ketanserin and mianserin

ketanserin has been researched along with mianserin in 84 studies

Research

Studies (84)

TimeframeStudies, this research(%)All Research%
pre-199028 (33.33)18.7374
1990's40 (47.62)18.2507
2000's11 (13.10)29.6817
2010's5 (5.95)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Amlaiky, N; Boschert, U; Hen, R; Maroteaux, L; Plassat, JL; Saudou, F1
Glennon, RA2
Janssen, CG; Laduron, PM; Thijssen, JB; Van Dun, J; Wouters, W1
Andrews, PR; Craik, DJ; Martin, JL1
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR1
Amlaiky, N; Hen, R; Plassat, JL1
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB1
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP1
Baez, M; Kursar, JD; Lucaites, VL; Nelson, DL; Sasso, DA; Wainscott, DB1
Egan, CT; Herrick-Davis, K; Teitler, M1
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP1
Booth, RG; Brown, RL; Bucholtz, EC; Tropsha, A; Wyrick, SD1
Itoh, H; Muramatsu, I; Taniguchi, T; Yoshio, R1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A1
Araki, H; Karasawa, Y; Otomo, S1
Miletic, V; Tan, H1
Barker, EL; Burris, KD; Sanders-Bush, E1
DeNoble, KF; DeNoble, VJ; Reigel, AL; Schrack, LM1
Agresta, CA; Freeman, GM; Liu, ZJ; Maitland-Heriot, RP; Puniak, MA; Salzman, SK1
Buckner, CK; Dea, D; Krell, RD; Liberati, N1
Giordano, J1
Gallager, DW; Goldman-Rakic, PS; Lidow, MS; Rakic, P1
Dewar, KM; Lima, L; Reader, TA1
Barrett, RJ; Sanders-Bush, E; Smith, RL1
Horst, D; Nakamura, Y; Saville, L; Terranova, PF; Uilenbroek, JT1
Battista, PJ; Condon, WA; Rexroad, CE1
Beni, M; Carla, V; Consolazione, A; Dall'Olio, R; Gandolfi, O; Lombardi, G; Moroni, F; Pellegrini-Giampietro, DE1
Dall'Olio, R; Gandolfi, O; Roncada, P1
DeNoble, VJ; Spencer, KR; Strek, KF1
North, RA; Uchimura, N1
Alexander, BS; Wood, MD1
Conn, PJ; Hartig, PR; Hoffman, BJ; Sanders-Bush, E1
Barbaccia, ML; Costa, E; Gandolfi, O2
Conn, PJ; Sanders-Bush, E1
Hole, DR; Hunter, AJ; Wilson, CA1
Frost, JJ; Hartig, PR; Scheffel, U; Wagner, HN1
Doğan, N; Ilhan, M; Kayaalp, SO; Tuncer, M1
Burvenich, C; Peeters, G; Vandeputte-Van Messon, G1
Doggrell, SA1
Kayaalp, SO; Tuncer, M; Uma, S1
Altman, HJ; Normile, HJ1
Bush, LR1
Helmeste, DM; Tang, SW2
Cheney, DL; Costa, E; Gandolfi, O; Hong, JS1
Köhler, C1
Anthony, M1
Heym, J; Jacobs, BL; Rasmussen, K1
Barbaccia, ML; Chuang, DM; Costa, E; Gandolfi, O1
Hartig, PR; Hoffman, BJ; Kaufman, MJ1
Altuğ, U; Erol, D; Germiyanoğlu, C; Gürdal, M; Kurt, U; Ozkardeş, H1
Blakely, RD; Davies, P; Pitt, BR; Reynolds, I; Steve, AR; Weng, W1
Ageel, AM; Alhaider, AA; Ginawi, OT1
Agresta, CA; Azim, S; Chavin, J; Kelly, G; Puniak, MA; Salzman, SK; Wang, L1
Hrdina, PD; Vu, TB1
Ferry, RC; Molinoff, PB; Unsworth, CD1
Gibbs, J; Greenberg, D; Poeschla, B; Simansky, KJ; Smith, GP1
Kaneko, M; Kumashiro, H; Mashiko, H; Ohsuka, N1
Caldarola-Pastuszka, M; Colon, L; Cox, A; Uphouse, L; Wolf, A1
Hartman, JL; Northup, JK1
Bishop-Robinson, C; Darmani, NA; Onaivi, ES; Sanders-Bush, E1
Marwood, JF; Okoro, EO1
Elliott, JM; Newton, RA1
Cowley, KC; MacLean, JN; Schmidt, BJ1
Burrows, GD; McGrath, C; Norman, TR1
Aguerre, S; Chaouloff, F; Mormede, P1
Harvey, JA; Hood, H; Romano, AG; Welsh, SE1
Fujiseki, Y; Inagaki, C; Kinoshita, T; Okugawa, G; Omori, K; Suzukawa, J1
Anji, A; Bryan, GL; Hensler, JG; Kumari, M; Sullivan Hanley, NR1
Davidson, C; Ellinwood, EH; Lazarus, C; Lee, TH; Xiong, X1
Lehr, T; Schipp, R1
Gatellier, L; Kanzaki, R; Nagao, T1
Matsumoto, K; Morishige, R; Murakami, Y; Sakakibara, I; Takayama, H; Tohda, M; Watanabe, H1
Pericić, D; Strac, DS; Vlainić, J1
Angle, JM; Dallimore, JE; Mackie, AR; McDaid, J; Mickiewicz, AL; Napier, TC; Shen, F; Tedford, CE1
Bhatia, KS; Fowler, JC; Lee, TH; Szabo, ST; Wetsel, WC1
Callado, LF; Díez-Alarcia, R; González-Maeso, J; Meana, JJ; Miranda-Azpiazu, P; Morentin, B; Muguruza, C1
Celeste, T; Persons, AL; Tedford, SE1

Reviews

3 review(s) available for ketanserin and mianserin

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003
Serotonin antagonists.
    Australian and New Zealand journal of medicine, 1984, Volume: 14, Issue:6

    Topics: Cyproheptadine; Depression; Ergotamine; Humans; Hypertension; Ketanserin; Lisuride; Methysergide; Mianserin; Migraine Disorders; Piperidines; Pizotyline; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Diseases

1984

Trials

1 trial(s) available for ketanserin and mianserin

ArticleYear
The efficacy of anti-serotoninergic agents in the treatment of erectile dysfunction.
    The Journal of urology, 1994, Volume: 152, Issue:2 Pt 1

    Topics: Adult; Aged; Double-Blind Method; Erectile Dysfunction; Humans; Ketanserin; Male; Mianserin; Middle Aged; Trazodone

1994

Other Studies

80 other study(ies) available for ketanserin and mianserin

ArticleYear
Mouse 5HT1B serotonin receptor: cloning, functional expression, and localization in motor control centers.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Apr-01, Volume: 89, Issue:7

    Topics: 3T3 Cells; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Cerebellum; Corpus Striatum; Gene Expression; Genes; GTP-Binding Proteins; Mice; Molecular Sequence Data; Nucleic Acid Hybridization; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Purkinje Cells; Receptors, Serotonin; RNA, Messenger; Serotonin

1992
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Frontal Lobe; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1986
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
    The Journal of biological chemistry, 1993, Aug-25, Volume: 268, Issue:24

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection

1993
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.
    Molecular pharmacology, 1993, Volume: 44, Issue:2

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Cyclic AMP; DNA; Drosophila; Enzyme Activation; Humans; Intestinal Mucosa; Mice; Molecular Sequence Data; Myocardium; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists

1993
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature

1993
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
    British journal of pharmacology, 1997, Volume: 122, Issue:1

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid

1997
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adrenergic alpha-Antagonists; Benzofurans; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Imidazoles; Radioligand Assay; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Yohimbine

1998
Creation of a constitutively activated state of the 5-hydroxytryptamine2A receptor by site-directed mutagenesis: inverse agonist activity of antipsychotic drugs.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:1

    Topics: Animals; Antipsychotic Agents; COS Cells; Mutagenesis, Site-Directed; Phosphatidylinositols; Protein Conformation; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship

1998
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
    Journal of neurochemistry, 1999, Volume: 72, Issue:5

    Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1999
Synthesis, evaluation, and comparative molecular field analysis of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for histamine H(1) receptors.
    Journal of medicinal chemistry, 1999, Aug-12, Volume: 42, Issue:16

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ligands; Models, Molecular; Pyrilamine; Radioligand Assay; Structure-Activity Relationship; Tetrahydronaphthalenes

1999
Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:2

    Topics: Animals; Aorta, Thoracic; Carotid Arteries; Dogs; Humans; Male; Organ Culture Techniques; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists

2001
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 101, Issue:2

    Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1992
Effects of ketanserin and mianserin on delayed neuronal death induced by cerebral ischemia in Mongolian gerbils.
    Psychopharmacology, 1992, Volume: 109, Issue:3

    Topics: Analysis of Variance; Animals; Behavior, Animal; Brain Ischemia; Cell Death; Gerbillinae; Hippocampus; Ketanserin; Male; Mianserin; Neurons; Scopolamine; Time Factors

1992
Diverse actions of 5-hydroxytryptamine on frog spinal dorsal horn neurons in vitro.
    Neuroscience, 1992, Volume: 49, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dioxanes; Electric Stimulation; Evoked Potentials; Female; In Vitro Techniques; Ketanserin; Kinetics; Male; Membrane Potentials; Methysergide; Mianserin; Neurons; Rana pipiens; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Synapses; Tetrodotoxin; Tropanes

1992
Phosphoinositide hydrolysis linked 5-HT2 receptors in fibroblasts from choroid plexus.
    Brain research, 1991, Jun-28, Volume: 552, Issue:2

    Topics: Animals; Cells, Cultured; Choroid Plexus; DOM 2,5-Dimethoxy-4-Methylamphetamine; Fibroblasts; Haloperidol; Hydrolysis; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Phosphatidylinositols; Prazosin; Rabbits; Receptors, Serotonin; Serotonin; Spiperone

1991
Visual recognition memory in squirrel monkeys: effects of serotonin antagonists on baseline and hypoxia-induced performance deficits.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:4

    Topics: Animals; Avoidance Learning; Cognition; Dose-Response Relationship, Drug; Hypoxia; Ketanserin; Male; Memory; Mianserin; Piperidines; Psychomotor Performance; Reinforcement Schedule; Saimiri; Serotonin Antagonists

1991
The serotonin antagonist mianserin improves functional recovery following experimental spinal trauma.
    Annals of neurology, 1991, Volume: 30, Issue:4

    Topics: Analysis of Variance; Animals; Cyproheptadine; Dose-Response Relationship, Drug; Ketanserin; Male; Mianserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spinal Cord Injuries

1991
Guinea pig pulmonary responses to serotonin (5-HT) and related agonists.
    Annals of the New York Academy of Sciences, 1991, Volume: 629

    Topics: Animals; Ergolines; Guinea Pigs; Ketanserin; Lung; Mianserin; Respiratory Function Tests; Serotonin

1991
Analgesic profile of centrally administered 2-methylserotonin against acute pain in rats.
    European journal of pharmacology, 1991, Jun-25, Volume: 199, Issue:2

    Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Mianserin; Motor Activity; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Respiration; Serotonin; Serotonin Antagonists; Tropanes

1991
Distribution of dopaminergic receptors in the primate cerebral cortex: quantitative autoradiographic analysis using [3H]raclopride, [3H]spiperone and [3H]SCH23390.
    Neuroscience, 1991, Volume: 40, Issue:3

    Topics: Animals; Benzazepines; Brain Mapping; Cerebral Cortex; Ketanserin; Macaca mulatta; Mianserin; Raclopride; Receptors, Dopamine; Salicylamides; Species Specificity; Spiperone

1991
[3H]ketanserin binds to non-5-HT2 sites in rabbit cerebral cortex and neostriatum.
    Neurochemical research, 1990, Volume: 15, Issue:5

    Topics: Animals; Binding, Competitive; Caudate Nucleus; Cell Membrane; Cerebral Cortex; Corpus Striatum; Frontal Lobe; Ketanserin; Kinetics; Male; Methysergide; Mianserin; Piperidines; Putamen; Rabbits; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1990
Adaptation of brain 5HT2 receptors after mianserin treatment: receptor sensitivity, not receptor binding, more accurately correlates with behavior.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:2

    Topics: Animals; Brain; Dose-Response Relationship, Drug; Injections, Subcutaneous; Ketanserin; Male; Mianserin; Phosphatidylinositols; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin

1990
Serotonin enhances oestradiol production by hamster preovulatory follicles in vitro: effects of experimentally induced atresia.
    The Journal of endocrinology, 1990, Volume: 125, Issue:3

    Topics: Androstenedione; Animals; Cells, Cultured; Cricetinae; Estradiol; Female; Follicular Atresia; Follicular Phase; Granulosa Cells; Ketanserin; Mesocricetus; Mianserin; Organ Culture Techniques; Ovarian Follicle; Phenobarbital; Serotonin

1990
Mechanisms involved in the action of serotonin-induced stimulation of progesterone production by bovine luteal cells in vitro.
    Molecular and cellular endocrinology, 1987, Volume: 51, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cattle; Corpus Luteum; Estrus; Female; In Vitro Techniques; Ketanserin; Mianserin; Progesterone; Receptors, Serotonin; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes

1987
Lesioning and recovery of the serotoninergic projections to the hippocampus.
    Brain research, 1987, May-19, Volume: 411, Issue:2

    Topics: Animals; Behavior, Animal; Brain; Hippocampus; Hydroxyindoleacetic Acid; Imipramine; Ketanserin; Kinetics; Mianserin; Nerve Regeneration; Neural Pathways; Rats; Receptors, Serotonin; Serotonin; Synaptosomes

1987
Single or repeated administrations of SCH 23390 fail to affect serotonergic neurotransmission.
    Neuroscience letters, 1988, Oct-05, Volume: 92, Issue:2

    Topics: Animals; Benzazepines; Dose-Response Relationship, Drug; Frontal Lobe; Hydroxyindoleacetic Acid; Ketanserin; Male; Methysergide; Mianserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Synaptic Transmission; Synaptosomes

1988
Manipulation of serotonin protects against an hypoxia-induced deficit of a passive avoidance response in rats.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:1

    Topics: Animals; Avoidance Learning; Cyproheptadine; Dose-Response Relationship, Drug; Fluoxetine; Hypoxia; Ketanserin; Male; Methysergide; Mianserin; Rats; Rats, Inbred Strains; Serotonin; Zimeldine

1989
5-Hydroxytryptamine acts at 5-HT2 receptors to decrease potassium conductance in rat nucleus accumbens neurones.
    The Journal of physiology, 1989, Volume: 417

    Topics: Animals; In Vitro Techniques; Ketanserin; Mianserin; Neurons; Nucleus Accumbens; Potassium Channels; Rats; Receptors, Serotonin; Septal Nuclei; Serotonin; Tetrodotoxin

1989
Stereoselective blockade of central [3H]5-hydroxytryptamine binding to multiple sites (5-HT1A, 5-HT1B and 5-HT1C) by mianserin and propranolol.
    The Journal of pharmacy and pharmacology, 1987, Volume: 39, Issue:8

    Topics: Animals; Brain Chemistry; Corpus Striatum; In Vitro Techniques; Ketanserin; Male; Membranes; Mianserin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Stereoisomerism

1987
A unique serotonin receptor in choroid plexus is linked to phosphatidylinositol turnover.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:11

    Topics: Animals; Cerebral Cortex; Choroid Plexus; In Vitro Techniques; Ketanserin; Mianserin; Phosphatidylinositols; Piperidines; Rats; Receptors, Serotonin; Spiperone

1986
Different effects of serotonin antagonists on 3H-mianserin and 3H-ketanserin recognition sites.
    Life sciences, 1985, Feb-25, Volume: 36, Issue:8

    Topics: Animals; Binding Sites; Cerebral Cortex; Cyclic AMP; Dibenzazepines; Ketanserin; Kinetics; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin Antagonists; Time Factors

1985
Regulation of serotonin-stimulated phosphoinositide hydrolysis: relation to the serotonin 5-HT-2 binding site.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1986, Volume: 6, Issue:12

    Topics: 5,7-Dihydroxytryptamine; Animals; Binding, Competitive; Cerebral Cortex; Fenclonine; Hydrolysis; Ketanserin; Male; Mianserin; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1986
Studies into the dual effects of serotonergic pharmacological agents on female sexual behaviour in the rat: preliminary evidence that endogenous 5HT is stimulatory.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:1

    Topics: 5-Hydroxytryptophan; Adrenalectomy; Alanine; Animals; Castration; Cinanserin; Female; Ketanserin; Metergoline; Methysergide; Mianserin; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal; Zimeldine

1985
In vivo binding of 125I-LSD to serotonin 5-HT2 receptors in mouse brain.
    Life sciences, 1985, Aug-19, Volume: 37, Issue:7

    Topics: Animals; Binding, Competitive; Brain; Cinanserin; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Mice; Piperidines; Receptors, Serotonin; Spiperone; Time Factors; Tissue Distribution

1985
Serotonin-induced contraction of canine saphenous vein: mediation by 5-HT1 receptors.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 274, Issue:2

    Topics: Animals; Clonidine; Dogs; Drug Interactions; Emetics; In Vitro Techniques; Ketanserin; Mianserin; Muscle Contraction; Naphthols; Piperidines; Receptors, Serotonin; Saphenous Vein; Serotonin; Yohimbine

1985
Effect of serotonin on the motility of smooth muscles in teats of lactating cows.
    The Journal of dairy research, 1985, Volume: 52, Issue:3

    Topics: Animals; Cattle; Female; Ketanserin; Lactation; Mammary Glands, Animal; Methysergide; Mianserin; Milk Ejection; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Piperidines; Pregnancy; Serotonin; Serotonin Antagonists

1985
Differential antagonism of the initial fast and secondary slow contractile responses of the rat isolated aorta to 5-hydroxytryptamine by mianserin and ketanserin.
    Journal of autonomic pharmacology, 1987, Volume: 7, Issue:2

    Topics: Animals; Drug Interactions; In Vitro Techniques; Ketanserin; Male; Mianserin; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists

1987
The subtype of serotonin (5-HT) receptors in the rat pulmonary artery.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 288, Issue:2

    Topics: Animals; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Mianserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Pizotyline; Prazosin; Pulmonary Artery; Rats; Receptors, Serotonin

1987
Different temporal effects of serotonergic antagonists on passive avoidance retention.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:3

    Topics: Animals; Avoidance Learning; Ketanserin; Male; Memory; Mianserin; Mice; Piperidines; Receptors, Serotonin; Retention, Psychology; Serotonin Antagonists; Time Factors

1987
Effects of the serotonin antagonists, cyproheptadine, ketanserin and mianserin, on cyclic flow reductions in stenosed canine coronary arteries.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:2

    Topics: Adenosine Diphosphate; Animals; Blood Flow Velocity; Coronary Circulation; Cyproheptadine; Dogs; Epinephrine; Female; Hemodynamics; Ketanserin; Male; Mianserin; Periodicity; Platelet Aggregation; Serotonin

1987
Unusual acute effects of antidepressants and neuroleptics on S2-serotonergic receptors.
    Life sciences, 1983, Dec-19, Volume: 33, Issue:25

    Topics: Amoxapine; Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Fenclonine; Frontal Lobe; Ketanserin; Loxapine; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1983
On the neurotoxicity of chlordecone: a role for gamma-aminobutyric acid and serotonin.
    Brain research, 1984, Jun-11, Volume: 303, Issue:1

    Topics: Acetylcholine; Animals; Binding Sites; Brain; Chlordecone; gamma-Aminobutyric Acid; Insecticides; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Spiperone

1984
Comparison of iprindole, imipramine and mianserin action on brain serotonergic and beta adrenergic receptors.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 229, Issue:3

    Topics: Animals; Axons; Brain; Cyclic AMP; Dibenzazepines; Imipramine; Indoles; Iprindole; Ketanserin; Male; Mianserin; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin

1984
Autoradiographic mapping of spirodecanone binding-sites in the hippocampal region of the rat. Evidence for a localization on intrinsic neurons.
    Neuroscience letters, 1984, May-04, Volume: 46, Issue:2

    Topics: Animals; Autoradiography; Binding, Competitive; Brain Mapping; Butyrophenones; Haloperidol; Hippocampus; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Serotonin; Spiperone; Tetrahydronaphthalenes

1984
Temperature-sensitive high affinity [3H]serotonin binding: characterization and effects of antidepressant treatment.
    Life sciences, 1984, Aug-13, Volume: 35, Issue:7

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Ketanserin; Kinetics; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Temperature; Tritium

1984
Some behavioral effects of hallucinogens are mediated by a postsynaptic serotonergic action: evidence from single unit studies in freely moving cats.
    European journal of pharmacology, 1984, May-18, Volume: 101, Issue:1-2

    Topics: Animals; Apomorphine; Behavior, Animal; Cats; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Female; Hallucinogens; Ketanserin; Lisuride; Lysergic Acid Diethylamide; Metergoline; Mianserin; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Synapses

1984
Differences in the regulatory adaptation of the 5HT recognition sites labelled by 3H-mianserin or 3H-ketanserin.
    Neuropharmacology, 1983, Volume: 22, Issue:1

    Topics: Animals; Axons; Dibenzazepines; Hippocampus; Imipramine; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Synapses; Tritium

1983
Serotonin 5-HT2C receptor stimulates cyclic GMP formation in choroid plexus.
    Journal of neurochemistry, 1995, Volume: 64, Issue:1

    Topics: Animals; Cattle; Choroid Plexus; Cyclic GMP; Ketanserin; Mianserin; Phosphatidylinositols; Receptors, Serotonin; Spiperone; Swine

1995
Serotonin increases DNA synthesis in rat proximal and distal pulmonary vascular smooth muscle cells in culture.
    The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 1

    Topics: Animals; Binding, Competitive; Blotting, Northern; Calcium; Cells, Cultured; DNA; Ketanserin; Lung; Lysergic Acid Diethylamide; Mianserin; Muscle, Smooth, Vascular; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA, Messenger; Serotonin; Thymidine

1994
The quipazine- and TFMPP-increased conditioned avoidance response in rats: role of 5HT1C/5-HT2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: Animals; Avoidance Learning; Conditioning, Operant; Ketanserin; Male; Mianserin; Nadolol; Pindolol; Piperazines; Prazosin; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tropanes

1993
Characterization of mianserin neuroprotection in experimental spinal trauma: dose/route response and late treatment.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Administration Routes; Edema; Ketanserin; Male; Mianserin; Oxidation-Reduction; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord Diseases; Spinal Cord Injuries

1994
Chronic fluoxetine treatment upregulates 5-HT uptake sites and 5-HT2 receptors in rat brain: an autoradiographic study.
    Synapse (New York, N.Y.), 1993, Volume: 14, Issue:4

    Topics: Animals; Autoradiography; Brain Chemistry; Fluoxetine; Image Processing, Computer-Assisted; Ketanserin; Male; Mianserin; Paroxetine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Up-Regulation

1993
Effects of agonists, partial agonists, and antagonists on the regulation of 5-hydroxytryptamine2 receptors in P11 cells.
    Molecular pharmacology, 1993, Volume: 43, Issue:5

    Topics: Amphetamines; Animals; Down-Regulation; Hydrolysis; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Phosphatidylinositols; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tumor Cells, Cultured

1993
Cholecystokinin-induced satiety depends on activation of 5-HT1C receptors.
    The American journal of physiology, 1993, Volume: 264, Issue:1 Pt 2

    Topics: Animals; Eating; Ketanserin; Male; Mianserin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Satiation; Serotonin Antagonists; Sincalide; Tropanes

1993
Effects of Antidepressants and antipsychotics on the 5HT2 receptor-mediated signal transducing system in human platelets.
    Psychopharmacology, 1995, Volume: 121, Issue:4

    Topics: Adult; Amoxapine; Antidepressive Agents; Antipsychotic Agents; Binding, Competitive; Blood Platelets; Female; Humans; Ketanserin; Male; Mianserin; Middle Aged; Signal Transduction

1995
Effects of mianserin and ketanserin on lordosis behavior after systemic treatment or infusion into the ventromedial nucleus of the hypothalamus.
    Brain research, 1996, Apr-29, Volume: 718, Issue:1-2

    Topics: Animals; Brain; Estradiol; Female; Injections; Ketanserin; Male; Mianserin; Ovariectomy; Posture; Proestrus; Progesterone; Rats; Rats, Inbred F344; Serotonin Antagonists; Sexual Behavior, Animal; Vagina; Ventromedial Hypothalamic Nucleus

1996
Functional reconstitution in situ of 5-hydroxytryptamine2c (5HT2c) receptors with alphaq and inverse agonism of 5HT2c receptor antagonists.
    The Journal of biological chemistry, 1996, Sep-13, Volume: 271, Issue:37

    Topics: Animals; Binding, Competitive; Cattle; Cell Line; Decapodiformes; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Ketanserin; Mianserin; Photoreceptor Cells, Invertebrate; Rats; Receptor, Serotonin, 5-HT2C; Receptors, Cell Surface; Receptors, Serotonin; Recombinant Proteins; Serotonin

1996
Behavioral effects of (+/-)-1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane, (DOI) in the elevated plus-maze test.
    Life sciences, 1995, Nov-17, Volume: 57, Issue:26

    Topics: Amphetamines; Animals; Behavior, Animal; Flumazenil; GABA Modulators; Hallucinogens; Ketanserin; Male; Mianserin; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Inbred ICR; Motor Activity; Rats; Receptors, Serotonin; Serotonin Antagonists

1995
Effects of 5HT2 receptor antagonists on responses to potassium depolarization in rat isolated aorta.
    Clinical and experimental pharmacology & physiology, 1997, Volume: 24, Issue:1

    Topics: Animals; Aorta, Thoracic; Cinnarizine; Cyproheptadine; Diltiazem; Drug Synergism; Felodipine; Female; In Vitro Techniques; Ketanserin; Male; Mianserin; Muscle Contraction; Nifedipine; Potassium; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reproducibility of Results; Ritanserin; Serotonin Antagonists; Verapamil

1997
Mianserin-induced down-regulation of human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors stably expressed in the human neuroblastoma cell line SH-SY5Y.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: Cell Membrane; DNA, Complementary; Down-Regulation; Ergolines; Humans; Ketanserin; Kinetics; Mianserin; Neuroblastoma; Phosphatidylinositols; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Serotonin; Time Factors; Transfection; Tumor Cells, Cultured

1997
NMDA receptor-mediated oscillatory activity in the neonatal rat spinal cord is serotonin dependent.
    Journal of neurophysiology, 1998, Volume: 79, Issue:5

    Topics: Acetylcholine; Animals; Animals, Newborn; Biological Clocks; Edrophonium; Hindlimb; Ketanserin; Locomotion; Mianserin; Motor Activity; Motor Neurons; N-Methylaspartate; Parasympathomimetics; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrodotoxin

1998
Neurochemical effects of the enantiomers of mirtazapine in normal rats.
    European journal of pharmacology, 1998, Sep-04, Volume: 356, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Antidepressive Agents, Tricyclic; Body Temperature; Injections, Intraperitoneal; Ketanserin; Male; Mianserin; Mirtazapine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism

1998
GR 127935 and (+)-WAY 100135 do not affect TFMPP-induced inhibition of 5-HT synthesis in the midbrain and hippocampus of Wistar-Kyoto rats.
    Neuropharmacology, 1998, Volume: 37, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Hippocampus; Idazoxan; Ketanserin; Male; Mesencephalon; Mianserin; Nerve Endings; Oxadiazoles; Piperazines; Rats; Rats, Inbred WKY; Rats, Wistar; Reserpine; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Tryptophan Hydroxylase

1998
Effect of 5-HT2 receptor antagonists on a cranial nerve reflex in the rabbit: evidence for inverse agonism.
    Psychopharmacology, 1999, Volume: 141, Issue:2

    Topics: Animals; Cranial Nerves; Ergolines; Female; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Piperidines; Rabbits; Receptors, Serotonin; Reflex; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Long-term treatment with antidepressants increases glucocorticoid receptor binding and gene expression in cultured rat hippocampal neurones.
    Journal of neuroendocrinology, 1999, Volume: 11, Issue:11

    Topics: Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cells, Cultured; Desipramine; Dexamethasone; Gene Expression Regulation; Haloperidol; Hippocampus; Ketanserin; Mianserin; Neurons; Paroxetine; Phentolamine; Propranolol; Radioligand Assay; Rats; Receptors, Glucocorticoid; Receptors, Mineralocorticoid; RNA, Messenger; Sulpiride; Transcription, Genetic; Tritium

1999
Regulation of 5-HT(2A) receptor mRNA levels and binding sites in rat frontal cortex by the agonist DOI and the antagonist mianserin.
    Neuropharmacology, 2000, Aug-23, Volume: 39, Issue:11

    Topics: Amphetamines; Animals; Frontal Lobe; Ketanserin; Male; Mianserin; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists; Serotonin Receptor Agonists

2000
5-HT2 receptor antagonists given in the acute withdrawal from daily cocaine injections can reverse established sensitization.
    European journal of pharmacology, 2002, Oct-25, Volume: 453, Issue:2-3

    Topics: Animals; Behavior, Animal; Clozapine; Cocaine; Injections; Ketanserin; Male; Mianserin; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Substance Withdrawal Syndrome

2002
Serotonergic regulation of the central heart auricles of Sepia officinalis L. (Mollusca, Cephalopoda).
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 2004, Volume: 138, Issue:1

    Topics: Animals; Atrial Function; Dose-Response Relationship, Drug; Fluorescence; Heart Atria; In Vitro Techniques; Ketanserin; Mianserin; Mollusca; Myocardial Contraction; Piperazines; Serotonin; Serotonin Antagonists

2004
Serotonin modifies the sensitivity of the male silkmoth to pheromone.
    The Journal of experimental biology, 2004, Volume: 207, Issue:Pt 14

    Topics: Analysis of Variance; Animals; Bombyx; Brain; Chromatography, High Pressure Liquid; Circadian Rhythm; Dose-Response Relationship, Drug; Ketanserin; Male; Mianserin; Olfactory Bulb; Olfactory Pathways; Serotonin; Serotonin Antagonists; Sex Attractants; Time Factors

2004
Suppressive effects of isorhynchophylline on 5-HT2A receptor function in the brain: behavioural and electrophysiological studies.
    European journal of pharmacology, 2005, Jul-11, Volume: 517, Issue:3

    Topics: Alkaloids; Aminopyridines; Animals; Behavior, Animal; Brain; Dose-Response Relationship, Drug; Female; Indole Alkaloids; Ketanserin; Male; Membrane Potentials; Methoxydimethyltryptamines; Mianserin; Mice; Mice, Inbred ICR; Motor Activity; Oocytes; Oxindoles; Patch-Clamp Techniques; Piperazines; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Xenopus

2005
Zimelidine decreases seizure susceptibility in stressed mice.
    Journal of neural transmission (Vienna, Austria : 1996), 2006, Volume: 113, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anticonvulsants; Behavior, Animal; Convulsants; Ketanserin; Male; Mianserin; Mice; Mice, Inbred CBA; Phenols; Picrotoxin; Piperazines; Pyridines; Seizures; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Stress, Psychological; Sulfonamides; Swimming; Zimeldine

2006
Nullifying drug-induced sensitization: behavioral and electrophysiological evaluations of dopaminergic and serotonergic ligands in methamphetamine-sensitized rats.
    Drug and alcohol dependence, 2007, Jan-05, Volume: 86, Issue:1

    Topics: Action Potentials; Adrenergic Agents; Adrenergic alpha-Antagonists; Animals; Dopamine; Electrochemistry; Globus Pallidus; Ketanserin; Locomotion; Male; Methamphetamine; Mianserin; Microelectrodes; Mirtazapine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Receptors, Dopamine D1; Receptors, Serotonin; Serotonin; Serotonin Antagonists

2007
Reversal of long-term methamphetamine sensitization by combination of pergolide with ondansetron or ketanserin, but not mirtazapine.
    Behavioural brain research, 2011, Sep-30, Volume: 223, Issue:1

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Infusion Pumps, Implantable; Ketanserin; Male; Methamphetamine; Mianserin; Mirtazapine; Ondansetron; Pergolide; Rats; Rats, Sprague-Dawley

2011
Evaluation of 5-HT2A and mGlu2/3 receptors in postmortem prefrontal cortex of subjects with major depressive disorder: effect of antidepressant treatment.
    Neuropharmacology, 2014, Volume: 86

    Topics: Amino Acids; Animals; Antidepressive Agents; Citalopram; Depressive Disorder, Major; Down-Regulation; Female; Humans; Ketanserin; Male; Mianserin; Middle Aged; Mirtazapine; Morpholines; Prefrontal Cortex; Radioligand Assay; Rats, Sprague-Dawley; Reboxetine; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; RNA, Messenger; Tritium; Xanthenes

2014
Mirtazapine and ketanserin alter preference for gambling-like schedules of reinforcement in rats.
    Progress in neuro-psychopharmacology & biological psychiatry, 2017, 07-03, Volume: 77

    Topics: Animals; Choice Behavior; Decision Making; Gambling; Ketanserin; Male; Mianserin; Mirtazapine; Rats; Reinforcement Schedule; Reward; Self Stimulation

2017