapine; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Sulpiride | 1986 |
[Ketanserin in association with a beta blocker and a diuretic in the treatment of essential hypertension].
Topics: Adrenergic beta-Antagonists; Blood Pressure; Diuretics; Drug Therapy, Combination; Humans; Hypertension; Ketanserin; Piperidines | 1985 |
Ketanserin in intermittent claudication.
Topics: Humans; Intermittent Claudication; Ketanserin; Piperidines | 1986 |
Serotonin receptor involvement in the avoidance learning deficit caused by p-chloroamphetamine-induced serotonin release.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Amphetamines; Animals; Avoidance Learning; Brain; Ketanserin; Male; p-Chloroamphetamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Histamine H1; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Serotonin | 1986 |
Studies on the receptor profile of bisoprolol.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Bisoprolol; Cattle; Dihydroalprenolol; Domperidone; Humans; In Vitro Techniques; Ketanserin; Male; Piperidines; Prazosin; Propanolamines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Histamine; Receptors, Muscarinic; Spiperone; Tetrahydronaphthalenes; Yohimbine | 1986 |
Characterization of flufylline, fluprofylline, ritanserin, butanserin and R 56413 with respect to in-vivo alpha 1-,alpha 2- and 5-HT2-receptor antagonism and in-vitro affinity for alpha 1-,alpha 2- and 5-HT2-receptors: comparison with ketanserin.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Decerebrate State; Histamine H2 Antagonists; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Theophylline; Vasoconstriction | 1986 |
Typical and atypical antipsychotic occupancy of D2 and S2 receptors: an autoradiographic analysis in rat brain.
Topics: Animals; Antipsychotic Agents; Autoradiography; Binding, Competitive; Brain; Caudate Nucleus; Haloperidol; Ketanserin; Kinetics; Male; Nucleus Accumbens; Olfactory Bulb; Piperidines; Putamen; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Spiperone | 1986 |
Permissive role of D-1 receptor stimulation by endogenous dopamine for the expression of postsynaptic D-2-mediated behavioural responses. Yawning in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Azepines; Benzazepines; Brain Chemistry; Dopamine; Ergolines; Kainic Acid; Ketanserin; Male; Metergoline; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sulpiride; Yawning | 1987 |
Quipazine reduces food intake in the rat by activation of 5-HT2-receptors.
Topics: Animals; Diet; Dose-Response Relationship, Drug; Eating; Histamine H2 Antagonists; Imidazoles; Ketanserin; Methysergide; Ondansetron; Pindolol; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1988 |
Antagonism of the LSD cue by putative serotonin antagonists: relationship to inhibition of in vivo [3H]spiroperidol binding.
Topics: Animals; Cerebellum; Corpus Striatum; Frontal Lobe; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Pizotyline; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1985 |
Behavioural stimulation is induced by separate dopamine D-1 and D-2 receptor sites in reserpine-pretreated but not in normal rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Catalepsy; Ergolines; Hydroxydopamines; Ketanserin; Male; Motor Activity; Oxidopamine; Pergolide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Stereotyped Behavior | 1985 |
The effects of ketanserin, methysergide and LY 53857 on sympathetic nerve activity.
Topics: Anesthesia; Animals; Blood Pressure; Cats; Ergolines; Heart Rate; Hemodynamics; Ketanserin; Lactates; Lactic Acid; Male; Methysergide; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Sympathetic Nervous System | 1985 |
Mechanisms involved in the vasodilator action of 5-hydroxytryptamine in the dog femoral arterial circulation in vivo.
Topics: Animals; Blood Pressure; Carbon Dioxide; Dogs; Dose-Response Relationship, Drug; Female; Femoral Artery; Hindlimb; Ketanserin; Male; Muscle, Smooth, Vascular; Ornipressin; Piperidines; Pizotyline; Regional Blood Flow; Serotonin; Sympathetic Nervous System; Vasodilator Agents | 1985 |
Solubilization of rat brain serotonin-S2 receptors using CHAPS/salt.
Topics: Animals; Brain Chemistry; Centrifugation, Density Gradient; Cholic Acids; Filtration; In Vitro Techniques; Ketanserin; Microsomes; Nerve Tissue Proteins; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Sodium Chloride | 1985 |
Analysis of the heart rate effects of 5-hydroxytryptamine in the cat; mediation of tachycardia by 5-HT1-like receptors.
Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Isoproterenol; Ketanserin; Male; Methysergide; Piperidines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tropanes; Vagus Nerve | 1985 |
Hemodynamic evaluation of endotoxic shock in anesthetized piglets: antagonism of endogenous vasoactive substances.
Topics: Adrenal Cortex Hormones; Anesthesia; Animals; Bacterial Toxins; Blood Pressure; Cardiac Output; Enterotoxins; Escherichia coli Proteins; Flurbiprofen; Heart Rate; Hemodynamics; Ketanserin; Narcotic Antagonists; Piperidines; Prednisone; Pulmonary Circulation; Serotonin Antagonists; Shock, Septic; Swine; Time Factors; Vascular Resistance | 1985 |
Spiperone differentiates multiple 5-hydroxytryptamine responses in rat hippocampal slices in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Butyrophenones; Hippocampus; In Vitro Techniques; Ketanserin; Piperidines; Rats; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes | 1985 |
Effect of serotonin and its antagonist ketanserin on pial vessels.
Topics: Administration, Topical; Animals; Arteries; Carbon Dioxide; Cats; Cerebrovascular Circulation; Ketanserin; Oxygen; Pia Mater; Piperidines; Rest; Serotonin; Serotonin Antagonists; Veins | 1985 |
Peripheral serotonin2 receptor blockade does not inhibit 5-hydroxytryptophan-induced aldosterone stimulation.
Topics: 5-Hydroxytryptophan; Adult; Aldosterone; Humans; Ketanserin; Male; Methysergide; Piperidines; Potassium; Renin; Serotonin; Serotonin Antagonists | 1985 |
Effects of ketanserin, a 5-HT2-receptor antagonist, on the blood flow response to temperature changes in the diabetic foot.
Topics: Adult; Aged; Diabetes Mellitus; Female; Foot; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Piperidines; Plethysmography; Regional Blood Flow; Serotonin Antagonists; Temperature | 1985 |
Effects of serotonin receptor agonists and antagonists on schedule-controlled behavior of squirrel monkeys.
Topics: 5-Hydroxytryptophan; Animals; Cinanserin; Conditioning, Operant; Cyproheptadine; Electroshock; Female; Ketanserin; Male; Metergoline; Methysergide; Piperazines; Piperidines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri | 1985 |
A comparison of cardiovascular and smooth muscle effects of 5-hydroxytryptamine and 5-carboxamidotryptamine, a selective agonist of 5-HT1 receptors.
Topics: Airway Resistance; Animals; Cyproheptadine; Guinea Pigs; Heart Rate; Hemodynamics; Ileum; In Vitro Techniques; Ketanserin; Male; Mecamylamine; Methysergide; Muscle, Smooth; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Urinary Bladder | 1985 |
Monoaminergic involvement in the pharmacological actions of buspirone.
Topics: Animals; Apomorphine; Behavior, Animal; Brain; Buspirone; Dopamine; Ketanserin; Male; Methoxydimethyltryptamines; Monoamine Oxidase; p-Chloroamphetamine; Piperazines; Piperidines; Psychotropic Drugs; Pyrimidines; Rats; Serotonin | 1985 |
A comparison of 5-hydroxytryptamine receptors mediating contraction in rabbit aorta and dog saphenous vein: evidence for different receptor types obtained by use of selective agonists and antagonists.
Topics: Animals; Aorta; Dogs; In Vitro Techniques; Ketanserin; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rabbits; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Antagonists; Spiperone | 1985 |
Relationship of increased lung serotonin levels to endotoxin-induced pulmonary hypertension in sheep. Effect of a serotonin antagonist.
Topics: Animals; Blood Pressure; Endotoxins; Escherichia coli; Hypertension, Pulmonary; Hypoxia; Ketanserin; Lung; Lymph; Oxygen; Piperidines; Platelet Count; Pulmonary Artery; Serotonin; Serotonin Antagonists; Sheep | 1985 |
Lack of effect of propranolol on the steady-state plasma levels of ketanserin.
Topics: Adult; Blood Pressure; Female; Heart Rate; Humans; Ketanserin; Liver; Male; Middle Aged; Piperidines; Propranolol; Time Factors | 1985 |
Chronic 5-HT2 receptor blockade with ritanserin does not reduce blood pressure in the spontaneously hypertensive rat.
Topics: Animals; Blood Pressure; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Heart Rate; Hypertension; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Receptors, Serotonin; Ritanserin; Time Factors | 1985 |
Different subcellular localization of muscarinic and serotonin (S2) receptors in human, dog, and rat brain.
Topics: Adult; Aged; Animals; Brain; Brain Chemistry; Centrifugation, Density Gradient; Dexetimide; Dogs; Humans; Ketanserin; Mathematics; Microscopy, Electron; Middle Aged; Piperidines; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Receptors, Serotonin; Species Specificity; Subcellular Fractions | 1986 |
In vitro and in vivo irreversible blockade of cortical S2 serotonin receptors by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline: a technique for investigating S2 serotonin receptor recovery.
Topics: Animals; Cerebral Cortex; Domperidone; Dose-Response Relationship, Drug; Ketanserin; Kinetics; Male; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin | 1986 |
Characterization of 5-hydroxytryptamine receptors in rat stomach fundus.
Topics: Animals; Binding, Competitive; Brain Chemistry; Gastric Fundus; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Piperazines; Piperidines; Propranolol; Pyrazines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium | 1985 |
Serotonin type 2 antagonists inhibit lordosis behavior in the female rat: reversal with quipazine.
Topics: Analysis of Variance; Animals; Butyrophenones; Cyproheptadine; Estradiol; Female; Ketanserin; Methiothepin; Piperidines; Pizotyline; Posture; Progesterone; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Sexual Behavior, Animal | 1986 |
Reactivity of the bronchial artery to 5-hydroxytryptamine.
Topics: Animals; Bronchial Arteries; Cattle; Female; Horses; In Vitro Techniques; Ketanserin; Male; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sheep; Vasoconstriction | 1985 |
Solubilized ketanserin binding sites from pig platelet membranes.
Topics: Animals; Binding Sites; Binding, Competitive; Blood Platelets; Cell Membrane; In Vitro Techniques; Ketanserin; Kinetics; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Solubility; Swine | 1985 |
Peripheral arterial diseases: treatment with ketanserin as i.v. infusion. An open study in 20 patients.
Topics: Arteriosclerosis; Humans; Infusions, Parenteral; Ketanserin; Piperidines; Regional Blood Flow | 1985 |
Subtypes of the 5-HT receptor mediating the behavioural responses to 5-methoxy-N,N-dimethyltryptamine in the rat.
Topics: Animals; Apomorphine; Behavior, Animal; Betaxolol; Haloperidol; Ketanserin; Male; Pindolol; Piperidines; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reserpine; Spiperone | 1985 |
Molecular pharmacology of 5-HT1 and 5-HT2 recognition sites in rat and pig brain membranes: radioligand binding studies with [3H]5-HT, [3H]8-OH-DPAT, (-)[125I]iodocyanopindolol, [3H]mesulergine and [3H]ketanserin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Chemistry; Choroid Plexus; Ergolines; In Vitro Techniques; Iodocyanopindolol; Ketanserin; Male; Membranes; Pindolol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tetrahydronaphthalenes | 1985 |
Drug treatment of claudication: vasodilators, hemorrheologic agents, and antiserotonin drugs.
Topics: Double-Blind Method; Erythrocyte Deformability; Humans; Intermittent Claudication; Ketanserin; Pentoxifylline; Piperidines; Serotonin Antagonists; Theobromine; Vasodilator Agents | 1986 |
In vivo regulation of the serotonin-2 receptor in rat brain.
Topics: Amitriptyline; Animals; Brain Chemistry; Electroshock; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tritium | 1986 |
[In vivo study of central serotoninergic receptors in man using positron tomography].
Topics: Brain; Cerebellum; Chlorpromazine; Frontal Lobe; Humans; Ketanserin; Kinetics; Piperidines; Receptors, Serotonin; Tomography, Emission-Computed | 1985 |
Dependence of the antagonism at human platelet 5-HT2 receptors by ketanserin on the reaction pH.
Topics: Amidines; Blood Platelets; Butyrophenones; Cyproheptadine; Female; Humans; Hydrogen-Ion Concentration; Ketanserin; Kinetics; Male; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone | 1985 |
Characterization and localization of serotonin receptors in human brain postmortem.
Topics: Adult; Aged; Autoradiography; Binding, Competitive; Diencephalon; Female; Frontal Lobe; Hippocampus; Humans; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin; Spiperone; Telencephalon | 1986 |
Serotonin as a mediator of cyclic flow variations in stenosed canine coronary arteries.
Topics: Animals; Coronary Circulation; Coronary Disease; Coronary Vessels; Dogs; Hemodynamics; Ketanserin; Male; Periodicity; Piperidines; Serotonin | 1986 |
Comparative effects of oxygen, nifedipine and ketanserin in hypoxic pulmonary hypertension.
Topics: Adult; Carbon Dioxide; Cardiac Output; Female; Heart Rate; Humans; Hypertension, Pulmonary; Hypoxia; Ketanserin; Lung Diseases, Obstructive; Lung Volume Measurements; Male; Middle Aged; Nifedipine; Oxygen; Oxygen Inhalation Therapy; Piperidines; Pulmonary Wedge Pressure; Serotonin Antagonists | 1985 |
Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites.
Topics: Animals; Cerebral Cortex; In Vitro Techniques; Isoproterenol; Ketanserin; Kinetics; Male; Pindolol; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Subcellular Fractions; Swine | 1986 |
Stereoselective blockade at the 5-HT autoreceptor and inhibition of radioligand binding to central 5-HT recognition sites by the optical isomers of methiothepin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dibenzothiepins; Frontal Lobe; In Vitro Techniques; Ketanserin; Male; Methiothepin; Piperidines; Rats; Receptors, Serotonin; Serotonin; Stereoisomerism; Tetrahydronaphthalenes | 1986 |
Effects of MK-212 (6-chloro-2[1-piperazinyl]pyrazine) on schedule-controlled behavior and their reversal by 5-HT antagonists in the pigeon.
Topics: Animals; Columbidae; Conditioning, Operant; Cues; Generalization, Stimulus; Ketanserin; Male; Metergoline; Methysergide; Piperidines; Pyrazines; Receptors, Serotonin; Reinforcement Schedule | 1986 |
Antimyoclonic properties of S2 serotonin receptor antagonists in the rat.
Topics: 5-Hydroxytryptophan; Animals; Brain Chemistry; Butyrophenones; Cinanserin; Ketanserin; Male; Myoclonus; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists | 1986 |
Catecholamine release and potentiation of thromboxane A2 production by nicotine in the greyhound.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Pressure; Catecholamines; Dioxanes; Dogs; Epinephrine; Female; Heart Rate; Idazoxan; Imidazoles; In Vitro Techniques; Ketanserin; Male; Nicotine; Phenoxybenzamine; Piperidines; Thromboxane A2; Vasoconstriction | 1986 |
5-Carboxamidotryptamine is a selective agonist at 5-hydroxytryptamine receptors mediating vasodilatation and tachycardia in anaesthetized cats.
Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Ketanserin; Male; Methiothepin; Methysergide; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasodilation | 1986 |
Ketanserin (S2-receptor blocking agent), platelet activity and chronic alcoholism.
Topics: Adult; Alcoholism; beta-Thromboglobulin; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Serotonin Antagonists | 1986 |
Ketanserin (S2-receptor blocking agents), hypertension and chronic alcoholism.
Topics: Adult; Alcoholism; Antihypertensive Agents; Blood Pressure; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Time Factors | 1986 |
Monocrotaline pyrrole-induced cardiopulmonary toxicity is not altered by metergoline or ketanserin.
Topics: Angiotensin II; Animals; Blood Platelets; Blood Pressure; Cardiomegaly; Ergolines; Ketanserin; Lung; Male; Metergoline; Monocrotaline; Organ Size; Piperidines; Pyrrolizidine Alkaloids; Rats; Receptors, Serotonin; Serotonin | 1986 |
Ketanserin and malignant hyperthermia in pigs.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Body Temperature; Carbon Dioxide; Halothane; Heart Rate; Hydrogen-Ion Concentration; Ketanserin; Lactates; Malignant Hyperthermia; Piperidines; Potassium; Serotonin Antagonists; Succinylcholine; Swine | 1986 |
Postnatal ontogeny of dopamine D2 receptors in rat striatum.
Topics: Age Factors; Animals; Animals, Newborn; Corpus Striatum; Ketanserin; Kinetics; Mathematics; Piperidines; Rats; Receptors, Dopamine; Spiperone | 1986 |
Symposium on serotonin and cardiovascular regulation: a new approach to hypertension. Satellite symposium of the Second European Meeting on Hypertension. 9 June 1985, Milan, Italy.
Topics: Animals; Humans; Hypertension; Ketanserin; Piperidines; Serotonin; Serotonin Antagonists | 1986 |
Nitroprusside and ketanserin in the treatment of postoperative hypertension following coronary artery bypass grafting: a haemodynamic and ventilatory comparison.
Topics: Blood Pressure; Coronary Artery Bypass; Female; Ferricyanides; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Nitroprusside; Piperidines; Postoperative Complications; Pulmonary Artery; Vascular Resistance | 1986 |
Potentiation of vasoconstrictor responses to serotonin in the limb of atherosclerotic monkeys.
Topics: Animals; Arteriosclerosis; Hindlimb; Hypercholesterolemia; Ketanserin; Macaca fascicularis; Methysergide; Piperidines; Serotonin; Vasoconstriction | 1986 |
Serotonin and the blood vessel wall.
Topics: Animals; Blood Platelets; Heart; Hypertension; Ketanserin; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred SHR; Serotonin; Vasoconstriction; Vasodilation | 1986 |
Serotonin and cardiovascular regulation: a new approach to hypertension.
Topics: Cardiovascular Diseases; Drug Therapy, Combination; Humans; Hypertension; Ketanserin; Piperidines; Serotonin | 1986 |
Augmentation of vasoconstrictor responses to serotonin by acute and chronic factors: inhibition by ketanserin.
Topics: Animals; Drug Synergism; Ketanserin; Norepinephrine; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Sheep; Vasoconstriction; Vasodilation | 1986 |
Renal effects of ketanserin in essential hypertension.
Topics: Adult; Angiotensins; Female; Glomerular Filtration Rate; Humans; Hypertension; Ketanserin; Kidney; Male; Middle Aged; Piperidines; Renin | 1986 |
Regional haemodynamics and antihypertensive effects during long-term ketanserin treatment.
Topics: Female; Hemodynamics; Humans; Hypertension; Ketanserin; Long-Term Care; Male; Middle Aged; Piperidines | 1986 |
Contractions of isolated canine coronary arteries resistant to S2-serotonergic blockade.
Topics: Angiotensin II; Animals; Blood Platelets; Cocaine; Coronary Vessels; Cyproheptadine; Dibenzothiepins; Dinoprost; Dogs; Drug Resistance; Endothelium; Femoral Artery; In Vitro Techniques; Ketanserin; Methiothepin; Piperidines; Potassium; Prostaglandins F; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sympathetic Nervous System; Vasoconstriction | 1986 |
Receptor-mediated effects of serotonin and 5-methoxytryptamine on noradrenaline release in the rat vena cava and in the heart of the pithed rat.
Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Decerebrate State; Desipramine; Electric Stimulation; Heart; Heart Rate; Ketanserin; Male; Myocardium; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Tryptamines; Vagotomy; Vena Cava, Inferior | 1986 |
Effects of ketanserin, a selective 5-HT2 serotonergic antagonist, on the secondary recruitment of human platelets in vitro.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Blood Platelets; Collagen; Epinephrine; Humans; Ketanserin; Kinetics; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1986 |
Binding sites for [3H]dopamine and dopamine-antagonists on cultured astrocytes of rat striatum and spinal cord: an autoradiographic study.
Topics: Animals; Astrocytes; Autoradiography; Binding Sites; Cells, Cultured; Corpus Striatum; Domperidone; Dopamine; Dopamine Antagonists; Flupenthixol; Ketanserin; Piperidines; Rats; Spinal Cord; Spiperone; Stereoisomerism; Tritium | 1986 |
A unique serotonin receptor in choroid plexus is linked to phosphatidylinositol turnover.
Topics: Animals; Cerebral Cortex; Choroid Plexus; In Vitro Techniques; Ketanserin; Mianserin; Phosphatidylinositols; Piperidines; Rats; Receptors, Serotonin; Spiperone | 1986 |
Continuous inhibition of the platelet S2-serotonergic receptors during the long term administration of ketanserin.
Topics: Blood Platelets; Humans; Ketanserin; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin | 1986 |
Serotonin receptors in the human brain. II. Characterization and autoradiographic localization of 5-HT1C and 5-HT2 recognition sites.
Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Cerebral Cortex; Choroid Plexus; Ergolines; Female; Humans; Ketanserin; Male; Membranes; Middle Aged; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tissue Distribution; Tritium | 1986 |
The effect of ketanserin on hypoxia-induced vasoconstriction in isolated lungs.
Topics: Animals; Hypoxia; In Vitro Techniques; Ketanserin; Lung; Perfusion; Piperidines; Pulmonary Circulation; Rats; Rats, Inbred Strains; Vasoconstriction | 1986 |
Cardiovascular effects of ketanserin in conscious rabbits.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension, Renovascular; Injections, Intravenous; Ketanserin; Male; Norepinephrine; Piperidines; Rabbits; Renin; Serotonin Antagonists | 1986 |
Regional and selective changes in blood flow of the feline small intestine induced by endoluminal serotonin.
Topics: Animals; Atropine; Cats; Intestinal Mucosa; Jejunum; Ketanserin; Male; Microspheres; Perfusion; Piperidines; Receptors, Muscarinic; Receptors, Serotonin; Regional Blood Flow; Serotonin | 1986 |
Peri-operative management of carcinoid syndrome using ketanserin.
Topics: Aged; Antihypertensive Agents; Embolization, Therapeutic; Female; Hepatic Artery; Humans; Hypertension; Intraoperative Period; Ketanserin; Malignant Carcinoid Syndrome; Piperidines | 1986 |
Effects of noradrenaline, serotonin, and selected antagonists on the vascular smooth muscle of normal and dystrophic chickens.
Topics: Animals; Chickens; Dose-Response Relationship, Drug; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Muscular Dystrophy, Animal; Norepinephrine; Organ Size; Piperidines; Prazosin; Reference Values; Serotonin; Serotonin Antagonists; Tetrodotoxin | 1986 |
Serotonin, norepinephrine, and histamine mediation of endothelial cell barrier function in vitro.
Topics: Animals; Aorta; Cattle; Cell Line; Cells, Cultured; Diffusion; Diphenhydramine; Endothelium; Histamine; Ketanserin; Norepinephrine; Phenoxybenzamine; Piperidines; Propranolol; Serotonin; Serum Albumin, Bovine; Trypan Blue | 1986 |
[3H]ketanserin (serotonin type 2) binding increases in rat cortex following basal forebrain lesions with ibotenic acid.
Topics: Animals; Cerebral Cortex; Choline O-Acetyltransferase; Diencephalon; Frontal Lobe; Hippocampus; Ibotenic Acid; Ketanserin; Male; Oxazoles; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Telencephalon | 1986 |
Comparative effects of ketanserin, atropine and methysergide on the gastrointestinal effects of hyperserotoninemia in the awake dog.
Topics: Animals; Atropine; Digestive System; Dogs; Gastrointestinal Motility; Ketanserin; Methysergide; Piperidines; Receptors, Serotonin; Serotonin; Water-Electrolyte Balance | 1986 |
The influence of ketanserin on hemostasis in vitro.
Topics: Adenosine Diphosphate; Adult; Blood Coagulation; Collagen; Epinephrine; Female; Fibrinolysis; Hemostasis; Humans; In Vitro Techniques; Ketanserin; Male; Piperidines; Platelet Aggregation; Serotonin Antagonists | 1986 |
Cold hands after exposure to arsenic or vibrating tools: effects of ketanserin on finger blood pressure and skin temperature.
Topics: Administration, Oral; Adult; Arsenic Poisoning; Blood Pressure; Double-Blind Method; Hand; Humans; Injections, Intravenous; Ketanserin; Male; Middle Aged; Piperidines; Random Allocation; Raynaud Disease; Regional Blood Flow; Skin Temperature; Vibration | 1986 |
Comparisons between the in vitro binding of two substituted benzamides and two butyrophenones to dopamine-D2 receptors in the rat striatum.
Topics: Animals; Benzamides; Butyrophenones; Corpus Striatum; Domperidone; In Vitro Techniques; Ketanserin; Kinetics; Male; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride | 1986 |
Intrapartum treatment of preeclamptic hypertension by ketanserin.
Topics: Blood Pressure; Female; Fetal Heart; Heart Rate; Humans; Hypertension; Ketanserin; Obstetric Labor Complications; Piperidines; Pre-Eclampsia; Pregnancy; Uterine Contraction | 1986 |
The increase in testicular vascular permeability induced by human chorionic gonadotrophin involves 5-hydroxytryptamine and possibly oestrogens, but not testosterone, prostaglandins, histamine or bradykinin.
Topics: Aminoglutethimide; Androstatrienes; Animals; Aromatase Inhibitors; Bradykinin; Capillary Permeability; Chorionic Gonadotropin; Dihydrotestosterone; Estrogens; Histamine; Ketanserin; Kinetics; Male; Piperidines; Prostaglandins; Rats; Rats, Inbred Strains; Serotonin; Testis; Testosterone | 1986 |
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
Topics: Animals; Aorta, Thoracic; In Vitro Techniques; Jugular Veins; Ketanserin; Male; Methysergide; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Trazodone | 1986 |
Allosteric properties of 5-HT2 receptors in tracheal smooth muscle.
Topics: Allosteric Regulation; Animals; Binding, Competitive; Cattle; Female; Guinea Pigs; Ketanserin; Kinetics; Male; Methysergide; Models, Biological; Muscle Relaxation; Muscle, Smooth; Piperidines; Potassium; Receptors, Serotonin; Serotonin; Species Specificity; Trachea | 1986 |
Serotonin increases the production of inositol phosphates and mobilises calcium via the 5-HT2 receptor in A7r5 smooth muscle cells.
Topics: Animals; Aorta; Calcium; Cell Line; Cerebral Cortex; Inositol Phosphates; Ketanserin; Kinetics; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sugar Phosphates; Time Factors | 1986 |
Modulation of the serotonin S2-receptor in brain after chronic lithium.
Topics: Animals; Cerebral Cortex; Corpus Striatum; Domperidone; Ketanserin; Kinetics; Lithium; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin | 1986 |
Hypertension and tachycardia produced by inhibition of reuptake of 5-hydroxytryptamine by fluoxetine in the rat.
Topics: Adrenalectomy; Animals; Blood Pressure; Brain; Female; Fluoxetine; Heart Rate; Injections, Intraventricular; Ketanserin; Piperidines; Propylamines; Rats; Rats, Inbred Strains; Serotonin; Vagotomy | 1986 |
Does ketanserin relieve frostbite?
Topics: Adult; Frostbite; Humans; Ketanserin; Male; Piperidines; Serotonin Antagonists | 1986 |
Harmine reverses the inhibition of lordosis by the 5-HT2 antagonists pirenperone and ketanserin in the female rat.
Topics: Alkaloids; Animals; Estradiol; Female; Harmine; Ketanserin; Ovariectomy; Piperidines; Posture; Progesterone; Rats; Rats, Inbred Strains; Receptors, Serotonin; Sexual Behavior, Animal | 1986 |
Discriminative stimulus properties of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH DPAT).
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Discrimination Learning; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ketanserin; Male; Naphthalenes; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes | 1986 |
A sensitive model of venous thrombosis in rats.
Topics: Animals; Anticoagulants; Aspirin; Dipyridamole; Disease Models, Animal; Female; Heparin; Ketanserin; Piperidines; Rats; Rats, Inbred Strains; Sulfinpyrazone; Thrombophlebitis; Time Factors | 1986 |
Antithrombotics in view of thrombosis models.
Topics: Animals; Anticoagulants; Arteries; Aspirin; Dipyridamole; Female; Hydroxyethylrutoside; Ketanserin; Piperidines; Pizotyline; Prenylamine; Rats; Rats, Inbred Strains; Sulfinpyrazone; Thrombophlebitis; Thrombosis | 1986 |
Adenosine-induced contractions of the isolated rat trachea are mediated by 5-hydroxytryptamine.
Topics: Adenosine; Animals; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Trachea | 1986 |
Ketanserin and the cardiovascular system. 1. Modification of the effects of pressor amines in patients undergoing myocardial revascularisation.
Topics: Angiotensin II; Antihypertensive Agents; Cardiopulmonary Bypass; Drug Evaluation; Hemodynamics; Humans; Ketanserin; Middle Aged; Myocardial Revascularization; Norepinephrine; Phenylephrine; Piperidines | 1986 |
Thermoregulatory responses to serotonin (5-HT) receptor stimulation in the rat. Evidence for opposing roles of 5-HT2 and 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature Regulation; Ketanserin; Male; Methoxydimethyltryptamines; Pindolol; Piperidines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes | 1986 |
Regional and subcellular localization in human brain of [3H]paroxetine binding, a marker of serotonin uptake sites.
Topics: Adult; Aged; Animals; Binding, Competitive; Brain; Brain Mapping; Cerebral Cortex; Corpus Striatum; Humans; Ketanserin; Male; Middle Aged; Paroxetine; Piperidines; Putamen; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Subcellular Fractions; Synaptosomes | 1988 |
[3H]vesamicol binding in brain: autoradiographic distribution, pharmacology, and effects of cholinergic lesions.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Autoradiography; Brain; Cholinergic Fibers; Frontal Lobe; Haloperidol; Hippocampus; Image Processing, Computer-Assisted; Ketanserin; Male; Neural Pathways; Neurotransmitter Uptake Inhibitors; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains | 1988 |
Changes in cortical 5-HT2 receptors following 5-HTP and paroxetine administration in rats.
Topics: Animals; Carbidopa; Cerebral Cortex; Ketanserin; Male; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin | 1988 |
Different effects of serotonin antagonists on 3H-mianserin and 3H-ketanserin recognition sites.
Topics: Animals; Binding Sites; Cerebral Cortex; Cyclic AMP; Dibenzazepines; Ketanserin; Kinetics; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin Antagonists; Time Factors | 1985 |
Serotonin, histamine, and norepinephrine mediation of endothelial and vascular smooth muscle cell movement.
Topics: Animals; Aorta; Cattle; Cell Movement; Cells, Cultured; Depression, Chemical; Diphenhydramine; Endothelium; Histamine; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Piperidines; Propranolol; Receptors, Adrenergic, beta; Receptors, Histamine H1; Serotonin; Time Factors | 1985 |
Ketanserin without effects on basal anterior pituitary hormone secretion in healthy subjects.
Topics: Adrenocorticotropic Hormone; Adult; Blood Glucose; Growth Hormone; Humans; Hydrocortisone; Ketanserin; Luteinizing Hormone; Male; Piperidines; Pituitary Hormones, Anterior; Prolactin; Serotonin Antagonists; Thyroid Hormones; Thyrotropin | 1985 |
5-Hydroxytryptamine-stimulated inositol phospholipid hydrolysis in rat cerebral cortex slices: pharmacological characterization and effects of antidepressants.
Topics: Affinity Labels; Animals; Antidepressive Agents; Cerebral Cortex; Hydrolysis; Imipramine; Iprindole; Ketanserin; Male; Phenoxybenzamine; Phosphatidylinositols; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin | 1985 |
Role of serotonin type 2 receptors in regulation of aldosterone production.
Topics: Adrenal Glands; Aldosterone; Angiotensin II; Animals; Cosyntropin; Cyclic AMP; Cyproheptadine; Female; In Vitro Techniques; Ketanserin; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1985 |
Antihypertensive mechanism of action of ketanserin and some ketanserin analogues in the spontaneously hypertensive rat.
Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension; Ketanserin; Phenylephrine; Piperidines; Prazosin; Pyrimidines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Ritanserin; Sympathetic Nervous System | 1985 |
Serotonergic agonists stimulate inositol lipid metabolism in rabbit platelets.
Topics: Animals; Blood Platelets; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Phosphatidylinositols; Piperidines; Quipazine; Rabbits; Receptors, Serotonin; Serotonin | 1985 |
Serotonin 5-HT1 receptors mediate inhibition of cyclic AMP production in neurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Brain; Cerebral Cortex; Corpus Striatum; Cyclic AMP; Female; Fetus; Indoles; Ketanserin; Metergoline; Mice; Neurons; Piperidines; Pregnancy; Receptors, Serotonin; Tetrahydronaphthalenes; Vasoactive Intestinal Peptide | 1986 |
Central alpha-2 adrenoceptor-mediated hypertensive response to clonidine in conscious, normotensive rats.
Topics: Animals; Azepines; Blood Pressure; Brain; Cimetidine; Clonidine; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Male; Methoxamine; Oxidopamine; Piperidines; Prazosin; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1986 |
A simple 'free 3H-ligand' assay for rapid screening of hybridoma monoclonal antibodies against neurotransmitter analogs and anti-idiotype antibodies.
Topics: Animals; Antibodies, Monoclonal; Haloperidol; Hybridomas; Immunoglobulin Idiotypes; Ketanserin; Mice; Pimozide; Piperidines; Receptors, Neurotransmitter | 1986 |
Studies on the antinociceptive effect of intrathecal salmon calcitonin.
Topics: Analgesics; Animals; Benzomorphans; Calcitonin; Enkephalin, Leucine; Haloperidol; Ketanserin; Male; Methysergide; Nociceptors; Phentolamine; Piperidines; Rats; Receptors, Opioid | 1985 |
Effect of ketanserin on the in vitro regulation of aldosterone.
Topics: Adrenocorticotropic Hormone; Angiotensin II; Animals; Female; In Vitro Techniques; Ketanserin; Mineralocorticoid Receptor Antagonists; Piperidines; Potassium; Rats; Rats, Inbred Strains | 1986 |
Down regulation of serotonin-S2 receptor sites in rat brain by chronic treatment with the serotonin-S2 antagonists: ritanserin and setoperone.
Topics: Animals; Brain; Corpus Striatum; Frontal Lobe; Ketanserin; Male; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Neurotransmitter; Receptors, Serotonin; Ritanserin | 1986 |
Evidence for separate receptors that mediate parallel effects of serotonin and small cardioactive peptideB (SCPB) on adenylate cyclase in Aplysia californica.
Topics: Adenylyl Cyclases; Animals; Aplysia; Enzyme Activation; Ketanserin; Neuropeptides; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1986 |
Antagonism by methysergide of neurogenic vasoconstriction in the dog forelimb.
Topics: Animals; Dogs; Electric Stimulation; Forelimb; Ketanserin; Median Nerve; Methysergide; Phentolamine; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasoconstriction; Vasodilation | 1987 |
Serotonin receptors in the rat nucleus tractus solitarii and cardiovascular regulation.
Topics: Animals; Blood Pressure; Body Temperature; Cardiovascular Physiological Phenomena; Heart Rate; Indoles; Ketanserin; Male; Medulla Oblongata; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1986 |
Ritanserin and serotonergic mechanisms in blood pressure and fluid regulation in sheep.
Topics: Animals; Blood Pressure; Cardiac Output; Heart Rate; Hypertension; Ketanserin; Phenylephrine; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Sheep; Water-Electrolyte Balance | 1987 |
Protection with phencyclidine against inactivation of 5-HT2 receptors by sulfhydryl-modifying reagents.
Topics: Animals; Behavior, Animal; Ethylmaleimide; Ketanserin; Male; Phencyclidine; Piperidines; Rats; Rats, Inbred F344; Receptors, Serotonin; Ritanserin; Serotonin; Sulfhydryl Reagents | 1988 |
Interference of ketanserin with baroreflex control of the circulation in the conscious spontaneously hypertensive rat.
Topics: Animals; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Piperidines; Prazosin; Pressoreceptors; Rats; Rats, Inbred SHR; Ritanserin; Serotonin Antagonists | 1988 |
Habituation of tactile startle is altered by drugs acting on serotonin-2 receptors.
Topics: Animals; Cinanserin; Cyproheptadine; Habituation, Psychophysiologic; Ketanserin; Male; Piperidines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reference Values; Reflex, Startle; Ritanserin; Serotonin; Serotonin Antagonists; Touch | 1988 |
Adrenergic and serotoninergic mechanisms in human hand arteries and veins studied by fluorescence histochemistry and in vitro pharmacology.
Topics: Arteries; Binding, Competitive; Biogenic Amines; Epinephrine; Female; Hand; Humans; Isoproterenol; Ketanserin; Male; Microscopy, Fluorescence; Muscle Contraction; Norepinephrine; Phentolamine; Piperidines; Receptors, Adrenergic; Serotonin; Sympathetic Nervous System; Veins | 1985 |
Studies into the dual effects of serotonergic pharmacological agents on female sexual behaviour in the rat: preliminary evidence that endogenous 5HT is stimulatory.
Topics: 5-Hydroxytryptophan; Adrenalectomy; Alanine; Animals; Castration; Cinanserin; Female; Ketanserin; Metergoline; Methysergide; Mianserin; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal; Zimeldine | 1985 |
Adenine nucleotides, serotonin, and endothelium-dependent relaxations to platelets.
Topics: Adenine Nucleotides; Animals; Apyrase; Blood Platelets; Coronary Vessels; Dogs; Endothelium; Female; Ketanserin; Male; Meclofenamic Acid; Methiothepin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists; Vasoconstriction | 1985 |
Pharmacological properties of mechanical responses of the rat oesophageal muscularis mucosae to vagal and field stimulation.
Topics: Animals; Dioxolanes; Electric Stimulation; Esophagus; Hexamethonium Compounds; In Vitro Techniques; Ketanserin; Male; Morphine; Muscle Contraction; Muscle, Smooth; N-Methylscopolamine; Naloxone; Piperidines; Rats; Rats, Inbred Strains; Scopolamine Derivatives; Serotonin; Tetrodotoxin; Tubocurarine; Vagus Nerve | 1985 |
Rapid intracellular release of calcium in human platelets by stimulation of 5-HT2-receptors.
Topics: Aminoquinolines; Blood Platelets; Calcium; Cytoplasm; Gallic Acid; Humans; In Vitro Techniques; Ketanserin; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1985 |
N-(3-acetylaminophenyl)piperazine hydrochloride (BEA 1654), a putative 5-HT1 agonist, causes constriction of arteriovenous anastomoses and dilatation of arterioles.
Topics: Animals; Arterioles; Arteriovenous Anastomosis; Carotid Arteries; Hemodynamics; In Vitro Techniques; Ketanserin; Phentolamine; Piperazines; Piperidines; Rats; Receptors, Serotonin; Regional Blood Flow; Swine; Vasoconstriction; Vasodilation | 1985 |
Verapamil, an antagonist at 5-hydroxytryptamine receptors of human blood platelets.
Topics: Adenosine Diphosphate; Binding, Competitive; Blood Platelets; Cerebral Cortex; Gallopamil; Humans; In Vitro Techniques; Ketanserin; Membranes; Piperidines; Receptors, Serotonin; Spiperone; Verapamil | 1985 |
Differentiation between the stimulus effects of l-5-hydroxytryptophan and LSD.
Topics: 5-Hydroxytryptophan; Animals; Benserazide; Cues; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains | 1985 |
A paradox: the 5-HT2-receptor antagonist ketanserin restores the 5-HT-induced contraction depressed by methysergide in large coronary arteries of calf. Allosteric regulation of 5-HT2-receptors.
Topics: Allosteric Regulation; Animals; Cattle; Coronary Vessels; In Vitro Techniques; Ketanserin; Methysergide; Models, Biological; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vasoconstriction | 1985 |
Ketanserin causes surmountable antagonism of 5-hydroxytryptamine-induced contractions of large coronary arteries of dog.
Topics: Animals; Coronary Vessels; Dogs; Female; In Vitro Techniques; Ketanserin; Male; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vasoconstriction | 1985 |
Cardiovascular and blood gas responses to ketanserin in canine pulmonary edema induced by oleic acid.
Topics: Animals; Blood Pressure; Carbon Dioxide; Cardiac Output; Dogs; Hemodynamics; Hydrogen-Ion Concentration; Ketanserin; Lung; Oleic Acid; Oleic Acids; Oxygen; Piperidines; Pulmonary Edema; Serotonin; Serotonin Antagonists; Vascular Resistance | 1985 |
Estradiol-induced increase of specific [3H]ketanserin binding sites on rat uterine membranes.
Topics: Animals; Binding Sites; Castration; Estradiol; Female; In Vitro Techniques; Ketanserin; Membranes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tritium; Uterus | 1985 |
Characterization of 5-hydroxytryptamine binding sites in the plasma membrane of pig blood platelets.
Topics: Animals; Binding Sites; Blood Platelets; Brain; Ketanserin; Lysergic Acid Diethylamide; Piperidines; Platelet Aggregation; Serotonin; Sodium; Swine | 1985 |
Complete conversion of brain D2 dopamine receptors from the high- to the low-affinity state for dopamine agonists, using sodium ions and guanine nucleotide.
Topics: Animals; Apomorphine; Brain; Guanine Nucleotides; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Tetrahydronaphthalenes; Tritium | 1985 |
A calcium-dependent reversible permeability increase in microvessels in frog brain, induced by serotonin.
Topics: Animals; Blood-Brain Barrier; Brain; Calcium; Capillary Permeability; Dose-Response Relationship, Drug; Electric Conductivity; Endothelium; Ketanserin; Piperidines; Rana temporaria; Serotonin; Serotonin Antagonists; Verapamil | 1985 |
The effect of prolonged treatment with tricyclic antidepressants on the actions of 5-hydroxytryptamine in the hippocampal slice of the rat.
Topics: Animals; Cyproheptadine; Desipramine; Evoked Potentials; Hippocampus; Imipramine; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin | 1985 |
Serotonin antagonist pirenperone inhibits sexual behavior in the male rat: attenuation by quipazine.
Topics: Animals; Dose-Response Relationship, Drug; Fenclonine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Serotonin Antagonists; Sexual Behavior, Animal; Tranquilizing Agents | 1985 |
Interaction of 5-hydroxytryptamine and ketanserin in rat vas deferens subjected to low frequency field stimulation.
Topics: Animals; Drug Interactions; Electric Stimulation; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth; Piperidines; Prazosin; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Vas Deferens | 1985 |
Effects of ketanserin on neuronal responses to serotonin in the prefrontal cortex, lateral geniculate and dorsal raphe nucleus.
Topics: Animals; Decerebrate State; Electrophysiology; Frontal Lobe; gamma-Aminobutyric Acid; Geniculate Bodies; Ketanserin; Male; Norepinephrine; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Tryptamines | 1985 |
Anti-aversive role of serotonin in the dorsal periaqueductal grey matter.
Topics: Animals; Avoidance Learning; Electric Stimulation; Electrodes, Implanted; Injections; Ketanserin; Male; Metergoline; Methoxydimethyltryptamines; Periaqueductal Gray; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Zimeldine | 1985 |
Serotonin-induced platelet aggregation in whole blood and the effects of ketanserin and mepyramine.
Topics: Aminopyridines; Dose-Response Relationship, Drug; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Serotonin; Time Factors | 1985 |
Tryptamine-induced vasoconstrictor responses in rat caudal arteries are mediated predominantly via 5-hydroxytryptamine receptors.
Topics: Animals; Arteries; In Vitro Techniques; Ketanserin; Male; Methysergide; Monoamine Oxidase Inhibitors; Phentolamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tryptamines; Vasoconstriction | 1985 |
Localization of 11C-radiopharmaceuticals in the Greene melanoma of hamsters.
Topics: Animals; Benzodiazepinones; Carbon Radioisotopes; Chlorpromazine; Cricetinae; Flumazenil; Flunitrazepam; Gallium Radioisotopes; Isotope Labeling; Ketanserin; Melanoma; Mesocricetus; Methionine; Neoplasm Transplantation; Pimozide; Piperidines; Quinuclidinyl Benzilate; Radionuclide Imaging; Tissue Distribution | 1985 |
Is waning of a 5-hydroxytryptamine (5-HT)-mediated syndrome due to 5-HT2 receptor down-regulation?
Topics: Animals; Cerebral Cortex; Ketanserin; Male; Myoclonus; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Syndrome; Time Factors; Tritium | 1985 |
Platelet-mediated vascular permeability in the rat: a predominant role for 5-hydroxytryptamine.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Capillary Permeability; Dose-Response Relationship, Drug; Histamine; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Suprofen; Thrombin | 1985 |
Raynaud's disease.
Topics: Antihypertensive Agents; Child; Dinoprostone; Epoprostenol; Female; Humans; Ketanserin; Male; Nifedipine; Nitroprusside; Phenoxybenzamine; Piperidines; Prostaglandins E, Synthetic; Raynaud Disease | 1985 |
Excitatory 5-hydroxytryptamine receptors in the cat urinary bladder are of the M- and 5-HT2-type.
Topics: Animals; Atropine; Cats; Cyproheptadine; Dimethylphenylpiperazinium Iodide; Drug Interactions; Female; Guanethidine; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Urinary Bladder | 1985 |
Simultaneous determination of ketanserin and ketanserinol in biological fluids using ion-pair liquid chromatography and fluorometric detection.
Topics: Aged; Antihypertensive Agents; Body Fluids; Chromatography, High Pressure Liquid; Female; Humans; Hydrogen-Ion Concentration; Ketanserin; Kinetics; Piperidines; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet | 1985 |
In vivo binding of 125I-LSD to serotonin 5-HT2 receptors in mouse brain.
Topics: Animals; Binding, Competitive; Brain; Cinanserin; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Mice; Piperidines; Receptors, Serotonin; Spiperone; Time Factors; Tissue Distribution | 1985 |
Binding of the putative anxiolytic TVX Q 7821 to hippocampal 5-hydroxytryptamine (5-HT) recognition sites.
Topics: Animals; Binding, Competitive; Cattle; Hippocampus; Ketanserin; Kinetics; Membranes; Piperidines; Pyrimidines; Rats; Receptors, Serotonin | 1985 |
Potentiation of motoneurone excitability by combined administration of 5-HT agonist and TRH analogue.
Topics: Animals; Anterior Horn Cells; Drug Synergism; Female; Fenclonine; Ketanserin; Methoxydimethyltryptamines; Methysergide; Motor Neurons; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Serotonin; Stimulation, Chemical; Thyrotropin-Releasing Hormone | 1985 |
A facilitatory role for serotonin in the sexual behavior of the female rat.
Topics: Animals; Castration; Estradiol; Female; Ketanserin; Methysergide; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Sexual Behavior, Animal; Spiperone | 1985 |
Serotonin-induced contraction of canine saphenous vein: mediation by 5-HT1 receptors.
Topics: Animals; Clonidine; Dogs; Drug Interactions; Emetics; In Vitro Techniques; Ketanserin; Mianserin; Muscle Contraction; Naphthols; Piperidines; Receptors, Serotonin; Saphenous Vein; Serotonin; Yohimbine | 1985 |
Cardiovascular effects of ketanserin in closed-chest anesthetized dogs.
Topics: Anesthesia; Animals; Blood Pressure; Dogs; Electrocardiography; Female; Heart Rate; Hemodynamics; Ketanserin; Male; Piperidines; Respiration; Serotonin; Serotonin Antagonists; Stroke Volume; Vascular Resistance | 1985 |
Two types of receptors for 5-hydroxytryptamine on the cholinergic nerves of the guinea-pig myenteric plexus.
Topics: Acetylcholine; Animals; Binding, Competitive; Cocaine; Electric Stimulation; Female; Guinea Pigs; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Myenteric Plexus; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes | 1985 |
[Ketanserin in the treatment of ischemic disease of the lower extremities].
Topics: Female; Humans; Ischemia; Ketanserin; Leg; Male; Middle Aged; Piperidines; Regional Blood Flow; Serotonin Antagonists | 1985 |
Selective 5-HT2 receptor blockade in exercise-induced asthma.
Topics: Adolescent; Adult; Asthma; Asthma, Exercise-Induced; Bronchi; Child; Humans; Ketanserin; Piperidines; Receptors, Serotonin; Sleep Stages | 1985 |
Bioavailability and pharmacokinetics of ketanserin in elderly subjects.
Topics: Age Factors; Aged; Biological Availability; Female; Half-Life; Humans; Ketanserin; Kinetics; Male; Middle Aged; Piperidines; Serotonin Antagonists | 1985 |
Evidence for serotoninergic control of exercise-induced prolactin secretion.
Topics: Adult; Heart Rate; Humans; Ketanserin; Male; Physical Exertion; Piperidines; Prolactin; Serotonin; Time Factors | 1985 |
Effect of serotonin on the motility of smooth muscles in teats of lactating cows.
Topics: Animals; Cattle; Female; Ketanserin; Lactation; Mammary Glands, Animal; Methysergide; Mianserin; Milk Ejection; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Piperidines; Pregnancy; Serotonin; Serotonin Antagonists | 1985 |
Changes of the striatal 3H-spiperone binding 3-6 weeks after nigrostriatal denervation and after two years.
Topics: Animals; Butyrophenones; Corpus Striatum; Denervation; Haloperidol; Hydroxydopamines; Ketanserin; Kinetics; Male; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Spiperone; Substantia Nigra; Time Factors | 1985 |
Target size analysis of serotonin 5-HT1 and 5-HT2 receptors in bovine brain membranes.
Topics: Animals; Binding, Competitive; Brain Chemistry; Cattle; Caudate Nucleus; Cerebral Cortex; Freeze Drying; Ketanserin; Molecular Weight; Piperidines; Radioligand Assay; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Synaptic Membranes | 1985 |
Attenuation of morphine analgesia by the S2 antagonists, pirenperone and ketanserin.
Topics: Analgesia; Animals; Dose-Response Relationship, Drug; Ketamine; Ketanserin; Male; Morphine; Piperidines; Rats; Reaction Time; Receptors, Serotonin; Serotonin Antagonists | 1988 |
Opposite regulation of serotonin-S2 and dopamine-D2 receptors in rat brain following chronic receptor blockade.
Topics: Animals; Apomorphine; Behavior, Animal; Corpus Striatum; Diazepam; Dopamine Antagonists; Frontal Lobe; Gene Expression Regulation; Ketanserin; Male; Models, Biological; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin Antagonists; Tryptamines | 1987 |
Different temporal effects of serotonergic antagonists on passive avoidance retention.
Topics: Animals; Avoidance Learning; Ketanserin; Male; Memory; Mianserin; Mice; Piperidines; Receptors, Serotonin; Retention, Psychology; Serotonin Antagonists; Time Factors | 1987 |
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Frontal Lobe; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1986 |
Ketanserin and pirenperone attenuate acute morphine withdrawal in rats.
Topics: Animals; Body Temperature; Conditioning, Operant; Ketanserin; Male; Morphine Dependence; Piperidines; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome | 1986 |
Photoaffinity probes for serotonin and histamine receptors. Synthesis and characterization of two azide analogues of ketanserin.
Topics: 4-Aminobenzoic Acid; Affinity Labels; Animals; Azides; Binding, Competitive; Cerebellum; Cerebral Cortex; Guinea Pigs; Histamine Antagonists; Ketanserin; Kinetics; Lysergic Acid Diethylamide; Photochemistry; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Receptors, Serotonin; Serotonin Antagonists; Ultraviolet Rays | 1985 |
Photoaffinity labelling of serotonin-S2 receptors with 7-azidoketanserin.
Topics: Affinity Labels; Animals; Azides; Female; Frontal Lobe; In Vitro Techniques; Ketanserin; Light; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1985 |
Differential photoaffinity labelling of serotonin-S2 receptors and histamine-H1 receptors using 7-azidoketanserin.
Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Butyrophenones; Cerebellum; Cerebral Cortex; Female; Guinea Pigs; Ketanserin; Photolysis; Piperidines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Serotonin; Spiperone | 1985 |
[Reciprocal potentiation of the bronchoconstrictor activity of histamine and 5-hydroxytryptamine in the guinea pig].
Topics: Animals; Bronchi; Drug Synergism; Female; Guinea Pigs; Histamine; Histamine Antagonists; Ketanserin; Male; Piperidines; Serotonin; Serotonin Antagonists | 1984 |
Acute effects of antagonist of S2-receptors.
Topics: Adult; Blood Pressure; Drug Evaluation; Female; Humans; Hydroxyindoleacetic Acid; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Serotonin Antagonists; Vanilmandelic Acid | 1984 |
Neurotransmitter receptors and monoamine metabolites in the brains of patients with Alzheimer-type dementia and depression, and suicides.
Topics: Aged; Aging; Alzheimer Disease; Binding, Competitive; Biogenic Amines; Brain; Choline O-Acetyltransferase; Depressive Disorder; Female; Humans; Hydroxyindoleacetic Acid; Ketanserin; Male; Middle Aged; Piperidines; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Serotonin; Serotonin; Sex Factors; Suicide | 1984 |
Regional and cortical laminar distributions of serotonin S2, benzodiazepine, muscarinic, and dopamine D2 receptors in human brain.
Topics: Adult; Aged; Brain; Cerebral Cortex; Diazepam; Humans; Ketanserin; Male; Middle Aged; Piperidines; Quinuclidinyl Benzilate; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Serotonin; Spiperone; Tissue Distribution | 1984 |
Colonic secretion mediated by prostaglandin E2 and 5-hydroxytryptamine may contribute to diarrhea due to morphine withdrawal in the rat.
Topics: Animals; Atropine; Clonidine; Colon; Cyclic AMP; Diarrhea; Dinoprostone; Female; Humans; Indomethacin; Ketanserin; Morphine Dependence; Naloxone; Piperidines; Prostaglandins E; Rats; Rats, Inbred Strains; Serotonin; Substance Withdrawal Syndrome | 1984 |
Assessment of sodium-potassium ATPase activity in human erythrocytes in vitro.
Topics: Erythrocytes; Humans; In Vitro Techniques; Ketanserin; Male; Ouabain; Piperidines; Rubidium; Sodium; Sodium-Potassium-Exchanging ATPase | 1984 |
Alpha 1 adrenergic receptors in the porcine pituitary neurointermediate lobe: detection with [3H]ketanserin.
Topics: Animals; Binding, Competitive; Brain; Cinanserin; In Vitro Techniques; Ketanserin; Kinetics; Piperidines; Pituitary Gland; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Swine | 1984 |
The specificity of ketanserin in the inhibition of serotonin-induced steroidogenesis in the rat adrenal zona glomerulosa.
Topics: Adrenal Cortex; Aldosterone; Animals; Corticosterone; Cyclic AMP; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Methysergide; Piperidines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1984 |
Acute blood-pressure-lowering effect of ketanserin.
Topics: Aged; Antihypertensive Agents; Blood Pressure; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Serotonin Antagonists | 1981 |
5-HT2-receptor blockade in the treatment of heart failure. A preliminary study.
Topics: Adult; Aged; Blood Pressure; Cardiac Output; Heart Failure; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Piperidines; Platelet Aggregation; Pulmonary Wedge Pressure; Serotonin Antagonists; Stroke Volume; Vascular Resistance; Vasoconstriction | 1981 |
Vascular effects of ketanserin (R 41 468), a novel antagonist of 5-HT2 serotonergic receptors.
Topics: Adrenergic alpha-Agonists; Animals; Arteries; Blood Pressure; Calcium; Dogs; Guinea Pigs; Hypertension; In Vitro Techniques; Ketanserin; Kidney; Male; Muscle, Smooth, Vascular; Norepinephrine; Organ Specificity; Piperidines; Rats; Serotonin Antagonists; Species Specificity; Stomach; Vasoconstriction; Veins | 1981 |
Solubilized serotonin receptors from rat and dog brain. Selective labelling with [3H]ketanserin.
Topics: Animals; Antipsychotic Agents; Binding, Competitive; Brain; Butyrophenones; Dogs; Isonipecotic Acids; Ketanserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Solubility; Species Specificity; Spiperone; Time Factors | 1982 |
Cardiovascular effects in the rat of ketanserin, a novel 5-hydroxytryptamine receptor blocking agent.
Topics: Animals; Blood Pressure; Heart Rate; Hemodynamics; Injections, Intraventricular; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Time Factors | 1982 |
Ketanserin--a novel antihypertensive drug?
Topics: Animals; Antihypertensive Agents; In Vitro Techniques; Ketanserin; Muscle, Smooth; Piperidines; Rats; Receptors, Histamine H2 | 1982 |
Ketanserin: a selective serotonin antagonist.
Topics: Cardiovascular System; Humans; Hypertension; Ketanserin; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1982 |
Mechanism of action of ketanserin.
Topics: Animals; Antihypertensive Agents; Humans; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Spiperone | 1982 |
Ketanserin: a selective antagonist of 5-HT2 serotoninergic receptors.
Topics: Animals; Binding Sites; Ketanserin; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists | 1983 |
Preliminary studies of human cortical 5-HT2 receptors and their involvement in schizophrenia and neuroleptic drug action.
Topics: Antipsychotic Agents; Cerebral Cortex; Humans; Ketanserin; Piperidines; Receptors, Serotonin; Schizophrenia; Spiperone; Substrate Specificity | 1983 |
Yohimbine and rauwolscine inhibit 5-hydroxytryptamine-induced contraction of large coronary arteries of calf through blockade of 5 HT2 receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Cattle; Coronary Vessels; Drug Combinations; Ketanserin; Muscle Contraction; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Yohimbine | 1983 |
Unusual acute effects of antidepressants and neuroleptics on S2-serotonergic receptors.
Topics: Amoxapine; Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Fenclonine; Frontal Lobe; Ketanserin; Loxapine; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone | 1983 |
Influence of ketanserin, an antihypertensive agent with specific 5-HT2-receptor blocking activity, on intracranial pressure.
Topics: Animals; Blood Gas Analysis; Cardiac Output; Cerebral Cortex; Dogs; Female; Hemodynamics; Histamine H2 Antagonists; Intermittent Positive-Pressure Ventilation; Intracranial Pressure; Ketanserin; Male; Piperidines | 1984 |
Ketanserin in intermittent claudication.
Topics: Appetite; Blood Pressure; Body Weight; Humans; Intermittent Claudication; Ketanserin; Piperidines | 1984 |
Serotoninergic control of somatostatin and gastrin release from the isolated rat stomach.
Topics: Animals; Gastric Mucosa; Gastrins; In Vitro Techniques; Ketanserin; Male; Methysergide; Perfusion; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Receptors, Serotonin; Serotonin; Somatostatin | 1984 |
The 5-hydroxytryptamine antagonist ketanserin inhibits the vasoconstrictor activity of per-operative CSF, from subarachnoid haemorrhage patients, on isolated tissues.
Topics: Adult; Aged; Animals; Female; Humans; Hydroxyindoleacetic Acid; Intracranial Aneurysm; Intraoperative Complications; Ischemic Attack, Transient; Ketanserin; Male; Middle Aged; Piperidines; Postoperative Complications; Rats; Rupture, Spontaneous; Serotonin; Serotonin Antagonists; Subarachnoid Hemorrhage; Vasoconstriction | 1983 |
[Thermogenic shivering in the anesthetized rat].
Topics: Animals; Body Temperature Regulation; Ketanserin; Pentobarbital; Piperidines; Rats; Shivering | 1982 |
On the neurotoxicity of chlordecone: a role for gamma-aminobutyric acid and serotonin.
Topics: Acetylcholine; Animals; Binding Sites; Brain; Chlordecone; gamma-Aminobutyric Acid; Insecticides; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Spiperone | 1984 |
Serotonin receptor changes in dementia of the Alzheimer type.
Topics: Aged; Alzheimer Disease; Choline O-Acetyltransferase; Female; Humans; Hydroxyindoleacetic Acid; Ketanserin; Male; Piperidines; Postmortem Changes; Receptors, Serotonin; Serotonin; Somatostatin; Tissue Distribution | 1984 |
Inhibition of 5-hydroxytryptamine-induced and -amplified human platelet aggregation by ketanserin (R 41 468), a selective 5-HT2-receptor antagonist.
Topics: beta-Thromboglobulin; Blood Platelets; Blood Proteins; Humans; In Vitro Techniques; Ketanserin; Malondialdehyde; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists; Thromboxane B2 | 1982 |
[Effect of ketanserin on various properties of pentobarbital in rats].
Topics: Animals; Body Temperature; Drug Interactions; Ketanserin; Pentobarbital; Piperidines; Rats; Rats, Inbred Strains; Sleep | 1983 |
Stimulation by serotonin of 40 kDa and 20 kDa protein phosphorylation in human platelets.
Topics: Blood Platelets; Blood Proteins; Humans; Ketanserin; Molecular Weight; Myosin-Light-Chain Kinase; Phosphatidic Acids; Phosphorylation; Piperidines; Protein Kinase C; Protein Kinases; Receptors, Serotonin; Serotonin | 1984 |
The role of serotonin (5-HT) in the control of TSH and prolactin release in euthyroid subjects as assessed by the administration of ketanserin (5-HT2 antagonist) and zimelidine (5-HT re-uptake inhibitor).
Topics: Female; Humans; Ketanserin; Male; Piperidines; Prolactin; Serotonin; Serotonin Antagonists; Thyrotropin; Thyrotropin-Releasing Hormone; Thyroxine; Zimeldine | 1984 |
Prolongation of rat tail bleeding time by ketanserin: mechanisms of action.
Topics: Animals; Bleeding Time; Blood Coagulation; Blood Platelets; Blood Pressure; Drug Interactions; Fenclonine; Ketanserin; Male; Metergoline; Piperidines; Platelet Aggregation; Prazosin; Rats; Serotonin; Serotonin Antagonists; Sympatholytics; Tail | 1984 |
Receptor binding profile of R 41 468, a novel antagonist at 5-HT2 receptors.
Topics: Animals; Brain; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Receptors, Adrenergic, alpha; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Serotonin; Serotonin Antagonists | 1981 |
Characterization of the antihypertensive properties of ketanserin (R 41 468) in rats.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Ketanserin; Male; Methoxamine; Piperidines; Rats; Receptors, Adrenergic, alpha; Receptors, Serotonin; Vasopressins | 1982 |
Principles of therapy for congestive heart failure.
Topics: Calcium; Calcium Channel Blockers; Calmodulin; Cardiotonic Agents; Clonidine; Cyclic AMP; Cytosol; Digitalis Glycosides; Diuretics; Heart Failure; Humans; Ketanserin; Models, Cardiovascular; Muscle, Smooth, Vascular; Myocardium; Myosins; Piperidines; Receptors, Adrenergic, alpha; Vasodilator Agents | 1983 |
Modulation of brain S2 serotonin receptors by lithium, sodium and potassium chloride.
Topics: Animals; Binding, Competitive; Brain; Chlorides; Dose-Response Relationship, Drug; Female; Ketanserin; Lithium; Lithium Chloride; Piperidines; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium Chloride | 1983 |
Mechanism of antihypertensive action of ketanserin in man.
Topics: Antihypertensive Agents; Blood Pressure; Humans; Ketanserin; Piperidines; Receptors, Adrenergic, alpha | 1983 |
Evidence for an alpha-1 receptor-mediated central sympathoinhibitory action of ketanserin.
Topics: Animals; Blood Pressure; Brain; Cats; Clonidine; Heart Rate; Ketanserin; Piperidines; Receptors, Adrenergic, alpha; Serotonin Antagonists; Sympathetic Nervous System; Sympatholytics | 1984 |
Comparison of iprindole, imipramine and mianserin action on brain serotonergic and beta adrenergic receptors.
Topics: Animals; Axons; Brain; Cyclic AMP; Dibenzazepines; Imipramine; Indoles; Iprindole; Ketanserin; Male; Mianserin; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin | 1984 |
Tryptaminergic receptors in the bovine pulmonary vasculature: effects of ketanserin.
Topics: Animals; Cattle; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pulmonary Artery; Pulmonary Veins; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists | 1984 |
Autoradiographic mapping of spirodecanone binding-sites in the hippocampal region of the rat. Evidence for a localization on intrinsic neurons.
Topics: Animals; Autoradiography; Binding, Competitive; Brain Mapping; Butyrophenones; Haloperidol; Hippocampus; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Serotonin; Spiperone; Tetrahydronaphthalenes | 1984 |
Effect of ketanserin, an inhibitor of 5-HT2 receptors, on the aldosterone-stimulating action of metoclopramide.
Topics: Adolescent; Adult; Aldosterone; Humans; Ketanserin; Kinetics; Male; Metoclopramide; Piperidines; Potassium; Prolactin; Receptors, Serotonin; Renin; Serotonin Antagonists | 1983 |
Role and localization of serotonin2 (S2)-receptor-binding sites: effects of neuronal lesions.
Topics: Animals; Catecholamines; Cerebral Cortex; Dogs; Female; Guinea Pigs; Kainic Acid; Ketanserin; Kinetics; Male; Nerve Tissue Proteins; Neurons; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Serotonin; Stereotaxic Techniques; Subcellular Fractions | 1983 |
The role of 5-hydroxytryptamine in the feline response to intravenous infusion of live E. coli.
Topics: Animals; Blood Pressure; Cats; Escherichia coli Infections; Hemodynamics; Intestines; Ketanserin; Lung; Piperidines; Premedication; Regional Blood Flow; Shock, Septic; Time Factors; Vascular Resistance | 1983 |
The effect of a selective 5-HT2 antagonist, ketanserin, on the pulmonary responses to Escherichia coli endotoxin.
Topics: Animals; Blood Gas Analysis; Cats; Endotoxins; Escherichia coli; Female; Hemodynamics; Ketanserin; Lung; Lung Compliance; Male; Piperidines; Serotonin; Serotonin Antagonists | 1983 |
Is 5-HT a mediator in the motor control of the feline pylorus?
Topics: Animals; Cats; Dose-Response Relationship, Drug; Electric Stimulation; Female; Fluorescent Antibody Technique; Histocytochemistry; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Pylorus; Serotonin; Serotonin Antagonists | 1984 |
Effects of dihydroergotamine on the feline cardiovascular response to intravenous infusion of live Escherichia coli bacteria.
Topics: Animals; Blood Pressure; Cardiovascular System; Cats; Dihydroergotamine; Escherichia coli Infections; Gastric Mucosa; Intestinal Mucosa; Ketanserin; Piperidines; Regional Blood Flow; Sepsis; Shock, Septic; Vascular Resistance | 1984 |
A role for serotonin in alpha-naphthylthiourea-induced pulmonary edema.
Topics: Animals; Blood Platelets; Clorgyline; Drug Interactions; Fluoxetine; Ketanserin; Lung; Male; Mice; Piperidines; Pulmonary Edema; Reserpine; Serotonin; Serotonin Antagonists; Thiourea; Thrombocytopenia | 1984 |
Treatment of Raynaud's phenomenon with ketanserin.
Topics: Adolescent; Humans; Ketanserin; Leg Ulcer; Male; Piperidines; Scleroderma, Systemic | 1984 |
Ketanserin treatment in essential hypertension.
Topics: Antihypertensive Agents; Humans; Hypertension; Ketanserin; Piperidines | 1984 |
Aggregating platelets contract isolated canine pulmonary arteries by releasing 5-hydroxytryptamine.
Topics: Animals; Blood Platelets; Dogs; Epinephrine; In Vitro Techniques; Ketanserin; Muscle Contraction; Norepinephrine; Piperidines; Platelet Aggregation; Pulmonary Artery; Serotonin; Serotonin Antagonists; Thromboxane B2 | 1984 |
Temperature-sensitive high affinity [3H]serotonin binding: characterization and effects of antidepressant treatment.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Ketanserin; Kinetics; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Temperature; Tritium | 1984 |
5-HT1 and 5-HT2 binding properties of derivatives of the hallucinogen 1-(2,5-dimethoxyphenyl)-2-aminopropane (2,5-DMA).
Topics: Amphetamines; Animals; Binding, Competitive; Cerebral Cortex; Guanylyl Imidodiphosphate; Hallucinogens; In Vitro Techniques; Ketanserin; Male; Membranes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Structure-Activity Relationship | 1984 |
Discriminative stimulus properties of the serotonin agonist 1-(3-trifluoromethylphenyl)piperazine (TFMPP).
Topics: Animals; Discrimination Learning; DOM 2,5-Dimethoxy-4-Methylamphetamine; Extinction, Psychological; Fenfluramine; Indoles; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin | 1984 |
Interaction of ketanserin and its metabolite ketanserinol with 5HT2 receptors in pulmonary and coronary arteries of calf.
Topics: Animals; Cattle; Coronary Vessels; In Vitro Techniques; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Pulmonary Artery; Receptors, Serotonin; Yohimbine | 1984 |
Selective 5HT-2 antagonists inhibit serotonin stimulated phosphatidylinositol metabolism in cerebral cortex.
Topics: Animals; Cerebral Cortex; In Vitro Techniques; Ketanserin; Phosphatidylinositols; Piperidines; Pizotyline; Rats; Serotonin; Serotonin Antagonists | 1984 |
Restoration of post-thrombotic peripheral collateral circulation in the cat by ketanserin, a selective 5-HT2-receptor antagonist.
Topics: Animals; Blood Platelets; Blood Pressure; Cats; Collateral Circulation; Ketanserin; Piperidines; Prostaglandins; Receptors, Serotonin; Serotonin Antagonists; Thrombosis; Vascular Resistance | 1984 |
Serotonin-induced blood flow changes in the rat hindlegs after unilateral ligation of the femoral artery. Inhibition by the S2 receptor antagonist ketanserin.
Topics: Angiography; Animals; Body Temperature; Collateral Circulation; Corrosion; Evans Blue; Femoral Artery; Hindlimb; Ketanserin; Ligation; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists | 1984 |
Effects of the antagonists MDL 72222 and ketanserin on responses of cat carotid body chemoreceptors to 5-hydroxytryptamine.
Topics: Action Potentials; Animals; Carotid Body; Cats; Chemoreceptor Cells; Domperidone; Dopamine; Electrophysiology; Female; Hypoxia; Ketanserin; Male; Piperidines; Serotonin; Serotonin Antagonists; Tropanes | 1984 |
Serotonin-2 binding sites in human frontal cortex and hippocampus. Selective loss of S-2A sites with age.
Topics: Adolescent; Adult; Aged; Aging; Cerebral Cortex; Hippocampus; Humans; Ketanserin; Kinetics; Methysergide; Middle Aged; Organ Specificity; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone | 1984 |
The effects of alpha 2-adrenergic and serotonergic receptor antagonists on cyclic blood flow alterations in stenosed canine coronary arteries.
Topics: Adenosine Diphosphate; Animals; Blood Flow Velocity; Coronary Circulation; Coronary Disease; Dogs; Female; Heart Rate; Hemodynamics; Ketanserin; Male; Piperidines; Platelet Aggregation; Prazosin; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Yohimbine | 1984 |
Guanyl nucleotide and divalent cation regulation of cortical S2 serotonin receptors.
Topics: Animals; Binding, Competitive; Calcium Chloride; Cations, Divalent; Cerebral Cortex; Chlorides; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Ketanserin; Magnesium; Magnesium Chloride; Male; Manganese; Manganese Compounds; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1984 |
Antihypertensive effects of chronic 5-hydroxytryptamine (5-HT2) receptor blockade with ketanserin in the spontaneously hypertensive rat.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Piperidines; Rats; Rats, Inbred SHR; Receptors, Serotonin; Serotonin Antagonists | 1984 |
Antagonism by ketanserin of 5-HT-induced vasoconstriction unmasks a 5-HT-induced vasodilation.
Topics: Amidines; Animals; Antihypertensive Agents; Blood Pressure; Hypertension; In Vitro Techniques; Ketanserin; Male; Norepinephrine; Piperidines; Rats; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation | 1984 |
Ketanserin alters [3H]serotonin uptake and release in rat hypothalamus.
Topics: Animals; Calcium; Dose-Response Relationship, Drug; Hypothalamus; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Tritium | 1984 |
Central serotonin antagonist activity of ketanserin.
Topics: Animals; Brain; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists | 1984 |
The haemodynamic effects of labetalol, ketanserin and a placebo at the end of a NLA. A double blind study.
Topics: Adolescent; Adult; Aged; Double-Blind Method; Ethanolamines; Female; Hemodynamics; Humans; Ketanserin; Labetalol; Middle Aged; Piperidines; Placebos; Random Allocation; Serotonin Antagonists; Sympatholytics | 1984 |
Mesulergine, a selective serotonin-2 ligand in the rat cortex, does not label these receptors in porcine and human cortex: evidence for species differences in brain serotonin-2 receptors.
Topics: Animals; Brain Chemistry; Cerebral Cortex; Ergolines; Humans; In Vitro Techniques; Ketanserin; Kinetics; Ligands; Male; Piperidines; Rats; Receptors, Serotonin; Species Specificity; Swine; Tritium | 1984 |
Aortic recognition sites for serotonin (5HT) are coupled to phospholipase C and modulate phosphatidylinositol turnover.
Topics: Animals; Aorta; Hydrolysis; Ketanserin; Male; Phosphatidylinositols; Phospholipases; Piperidines; Rats; Receptors, Serotonin; Serotonin; Type C Phospholipases; Vasoconstriction | 1984 |
The effects of serotonin antagonists in a behavioral despair procedure in mice.
Topics: Animals; Behavior, Animal; Cyproheptadine; Guinea Pigs; Ketanserin; Male; Methysergide; Mice; Muscle, Smooth; Piperidines; Pizotyline; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Trazodone; Tritium | 1984 |
Identification of 5HT2-receptors on longitudinal muscle of the guinea pig ileum.
Topics: Animals; Cerebral Cortex; Female; Guinea Pigs; Ileum; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Muscle, Smooth; Piperidines; Rats; Receptors, Serotonin | 1984 |
Guanine nucleotides modulate cortical S2 serotonin receptors.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone | 1984 |
The distribution of serotonin binding sites in the hippocampal region of the rat brain. An autoradiographic study.
Topics: Animals; Autoradiography; Binding Sites; Binding, Competitive; Hippocampus; Ketanserin; Male; Methoxydimethyltryptamines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone | 1984 |
Excitatory and inhibitory effects of 5-hydroxytryptamine in mesenteric arteries of spontaneously hypertensive rats.
Topics: Animals; Blood Pressure; Cyproheptadine; Drug Synergism; Hypertension; In Vitro Techniques; Ketanserin; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Norepinephrine; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Serotonin; Synapses | 1984 |
Role of serotonin in patients with acute respiratory failure.
Topics: 6-Ketoprostaglandin F1 alpha; Acute Disease; Adult; Aged; Blood Platelets; Blood Pressure; Cardiac Output; Female; Humans; Intubation, Intratracheal; Ketanserin; Male; Middle Aged; Piperidines; Platelet Count; Pulmonary Wedge Pressure; Respiratory Function Tests; Respiratory Insufficiency; Serotonin; Serotonin Antagonists; Thromboxane B2 | 1984 |
Redistribution of carotid artery blood flow by 5-HT: effects of the 5-HT2 receptor antagonists ketanserin and Wal 1307.
Topics: Animals; Carotid Arteries; Dibenzoxazepines; Hemodynamics; Ketanserin; Piperidines; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Swine | 1984 |
Three distinct subtypes of serotonergic receptors mediate the triphasic blood pressure response to serotonin in rats.
Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Indoles; Ketanserin; Mice; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Tropisetron | 1984 |
The use of ketanserin, a 5-hydroxytryptamine receptor antagonist, for treatment of postoperative hypertension following coronary artery bypass surgery.
Topics: Coronary Artery Bypass; Female; Heart Rate; Hemodynamics; Humans; Hypertension; Infusions, Parenteral; Injections, Intravenous; Ketanserin; Male; Middle Aged; Piperidines; Postoperative Complications; Serotonin Antagonists | 1983 |
Involvement of 5-HT2 receptors in the wet-dog shake behaviour induced by 5-hydroxytryptophan in the rat.
Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Female; Ketanserin; Methysergide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists | 1983 |
Ketanserin in the treatment of hypertension following coronary artery bypass surgery. A preliminary study.
Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Coronary Artery Bypass; Humans; Hypertension; Ketanserin; Middle Aged; Piperidines; Postoperative Care; Postoperative Complications | 1983 |
Effects of ketanserin and mepyramine on platelet aggregation and on the uptake of 5-hydroxytryptamine into platelets.
Topics: Adenosine Diphosphate; Aminopyridines; Blood Platelets; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1983 |
Antagonism of the 5-HT-induced bronchoconstriction in the cat.
Topics: Animals; Bronchi; Carbachol; Cats; Clenbuterol; Cyproheptadine; Female; Hemodynamics; Ketanserin; Male; Piperidines; Pregnancy; Serotonin; Serotonin Antagonists; Theophylline | 1983 |
Prophylactic use of ketanserin in a patient with carcinoid syndrome.
Topics: Female; Humans; Hypertension; Intraoperative Complications; Ketanserin; Malignant Carcinoid Syndrome; Middle Aged; Piperidines; Serotonin Antagonists | 1983 |
Ketanserin, a novel 5-hydroxytryptamine antagonist: monotherapy in essential hypertension.
Topics: Adult; Aged; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Ketanserin; Kinetics; Male; Middle Aged; Piperidines; Serotonin Antagonists | 1983 |
Pharmacokinetics of ketanserin in man.
Topics: Administration, Oral; Adult; Blood Pressure; Blood Proteins; Female; Half-Life; Heart Rate; Humans; Injections, Intravenous; Ketanserin; Kinetics; Male; Piperidines; Protein Binding | 1983 |
Antagonism of the effects of the hallucinogen DOM and the purported 5-HT agonist quipazine by 5-HT2 antagonists.
Topics: Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists | 1983 |
The effect of a 5-HT antagonist, ketanserin, on blood pressure, the renin-angiotensin system and sympathoadrenal function in normal man.
Topics: Adrenal Glands; Adult; Blood Pressure; Diet; Heart Rate; Humans; Ketanserin; Male; Phenylephrine; Piperidines; Posture; Renin-Angiotensin System; Serotonin Antagonists; Sympathetic Nervous System; Time Factors | 1983 |
Characterization and regional distribution of serotonin S2-receptors in human brain.
Topics: Brain; Brain Chemistry; Humans; Ketanserin; Kinetics; Piperidines; Receptors, Serotonin | 1983 |
Effects of pirenperone and ketanserin on rat prolactin secretion in vivo and in vitro.
Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin Antagonists; Tranquilizing Agents | 1983 |
Autoradiographic distribution of serotonin2 receptors in rat brain.
Topics: Animals; Brain Chemistry; Ketanserin; Male; Piperidines; Rats; Receptors, Serotonin; Tissue Distribution | 1983 |
The effect of ketanserin, a specific serotonin antagonist, on burn shock hemodynamic parameters in a porcine burn model.
Topics: Animals; Blood Pressure; Body Temperature; Burns; Disease Models, Animal; Heart Rate; Hemodynamics; Ketanserin; Piperidines; Serotonin Antagonists; Shock, Traumatic; Swine | 1983 |
Determination of ketanserin and its major metabolite (reduced ketanserin) in human plasma by high-performance liquid chromatography.
Topics: Adult; Chromatography, High Pressure Liquid; Female; Humans; Ketanserin; Oxidation-Reduction; Piperidines; Spectrophotometry, Ultraviolet | 1983 |
pH-dependent modulation of agonist interactions with [3H]-ketanserin-labelled S2 serotonin receptors.
Topics: Animals; Binding, Competitive; Frontal Lobe; Hydrogen-Ion Concentration; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1983 |
Characterization of serotonin binding sites on human platelets.
Topics: Adult; Binding, Competitive; Blood Platelets; Frontal Lobe; Humans; Ketanserin; Male; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone | 1983 |
Inhibitory effect of ketanserin on ergonovine-induced contractions of isolated canine coronary arteries.
Topics: Animals; Coronary Vessels; Dogs; Ergonovine; In Vitro Techniques; Ketanserin; Methysergide; Piperidines; Serotonin Antagonists; Vasoconstriction | 1983 |
The 5-hydroxytryptamine receptor of blood platelets.
Topics: Animals; Binding, Competitive; Blood Platelets; Brain; Calcium; Cell Membrane; Ketanserin; Kinetics; Lysergic Acid Diethylamide; Models, Neurological; Neurons; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship | 1983 |
5-Hydroxytryptamine can mediate endothelium-dependent relaxation of coronary arteries.
Topics: Animals; Blood Platelets; Coronary Vessels; Dogs; In Vitro Techniques; Isometric Contraction; Ketanserin; Methysergide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Piperidines; Serotonin; Serotonin Antagonists; Thromboxane B2 | 1983 |
Selective inhibition by ketanserin and spiroperidol of 5-HT-induced myometrial contraction.
Topics: Animals; Butyrophenones; Estradiol; Female; Ketanserin; Ovary; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Spiperone; Uterine Contraction | 1983 |
Evidence for mediation by 5-HT2 receptors of 5-hydroxytryptamine-induced contraction of canine basilar artery.
Topics: Animals; Basilar Artery; Cerebral Cortex; Dogs; Female; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium | 1983 |
Haemodynamic response to ketanserin in rabbits with Page hypertension: comparison with prazosin.
Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Hypertension; Ketanserin; Male; Methoxamine; Piperidines; Prazosin; Quinazolines; Rabbits; Receptors, Serotonin; Serotonin Antagonists | 1983 |
Long-term effects on central haemodynamics and body fluid volumes of ketanserin in essential hypertension studies at rest and during dynamic exercise.
Topics: Adult; Blood Pressure; Body Fluids; Body Weight; Cardiac Output; Female; Heart Rate; Hemodynamics; Humans; Hypertension; Ketanserin; Male; Middle Aged; Oxygen Consumption; Physical Exertion; Piperidines; Rest; Time Factors; Vascular Resistance | 1983 |
The influence of antiserotonin treatment with ketanserin on the pulmonary lodgement of circulating tumour cells in normal and traumatized rats.
Topics: Animals; Femoral Fractures; Fibrosarcoma; Ketanserin; Lung Neoplasms; Neoplasm Transplantation; Neoplastic Cells, Circulating; Piperidines; Rats; Sarcoma, Experimental; Serotonin Antagonists | 1983 |
Differential actions of serotonin antagonists on two behavioral models of serotonin receptor activation in the rat.
Topics: Animals; Behavior, Animal; Butyrophenones; Ketanserin; Male; Metergoline; Methysergide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists | 1984 |
The effects of platelet-derived contractile agents on human digital arteries.
Topics: Arteries; Blood Platelets; Humans; Imidazoles; In Vitro Techniques; Indomethacin; Ketanserin; Muscle Contraction; Piperidines; Platelet Aggregation; Serotonin Antagonists; Thromboxane A2; Time Factors | 1984 |
Ketanserin, a serotonin antagonist. Administration in patients with acute respiratory failure.
Topics: Adult; Aged; Blood Proteins; Erythrocyte Indices; Female; Humans; Ketanserin; Male; Middle Aged; Piperidines; Pulmonary Wedge Pressure; Respiratory Insufficiency; Stroke Volume; Vascular Resistance | 1984 |
The involvement of 5-HT2-receptor sites in the activation of cat platelets.
Topics: Adenosine Diphosphate; Animals; Blood Platelets; Cats; Collagen; Dose-Response Relationship, Drug; Ketanserin; Kinetics; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin | 1984 |
Interactions of agonists with D-2 dopamine receptors: evidence for a single receptor population existing in multiple agonist affinity-states in rat striatal membranes.
Topics: Animals; Binding, Competitive; Butyrophenones; Corpus Striatum; Domperidone; Dopamine Antagonists; Guanine Nucleotides; Ketanserin; Metoclopramide; Piperidines; Radioligand Assay; Rats; Receptors, Dopamine; Sodium; Spiperone; Temperature | 1984 |
Acute effects of ketanserin on left ventricular function, metabolism and coronary blood flow.
Topics: Adult; Blood Pressure; Cardiac Catheterization; Coronary Circulation; Female; Heart; Heart Rate; Heart Ventricles; Humans; Ketanserin; Male; Middle Aged; Myocardium; Piperidines; Pulmonary Artery; Vascular Resistance | 1984 |
Reduced binding of [3H]ketanserin to cortical 5-ht2 receptors in senile dementia of the Alzheimer type.
Topics: Age Factors; Aged; Alzheimer Disease; Cerebral Cortex; Humans; Ketanserin; Piperidines; Receptors, Serotonin; Serotonin Antagonists | 1984 |
Ergonovine-induced myocardial ischemia: no role for serotonergic receptors?
Topics: Aged; Angina Pectoris; Coronary Vasospasm; Coronary Vessels; Ergonovine; Hand; Humans; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Vasoconstriction | 1984 |
Solubilization of serotonin S2-receptors from human brain.
Topics: Animals; Brain Chemistry; Dogs; Humans; In Vitro Techniques; Ketanserin; Kinetics; Lysophosphatidylcholines; Membranes; Piperidines; Rats; Receptors, Serotonin; Species Specificity | 1984 |
Ketanserin and vascular contractions in response to cooling.
Topics: Animals; Arteries; Cold Temperature; In Vitro Techniques; Ketanserin; Piperidines; Rabbits; Serotonin; Serotonin Antagonists; Vasoconstriction | 1984 |
Intrapartum treatment of preeclamptic hypertension by ketanserin--a serotonin receptor antagonist.
Topics: Adult; Antihypertensive Agents; Delivery, Obstetric; Female; Humans; Hydralazine; Hypertension; Infant, Newborn; Ketanserin; Piperidines; Pre-Eclampsia; Pregnancy; Serotonin Antagonists; Time Factors; Vascular Resistance | 1984 |
Serotonergic regulation of cortisol secretion in dogs.
Topics: Animals; Dogs; Fenfluramine; Hydrocortisone; Ketanserin; Piperidines; Quipazine; Serotonin; Time Factors | 1984 |
Some behavioral effects of hallucinogens are mediated by a postsynaptic serotonergic action: evidence from single unit studies in freely moving cats.
Topics: Animals; Apomorphine; Behavior, Animal; Cats; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Female; Hallucinogens; Ketanserin; Lisuride; Lysergic Acid Diethylamide; Metergoline; Mianserin; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Synapses | 1984 |
Effects of tryptamine antagonists on the anaphylactic contractions of the bovine pulmonary smooth muscles.
Topics: Anaphylaxis; Animals; Cattle; Horses; In Vitro Techniques; Ketanserin; Lung; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Pulmonary Artery; Pulmonary Veins; Serotonin Antagonists; Trachea; Tryptamines | 1984 |
Restoration of pulmonary perfusion by a serotonin antagonist.
Topics: Adult; Aged; Blood Pressure; Carbon Dioxide; Embolism, Air; Female; Humans; Infant, Newborn; Intraoperative Complications; Ketanserin; Male; Piperidines; Pulmonary Circulation; Respiration; Respiratory Distress Syndrome; Serotonin Antagonists; Vasodilator Agents | 1981 |
Treatment of hypertension with ketanserin, a new selective 5-HT2 receptor antagonist.
Topics: Adult; Aged; Cardiac Output; Female; Heart Rate; Humans; Hypertension; Ketanserin; Kidney; Male; Middle Aged; Norepinephrine; Piperidines; Receptors, Serotonin; Vascular Resistance | 1982 |
Platelet-mediated vascular contractions: inhibition of the serotonergic component by ketanserin.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Depression, Chemical; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Suprofen; Thrombin | 1982 |
An assessment of the participatory role of prostaglandins and serotonin in the pathophysiology of endotoxic shock.
Topics: Animals; Dogs; Hemodynamics; Indomethacin; Ketanserin; Oxygen; Piperidines; Prostaglandins; Pulmonary Circulation; Serotonin; Serotonin Antagonists; Shock, Septic | 1983 |
Therapeutic benefits of 5-hydroxytryptamine inhibition following pulmonary embolism.
Topics: Animals; Dogs; Female; Ketanserin; Male; Piperidines; Platelet Count; Prostaglandins; Pulmonary Embolism; Pulmonary Wedge Pressure; Receptors, Serotonin; Respiratory Dead Space; Serotonin; Serotonin Antagonists; Vascular Resistance | 1983 |
The effect of thrombocytopenia and antiserotonin treatment on the lodgement of circulating tumor cells. A vital fluorescence microscopic, electron microscopic and isotope study in the rat.
Topics: Animals; Female; Fibrosarcoma; Ketanserin; Liver Neoplasms; Male; Microscopy, Electron; Microscopy, Fluorescence; Neoplasm Transplantation; Neoplastic Cells, Circulating; Phagocytosis; Piperidines; Rats; Sarcoma, Experimental; Serotonin Antagonists; Thrombocytopenia | 1983 |
High-performance liquid chromatographic assay with fluorometric detection of ketanserin, a new antihypertensive agent and serotonin S2 antagonist in human plasma, blood and urine.
Topics: Antihypertensive Agents; Chromatography, High Pressure Liquid; Half-Life; Humans; Ketanserin; Piperidines; Radioimmunoassay; Serotonin Antagonists; Spectrometry, Fluorescence | 1983 |
Determination of ketanserin in human plasma by high-performance liquid chromatography.
Topics: Chromatography, High Pressure Liquid; Humans; Hypertension; Ketanserin; Piperidines; Time Factors | 1983 |
Ketanserin, a new selective 5-HT2 receptor blocking agent, inhibits the antidiuretic effect of 5-hydroxytryptamine (5-HT) in Wistar rats.
Topics: Animals; Diuresis; Ketanserin; Kidney; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Time Factors | 1983 |
Differences in the regulatory adaptation of the 5HT recognition sites labelled by 3H-mianserin or 3H-ketanserin.
Topics: Animals; Axons; Dibenzazepines; Hippocampus; Imipramine; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Synapses; Tritium | 1983 |
Continuous imaging of regional blood flow in peripheral vascular disease using Krypton-81m: effect of Ketanserin, a new selective serotonin antagonist.
Topics: Animals; Arteriosclerosis Obliterans; Cats; Diabetic Angiopathies; Female; Humans; Hyperemia; Ketanserin; Krypton; Leg; Male; Piperidines; Radioisotopes; Radionuclide Imaging; Regional Blood Flow; Serotonin; Serotonin Antagonists; Thromboangiitis Obliterans; Vascular Diseases | 1983 |
Demonstration of S2-receptor binding sites on cat blood platelets using [3H]ketanserin.
Topics: Animals; Binding Sites; Blood Platelets; Cats; Corpus Striatum; Female; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Tritium | 1983 |
Ketanserin prevents platelet aggregation and endotoxin-induced pulmonary vasoconstriction.
Topics: Animals; Dogs; Epinephrine; Hemodynamics; Hypertension, Pulmonary; Ketanserin; Male; Oxygen; Piperidines; Platelet Aggregation; Serotonin; Serotonin Antagonists; Shock, Septic | 1983 |
Chronic clozapine treatment of rats down-regulates cortical 5-HT2 receptors.
Topics: Animals; Cerebral Cortex; Clozapine; Dibenzazepines; Ketanserin; Male; Piperidines; Rats; Receptors, Serotonin; Time Factors | 1983 |
Determination of ketanserin in plasma by reversed-phase high-performance liquid chromatography.
Topics: Chromatography, High Pressure Liquid; Humans; Ketanserin; Piperidines | 1983 |
The effect of serotonin inhibition on initial microvessel hemostasis and platelet aggregation in vivo.
Topics: Animals; Bleeding Time; Dihydroergotamine; Female; Hemostasis; Ketanserin; Male; Mesenteric Arteries; Mesenteric Veins; Microcirculation; Piperidines; Platelet Aggregation; Rabbits; Serotonin Antagonists | 1983 |
3H-Ketanserin labels serotonin S2-receptor binding sites on cat blood platelets.
Topics: Animals; Blood Platelets; Cats; Cell Membrane; In Vitro Techniques; Ketanserin; Kinetics; Piperidines; Receptors, Serotonin | 1983 |
On the mechanism of action of ketanserin, a selective antagonist of the S2 receptors with antihypertensive activity.
Topics: Animals; Antihypertensive Agents; Dogs; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Norepinephrine; Piperidines; Rats; Serotonin Antagonists; Vasodilation | 1983 |
Is prevention of hypertension after open heart surgery possible by blocking 5HT2-receptors with ketanserin?
Topics: Adult; Aged; Anesthesia; Aortic Valve; Coronary Artery Bypass; Heart Valve Prosthesis; Hemodynamics; Humans; Hypertension; Injections, Intravenous; Ketanserin; Middle Aged; Nitrous Oxide; Piperidines; Postoperative Complications; Serotonin Antagonists | 1982 |
Interaction between 5-hydroxytryptamine and other vasoconstrictor substances in the isolated femoral artery of the rabbit; effect of ketanserin (R 41 468).
Topics: Animals; Drug Interactions; Evoked Potentials; Femoral Artery; In Vitro Techniques; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rabbits; Serotonin; Vasoconstrictor Agents | 1982 |
The effects of serotonin-receptor blockade after cardiopulmonary by-pass. A pilot study.
Topics: Aged; Cardiopulmonary Bypass; Female; Hemodynamics; Humans; Ketanserin; Male; Middle Aged; Pilot Projects; Piperidines; Postoperative Complications; Serotonin Antagonists | 1982 |
[3H]Ketanserin (R 41 468), a selective 3H-ligand for serotonin2 receptor binding sites. Binding properties, brain distribution, and functional role.
Topics: Animals; Binding, Competitive; Brain; Cerebral Cortex; Female; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Species Specificity | 1982 |
Regional distribution of serotonin-2 receptor binding sites in the brain and effects of neuronal lesions.
Topics: Animals; Brain; Dogs; Guinea Pigs; Ketanserin; Microsomes; Mitochondria; Neurons; Neurotoxins; Piperidines; Rabbits; Rats; Receptors, Serotonin; Serotonin Antagonists; Species Specificity | 1982 |
In vivo binding of [3H]ketanserin on serotonin S2-receptors in rat brain.
Topics: Animals; Brain; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Tritium | 1982 |
Haemorheological effects of ketanserin, a selective 5-HT2 receptor antagonist, in aged, spontaneously hypertensive dogs.
Topics: Aging; Animals; Blood Cell Count; Blood Pressure; Blood Viscosity; Dogs; Erythrocyte Membrane; Hypertension; Ketanserin; Piperidines; Serotonin Antagonists; Vascular Resistance | 1982 |
Comparative effects of ketanserin, a novel serotonergic receptor antagonist, on 5HT-induced shape change and 5HT uptake in rat and human platelets.
Topics: Adenosine Diphosphate; Animals; Blood Platelets; Clomipramine; Female; Humans; In Vitro Techniques; Ketanserin; Kinetics; Male; Methysergide; Piperidines; Rats; Serotonin; Serotonin Antagonists | 1982 |
Rapid method for determination of ketanserin, a novel antiserotonin drug, by high-performance liquid chromatography.
Topics: Autoanalysis; Chromatography, High Pressure Liquid; Humans; Ketanserin; Piperidines; Serotonin Antagonists | 1982 |
Effects of Ketanserine on rumino-reticular motility and eructation in sheep: a possible application as an anti-bloating substance.
Topics: Animals; Eructation; Gastrointestinal Motility; Ketanserin; Piperidines; Rumen; Serotonin Antagonists; Sheep | 1982 |
Selectivity of calcium antagonism and serotonin antagonism with respect to venous and arterial tissues.
Topics: Animals; Arteries; Calcium; Cinnarizine; Dogs; Flunarizine; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rabbits; Rats; Serotonin; Serotonin Antagonists; Veins | 1981 |
Vascular activity of ketanserin (R 41 468), a selective 5-HT2 receptor antagonist.
Topics: Animals; Blood Pressure; Dogs; Guinea Pigs; Humans; In Vitro Techniques; Ketanserin; Piperidines; Rabbits; Rats; Serotonin Antagonists; Vasoconstriction | 1981 |
Plethysmographic registration of volume changes in a hand vein. Effects of serotonin and of a specific antagonist.
Topics: Blood Pressure; Blood Volume; Hand; Heart Rate; Humans; Ketanserin; Piperidines; Plethysmography; Serotonin; Serotonin Antagonists; Veins | 1980 |
Neurochemical and behavioral evidence that quipazine-ketanserin discrimination is mediated by serotonin2A receptor.
Topics: Animals; Brain Mapping; Discrimination Learning; Dose-Response Relationship, Drug; Fluorobenzenes; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1995 |
In vivo dopamine-D2 and serotonin-5-HT2 receptor binding study of risperidone and haloperidol.
Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Cerebellum; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; In Vitro Techniques; Isoxazoles; Ketanserin; Ligands; Male; Neostriatum; Piperidines; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone | 1994 |
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach | 1995 |
Ketanserin analogues: the effect of structural modification on 5-HT2 serotonin receptor binding.
Topics: Animals; Binding Sites; Cerebral Cortex; Chemical Phenomena; Chemistry, Physical; In Vitro Techniques; Ketanserin; Magnetic Resonance Spectroscopy; Male; Molecular Structure; Piperazines; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Structure-Activity Relationship | 1995 |
Antinociceptive effects of the kappa opioid, U50,488: lack of modulation by 5-HT2 antagonists.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Ergolines; Ketanserin; Male; Piperidines; Pyrrolidines; Receptors, Opioid, kappa; Saimiri; Serotonin Antagonists | 1993 |
5-HT receptor subtypes involved in luminal serotonin-induced secretion in rat intestine in vivo.
Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Ileum; Indoles; Jejunum; Ketanserin; Male; Methysergide; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Tropisetron; Water-Electrolyte Balance | 1994 |
Monoamine systems in the discriminative effects of spiradoline, a kappa-opioid agonist.
Topics: Analgesics; Animals; Avoidance Learning; Biogenic Monoamines; Discrimination, Psychological; Dopamine Antagonists; Fenfluramine; Fluoxetine; Generalization, Stimulus; Ketanserin; Male; Piperidines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Selective Serotonin Reuptake Inhibitors; Serotonin; Synaptic Transmission | 1994 |
Antiserotoninergic activity of 2-aminoethylbenzocyclanones in rat aorta: structure-activity relationships.
Topics: Animals; Aorta, Thoracic; Butyrophenones; In Vitro Techniques; Ketanserin; Ketones; Molecular Conformation; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Structure-Activity Relationship | 1993 |
Investigation of the mechanism by which ketanserin prolongs the duration of the cardiac action potential.
Topics: Action Potentials; Amphetamines; Animals; Guinea Pigs; Heart; Ketanserin; Male; Piperidines; Potassium Channels; Serotonin Antagonists | 1995 |
Inhibition of noradrenaline release via presynaptic 5-HT1D alpha receptors in human atrium.
Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Cisapride; Corticosterone; Desipramine; Heart Atria; Humans; Indoles; Ketanserin; Male; Middle Aged; Norepinephrine; Oxadiazoles; Piperidines; Receptors, Presynaptic; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tritium; Tryptamines | 1996 |
[3H]MDL 100,907: a novel selective 5-HT2A receptor ligand.
Topics: Animals; Fluorobenzenes; Frontal Lobe; Ketanserin; Ligands; Male; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists | 1996 |
Novel potent sigma 1 ligands: N-[omega-(tetralin-1-yl)alkyl]piperidine derivatives.
Topics: Animals; Hippocampus; Ketanserin; Phencyclidine; Piperidines; Rats; Receptors, Phencyclidine; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, sigma; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes | 1996 |
Preclinical evaluation of [123I]R93274 as a SPECT radiotracer for imaging 5-HT2A receptors.
Topics: Animals; Benzamides; Brain; Dopamine Antagonists; Female; Iodine Radioisotopes; Ketanserin; Papio; Piperidines; Raclopride; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Salicylamides; Serotonin Antagonists; Tomography, Emission-Computed, Single-Photon | 1997 |
Pharmacological characterization of in vivo properties of putative mixed 5-HT1A agonist/5-HT(2A/2C) antagonist anxiolytics. II. Drug discrimination and behavioral observation studies in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzopyrans; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Nicotinic Acids; Piperazines; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 1997 |
Selective visualization of rat brain 5-HT2A receptors by autoradiography with [3H]MDL 100,907.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Fluorobenzenes; Guanylyl Imidodiphosphate; In Situ Hybridization; In Vitro Techniques; Ketanserin; Male; Naphthalenes; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists | 1997 |
A potent 5-hydroxytryptamine receptor (5-HT2A) antagonist, DV-7028, delays arterial thrombosis development in rats.
Topics: Animals; Aorta, Abdominal; Bleeding Time; Ketanserin; Male; Piperidines; Platelet Aggregation; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Thrombophlebitis; Thrombosis; Triazines | 1998 |
Vascular and cardiac effects of DV-7028, a selective, 5-HT2-receptor antagonist in rats.
Topics: Animals; Baroreflex; Blood Pressure; Cardiovascular System; Coronary Circulation; Heart; Heart Rate; Hindlimb; Injections, Intravenous; Ketanserin; Male; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Triazines; Vagotomy | 1998 |
5-HT2A receptor antagonists block MK-801-induced stereotypy and hyperlocomotion.
Topics: Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Histamine H2 Antagonists; Ketanserin; Locomotion; Male; Mice; Mice, Inbred BALB C; Neuroprotective Agents; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Stereotypic Movement Disorder | 1998 |
[3H]MDL 100,907 labels 5-HT2A serotonin receptors selectively in primate brain.
Topics: Aged; Aged, 80 and over; Animals; Binding Sites; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Male; Naphthalenes; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Tritium | 1998 |
Agonist and antagonist binding to rabbit cortical 5-HT2A receptors: opposite effects of magnesium.
Topics: Amphetamines; Animals; Cerebral Cortex; Fluorobenzenes; Guanylyl Imidodiphosphate; Ketanserin; Magnesium; Methysergide; Piperidines; Prazosin; Rabbits; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone | 1998 |
Effect of 5-HT2 receptor antagonists on a cranial nerve reflex in the rabbit: evidence for inverse agonism.
Topics: Animals; Cranial Nerves; Ergolines; Female; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Piperidines; Rabbits; Receptors, Serotonin; Reflex; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 1999 |
Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach.
Topics: Animals; Atropine; Dioxanes; Enzyme Inhibitors; Female; Gastric Fundus; Granisetron; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscarinic Antagonists; Muscle Relaxation; Muscle Tonus; Nitroarginine; Piperidines; Pyloric Antrum; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Tetrodotoxin | 1999 |
5-HT2C receptor involvement in female rat lordosis behavior.
Topics: Animals; Estradiol; Female; Fluorobenzenes; Indoles; Indophenol; Ketanserin; Ovariectomy; Piperidines; Posture; Pyridines; Rats; Rats, Inbred Strains; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sexual Behavior, Animal; Ventromedial Hypothalamic Nucleus | 1999 |
Ketanserin and tetrabenazine abolish aggression in mice lacking monoamine oxidase A.
Topics: Adrenergic Uptake Inhibitors; Aggression; Animals; Brain; Corpus Striatum; Drug Evaluation, Preclinical; Fluorobenzenes; Frontal Lobe; Ketanserin; Male; Mice; Mice, Knockout; Monoamine Oxidase; Neurotransmitter Agents; Piperidines; Radioligand Assay; Serotonin Antagonists; Tetrabenazine | 1999 |
Human striosomes are enriched in 5-HT2A receptors: autoradiographical visualization with [3H]MDL100,907,[125I](+/-)DOI and [3H]ketanserin.
Topics: Adult; Aged; Autoradiography; Female; Fluorobenzenes; Humans; Indophenol; Iodine Radioisotopes; Ketanserin; Male; Middle Aged; Neostriatum; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Tritium | 1999 |
[2-(omega-phenylalkyl)phenoxy]alkylamines.II: Synthesis and selective serotonin-2 receptor binding.
Topics: Animals; Blood Platelets; Blood Vessels; Humans; In Vitro Techniques; Ketanserin; Phenyl Ethers; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Pyrroles; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Structure-Activity Relationship; Succinates; Vasoconstriction | 2000 |
In vitro autoradiography of serotonin 5-HT(2A/2C) receptor-activated G protein: guanosine-5'-(gamma-[(35)S]thio)triphosphate binding in rat brain.
Topics: Amphetamines; Animals; Autoradiography; Brain Chemistry; Dose-Response Relationship, Drug; Fluorobenzenes; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Image Processing, Computer-Assisted; Indoles; Ketanserin; Male; Membrane Proteins; Piperidines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Subcellular Fractions; Sulfur Radioisotopes | 2000 |
Mapping of 5-HT2A receptors and their mRNA in monkey brain: [3H]MDL100,907 autoradiography and in situ hybridization studies.
Topics: Animals; Autoradiography; Brain; Brain Mapping; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Macaca mulatta; Male; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists | 2001 |
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron | 2000 |
Antagonism of 5-hydroxytryptamine(2a) receptors attenuates the behavioral effects of cocaine in rats.
Topics: Animals; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Discrimination Learning; Dopamine; Fluorobenzenes; Ketanserin; Male; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists | 2001 |
Assessment of affinity and dissociation ability of a newly synthesized 5-HT2 antagonist, AT-1015: comparison with other 5-HT2 antagonists.
Topics: Animals; Cerebral Cortex; Isonipecotic Acids; Ketanserin; Male; Piperidines; Rabbits; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists | 2001 |
Multiple 5-HT receptors are involved in the effects of acute MDMA treatment: studies on locomotor activity and responding for conditioned reinforcement.
Topics: 3,4-Methylenedioxyamphetamine; Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Ethylamines; Indoles; Ketanserin; Male; Motor Activity; Oxadiazoles; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2002 |
Biodistribution and displacement studies of the selective 5-HT2A receptor antagonist 123I-5-I-R91150 in the normal dog.
Topics: Animals; Binding, Competitive; Brain; Dogs; Ketanserin; Piperidines; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Tissue Distribution; Tomography, Emission-Computed, Single-Photon; Whole-Body Counting | 2002 |
Pharmacological characterization of the effects of 3,4-methylenedioxymethamphetamine ("ecstasy") and its enantiomers on lethality, core temperature, and locomotor activity in singly housed and crowded mice.
Topics: Animals; Body Temperature; Cold Temperature; Crowding; Dose-Response Relationship, Drug; Fluorobenzenes; Fluoxetine; Hallucinogens; Ketanserin; Lethal Dose 50; Male; Mice; Motor Activity; N-Methyl-3,4-methylenedioxyamphetamine; Piperidines; Platelet Aggregation Inhibitors; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Social Isolation; Stereoisomerism; Telemetry | 2003 |
Discriminative stimulus properties of (+/-)-fenfluramine: the role of 5-HT2 receptor subtypes.
Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Fenfluramine; Fluorobenzenes; Indoles; Ketanserin; Male; Piperidines; Pyrazines; Pyridines; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Thiophenes | 2003 |
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides | 2003 |
Serotonin induces tonic firing in layer V pyramidal neurons of rat prefrontal cortex during postnatal development.
Topics: Age Factors; Animals; Down-Regulation; Female; In Vitro Techniques; Ketanserin; Male; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Signal Transduction | 2003 |
Diverse regulation of atrial natriuretic peptide secretion by serotonin receptor subtypes.
Topics: Adenylyl Cyclase Inhibitors; Alkaloids; Aminobenzoates; Animals; Atrial Natriuretic Factor; Benzophenanthridines; Benzothiazoles; Calcium; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Dose-Response Relationship, Drug; Heart; Heart Atria; Imines; Indoles; Isoquinolines; Ketanserin; Male; Myocytes, Cardiac; Neomycin; para-Aminobenzoates; Perfusion; Phenanthridines; Piperazines; Piperidines; Protein Kinase C; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Staurosporine; Sulfonamides; Thiazoles; Type C Phospholipases | 2003 |
Fenfluramine evokes 5-HT2A receptor-mediated responses but does not displace [11C]MDL 100907: small animal PET and gene expression studies.
Topics: Animals; Carbon Radioisotopes; Cerebellum; Fenfluramine; Fluorobenzenes; Gene Expression; Genes, Immediate-Early; In Situ Hybridization; Ketanserin; Male; Neurons; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Time Factors; Tomography, Emission-Computed | 2003 |
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery.
Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines | 2004 |
Functional role of the endocannabinoid system and AMPA/kainate receptors in 5-HT2A receptor-mediated wet dog shakes.
Topics: Amphetamines; Animals; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Dose-Response Relationship, Drug; Endocannabinoids; Excitatory Amino Acid Antagonists; Injections, Intraperitoneal; Ketanserin; Male; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, Kainic Acid; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists | 2005 |
Effects of donepezil, nicotine and haloperidol on the central serotonergic system in mice: implications for Tourette's syndrome.
Topics: Amphetamines; Animals; Behavior, Animal; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Donepezil; Dose-Response Relationship, Drug; Frontal Lobe; Gene Expression; Haloperidol; Humans; Indans; Ketanserin; Male; Mesencephalon; Mice; Mice, Inbred ICR; Nicotine; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin Antagonists; Tourette Syndrome | 2005 |
Binding characteristics of the 5-HT2A receptor antagonists altanserin and MDL 100907.
Topics: Animals; Binding, Competitive; Brain; Carbon Radioisotopes; Fluorine Radioisotopes; Fluorobenzenes; Ketanserin; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists | 2005 |
Effects of 5-HT2A receptor stimulation on the discrimination of durations by rats.
Topics: Amphetamines; Animals; Association Learning; Brain; Discrimination Learning; Female; Fluorobenzenes; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Piperidines; Psychophysics; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Serotonin Receptor Agonists; Time Perception | 2006 |
Functional characterization of serotonin receptor subtypes in human duodenal secretion.
Topics: Adult; Aged; Bumetanide; Dioxanes; Duodenum; Female; Helicobacter Infections; Helicobacter pylori; Humans; In Vitro Techniques; Intestinal Secretions; Ion Transport; Ketanserin; Male; Middle Aged; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium Potassium Chloride Symporter Inhibitors | 2006 |
Gasping activity in vitro: a rhythm dependent on 5-HT2A receptors.
Topics: Action Potentials; Analysis of Variance; Animals; Animals, Newborn; Biological Clocks; Dose-Response Relationship, Drug; Drug Interactions; Flufenamic Acid; In Vitro Techniques; Ketanserin; Mice; Nerve Net; Neurons; Oxygen; Patch-Clamp Techniques; Piperidines; Receptor, Serotonin, 5-HT2A; Respiratory Burst; Respiratory Center; Respiratory Mechanics; Serotonin Antagonists; Substance P; Synaptic Transmission; Time Factors | 2006 |
Rewarding properties of 1-benzylpiperazine, a new drug of abuse, in rats.
Topics: Animals; Behavior, Animal; Benzazepines; Conditioning, Psychological; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ketanserin; Male; Piperidines; Psychotropic Drugs; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT3; Reward; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Substance-Related Disorders; Tropanes | 2006 |
Cardiac baroreflex facilitation evoked by hypothalamus and prefrontal cortex stimulation: role of the nucleus tractus solitarius 5-HT2A receptors.
Topics: Animals; Atenolol; Atropine Derivatives; Baroreflex; Brain; Electric Stimulation; Fluorobenzenes; Heart; Ketanserin; Male; Microinjections; Neural Inhibition; Neural Pathways; Parasympatholytics; Piperidines; Prefrontal Cortex; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Solitary Nucleus; Stimulation, Chemical; Sympatholytics | 2006 |
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin | 2007 |
Opposing effects of 5-HT(2A) and 5-HT(2C) receptor antagonists in the rat and mouse on premature responding in the five-choice serial reaction time test.
Topics: Aminopyridines; Amphetamines; Animals; Conditioning, Operant; Ethylamines; Fluorobenzenes; Impulsive Behavior; Indoles; Ketanserin; Male; Mice; Mice, Inbred C57BL; Piperidines; Quinolines; Rats; Reaction Time; Serial Learning; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Species Specificity | 2007 |
Total synthesis and evaluation of [18F]MHMZ.
Topics: Animals; Binding, Competitive; Brain; Fluorine Radioisotopes; Fluorobenzenes; Isotope Labeling; Ketanserin; Kinetics; Piperidines; Radioligand Assay; Radionuclide Imaging; Radiopharmaceuticals; Rats; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists | 2008 |
Evidence that genetic variation in 5-HT transporter expression is linked to changes in 5-HT2A receptor function.
Topics: Amphetamines; Analysis of Variance; Animals; Brain; Cytoskeletal Proteins; Dose-Response Relationship, Drug; Fluorobenzenes; Gene Expression; Genetic Variation; Head Movements; Ketanserin; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Nerve Tissue Proteins; Piperidines; Protein Binding; Proto-Oncogene Proteins c-fos; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists | 2008 |
Aripiprazole inhibits marble-burying behavior via 5-hydroxytryptamine (5-HT)1A receptor-independent mechanisms.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Anxiety; Aripiprazole; Behavior, Animal; Benzodiazepines; Catalepsy; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Ketanserin; Male; Mice; Mice, Inbred ICR; Olanzapine; Piperazines; Piperidines; Postural Balance; Psychomotor Performance; Pyridines; Quinolones; Quinpirole; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists | 2008 |
Effect of cyclosporin A administration on the biodistribution and multipinhole muSPECT imaging of [123I]R91150 in rodent brain.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Brain; Cyclosporine; Iodine Radioisotopes; Ketanserin; Ligands; Male; Mice; Piperidines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tomography, Emission-Computed, Single-Photon | 2009 |
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane in rhesus monkeys: antagonism and apparent pA2 analyses.
Topics: Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Electroshock; Fluorobenzenes; Hallucinogens; Ketanserin; Macaca mulatta; Phenethylamines; Piperidines; Reaction Time; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Regression Analysis; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 2009 |
Genetic deletion of MAO-A promotes serotonin-dependent ventricular hypertrophy by pressure overload.
Topics: Animals; Aorta; Blood Pressure; Cardiomegaly; Fibrosis; Fluorobenzenes; Gene Deletion; Gene Expression Regulation; Heart Ventricles; Ketanserin; Mice; Mice, Knockout; Monoamine Oxidase; Myocardium; Piperidines; Pressure; Receptors, Serotonin; Serotonin; Stress, Physiological; Ultrasonography | 2009 |
Enhanced 5-HT(2A) receptors in brain stem and ALDH activity in brain stem and liver: 5-HT(2A) regulation on ALDH in primary hepatocytes cultures in vitro.
Topics: Aldehyde Dehydrogenase; Animals; Brain Stem; Ethanol; Fluorobenzenes; Hepatocytes; Ketanserin; Liver; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin | 2009 |
Age-dependent effects of the cannabinoid CB1 antagonist SR141716A on food intake, body weight change, and pruritus in rats.
Topics: Age Factors; Animals; Brain; Dose-Response Relationship, Drug; Drinking; Eating; Feeding Behavior; Ketanserin; Male; Piperidines; Pruritus; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Serotonin Antagonists; Weight Gain | 2009 |
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM), ketanserin, and (R)-(+)-{alpha}-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-pipidinemethanol (MDL100907) in rats.
Topics: Analgesics, Opioid; Anesthetics, Dissociative; Animals; Conditioning, Operant; Discrimination, Psychological; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorobenzenes; Ketamine; Ketanserin; Male; Morphine; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 2009 |
State-dependent interactions between excitatory neuromodulators in the neuronal control of breathing.
Topics: Action Potentials; Adrenergic alpha-1 Receptor Antagonists; Animals; Animals, Newborn; Electric Stimulation; Electromyography; Hypoglossal Nerve; In Vitro Techniques; Isoindoles; Ketanserin; Locus Coeruleus; Mice; Microinjections; Neural Inhibition; Neural Pathways; Neurokinin-1 Receptor Antagonists; Neurons; Neurotransmitter Agents; Piperidines; Raphe Nuclei; Receptors, Adrenergic, alpha-1; Receptors, Neurokinin-1; Receptors, Serotonin, 5-HT2; Respiration; Respiratory Center; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists | 2010 |
Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode.
Topics: Binding, Competitive; Combinatorial Chemistry Techniques; Fluorobenzenes; Hydrophobic and Hydrophilic Interactions; Ketanserin; Ligands; Phenols; Piperidines; Protein Binding; Pyridines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists | 2010 |
Oleamide administered into the nucleus accumbens shell regulates feeding behaviour via CB1 and 5-HT2C receptors.
Topics: Aminopyridines; Animals; Eating; Feeding Behavior; Hyperphagia; Hypothalamus; Indoles; Ketanserin; Male; Motor Activity; Nucleus Accumbens; Oleic Acids; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Antagonists | 2010 |
Interaction of 5-HT2A and 5-HT2C receptors in R(-)-2,5-dimethoxy-4-iodoamphetamine-elicited head twitch behavior in mice.
Topics: Aminopyridines; Amphetamines; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Ethylamines; Fluorobenzenes; Hallucinogens; Head; Indoles; Ketanserin; Male; Mice; Mice, Inbred Strains; Movement; Piperidines; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Spiro Compounds; Sulfonamides | 2010 |
Effects of 5-HT(2A) and 5-HT(2C) receptor antagonists on acute and chronic dyskinetic effects induced by haloperidol in rats.
Topics: Aminopyridines; Animals; Antipsychotic Agents; Brain Chemistry; Catalepsy; Dyskinesia, Drug-Induced; Fluorobenzenes; Gene Expression Regulation; Haloperidol; Immunohistochemistry; In Situ Hybridization; Indoles; Ketanserin; Male; Mouth; Piperidines; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; RNA, Messenger; Serotonin Antagonists | 2011 |
p-Hydroxyamphetamine causes prepulse inhibition disruption in mice: contribution of serotonin neurotransmission.
Topics: 5,7-Dihydroxytryptamine; Acoustic Stimulation; Analysis of Variance; Animals; Autoradiography; Brain; Dose-Response Relationship, Drug; Fenclonine; Fluorobenzenes; Inhibition, Psychological; Ketanserin; Male; Mice; p-Hydroxyamphetamine; Piperidines; Reflex, Startle; Serotonin; Serotonin Agents; Serotonin Plasma Membrane Transport Proteins; Time Factors | 2011 |
Reduced levels of serotonin 2A receptors underlie resistance of Egr3-deficient mice to locomotor suppression by clozapine.
Topics: Animals; Clozapine; Disease Models, Animal; Early Growth Response Protein 3; Humans; Hypnotics and Sedatives; Ketanserin; Male; Mice; Mice, Transgenic; Motor Activity; Piperidines; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin 5-HT2 Receptor Agonists; Serotonin Antagonists | 2012 |
Direct comparison of [(18) F]MH.MZ and [(18) F] altanserin for 5-HT2A receptor imaging with PET.
Topics: Animals; Brain; Fluorine Radioisotopes; Fluorobenzenes; Ketanserin; Piperidines; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Swine; Tissue Distribution; Tritium | 2013 |
Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT₂A receptors, in mice.
Topics: Amphetamines; Animals; Dose-Response Relationship, Drug; Fluorobenzenes; Hallucinogens; Head Movements; Ketanserin; Male; Mice; Phenethylamines; Piperidines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists | 2015 |
Involvement of Descending Serotonergic and Noradrenergic Systems and their Spinal Receptor Subtypes in the Antinociceptive Effect of Dipyrone.
Topics: 5,7-Dihydroxytryptamine; Adrenergic Neurons; Analgesics; Animals; Dipyrone; Dose-Response Relationship, Drug; Injections, Spinal; Ketanserin; Mice; Ondansetron; Oxidopamine; Pain Measurement; Piperidines; Prazosin; Propranolol; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonergic Neurons; Spinal Cord; Sulfonamides; Yohimbine | 2015 |
Individual Differences in Impulsive Action Reflect Variation in the Cortical Serotonin 5-HT2A Receptor System.
Topics: Animals; Choice Behavior; Dimethoxyphenylethylamine; Fluorobenzenes; Head Movements; Immunoprecipitation; Impulsive Behavior; Individuality; Ketanserin; Male; Piperidines; Prefrontal Cortex; Protein Binding; Rats; Rats, Sprague-Dawley; Reaction Time; Receptor, Serotonin, 5-HT2A; Serotonin Agents; Tritium | 2015 |