ketanserin has been researched along with mianserin in 84 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 28 (33.33) | 18.7374 |
1990's | 40 (47.62) | 18.2507 |
2000's | 11 (13.10) | 29.6817 |
2010's | 5 (5.95) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Amlaiky, N; Boschert, U; Hen, R; Maroteaux, L; Plassat, JL; Saudou, F | 1 |
Glennon, RA | 2 |
Janssen, CG; Laduron, PM; Thijssen, JB; Van Dun, J; Wouters, W | 1 |
Andrews, PR; Craik, DJ; Martin, JL | 1 |
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR | 1 |
Amlaiky, N; Hen, R; Plassat, JL | 1 |
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP | 1 |
Baez, M; Kursar, JD; Lucaites, VL; Nelson, DL; Sasso, DA; Wainscott, DB | 1 |
Egan, CT; Herrick-Davis, K; Teitler, M | 1 |
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP | 1 |
Booth, RG; Brown, RL; Bucholtz, EC; Tropsha, A; Wyrick, SD | 1 |
Itoh, H; Muramatsu, I; Taniguchi, T; Yoshio, R | 1 |
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A | 1 |
Araki, H; Karasawa, Y; Otomo, S | 1 |
Miletic, V; Tan, H | 1 |
Barker, EL; Burris, KD; Sanders-Bush, E | 1 |
DeNoble, KF; DeNoble, VJ; Reigel, AL; Schrack, LM | 1 |
Agresta, CA; Freeman, GM; Liu, ZJ; Maitland-Heriot, RP; Puniak, MA; Salzman, SK | 1 |
Buckner, CK; Dea, D; Krell, RD; Liberati, N | 1 |
Giordano, J | 1 |
Gallager, DW; Goldman-Rakic, PS; Lidow, MS; Rakic, P | 1 |
Dewar, KM; Lima, L; Reader, TA | 1 |
Barrett, RJ; Sanders-Bush, E; Smith, RL | 1 |
Horst, D; Nakamura, Y; Saville, L; Terranova, PF; Uilenbroek, JT | 1 |
Battista, PJ; Condon, WA; Rexroad, CE | 1 |
Beni, M; Carla, V; Consolazione, A; Dall'Olio, R; Gandolfi, O; Lombardi, G; Moroni, F; Pellegrini-Giampietro, DE | 1 |
Dall'Olio, R; Gandolfi, O; Roncada, P | 1 |
DeNoble, VJ; Spencer, KR; Strek, KF | 1 |
North, RA; Uchimura, N | 1 |
Alexander, BS; Wood, MD | 1 |
Conn, PJ; Hartig, PR; Hoffman, BJ; Sanders-Bush, E | 1 |
Barbaccia, ML; Costa, E; Gandolfi, O | 2 |
Conn, PJ; Sanders-Bush, E | 1 |
Hole, DR; Hunter, AJ; Wilson, CA | 1 |
Frost, JJ; Hartig, PR; Scheffel, U; Wagner, HN | 1 |
Doğan, N; Ilhan, M; Kayaalp, SO; Tuncer, M | 1 |
Burvenich, C; Peeters, G; Vandeputte-Van Messon, G | 1 |
Doggrell, SA | 1 |
Kayaalp, SO; Tuncer, M; Uma, S | 1 |
Altman, HJ; Normile, HJ | 1 |
Bush, LR | 1 |
Helmeste, DM; Tang, SW | 2 |
Cheney, DL; Costa, E; Gandolfi, O; Hong, JS | 1 |
Köhler, C | 1 |
Anthony, M | 1 |
Heym, J; Jacobs, BL; Rasmussen, K | 1 |
Barbaccia, ML; Chuang, DM; Costa, E; Gandolfi, O | 1 |
Hartig, PR; Hoffman, BJ; Kaufman, MJ | 1 |
Altuğ, U; Erol, D; Germiyanoğlu, C; Gürdal, M; Kurt, U; Ozkardeş, H | 1 |
Blakely, RD; Davies, P; Pitt, BR; Reynolds, I; Steve, AR; Weng, W | 1 |
Ageel, AM; Alhaider, AA; Ginawi, OT | 1 |
Agresta, CA; Azim, S; Chavin, J; Kelly, G; Puniak, MA; Salzman, SK; Wang, L | 1 |
Hrdina, PD; Vu, TB | 1 |
Ferry, RC; Molinoff, PB; Unsworth, CD | 1 |
Gibbs, J; Greenberg, D; Poeschla, B; Simansky, KJ; Smith, GP | 1 |
Kaneko, M; Kumashiro, H; Mashiko, H; Ohsuka, N | 1 |
Caldarola-Pastuszka, M; Colon, L; Cox, A; Uphouse, L; Wolf, A | 1 |
Hartman, JL; Northup, JK | 1 |
Bishop-Robinson, C; Darmani, NA; Onaivi, ES; Sanders-Bush, E | 1 |
Marwood, JF; Okoro, EO | 1 |
Elliott, JM; Newton, RA | 1 |
Cowley, KC; MacLean, JN; Schmidt, BJ | 1 |
Burrows, GD; McGrath, C; Norman, TR | 1 |
Aguerre, S; Chaouloff, F; Mormede, P | 1 |
Harvey, JA; Hood, H; Romano, AG; Welsh, SE | 1 |
Fujiseki, Y; Inagaki, C; Kinoshita, T; Okugawa, G; Omori, K; Suzukawa, J | 1 |
Anji, A; Bryan, GL; Hensler, JG; Kumari, M; Sullivan Hanley, NR | 1 |
Davidson, C; Ellinwood, EH; Lazarus, C; Lee, TH; Xiong, X | 1 |
Lehr, T; Schipp, R | 1 |
Gatellier, L; Kanzaki, R; Nagao, T | 1 |
Matsumoto, K; Morishige, R; Murakami, Y; Sakakibara, I; Takayama, H; Tohda, M; Watanabe, H | 1 |
Pericić, D; Strac, DS; Vlainić, J | 1 |
Angle, JM; Dallimore, JE; Mackie, AR; McDaid, J; Mickiewicz, AL; Napier, TC; Shen, F; Tedford, CE | 1 |
Bhatia, KS; Fowler, JC; Lee, TH; Szabo, ST; Wetsel, WC | 1 |
Callado, LF; Díez-Alarcia, R; González-Maeso, J; Meana, JJ; Miranda-Azpiazu, P; Morentin, B; Muguruza, C | 1 |
Celeste, T; Persons, AL; Tedford, SE | 1 |
3 review(s) available for ketanserin and mianserin
Article | Year |
---|---|
Central serotonin receptors as targets for drug research.
Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin | 1987 |
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists | 2003 |
Serotonin antagonists.
Topics: Cyproheptadine; Depression; Ergotamine; Humans; Hypertension; Ketanserin; Lisuride; Methysergide; Mianserin; Migraine Disorders; Piperidines; Pizotyline; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Diseases | 1984 |
1 trial(s) available for ketanserin and mianserin
Article | Year |
---|---|
The efficacy of anti-serotoninergic agents in the treatment of erectile dysfunction.
Topics: Adult; Aged; Double-Blind Method; Erectile Dysfunction; Humans; Ketanserin; Male; Mianserin; Middle Aged; Trazodone | 1994 |
80 other study(ies) available for ketanserin and mianserin
Article | Year |
---|---|
Mouse 5HT1B serotonin receptor: cloning, functional expression, and localization in motor control centers.
Topics: 3T3 Cells; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Cerebellum; Corpus Striatum; Gene Expression; Genes; GTP-Binding Proteins; Mice; Molecular Sequence Data; Nucleic Acid Hybridization; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Purkinje Cells; Receptors, Serotonin; RNA, Messenger; Serotonin | 1992 |
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Frontal Lobe; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1986 |
Functional group contributions to drug-receptor interactions.
Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship | 1984 |
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection | 1993 |
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Cyclic AMP; DNA; Drosophila; Enzyme Activation; Humans; Intestinal Mucosa; Mice; Molecular Sequence Data; Myocardium; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists | 1993 |
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid | 1997 |
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.
Topics: Adrenergic alpha-Antagonists; Benzofurans; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Imidazoles; Radioligand Assay; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Yohimbine | 1998 |
Creation of a constitutively activated state of the 5-hydroxytryptamine2A receptor by site-directed mutagenesis: inverse agonist activity of antipsychotic drugs.
Topics: Animals; Antipsychotic Agents; COS Cells; Mutagenesis, Site-Directed; Phosphatidylinositols; Protein Conformation; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship | 1998 |
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone | 1999 |
Synthesis, evaluation, and comparative molecular field analysis of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for histamine H(1) receptors.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ligands; Models, Molecular; Pyrilamine; Radioligand Assay; Structure-Activity Relationship; Tetrahydronaphthalenes | 1999 |
Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.
Topics: Animals; Aorta, Thoracic; Carotid Arteries; Dogs; Humans; Male; Organ Culture Techniques; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists | 2001 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Physical binding pocket induction for affinity prediction.
Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1992 |
Effects of ketanserin and mianserin on delayed neuronal death induced by cerebral ischemia in Mongolian gerbils.
Topics: Analysis of Variance; Animals; Behavior, Animal; Brain Ischemia; Cell Death; Gerbillinae; Hippocampus; Ketanserin; Male; Mianserin; Neurons; Scopolamine; Time Factors | 1992 |
Diverse actions of 5-hydroxytryptamine on frog spinal dorsal horn neurons in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dioxanes; Electric Stimulation; Evoked Potentials; Female; In Vitro Techniques; Ketanserin; Kinetics; Male; Membrane Potentials; Methysergide; Mianserin; Neurons; Rana pipiens; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Synapses; Tetrodotoxin; Tropanes | 1992 |
Phosphoinositide hydrolysis linked 5-HT2 receptors in fibroblasts from choroid plexus.
Topics: Animals; Cells, Cultured; Choroid Plexus; DOM 2,5-Dimethoxy-4-Methylamphetamine; Fibroblasts; Haloperidol; Hydrolysis; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Phosphatidylinositols; Prazosin; Rabbits; Receptors, Serotonin; Serotonin; Spiperone | 1991 |
Visual recognition memory in squirrel monkeys: effects of serotonin antagonists on baseline and hypoxia-induced performance deficits.
Topics: Animals; Avoidance Learning; Cognition; Dose-Response Relationship, Drug; Hypoxia; Ketanserin; Male; Memory; Mianserin; Piperidines; Psychomotor Performance; Reinforcement Schedule; Saimiri; Serotonin Antagonists | 1991 |
The serotonin antagonist mianserin improves functional recovery following experimental spinal trauma.
Topics: Analysis of Variance; Animals; Cyproheptadine; Dose-Response Relationship, Drug; Ketanserin; Male; Mianserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spinal Cord Injuries | 1991 |
Guinea pig pulmonary responses to serotonin (5-HT) and related agonists.
Topics: Animals; Ergolines; Guinea Pigs; Ketanserin; Lung; Mianserin; Respiratory Function Tests; Serotonin | 1991 |
Analgesic profile of centrally administered 2-methylserotonin against acute pain in rats.
Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Mianserin; Motor Activity; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Respiration; Serotonin; Serotonin Antagonists; Tropanes | 1991 |
Distribution of dopaminergic receptors in the primate cerebral cortex: quantitative autoradiographic analysis using [3H]raclopride, [3H]spiperone and [3H]SCH23390.
Topics: Animals; Benzazepines; Brain Mapping; Cerebral Cortex; Ketanserin; Macaca mulatta; Mianserin; Raclopride; Receptors, Dopamine; Salicylamides; Species Specificity; Spiperone | 1991 |
[3H]ketanserin binds to non-5-HT2 sites in rabbit cerebral cortex and neostriatum.
Topics: Animals; Binding, Competitive; Caudate Nucleus; Cell Membrane; Cerebral Cortex; Corpus Striatum; Frontal Lobe; Ketanserin; Kinetics; Male; Methysergide; Mianserin; Piperidines; Putamen; Rabbits; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Adaptation of brain 5HT2 receptors after mianserin treatment: receptor sensitivity, not receptor binding, more accurately correlates with behavior.
Topics: Animals; Brain; Dose-Response Relationship, Drug; Injections, Subcutaneous; Ketanserin; Male; Mianserin; Phosphatidylinositols; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1990 |
Serotonin enhances oestradiol production by hamster preovulatory follicles in vitro: effects of experimentally induced atresia.
Topics: Androstenedione; Animals; Cells, Cultured; Cricetinae; Estradiol; Female; Follicular Atresia; Follicular Phase; Granulosa Cells; Ketanserin; Mesocricetus; Mianserin; Organ Culture Techniques; Ovarian Follicle; Phenobarbital; Serotonin | 1990 |
Mechanisms involved in the action of serotonin-induced stimulation of progesterone production by bovine luteal cells in vitro.
Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cattle; Corpus Luteum; Estrus; Female; In Vitro Techniques; Ketanserin; Mianserin; Progesterone; Receptors, Serotonin; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes | 1987 |
Lesioning and recovery of the serotoninergic projections to the hippocampus.
Topics: Animals; Behavior, Animal; Brain; Hippocampus; Hydroxyindoleacetic Acid; Imipramine; Ketanserin; Kinetics; Mianserin; Nerve Regeneration; Neural Pathways; Rats; Receptors, Serotonin; Serotonin; Synaptosomes | 1987 |
Single or repeated administrations of SCH 23390 fail to affect serotonergic neurotransmission.
Topics: Animals; Benzazepines; Dose-Response Relationship, Drug; Frontal Lobe; Hydroxyindoleacetic Acid; Ketanserin; Male; Methysergide; Mianserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Synaptic Transmission; Synaptosomes | 1988 |
Manipulation of serotonin protects against an hypoxia-induced deficit of a passive avoidance response in rats.
Topics: Animals; Avoidance Learning; Cyproheptadine; Dose-Response Relationship, Drug; Fluoxetine; Hypoxia; Ketanserin; Male; Methysergide; Mianserin; Rats; Rats, Inbred Strains; Serotonin; Zimeldine | 1989 |
5-Hydroxytryptamine acts at 5-HT2 receptors to decrease potassium conductance in rat nucleus accumbens neurones.
Topics: Animals; In Vitro Techniques; Ketanserin; Mianserin; Neurons; Nucleus Accumbens; Potassium Channels; Rats; Receptors, Serotonin; Septal Nuclei; Serotonin; Tetrodotoxin | 1989 |
Stereoselective blockade of central [3H]5-hydroxytryptamine binding to multiple sites (5-HT1A, 5-HT1B and 5-HT1C) by mianserin and propranolol.
Topics: Animals; Brain Chemistry; Corpus Striatum; In Vitro Techniques; Ketanserin; Male; Membranes; Mianserin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Stereoisomerism | 1987 |
A unique serotonin receptor in choroid plexus is linked to phosphatidylinositol turnover.
Topics: Animals; Cerebral Cortex; Choroid Plexus; In Vitro Techniques; Ketanserin; Mianserin; Phosphatidylinositols; Piperidines; Rats; Receptors, Serotonin; Spiperone | 1986 |
Different effects of serotonin antagonists on 3H-mianserin and 3H-ketanserin recognition sites.
Topics: Animals; Binding Sites; Cerebral Cortex; Cyclic AMP; Dibenzazepines; Ketanserin; Kinetics; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin Antagonists; Time Factors | 1985 |
Regulation of serotonin-stimulated phosphoinositide hydrolysis: relation to the serotonin 5-HT-2 binding site.
Topics: 5,7-Dihydroxytryptamine; Animals; Binding, Competitive; Cerebral Cortex; Fenclonine; Hydrolysis; Ketanserin; Male; Mianserin; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1986 |
Studies into the dual effects of serotonergic pharmacological agents on female sexual behaviour in the rat: preliminary evidence that endogenous 5HT is stimulatory.
Topics: 5-Hydroxytryptophan; Adrenalectomy; Alanine; Animals; Castration; Cinanserin; Female; Ketanserin; Metergoline; Methysergide; Mianserin; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal; Zimeldine | 1985 |
In vivo binding of 125I-LSD to serotonin 5-HT2 receptors in mouse brain.
Topics: Animals; Binding, Competitive; Brain; Cinanserin; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Mice; Piperidines; Receptors, Serotonin; Spiperone; Time Factors; Tissue Distribution | 1985 |
Serotonin-induced contraction of canine saphenous vein: mediation by 5-HT1 receptors.
Topics: Animals; Clonidine; Dogs; Drug Interactions; Emetics; In Vitro Techniques; Ketanserin; Mianserin; Muscle Contraction; Naphthols; Piperidines; Receptors, Serotonin; Saphenous Vein; Serotonin; Yohimbine | 1985 |
Effect of serotonin on the motility of smooth muscles in teats of lactating cows.
Topics: Animals; Cattle; Female; Ketanserin; Lactation; Mammary Glands, Animal; Methysergide; Mianserin; Milk Ejection; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Piperidines; Pregnancy; Serotonin; Serotonin Antagonists | 1985 |
Differential antagonism of the initial fast and secondary slow contractile responses of the rat isolated aorta to 5-hydroxytryptamine by mianserin and ketanserin.
Topics: Animals; Drug Interactions; In Vitro Techniques; Ketanserin; Male; Mianserin; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists | 1987 |
The subtype of serotonin (5-HT) receptors in the rat pulmonary artery.
Topics: Animals; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Mianserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Pizotyline; Prazosin; Pulmonary Artery; Rats; Receptors, Serotonin | 1987 |
Different temporal effects of serotonergic antagonists on passive avoidance retention.
Topics: Animals; Avoidance Learning; Ketanserin; Male; Memory; Mianserin; Mice; Piperidines; Receptors, Serotonin; Retention, Psychology; Serotonin Antagonists; Time Factors | 1987 |
Effects of the serotonin antagonists, cyproheptadine, ketanserin and mianserin, on cyclic flow reductions in stenosed canine coronary arteries.
Topics: Adenosine Diphosphate; Animals; Blood Flow Velocity; Coronary Circulation; Cyproheptadine; Dogs; Epinephrine; Female; Hemodynamics; Ketanserin; Male; Mianserin; Periodicity; Platelet Aggregation; Serotonin | 1987 |
Unusual acute effects of antidepressants and neuroleptics on S2-serotonergic receptors.
Topics: Amoxapine; Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Fenclonine; Frontal Lobe; Ketanserin; Loxapine; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone | 1983 |
On the neurotoxicity of chlordecone: a role for gamma-aminobutyric acid and serotonin.
Topics: Acetylcholine; Animals; Binding Sites; Brain; Chlordecone; gamma-Aminobutyric Acid; Insecticides; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Spiperone | 1984 |
Comparison of iprindole, imipramine and mianserin action on brain serotonergic and beta adrenergic receptors.
Topics: Animals; Axons; Brain; Cyclic AMP; Dibenzazepines; Imipramine; Indoles; Iprindole; Ketanserin; Male; Mianserin; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin | 1984 |
Autoradiographic mapping of spirodecanone binding-sites in the hippocampal region of the rat. Evidence for a localization on intrinsic neurons.
Topics: Animals; Autoradiography; Binding, Competitive; Brain Mapping; Butyrophenones; Haloperidol; Hippocampus; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Serotonin; Spiperone; Tetrahydronaphthalenes | 1984 |
Temperature-sensitive high affinity [3H]serotonin binding: characterization and effects of antidepressant treatment.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Ketanserin; Kinetics; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Temperature; Tritium | 1984 |
Some behavioral effects of hallucinogens are mediated by a postsynaptic serotonergic action: evidence from single unit studies in freely moving cats.
Topics: Animals; Apomorphine; Behavior, Animal; Cats; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Female; Hallucinogens; Ketanserin; Lisuride; Lysergic Acid Diethylamide; Metergoline; Mianserin; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Synapses | 1984 |
Differences in the regulatory adaptation of the 5HT recognition sites labelled by 3H-mianserin or 3H-ketanserin.
Topics: Animals; Axons; Dibenzazepines; Hippocampus; Imipramine; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Synapses; Tritium | 1983 |
Serotonin 5-HT2C receptor stimulates cyclic GMP formation in choroid plexus.
Topics: Animals; Cattle; Choroid Plexus; Cyclic GMP; Ketanserin; Mianserin; Phosphatidylinositols; Receptors, Serotonin; Spiperone; Swine | 1995 |
Serotonin increases DNA synthesis in rat proximal and distal pulmonary vascular smooth muscle cells in culture.
Topics: Animals; Binding, Competitive; Blotting, Northern; Calcium; Cells, Cultured; DNA; Ketanserin; Lung; Lysergic Acid Diethylamide; Mianserin; Muscle, Smooth, Vascular; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA, Messenger; Serotonin; Thymidine | 1994 |
The quipazine- and TFMPP-increased conditioned avoidance response in rats: role of 5HT1C/5-HT2 receptors.
Topics: Animals; Avoidance Learning; Conditioning, Operant; Ketanserin; Male; Mianserin; Nadolol; Pindolol; Piperazines; Prazosin; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tropanes | 1993 |
Characterization of mianserin neuroprotection in experimental spinal trauma: dose/route response and late treatment.
Topics: Animals; Dose-Response Relationship, Drug; Drug Administration Routes; Edema; Ketanserin; Male; Mianserin; Oxidation-Reduction; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord Diseases; Spinal Cord Injuries | 1994 |
Chronic fluoxetine treatment upregulates 5-HT uptake sites and 5-HT2 receptors in rat brain: an autoradiographic study.
Topics: Animals; Autoradiography; Brain Chemistry; Fluoxetine; Image Processing, Computer-Assisted; Ketanserin; Male; Mianserin; Paroxetine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Up-Regulation | 1993 |
Effects of agonists, partial agonists, and antagonists on the regulation of 5-hydroxytryptamine2 receptors in P11 cells.
Topics: Amphetamines; Animals; Down-Regulation; Hydrolysis; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Phosphatidylinositols; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tumor Cells, Cultured | 1993 |
Cholecystokinin-induced satiety depends on activation of 5-HT1C receptors.
Topics: Animals; Eating; Ketanserin; Male; Mianserin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Satiation; Serotonin Antagonists; Sincalide; Tropanes | 1993 |
Effects of Antidepressants and antipsychotics on the 5HT2 receptor-mediated signal transducing system in human platelets.
Topics: Adult; Amoxapine; Antidepressive Agents; Antipsychotic Agents; Binding, Competitive; Blood Platelets; Female; Humans; Ketanserin; Male; Mianserin; Middle Aged; Signal Transduction | 1995 |
Effects of mianserin and ketanserin on lordosis behavior after systemic treatment or infusion into the ventromedial nucleus of the hypothalamus.
Topics: Animals; Brain; Estradiol; Female; Injections; Ketanserin; Male; Mianserin; Ovariectomy; Posture; Proestrus; Progesterone; Rats; Rats, Inbred F344; Serotonin Antagonists; Sexual Behavior, Animal; Vagina; Ventromedial Hypothalamic Nucleus | 1996 |
Functional reconstitution in situ of 5-hydroxytryptamine2c (5HT2c) receptors with alphaq and inverse agonism of 5HT2c receptor antagonists.
Topics: Animals; Binding, Competitive; Cattle; Cell Line; Decapodiformes; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Ketanserin; Mianserin; Photoreceptor Cells, Invertebrate; Rats; Receptor, Serotonin, 5-HT2C; Receptors, Cell Surface; Receptors, Serotonin; Recombinant Proteins; Serotonin | 1996 |
Behavioral effects of (+/-)-1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane, (DOI) in the elevated plus-maze test.
Topics: Amphetamines; Animals; Behavior, Animal; Flumazenil; GABA Modulators; Hallucinogens; Ketanserin; Male; Mianserin; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Inbred ICR; Motor Activity; Rats; Receptors, Serotonin; Serotonin Antagonists | 1995 |
Effects of 5HT2 receptor antagonists on responses to potassium depolarization in rat isolated aorta.
Topics: Animals; Aorta, Thoracic; Cinnarizine; Cyproheptadine; Diltiazem; Drug Synergism; Felodipine; Female; In Vitro Techniques; Ketanserin; Male; Mianserin; Muscle Contraction; Nifedipine; Potassium; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reproducibility of Results; Ritanserin; Serotonin Antagonists; Verapamil | 1997 |
Mianserin-induced down-regulation of human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors stably expressed in the human neuroblastoma cell line SH-SY5Y.
Topics: Cell Membrane; DNA, Complementary; Down-Regulation; Ergolines; Humans; Ketanserin; Kinetics; Mianserin; Neuroblastoma; Phosphatidylinositols; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Serotonin; Time Factors; Transfection; Tumor Cells, Cultured | 1997 |
NMDA receptor-mediated oscillatory activity in the neonatal rat spinal cord is serotonin dependent.
Topics: Acetylcholine; Animals; Animals, Newborn; Biological Clocks; Edrophonium; Hindlimb; Ketanserin; Locomotion; Mianserin; Motor Activity; Motor Neurons; N-Methylaspartate; Parasympathomimetics; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrodotoxin | 1998 |
Neurochemical effects of the enantiomers of mirtazapine in normal rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Antidepressive Agents, Tricyclic; Body Temperature; Injections, Intraperitoneal; Ketanserin; Male; Mianserin; Mirtazapine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism | 1998 |
GR 127935 and (+)-WAY 100135 do not affect TFMPP-induced inhibition of 5-HT synthesis in the midbrain and hippocampus of Wistar-Kyoto rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Hippocampus; Idazoxan; Ketanserin; Male; Mesencephalon; Mianserin; Nerve Endings; Oxadiazoles; Piperazines; Rats; Rats, Inbred WKY; Rats, Wistar; Reserpine; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Tryptophan Hydroxylase | 1998 |
Effect of 5-HT2 receptor antagonists on a cranial nerve reflex in the rabbit: evidence for inverse agonism.
Topics: Animals; Cranial Nerves; Ergolines; Female; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Piperidines; Rabbits; Receptors, Serotonin; Reflex; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 1999 |
Long-term treatment with antidepressants increases glucocorticoid receptor binding and gene expression in cultured rat hippocampal neurones.
Topics: Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cells, Cultured; Desipramine; Dexamethasone; Gene Expression Regulation; Haloperidol; Hippocampus; Ketanserin; Mianserin; Neurons; Paroxetine; Phentolamine; Propranolol; Radioligand Assay; Rats; Receptors, Glucocorticoid; Receptors, Mineralocorticoid; RNA, Messenger; Sulpiride; Transcription, Genetic; Tritium | 1999 |
Regulation of 5-HT(2A) receptor mRNA levels and binding sites in rat frontal cortex by the agonist DOI and the antagonist mianserin.
Topics: Amphetamines; Animals; Frontal Lobe; Ketanserin; Male; Mianserin; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
5-HT2 receptor antagonists given in the acute withdrawal from daily cocaine injections can reverse established sensitization.
Topics: Animals; Behavior, Animal; Clozapine; Cocaine; Injections; Ketanserin; Male; Mianserin; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Substance Withdrawal Syndrome | 2002 |
Serotonergic regulation of the central heart auricles of Sepia officinalis L. (Mollusca, Cephalopoda).
Topics: Animals; Atrial Function; Dose-Response Relationship, Drug; Fluorescence; Heart Atria; In Vitro Techniques; Ketanserin; Mianserin; Mollusca; Myocardial Contraction; Piperazines; Serotonin; Serotonin Antagonists | 2004 |
Serotonin modifies the sensitivity of the male silkmoth to pheromone.
Topics: Analysis of Variance; Animals; Bombyx; Brain; Chromatography, High Pressure Liquid; Circadian Rhythm; Dose-Response Relationship, Drug; Ketanserin; Male; Mianserin; Olfactory Bulb; Olfactory Pathways; Serotonin; Serotonin Antagonists; Sex Attractants; Time Factors | 2004 |
Suppressive effects of isorhynchophylline on 5-HT2A receptor function in the brain: behavioural and electrophysiological studies.
Topics: Alkaloids; Aminopyridines; Animals; Behavior, Animal; Brain; Dose-Response Relationship, Drug; Female; Indole Alkaloids; Ketanserin; Male; Membrane Potentials; Methoxydimethyltryptamines; Mianserin; Mice; Mice, Inbred ICR; Motor Activity; Oocytes; Oxindoles; Patch-Clamp Techniques; Piperazines; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Xenopus | 2005 |
Zimelidine decreases seizure susceptibility in stressed mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anticonvulsants; Behavior, Animal; Convulsants; Ketanserin; Male; Mianserin; Mice; Mice, Inbred CBA; Phenols; Picrotoxin; Piperazines; Pyridines; Seizures; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Stress, Psychological; Sulfonamides; Swimming; Zimeldine | 2006 |
Nullifying drug-induced sensitization: behavioral and electrophysiological evaluations of dopaminergic and serotonergic ligands in methamphetamine-sensitized rats.
Topics: Action Potentials; Adrenergic Agents; Adrenergic alpha-Antagonists; Animals; Dopamine; Electrochemistry; Globus Pallidus; Ketanserin; Locomotion; Male; Methamphetamine; Mianserin; Microelectrodes; Mirtazapine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Receptors, Dopamine D1; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 2007 |
Reversal of long-term methamphetamine sensitization by combination of pergolide with ondansetron or ketanserin, but not mirtazapine.
Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Infusion Pumps, Implantable; Ketanserin; Male; Methamphetamine; Mianserin; Mirtazapine; Ondansetron; Pergolide; Rats; Rats, Sprague-Dawley | 2011 |
Evaluation of 5-HT2A and mGlu2/3 receptors in postmortem prefrontal cortex of subjects with major depressive disorder: effect of antidepressant treatment.
Topics: Amino Acids; Animals; Antidepressive Agents; Citalopram; Depressive Disorder, Major; Down-Regulation; Female; Humans; Ketanserin; Male; Mianserin; Middle Aged; Mirtazapine; Morpholines; Prefrontal Cortex; Radioligand Assay; Rats, Sprague-Dawley; Reboxetine; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; RNA, Messenger; Tritium; Xanthenes | 2014 |
Mirtazapine and ketanserin alter preference for gambling-like schedules of reinforcement in rats.
Topics: Animals; Choice Behavior; Decision Making; Gambling; Ketanserin; Male; Mianserin; Mirtazapine; Rats; Reinforcement Schedule; Reward; Self Stimulation | 2017 |