ketanserin and mdl 100907

ketanserin has been researched along with mdl 100907 in 145 studies

Research

Studies (145)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (5.52)18.2507
2000's66 (45.52)29.6817
2010's63 (43.45)24.3611
2020's8 (5.52)2.80

Authors

AuthorsStudies
Bristow, LJ; Hutson, PH; Rowley, M1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Chen, Z; Collier, T; Fu, H; Liang, SH; Rong, J; Zhou, J1
Barrett, RJ; Sanders-Bush, E; Smith, RL1
Carr, AA; Johnson, MP; Siegel, BW1
López-Giménez, JF; Mengod, G; Palacios, JM; Vilaró, MT4
Aloyo, VJ; Harvey, JA; Hoffman, ME; Salt, GL1
Caldarola-Pastuszka, M; DeLashaw, M; Uphouse, L; Wolf, A1
Chen, K; De Maeyer, E; Kung, MP; Meehan, WP; Ridd, MJ; Seif, I; Shih, JC1
Adlersberg, M; Arango, V; Hsiung, S; Kassir, SA; Liu, K; Mann, JJ; Ruggiero, DA; Tamir, H; Underwood, MD1
Cunningham, KA; McMahon, LR1
Fantegrossi, WE; Godlewski, T; Karabenick, RL; Rice, KC; Stephens, JM; Ullrich, T; Woods, JH1
Cunningham, KA; Filip, M; McCreary, AC1
Grasby, P; Hirani, E; Hume, S; Sharp, T; Sprakes, M1
Holland, PJ; Johnson, MS; Lutz, EM; Mitchell, R; Moggach, LO; Robertson, DN1
Fink, GD; Li, MW; Ni, W; Thakali, K; Watts, SW1
Bailer, UF; Barbarich, NC; Brooks-Achenbach, S; Frank, GK; Henry, SE; Kaye, WH; Mathis, CA; McConaha, CW; Meltzer, CC; Price, JC; Weissfeld, L1
Goto, F; Obata, H; Saito, S; Sakurazawa, S; Sasaki, M; Usui, T1
Blake, BL; Breese, GR; Knapp, DJ; Papadeas, ST1
Hirano, S; Kamei, J; Miyata, S1
Dubreuil, B; Guilbert, F; Herbert, JM; Janiak, P; Lainée, P; McCort, G; O'Connor, SE1
Caldwell, DP; Levin, ED; Rezvani, AH1
Jacono, FJ; Kumar, GK; Peng, YJ; Prabhakar, NR1
Cao, YX; Edvinsson, L; He, LC; Luo, GG; Xu, CB1
Lutterschmidt, DI; Mason, RT1
Asgari, K; Body, S; Bradshaw, CM; Fone, KC; Rickard, JF; Szabadi, E; Zhang, Z1
Angers, P; Dalbó, S; Jürgensen, S; Ribeiro-do-Valle, RM; Santos, AR1
Gorzalka, BB; Hill, MN; Sun, JC1
Bourin, M; Dailly, E; Hascoët, M; Masse, F1
da Silva, SP; de Almeida, RM; de Oliveira, VP; Giovenardi, M; Stein, DJ1
Matsumoto, K; Morishige, R; Murakami, Y; Sakakibara, I; Takayama, H; Tohda, M; Watanabe, H1
Fujii, H; Hirai, T; Nishio, H; Nitanda, A; Tokumo, K; Yasunami, N1
Elfving, B; Gillings, N; Knudsen, GM; Kristiansen, H; Pinborg, LH; Plenge, P1
Jazvinsćak Jembrek, M; Lazić, J; Pericić, D; Svob Strac, D1
Asgari, K; Bak, VK; Body, S; Bradshaw, CM; Fone, KC; Glennon, JC; Rickard, JF; Szabadi, E; Zhang, ZQ1
Chapman, ME; Wideman, RF1
Kajos, M; Kankaanpää, A; Meririnne, E; Seppälä, T1
Günther, S; Maroteaux, L; Schwarzacher, SW1
Bernard, JF; Comet, MA; Hamon, M; Laguzzi, R; Sévoz-Couche, C1
Crespo, MJ; Dunbar, DC; Quidgley, J1
Elfrey, JE; Finkelman, FD; Madden, KB; Morimoto, M; Shea-Donohue, T; Urban, JF; Zhao, A1
Kuypers, KP; Ramaekers, JG; Wingen, M2
Harris, MB; Kober, AM; Leiter, JC; St-John, WM; Toppin, VA1
Alexandropoulou, KN; Demonakou, MD; Hereti, RI; Kourentzi, KT; Manta, GA; Mykoniatis, MG; Panoutsopoulos, GI; Papadimas, GK; Skaltsas, SD; Tzirogiannis, KN1
Ni, CR; Shen, FM; Su, DF; Wang, J; Wang, WZ; Yu, JG1
Aranda, E; Downey, P; Giacaman, A; Mezzano, D; Romero, W; Salas, SP; Vío, CP1
Chang, FC; Lin, CP; Lin, JG; Tsai, CH; Yi, PL1
Birkeland, JA; Enger, U; Levy, FO; Lunde, PK; Qvigstad, E; Sejersted, OM; Sjaastad, I; Swift, F; Tovsrud, N1
Fletcher, PJ; Higgins, GA; Sinyard, J; Tampakeras, M1
Carter, OL; Hasler, F; Liu, GB; Pettigrew, JD; Vollenweider, FX; Wallis, GM1
Ballabeni, V; Barocelli, E; Bertoni, S; Cattaruzza, F; Ghizzardi, P; Impicciatore, M; Lagrasta, CA; Tognolini, M1
Leiter, JC; St-John, WM1
Debus, F; Herth, MM; Knudsen, GM; Lüddens, H; Palner, M; Piel, M; Rösch, F1
Harmar, AJ; Jennings, KA; Sharp, T; Sheward, WJ1
Agrawal, AK; Bhattamisra, SK; Khanna, VK; Singh, PN; Singh, SK1
Chemel, BR; Frescas, SP; Lewin, AH; Nichols, DE; Rehder, KS; Zhong, D1
Baumeister, AA; Hawkins, MF; Hearn, JK; Uzelac, SM1
Atwood, WJ; Lane, TE; O'Hara, BA; Schaumburg, C1
Ahmad, R; Egerton, A; Grasby, PM; Hirani, E1
Bras, H; Coulon, P; Gaytán, SP; Hilaire, G; Pásaro, R; Portalier, P; Zanella, S1
Horton, K; Johnson, M; Levin, ED; Petro, A; Rezvani, AH; Rose, JE; Slade, S; Williams, P1
Becnel, J; Johnson, O; Nichols, CD1
Araki, H; Cui, R; Li, B; Suemaru, K; Tanaka, M; Watanabe, S1
France, CP; Li, JX; Rice, KC1
Bianchi, P; Calise, D; Escourrou, G; Galinier, M; Guilbeau-Frugier, C; Lairez, O; Mialet-Perez, J; Ordener, C; Parini, A; Pizzinat, N; Roncalli, J; Seif, I; Spreux-Varoquaux, O1
Anju, TR; George, AK; Paulose, CS1
Huang, X; Krishnamoorthy, S; Ma, Z; Tao, R; Vukovich, NP; Zhang, G1
Hadamitzky, M; Koch, M1
France, CP; Javors, MA; Koek, W; Li, JX; Rice, KC; Unzeitig, A1
Nakamichi, K; Nukuzuma, C; Nukuzuma, S; Takegami, T1
Becker, T; Feja, M; Hadamitzky, M; Koch, M1
Anselmo-Franci, JA; Bícego, KC; de Souza Moreno, V; Gargaglioni, LH; Szawka, RE1
Doyle, JR; Yamamoto, BK1
Bullich, S; Catafau, AM; Farre, M; Gunn, RN; Herance, R; Laruelle, M; Rabiner, EA; Radua, J; Searle, GE1
le Grand, SM; Srikiatkhachorn, A; Supornsilpchai, W1
Eriksson, AC; Felixsson, E; Persson, IA; Persson, K1
Auerbach, SB; Krishnamoorthy, S; Ma, Z; Tao, R; Wei, J; Zhang, G1
Pobbe, RL; Zangrossi, H1
Doi, A; Ramirez, JM1
Herth, MM; Knudsen, GM; Kramer, V; Palner, M; Rösch, F; Santini, MA1
Estrada-González, V; Márquez-Diosdado, MI; Montes-Rodríguez, CJ; Prospéro-García, O; Soria-Gómez, E1
Larrauri, JA; Levin, ED1
Abe, C; Iwata, C; Morita, H; Tanaka, K1
Cohen, MS; Fantegrossi, WE; Henson, CM; Rice, KC; Simoneau, J; Woods, JH; Zimmerman, SM1
Fan, Y; Hong, Y; Huang, J; Jia, Y1
MacFarlane, PM; Mitchell, GS; Vinit, S1
Creed-Carson, M; Nobrega, JN; Oraha, A1
Nagatani, H; Nakata, Y; Oshima, T; Saitoh, Y; Urano, A; Yokota, M1
Jolivalt, CG; Mixcoatl-Zecuatl, T1
Pazos, A; Pilar-Cuéllar, F; Vidal, R1
Arai, Y; Kikuchi, T; Mitazaki, S; Nakagawasai, O; Nakaya, K; Niijima-Yaoita, F; Onogi, H; Sato, A; Tadano, T; Tan-No, K; Watanabe, K1
Grandt, R; Hautzel, H; Herzog, H; Müller, HW1
Abman, SH; Delaney, C; Gien, J; Grover, TR; Roe, G1
Bennett, A; Blood, AB; Blood, Q; Dawson, A; Goyal, R; Longo, LD; Osman, NJ; Papamatheakis, DG; Pearce, WJ; Rubalcava, M; Vemulakonda, S; Vrancken, K; Wilson, SM1
Chan, SC; Ip, MS; Lau, WK; Law, AC; Mak, JC1
Glusa, E; Görnemann, T; Jantschak, F; Kekewska, A; Pertz, HH1
Hackett, A; Hanania, T; Paterson, NE; Wetzler, C1
Maraschin, M; Rodrigues, AL; Tasca, CI; Zeni, AL; Zomkowski, AD1
Chen, T; Gao, Y; Hong, Y; Quirion, R; Wang, D1
Bachmann, R; Kometer, M; Schmidt, A; Seifritz, E; Studerus, E; Vollenweider, FX1
Bhattacharyya, S; Panicker, MM; Raote, I1
Chen, GS; Li, XQ; Liu, G; Liu, SB; Ma, L; Wu, YM; Xu, ZH; Yang, Q; Zhao, MG1
Fan, F; Han, J; Liu, Y; Tian, H; Wang, W; Yan, X1
Choi, HS; Jun, DW; Kim, DC; Kim, EK; Kwon, YI; Lee, HL; Lee, KN; Lee, OY; Yoon, BC1
Dyssegaard, A; Ettrup, A; Gillings, N; Hansen, HD; Herth, MM; Knudsen, GM; Ratner, C1
Corcoran, AE; Harris, MB; Richerson, GB1
Fedotova, IuO; Frolova, HO; Ordian, NE; Soboliev, VI1
Abman, SH; Delaney, C; Gien, J; Isenberg, N; Kailey, J; Roe, G1
Elliott, R; Hornboll, B; Knudsen, GM; Macoveanu, J; Paulson, OB; Rowe, J; Siebner, HR1
Couppis, MH; Juárez, P; Kennedy, CH; Lloyd, BP; May, ME; Valdovinos, MG1
Agnati, LF; Borroto-Escuela, DO; Fuxe, K; Narvaez, M; Oflijan, J; Romero-Fernandez, W1
Bae, YM; Cho, H; Kim, B; Kim, JG; Noh, HJ; Park, SW; Sung, DJ1
Dong, YL; Hu, W; Li, HS; Lu, GJ; Sun, YH; Wu, SX; Yang, J; Zhao, GL; Zhu, C1
Chacron, MJ; Larson, EA; Metzen, MG1
Ganev, EG; Hiruma-Lima, CA; Martins, DF; Mazzardo-Martins, L; Nishijima, CM; Rocha, LR; Santos, AR1
Chen, G; Chen, L; Fan, W; Guo, Y; Liu, L; Qian, Y; Shi, B; Xiao, L1
Anisimova, VA; Mal'tsev, DV; Spasov, AA; Yakovlev, DS1
Bailey, JM; Fantegrossi, WE; Gray, BW; Hansen, M; Kristensen, JL; Smith, DA1
Gerlai, R; Markovic, S; Muraleetharan, A; Nowicki, M; Tran, S1
Fukushima, S; Hagino, Y; Hall, FS; Igari, M; Ikeda, K; Kasahara, Y; Lesch, KP; Murphy, DL; Shen, HW; Sora, I; Uhl, GR; Yaegashi, N1
Anastasio, NC; Cunningham, KA; Fink, LH; Fox, RG; Moeller, FG; Rice, KC1
Hernekamp, JF; Klein, H; Kneser, U; Kremer, T; Schmidt, K1
Hu, K; Kang, J; Mei, Y; Tu, X; Wang, N; Zuo, J1
Hong, Y; Hu, W; Huang, BQ; Wu, B1
Ahangari, G; Deezagi, A; Hejazi, SH1
Beliveau, V; da Cunha-Bang, S; Dyssegaard, A; Ettrup, A; Ganz, M; Gillings, N; Jørgensen, LM; Knudsen, GM; Lehel, S; McMahon, B; Møller, K; Svarer, C1
Cai, Q; Hong, Y; Hu, W; Wang, D; Zhang, Y1
de Paula, BB; Leite-Panissi, CR1
Baki, L; Drossopoulos, P; Dukat, M; Ellaithy, A; Eltit, JM; Gaitonde, SA; Glennon, RA; González-Maeso, J; Hideshima, KS; Logothetis, DE; Moreno, JL; Shah, S; Vekariya, R; Younkin, J1
Barresi, M; Grasso, C; Li Volsi, G1
Kraehenmann, R; Pokorny, D; Pokorny, T; Preller, KH; Seifritz, E; Vollenweider, FX; Vollenweider, L1
Barrett, FS; Herdener, M; Janata, P; Preller, KH; Vollenweider, FX1
de la Torre, R; Farre, M; Haijen, E; Kuypers, KPC; Olesti, E; Pastor, A; Pizarro, N; Ramaekers, JG1
Cao, N; Gu, B; Karl-Erik, A; Ni, J; Si, J; Wang, X1
Chen, L; Dong, J; Li, Y; Shen, Y; Wan, C; Wang, H; Wen, F; Wu, Y; Yang, T; Zeng, Z1
Bova, S; Fusi, F; Saponara, S; Sgaragli, G; Spiga, O; Trezza, A1
Kubilis, PS; Mitchell, GS; Perim, RR; Seven, YB1
Makiguchi, A; Okada, T; Shioda, K; Suda, S1
Mendonça-Junior, BA; V Fernandes, M; Zoccal, DB1
Li, K; Liu, X; Su, R; Zhang, M1
Garza, G; Moghaddam, B; Olson, RJ; Torrado Pacheco, A1

Reviews

2 review(s) available for ketanserin and mdl 100907

ArticleYear
Current and novel approaches to the drug treatment of schizophrenia.
    Journal of medicinal chemistry, 2001, Feb-15, Volume: 44, Issue:4

    Topics: Animals; Antipsychotic Agents; Cholinergic Agonists; Disease Models, Animal; Dopamine Antagonists; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Humans; Mice; Mice, Transgenic; Nitric Oxide Synthase; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotensin; Receptors, Serotonin; Schizophrenia; Serotonin Antagonists

2001
Positron Emission Tomography (PET) Imaging Tracers for Serotonin Receptors.
    Journal of medicinal chemistry, 2022, 08-25, Volume: 65, Issue:16

    Topics: Brain; Humans; Ligands; Positron-Emission Tomography; Radiopharmaceuticals; Receptors, Serotonin

2022

Trials

6 trial(s) available for ketanserin and mdl 100907

ArticleYear
Evaluation of the serotonin receptor blockers ketanserin and methiothepin on the pulmonary hypertensive responses of broilers to intravenously infused serotonin.
    Poultry science, 2006, Volume: 85, Issue:4

    Topics: Animals; Blood Pressure; Chickens; Hypertension, Pulmonary; Injections, Intravenous; Ketanserin; Male; Methiothepin; Poultry Diseases; Prostaglandin Endoperoxides, Synthetic; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT2; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2006
Selective verbal and spatial memory impairment after 5-HT1A and 5-HT2A receptor blockade in healthy volunteers pre-treated with an SSRI.
    Journal of psychopharmacology (Oxford, England), 2007, Volume: 21, Issue:5

    Topics: Administration, Oral; Adult; Affect; Brain; Citalopram; Cognition; Cross-Over Studies; Double-Blind Method; Female; Humans; Ketanserin; Male; Mental Recall; Pindolol; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Reference Values; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Space Perception; Verbal Learning

2007
The role of 5-HT1a and 5-HT2a receptors in attention and motor control: a mechanistic study in healthy volunteers.
    Psychopharmacology, 2007, Volume: 190, Issue:3

    Topics: Administration, Oral; Adult; Attention; Citalopram; Cognition; Cross-Over Studies; Double-Blind Method; Female; Humans; Ketanserin; Male; Pindolol; Psychomotor Performance; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Sleep

2007
Psilocybin biases facial recognition, goal-directed behavior, and mood state toward positive relative to negative emotions through different serotonergic subreceptors.
    Biological psychiatry, 2012, Dec-01, Volume: 72, Issue:11

    Topics: Adult; Affect; Cerebral Cortex; Double-Blind Method; Electroencephalography; Emotions; Evoked Potentials; Female; Goals; Hallucinogens; Humans; Ketanserin; Male; Neuropsychological Tests; Psilocybin; Receptors, Serotonin; Recognition, Psychology; Serotonin 5-HT2 Receptor Antagonists

2012
Acute serotonin 2A receptor blocking alters the processing of fearful faces in the orbitofrontal cortex and amygdala.
    Journal of psychopharmacology (Oxford, England), 2013, Volume: 27, Issue:10

    Topics: Adult; Amygdala; Anger; Citalopram; Facial Expression; Fear; Female; Frontal Lobe; Functional Neuroimaging; Healthy Volunteers; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Neural Pathways; Photic Stimulation; Radioligand Assay; Reaction Time; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT2 Receptor Antagonists; Sex Factors; Tryptophan; Visual Perception

2013
Peripheral endocannabinoid concentrations are not associated with verbal memory impairment during MDMA intoxication.
    Psychopharmacology, 2018, Volume: 235, Issue:3

    Topics: Adult; Arachidonic Acids; Double-Blind Method; Endocannabinoids; Female; Humans; Ketanserin; Male; Memory Disorders; N-Methyl-3,4-methylenedioxyamphetamine; Polyunsaturated Alkamides; Serotonin 5-HT2 Receptor Antagonists; Serotonin Agents; Verbal Learning; Young Adult

2018

Other Studies

137 other study(ies) available for ketanserin and mdl 100907

ArticleYear
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Neurochemical and behavioral evidence that quipazine-ketanserin discrimination is mediated by serotonin2A receptor.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: Animals; Brain Mapping; Discrimination Learning; Dose-Response Relationship, Drug; Fluorobenzenes; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
[3H]MDL 100,907: a novel selective 5-HT2A receptor ligand.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:2

    Topics: Animals; Fluorobenzenes; Frontal Lobe; Ketanserin; Ligands; Male; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists

1996
Selective visualization of rat brain 5-HT2A receptors by autoradiography with [3H]MDL 100,907.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:4

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Fluorobenzenes; Guanylyl Imidodiphosphate; In Situ Hybridization; In Vitro Techniques; Ketanserin; Male; Naphthalenes; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists

1997
[3H]MDL 100,907 labels 5-HT2A serotonin receptors selectively in primate brain.
    Neuropharmacology, 1998, Volume: 37, Issue:9

    Topics: Aged; Aged, 80 and over; Animals; Binding Sites; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Male; Naphthalenes; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Tritium

1998
Agonist and antagonist binding to rabbit cortical 5-HT2A receptors: opposite effects of magnesium.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: Amphetamines; Animals; Cerebral Cortex; Fluorobenzenes; Guanylyl Imidodiphosphate; Ketanserin; Magnesium; Methysergide; Piperidines; Prazosin; Rabbits; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1998
5-HT2C receptor involvement in female rat lordosis behavior.
    Brain research, 1999, Apr-17, Volume: 825, Issue:1-2

    Topics: Animals; Estradiol; Female; Fluorobenzenes; Indoles; Indophenol; Ketanserin; Ovariectomy; Piperidines; Posture; Pyridines; Rats; Rats, Inbred Strains; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sexual Behavior, Animal; Ventromedial Hypothalamic Nucleus

1999
Ketanserin and tetrabenazine abolish aggression in mice lacking monoamine oxidase A.
    Brain research, 1999, Jul-24, Volume: 835, Issue:2

    Topics: Adrenergic Uptake Inhibitors; Aggression; Animals; Brain; Corpus Striatum; Drug Evaluation, Preclinical; Fluorobenzenes; Frontal Lobe; Ketanserin; Male; Mice; Mice, Knockout; Monoamine Oxidase; Neurotransmitter Agents; Piperidines; Radioligand Assay; Serotonin Antagonists; Tetrabenazine

1999
Human striosomes are enriched in 5-HT2A receptors: autoradiographical visualization with [3H]MDL100,907,[125I](+/-)DOI and [3H]ketanserin.
    The European journal of neuroscience, 1999, Volume: 11, Issue:10

    Topics: Adult; Aged; Autoradiography; Female; Fluorobenzenes; Humans; Indophenol; Iodine Radioisotopes; Ketanserin; Male; Middle Aged; Neostriatum; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Tritium

1999
In vitro autoradiography of serotonin 5-HT(2A/2C) receptor-activated G protein: guanosine-5'-(gamma-[(35)S]thio)triphosphate binding in rat brain.
    Journal of neuroscience research, 2000, Sep-15, Volume: 61, Issue:6

    Topics: Amphetamines; Animals; Autoradiography; Brain Chemistry; Dose-Response Relationship, Drug; Fluorobenzenes; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Image Processing, Computer-Assisted; Indoles; Ketanserin; Male; Membrane Proteins; Piperidines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Subcellular Fractions; Sulfur Radioisotopes

2000
Mapping of 5-HT2A receptors and their mRNA in monkey brain: [3H]MDL100,907 autoradiography and in situ hybridization studies.
    The Journal of comparative neurology, 2001, Jan-22, Volume: 429, Issue:4

    Topics: Animals; Autoradiography; Brain; Brain Mapping; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Macaca mulatta; Male; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists

2001
Antagonism of 5-hydroxytryptamine(2a) receptors attenuates the behavioral effects of cocaine in rats.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 297, Issue:1

    Topics: Animals; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Discrimination Learning; Dopamine; Fluorobenzenes; Ketanserin; Male; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists

2001
Pharmacological characterization of the effects of 3,4-methylenedioxymethamphetamine ("ecstasy") and its enantiomers on lethality, core temperature, and locomotor activity in singly housed and crowded mice.
    Psychopharmacology, 2003, Volume: 166, Issue:3

    Topics: Animals; Body Temperature; Cold Temperature; Crowding; Dose-Response Relationship, Drug; Fluorobenzenes; Fluoxetine; Hallucinogens; Ketanserin; Lethal Dose 50; Male; Mice; Motor Activity; N-Methyl-3,4-methylenedioxyamphetamine; Piperidines; Platelet Aggregation Inhibitors; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Social Isolation; Stereoisomerism; Telemetry

2003
Discriminative stimulus properties of (+/-)-fenfluramine: the role of 5-HT2 receptor subtypes.
    Behavioral neuroscience, 2003, Volume: 117, Issue:2

    Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Fenfluramine; Fluorobenzenes; Indoles; Ketanserin; Male; Piperidines; Pyrazines; Pyridines; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Thiophenes

2003
Fenfluramine evokes 5-HT2A receptor-mediated responses but does not displace [11C]MDL 100907: small animal PET and gene expression studies.
    Synapse (New York, N.Y.), 2003, Dec-01, Volume: 50, Issue:3

    Topics: Animals; Carbon Radioisotopes; Cerebellum; Fenfluramine; Fluorobenzenes; Gene Expression; Genes, Immediate-Early; In Situ Hybridization; Ketanserin; Male; Neurons; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Time Factors; Tomography, Emission-Computed

2003
Selective interaction of ARF1 with the carboxy-terminal tail domain of the 5-HT2A receptor.
    Molecular pharmacology, 2003, Volume: 64, Issue:5

    Topics: ADP-Ribosylation Factor 1; Amino Acid Sequence; Animals; COS Cells; Humans; Ketanserin; Molecular Sequence Data; Mutation; Protein Binding; Protein Structure, Tertiary; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2003
The fenfluramine metabolite (+)-norfenfluramine is vasoactive.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 309, Issue:2

    Topics: Animals; Aorta; Blood Pressure; Ergolines; Fenfluramine; In Vitro Techniques; Ketanserin; Male; Norfenfluramine; Prazosin; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Adrenergic, alpha; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Sympathectomy; Sympathetic Nervous System; Vasoconstriction

2004
Altered 5-HT(2A) receptor binding after recovery from bulimia-type anorexia nervosa: relationships to harm avoidance and drive for thinness.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2004, Volume: 29, Issue:6

    Topics: Adult; Age Factors; Anorexia Nervosa; Brain; Brain Mapping; Bulimia; Drive; Female; Fluorine Radioisotopes; Harm Reduction; Humans; Ketanserin; Protein Binding; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Thinness; Time Factors; Tomography, Emission-Computed

2004
Antiallodynic effects of intrathecally administered 5-HT(2C) receptor agonists in rats with nerve injury.
    Pain, 2004, Volume: 108, Issue:1-2

    Topics: Amphetamines; Animals; Indoles; Injections, Spinal; Ketanserin; Ligation; Lumbar Vertebrae; Male; Neuralgia; Nociceptors; Piperazines; Pyrazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Nerves; Spiro Compounds; Sulfonamides; Thiophenes

2004
Sustained extracellular signal-regulated kinase 1/2 phosphorylation in neonate 6-hydroxydopamine-lesioned rats after repeated D1-dopamine receptor agonist administration: implications for NMDA receptor involvement.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Jun-30, Volume: 24, Issue:26

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aminoacetonitrile; Animals; Animals, Newborn; Benzazepines; Corpus Striatum; Cyclic AMP Response Element-Binding Protein; Dopamine Agonists; Dopamine Antagonists; Enzyme Inhibitors; Female; Ketanserin; Male; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Nerve Tissue Proteins; Nucleus Accumbens; Oxidopamine; Phosphorylation; Prefrontal Cortex; Protease Inhibitors; Protein Processing, Post-Translational; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate; Serotonin 5-HT2 Receptor Antagonists

2004
Diabetes inhibits the DOI-induced head-twitch response in mice.
    Psychopharmacology, 2004, Volume: 177, Issue:1-2

    Topics: Amphetamines; Animals; Corticosterone; Diabetes Mellitus, Experimental; Head Movements; Ketanserin; Male; Mice; Mice, Inbred ICR; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2004
Serotonin aggravates exercise-induced cardiac ischemia in the dog: effect of serotonin receptor antagonists.
    European journal of pharmacology, 2004, Aug-16, Volume: 497, Issue:1

    Topics: Animals; Dogs; Endothelium, Vascular; Female; Hemodynamics; Hypercholesterolemia; Infusions, Intravenous; Ketanserin; Myocardial Ischemia; Physical Conditioning, Animal; Piperazines; Quinolines; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2004
Nicotinic-serotonergic drug interactions and attentional performance in rats.
    Psychopharmacology, 2005, Volume: 179, Issue:3

    Topics: Animals; Attention; Dose-Response Relationship, Drug; Drug Interactions; Female; Ketanserin; Nicotine; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2005
Modulation of the hypoxic sensory response of the carotid body by 5-hydroxytryptamine: role of the 5-HT2 receptor.
    Respiratory physiology & neurobiology, 2005, Feb-15, Volume: 145, Issue:2-3

    Topics: Action Potentials; Animals; Carotid Body; Chromatography, High Pressure Liquid; Dopamine; Electrochemistry; Free Radical Scavengers; Hypoxia; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT2; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Time Factors

2005
Enhanced transcription of contractile 5-hydroxytryptamine 2A receptors via extracellular signal-regulated kinase 1/2 after organ culture of rat mesenteric artery.
    Basic & clinical pharmacology & toxicology, 2005, Volume: 96, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Ketanserin; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; RNA, Messenger; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Time Factors; Transcription, Genetic; Up-Regulation; Vasoconstriction

2005
A serotonin receptor antagonist, but not melatonin, modulates hormonal responses to capture stress in two populations of garter snakes (Thamnophis sirtalis parietalis and Thamnophis sirtalis concinnus).
    General and comparative endocrinology, 2005, May-01, Volume: 141, Issue:3

    Topics: 5-Hydroxytryptophan; Adjuvants, Immunologic; Androgens; Animals; Colubridae; Corticosterone; Endocrine System; Ketanserin; Melatonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Stress, Physiological

2005
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on temporal differentiation: evidence for the involvement of 5-HT2A but not 5-HT3 receptors in interval timing behaviour.
    Psychopharmacology, 2005, Volume: 181, Issue:2

    Topics: Animals; Biguanides; Conditioning, Operant; Dose-Response Relationship, Drug; Female; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Psychometrics; Quipazine; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Task Performance and Analysis; Time Perception; Tropanes

2005
Involvement of 5-HT2 receptors in the antinociceptive effect of Uncaria tomentosa.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:3

    Topics: Acetic Acid; Analgesics; Animals; Arginine; Atropine; Behavior, Animal; Capsaicin; Cat's Claw; Dose-Response Relationship, Drug; Formaldehyde; Ketanserin; Male; Mice; Motor Activity; Naltrexone; Pain; Pain Measurement; Phytotherapy; Plant Preparations; Prazosin; Receptors, Serotonin, 5-HT2; Reserpine; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Yohimbine

2005
Functional role of the endocannabinoid system and AMPA/kainate receptors in 5-HT2A receptor-mediated wet dog shakes.
    European journal of pharmacology, 2005, May-23, Volume: 516, Issue:1

    Topics: Amphetamines; Animals; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Dose-Response Relationship, Drug; Endocannabinoids; Excitatory Amino Acid Antagonists; Injections, Intraperitoneal; Ketanserin; Male; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, Kainic Acid; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists

2005
Anxiolytic-like effect of milnacipran in the four-plate test in mice: mechanism of action.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzylamines; Brain; Cyclopropanes; Dopamine; Dose-Response Relationship, Drug; Fenclonine; Flumazenil; Fluorobenzenes; Idazoxan; Indoles; Ketanserin; Male; Mice; Milnacipran; Motor Activity; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phenols; Prazosin; Punishment; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2005
Maternal aggression in Wistar rats: effect of 5-HT2A/2C receptor agonist and antagonist microinjected into the dorsal periaqueductal gray matter and medial septum.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 2005, Volume: 38, Issue:4

    Topics: Aggression; Animals; Animals, Newborn; Female; Ketanserin; Male; Maternal Behavior; Microinjections; Periaqueductal Gray; Pregnancy; Rats; Rats, Wistar; Septum of Brain; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2005
Suppressive effects of isorhynchophylline on 5-HT2A receptor function in the brain: behavioural and electrophysiological studies.
    European journal of pharmacology, 2005, Jul-11, Volume: 517, Issue:3

    Topics: Alkaloids; Aminopyridines; Animals; Behavior, Animal; Brain; Dose-Response Relationship, Drug; Female; Indole Alkaloids; Ketanserin; Male; Membrane Potentials; Methoxydimethyltryptamines; Mianserin; Mice; Mice, Inbred ICR; Motor Activity; Oocytes; Oxindoles; Patch-Clamp Techniques; Piperazines; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Xenopus

2005
Contribution of the peripheral 5-HT 2A receptor to mechanical hyperalgesia in a rat model of neuropathic pain.
    Neurochemistry international, 2005, Volume: 47, Issue:6

    Topics: Animals; Binding Sites; Binding, Competitive; Denervation; Disease Models, Animal; Drug Interactions; Hyperalgesia; Ketanserin; Ligation; Male; Neuralgia; Pain Threshold; Peripheral Nerves; Peripheral Nervous System Diseases; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Sciatic Neuropathy; Sensory Receptor Cells; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Succinates

2005
Binding characteristics of the 5-HT2A receptor antagonists altanserin and MDL 100907.
    Synapse (New York, N.Y.), 2005, Dec-15, Volume: 58, Issue:4

    Topics: Animals; Binding, Competitive; Brain; Carbon Radioisotopes; Fluorine Radioisotopes; Fluorobenzenes; Ketanserin; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2005
Stimulation of 5-HT 1A receptors increases the seizure threshold for picrotoxin in mice.
    European journal of pharmacology, 2005, Dec-19, Volume: 527, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Drug Administration Schedule; Drug Therapy, Combination; Ketanserin; Male; Mice; Mice, Inbred CBA; Picrotoxin; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Seizures; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Stress, Physiological; Swimming

2005
Effects of 5-HT2A receptor stimulation on the discrimination of durations by rats.
    Behavioural pharmacology, 2006, Volume: 17, Issue:1

    Topics: Amphetamines; Animals; Association Learning; Brain; Discrimination Learning; Female; Fluorobenzenes; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Piperidines; Psychophysics; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Serotonin Receptor Agonists; Time Perception

2006
Rewarding properties of 1-benzylpiperazine, a new drug of abuse, in rats.
    Basic & clinical pharmacology & toxicology, 2006, Volume: 98, Issue:4

    Topics: Animals; Behavior, Animal; Benzazepines; Conditioning, Psychological; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ketanserin; Male; Piperidines; Psychotropic Drugs; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT3; Reward; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Substance-Related Disorders; Tropanes

2006
Endogenous 5-HT2B receptor activation regulates neonatal respiratory activity in vitro.
    Journal of neurobiology, 2006, Volume: 66, Issue:9

    Topics: Animals; Animals, Newborn; In Vitro Techniques; Indoles; Ketanserin; Kinetics; Mice; Microinjections; Organic Chemicals; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Respiration; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Thiophenes

2006
Cardiac baroreflex facilitation evoked by hypothalamus and prefrontal cortex stimulation: role of the nucleus tractus solitarius 5-HT2A receptors.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2006, Volume: 291, Issue:4

    Topics: Animals; Atenolol; Atropine Derivatives; Baroreflex; Brain; Electric Stimulation; Fluorobenzenes; Heart; Ketanserin; Male; Microinjections; Neural Inhibition; Neural Pathways; Parasympatholytics; Piperidines; Prefrontal Cortex; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Solitary Nucleus; Stimulation, Chemical; Sympatholytics

2006
Differential regulation of the left and right coronary arteries of swine.
    Pharmacology, 2006, Volume: 77, Issue:3

    Topics: Animals; Coronary Vessels; In Vitro Techniques; Ketanserin; Male; Potassium Chloride; Propranolol; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT2; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Swine; Vasoconstriction

2006
Contribution of 5-HT2A receptor in nematode infection-induced murine intestinal smooth muscle hypercontractility.
    Gastroenterology, 2006, Volume: 131, Issue:2

    Topics: Animals; Disease Models, Animal; Female; Gene Expression; Ketanserin; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle Hypertonia; Muscle, Smooth; Nematode Infections; Nippostrongylus; Polymerase Chain Reaction; Receptor, Serotonin, 5-HT2A; RNA, Messenger; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2006
Persistence of eupnea and gasping following blockade of both serotonin type 1 and 2 receptors in the in situ juvenile rat preparation.
    Journal of applied physiology (Bethesda, Md. : 1985), 2007, Volume: 103, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Decerebrate State; Disease Models, Animal; Dose-Response Relationship, Drug; Hypoglossal Nerve; Ischemia; Ketanserin; Lung; Methysergide; Peripheral Nerves; Phrenic Nerve; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT1; Respiratory Mechanics; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors; Vagus Nerve

2007
Effect of 5-HT(2) receptor blockade on cadmium-induced acute toxicity.
    Digestive diseases and sciences, 2007, Volume: 52, Issue:9

    Topics: Animals; Apoptosis; Cadmium; Disease Models, Animal; In Situ Nick-End Labeling; Ketanserin; Liver Failure, Acute; Male; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT2; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Treatment Outcome

2007
Ketanserin-induced baroreflex enhancement in spontaneously hypertensive rats depends on central 5-HT(2A) receptors.
    Clinical and experimental pharmacology & physiology, 2007, Volume: 34, Issue:8

    Topics: Animals; Antibodies, Monoclonal; Antihypertensive Agents; Baroreflex; Blood Pressure; Brain; Disease Models, Animal; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Immunotoxins; Ketanserin; N-Glycosyl Hydrolases; Neurons; Plant Proteins; Rats; Rats, Inbred SHR; Receptor, Serotonin, 5-HT2A; Ribosome Inactivating Proteins, Type 1; Saporins; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins

2007
Pregnant rats treated with a serotonin precursor have reduced fetal weight and lower plasma volume and kallikrein levels.
    Hypertension (Dallas, Tex. : 1979), 2007, Volume: 50, Issue:4

    Topics: 5-Hydroxytryptophan; Aldosterone; Animals; Blood Pressure; Creatinine; Disease Models, Animal; Female; Fetal Weight; Kallikreins; Ketanserin; Plasma Volume; Pre-Eclampsia; Pregnancy; Pregnancy, Animal; Random Allocation; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists

2007
The involvement of serotonin receptors in suanzaorentang-induced sleep alteration.
    Journal of biomedical science, 2007, Volume: 14, Issue:6

    Topics: Animals; Drugs, Chinese Herbal; Ketanserin; Piperazines; Plant Extracts; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin; Receptors, Serotonin, 5-HT2; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Sleep; Time Factors

2007
Serotonin increases L-type Ca2+ current and SR Ca2+ content through 5-HT4 receptors in failing rat ventricular cardiomyocytes.
    American journal of physiology. Heart and circulatory physiology, 2007, Volume: 293, Issue:4

    Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Calcium Channels, L-Type; Calcium Signaling; Calcium-Binding Proteins; Cardiac Myosins; Cardiotonic Agents; Coronary Vessels; Disease Models, Animal; Heart Failure; Indoles; Isoproterenol; Ketanserin; Ligation; Male; Myocardial Contraction; Myocardial Infarction; Myocytes, Cardiac; Myosin Light Chains; Phosphorylation; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT4; Sarcoplasmic Reticulum; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides; Time Factors; Troponin I; Ventricular Function

2007
Opposing effects of 5-HT(2A) and 5-HT(2C) receptor antagonists in the rat and mouse on premature responding in the five-choice serial reaction time test.
    Psychopharmacology, 2007, Volume: 195, Issue:2

    Topics: Aminopyridines; Amphetamines; Animals; Conditioning, Operant; Ethylamines; Fluorobenzenes; Impulsive Behavior; Indoles; Ketanserin; Male; Mice; Mice, Inbred C57BL; Piperidines; Quinolines; Rats; Reaction Time; Serial Learning; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Species Specificity

2007
Psilocybin links binocular rivalry switch rate to attention and subjective arousal levels in humans.
    Psychopharmacology, 2007, Volume: 195, Issue:3

    Topics: Adult; Arousal; Attention; Double-Blind Method; Drug Combinations; Female; Hallucinogens; Humans; Ketanserin; Male; Psilocybin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Vision Disparity; Vision, Binocular

2007
Evidence for the involvement of 5-HT2A receptors in mild mesenteric ischemia/reperfusion dysfunctions in mice.
    Pharmacological research, 2007, Volume: 56, Issue:6

    Topics: Amphetamines; Animals; Capillary Permeability; Female; Gastrointestinal Transit; Intestines; Ketanserin; Leukocytes; Lipid Peroxidation; Lung; Malondialdehyde; Mesenteric Artery, Superior; Mice; Peroxidase; Platelet Aggregation; Receptor, Serotonin, 5-HT2A; Reperfusion Injury; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Tumor Necrosis Factor-alpha

2007
Maintenance of gasping and restoration of eupnea after hypoxia is impaired following blockers of alpha1-adrenergic receptors and serotonin 5-HT2 receptors.
    Journal of applied physiology (Bethesda, Md. : 1985), 2008, Volume: 104, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amphetamines; Animals; Decerebrate State; Diaphragm; Dioxanes; Disease Models, Animal; Dose-Response Relationship, Drug; Hypoxia; Ketanserin; Methoxamine; Methysergide; Periodicity; Phrenic Nerve; Rats; Receptors, Adrenergic, alpha-1; Receptors, Serotonin, 5-HT2; Respiratory Mechanics; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2008
Total synthesis and evaluation of [18F]MHMZ.
    Bioorganic & medicinal chemistry letters, 2008, Feb-15, Volume: 18, Issue:4

    Topics: Animals; Binding, Competitive; Brain; Fluorine Radioisotopes; Fluorobenzenes; Isotope Labeling; Ketanserin; Kinetics; Piperidines; Radioligand Assay; Radionuclide Imaging; Radiopharmaceuticals; Rats; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2008
Evidence that genetic variation in 5-HT transporter expression is linked to changes in 5-HT2A receptor function.
    Neuropharmacology, 2008, Volume: 54, Issue:5

    Topics: Amphetamines; Analysis of Variance; Animals; Brain; Cytoskeletal Proteins; Dose-Response Relationship, Drug; Fluorobenzenes; Gene Expression; Genetic Variation; Head Movements; Ketanserin; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Nerve Tissue Proteins; Piperidines; Protein Binding; Proto-Oncogene Proteins c-fos; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists

2008
Antidepressant activity of standardised extract of Marsilea minuta Linn.
    Journal of ethnopharmacology, 2008, Apr-17, Volume: 117, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Antidepressive Agents; Female; Flunitrazepam; Hindlimb Suspension; Ketanserin; Male; Marsileaceae; Mice; Plant Extracts; Rats; Rats, Wistar; Serotonin 5-HT2 Receptor Antagonists; Swimming

2008
High specific activity tritium-labeled N-(2-methoxybenzyl)-2,5-dimethoxy-4-iodophenethylamine (INBMeO): a high-affinity 5-HT2A receptor-selective agonist radioligand.
    Bioorganic & medicinal chemistry, 2008, Jun-01, Volume: 16, Issue:11

    Topics: Binding Sites; Cell Line; Cell Line, Tumor; DNA-Binding Proteins; Ethylamines; Humans; Intracellular Signaling Peptides and Proteins; Iodine Radioisotopes; Iodobenzenes; Ketanserin; Nuclear Proteins; Radioligand Assay; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Tritium; Tumor Necrosis Factor alpha-Induced Protein 3

2008
Effects of selective serotonin2 ligands on behaviors evoked by stress in the rat.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 90, Issue:4

    Topics: Animals; Behavior, Animal; Dopamine Antagonists; Dose-Response Relationship, Drug; Ketanserin; Male; Motor Activity; Pain Measurement; Postural Balance; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT2; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Stress, Psychological; Vocalization, Animal

2008
Human embryonic stem cell-derived oligodendrocyte progenitor cells express the serotonin receptor and are susceptible to JC virus infection.
    Journal of virology, 2008, Volume: 82, Issue:17

    Topics: Antibodies, Monoclonal; Antigens; Biomarkers; Cell Line; Embryonic Stem Cells; Fetus; Humans; JC Virus; Ketanserin; Leukoencephalopathy, Progressive Multifocal; Oligodendroglia; Proteoglycans; Receptor, Serotonin, 5-HT2A; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2008
Modulation of striatal dopamine release by 5-HT2A and 5-HT2C receptor antagonists: [11C]raclopride PET studies in the rat.
    Psychopharmacology, 2008, Volume: 200, Issue:4

    Topics: Amphetamine; Animals; Binding, Competitive; Carbon Radioisotopes; Corpus Striatum; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Indoles; Ketanserin; Male; Positron-Emission Tomography; Protein Binding; Pyridines; Raclopride; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2008
Prenatal activation of 5-HT2A receptor induces expression of 5-HT1B receptor in phrenic motoneurons and alters the organization of their premotor network in newborn mice.
    The European journal of neuroscience, 2008, Volume: 28, Issue:6

    Topics: Amphetamines; Animals; Animals, Newborn; Embryo, Mammalian; Female; Ketanserin; Mice; Mice, Inbred C3H; Mice, Transgenic; Motor Neurons; Nerve Net; Phrenic Nerve; Pregnancy; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2008
Ketanserin, a 5-HT2 receptor antagonist, decreases nicotine self-administration in rats.
    European journal of pharmacology, 2008, Dec-14, Volume: 600, Issue:1-3

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Ketanserin; Male; Nicotine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Self Administration; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Tobacco Use Disorder

2008
Serotonin 5-HT(2) and 5-HT(1A)-like receptors differentially modulate aggressive behaviors in Drosophila melanogaster.
    Neuroscience, 2009, Feb-18, Volume: 158, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Amphetamines; Analysis of Variance; Animals; Drosophila melanogaster; Drosophila Proteins; Drug Interactions; Female; Gene Expression; Ketanserin; Male; Membrane Glycoproteins; Motor Activity; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin; Receptors, Serotonin, 5-HT2; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Social Behavior

2009
Behavioral pharmacological properties after recovery from the loss of righting reflex induced by benzodiazepine receptor agonists in mice.
    Methods and findings in experimental and clinical pharmacology, 2008, Volume: 30, Issue:8

    Topics: Animals; Azepines; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Flunitrazepam; GABA Agonists; GABA-A Receptor Agonists; Hypnotics and Sedatives; Ketanserin; Male; Mice; Mice, Inbred Strains; Pyridines; Reflex; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Time Factors; Zolpidem

2008
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane in rhesus monkeys: antagonism and apparent pA2 analyses.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 328, Issue:3

    Topics: Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Electroshock; Fluorobenzenes; Hallucinogens; Ketanserin; Macaca mulatta; Phenethylamines; Piperidines; Reaction Time; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Regression Analysis; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

2009
Genetic deletion of MAO-A promotes serotonin-dependent ventricular hypertrophy by pressure overload.
    Journal of molecular and cellular cardiology, 2009, Volume: 46, Issue:4

    Topics: Animals; Aorta; Blood Pressure; Cardiomegaly; Fibrosis; Fluorobenzenes; Gene Deletion; Gene Expression Regulation; Heart Ventricles; Ketanserin; Mice; Mice, Knockout; Monoamine Oxidase; Myocardium; Piperidines; Pressure; Receptors, Serotonin; Serotonin; Stress, Physiological; Ultrasonography

2009
Enhanced 5-HT(2A) receptors in brain stem and ALDH activity in brain stem and liver: 5-HT(2A) regulation on ALDH in primary hepatocytes cultures in vitro.
    Neurochemical research, 2009, Volume: 34, Issue:9

    Topics: Aldehyde Dehydrogenase; Animals; Brain Stem; Ethanol; Fluorobenzenes; Hepatocytes; Ketanserin; Liver; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin

2009
Assessment of 5-hydroxytryptamine efflux in rat brain during a mild, moderate and severe serotonin-toxicity syndrome.
    European journal of pharmacology, 2009, Aug-01, Volume: 615, Issue:1-3

    Topics: 5-Hydroxytryptophan; Animals; Antidepressive Agents; Body Temperature; Clorgyline; Cyproheptadine; Disease Models, Animal; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketanserin; Male; Microdialysis; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Syndrome

2009
Effects of acute intra-cerebral administration of the 5-HT(2A/C) receptor ligands DOI and ketanserin on impulse control in rats.
    Behavioural brain research, 2009, Dec-01, Volume: 204, Issue:1

    Topics: Amygdala; Analysis of Variance; Animals; Frontal Lobe; Impulsive Behavior; Indophenol; Ketanserin; Ligands; Male; Microinjections; Neuropsychological Tests; Psychomotor Performance; Rats; Rats, Wistar; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2009
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM), ketanserin, and (R)-(+)-{alpha}-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-pipidinemethanol (MDL100907) in rats.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:2

    Topics: Analgesics, Opioid; Anesthetics, Dissociative; Animals; Conditioning, Operant; Discrimination, Psychological; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorobenzenes; Ketamine; Ketanserin; Male; Morphine; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

2009
Inhibitory effect of serotonin antagonists on JC virus propagation in a carrier culture of human neuroblastoma cells.
    Microbiology and immunology, 2009, Volume: 53, Issue:9

    Topics: Cell Line, Tumor; Down-Regulation; Humans; JC Virus; Ketanserin; Neuroblastoma; Receptor, Serotonin, 5-HT2A; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Virus Cultivation; Virus Replication

2009
Effects of acute systemic administration of serotonin2A/C receptor ligands in a delay-based decision-making task in rats.
    Behavioural pharmacology, 2009, Volume: 20, Issue:5-6

    Topics: Amphetamines; Animals; Behavior, Animal; Decision Making; Dose-Response Relationship, Drug; Drug Interactions; Ketanserin; Male; Maze Learning; Rats; Rats, Wistar; Reaction Time; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Reinforcement Schedule; Reward; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Agents

2009
Serotonergic mechanisms on breathing modulation in the rat locus coeruleus.
    Pflugers Archiv : European journal of physiology, 2010, Volume: 459, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Amphetamines; Animals; Hydroxyindoleacetic Acid; Hypercapnia; Idazoxan; Ketanserin; Locus Coeruleus; Male; Microinjections; Piperazines; Pulmonary Ventilation; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Respiration; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2010
Serotonin 2 receptor modulation of hyperthermia, corticosterone, and hippocampal serotonin depletions following serial exposure to chronic stress and methamphetamine.
    Psychoneuroendocrinology, 2010, Volume: 35, Issue:4

    Topics: Amphetamine-Related Disorders; Animals; Behavior, Animal; Body Temperature Regulation; Central Nervous System Stimulants; Corticosterone; Drug Administration Schedule; Fever; Hippocampus; Ketanserin; Male; Methamphetamine; Periodicity; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT2; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Stress, Psychological

2010
Imaging cortical dopamine D1 receptors using [11C]NNC112 and ketanserin blockade of the 5-HT 2A receptors.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2010, Volume: 30, Issue:5

    Topics: Adult; Animals; Benzazepines; Benzofurans; Brain; Carbon Radioisotopes; Humans; Image Interpretation, Computer-Assisted; Ketanserin; Magnetic Resonance Imaging; Male; Positron-Emission Tomography; Receptors, Dopamine D1; Serotonin 5-HT2 Receptor Antagonists; Staining and Labeling; Young Adult

2010
Involvement of pro-nociceptive 5-HT2A receptor in the pathogenesis of medication-overuse headache.
    Headache, 2010, Volume: 50, Issue:2

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Animals; Cerebral Cortex; Cerebrovascular Circulation; Disease Models, Animal; Headache Disorders, Secondary; Hyperalgesia; Inflammation; Inflammation Mediators; Ketanserin; Male; Neuronal Plasticity; Nociceptors; Pain Measurement; Pain Threshold; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Reaction Time; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Trigeminal Nerve

2010
Horse chestnut extract contracts bovine vessels and affects human platelet aggregation through 5-HT(2A) receptors: an in vitro study.
    Phytotherapy research : PTR, 2010, Volume: 24, Issue:9

    Topics: Adenosine Diphosphate; Adrenergic alpha-1 Receptor Antagonists; Aesculus; Angiotensin II Type 1 Receptor Blockers; Animals; Cattle; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Humans; Ketanserin; Mesenteric Arteries; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Plant Bark; Plant Extracts; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptor, Serotonin, 5-HT2A; Seeds; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2010
Involvement of 5-HT2A receptors in the serotonin (5-HT) syndrome caused by excessive 5-HT efflux in rat brain.
    Basic & clinical pharmacology & toxicology, 2010, Volume: 107, Issue:4

    Topics: 5-Hydroxytryptophan; Animals; Body Temperature; Brain; Clorgyline; Hypothermia, Induced; Ketanserin; Male; Microdialysis; Monoamine Oxidase Inhibitors; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Syndrome

2010
The lateral habenula regulates defensive behaviors through changes in 5-HT-mediated neurotransmission in the dorsal periaqueductal gray matter.
    Neuroscience letters, 2010, Jul-26, Volume: 479, Issue:2

    Topics: Animals; Avoidance Learning; Habenula; Kainic Acid; Ketanserin; Male; Maze Learning; Motor Activity; Neurons; Periaqueductal Gray; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Synaptic Transmission

2010
State-dependent interactions between excitatory neuromodulators in the neuronal control of breathing.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Jun-16, Volume: 30, Issue:24

    Topics: Action Potentials; Adrenergic alpha-1 Receptor Antagonists; Animals; Animals, Newborn; Electric Stimulation; Electromyography; Hypoglossal Nerve; In Vitro Techniques; Isoindoles; Ketanserin; Locus Coeruleus; Mice; Microinjections; Neural Inhibition; Neural Pathways; Neurokinin-1 Receptor Antagonists; Neurons; Neurotransmitter Agents; Piperidines; Raphe Nuclei; Receptors, Adrenergic, alpha-1; Receptors, Neurokinin-1; Receptors, Serotonin, 5-HT2; Respiration; Respiratory Center; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2010
Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode.
    Chemical biology & drug design, 2010, Volume: 76, Issue:4

    Topics: Binding, Competitive; Combinatorial Chemistry Techniques; Fluorobenzenes; Hydrophobic and Hydrophilic Interactions; Ketanserin; Ligands; Phenols; Piperidines; Protein Binding; Pyridines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists

2010
Oleamide administered into the nucleus accumbens shell regulates feeding behaviour via CB1 and 5-HT2C receptors.
    The international journal of neuropsychopharmacology, 2010, Volume: 13, Issue:9

    Topics: Aminopyridines; Animals; Eating; Feeding Behavior; Hyperphagia; Hypothalamus; Indoles; Ketanserin; Male; Motor Activity; Nucleus Accumbens; Oleic Acids; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Antagonists

2010
PPI deficit induced by amphetamine is attenuated by the histamine H1 antagonist pyrilamine, but is exacerbated by the serotonin 5-HT2 antagonist ketanserin.
    Psychopharmacology, 2010, Volume: 212, Issue:4

    Topics: Acoustic Stimulation; Amphetamine; Animals; Behavior, Animal; Central Nervous System Stimulants; Female; Histamine H1 Antagonists; Inhibition, Psychological; Ketanserin; Physical Stimulation; Pyrilamine; Rats; Rats, Sprague-Dawley; Reflex, Startle; Sensory Gating; Serotonin 5-HT2 Receptor Antagonists

2010
Vestibular-mediated increase in central serotonin plays an important role in hypergravity-induced hypophagia in rats.
    Journal of applied physiology (Bethesda, Md. : 1985), 2010, Volume: 109, Issue:6

    Topics: Animals; Arsanilic Acid; Body Weight; Drinking; Eating; Feeding Behavior; Hypergravity; Ketanserin; Male; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Signal Transduction; Time Factors; Up-Regulation; Vestibular Nuclei

2010
Interaction of 5-HT2A and 5-HT2C receptors in R(-)-2,5-dimethoxy-4-iodoamphetamine-elicited head twitch behavior in mice.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 335, Issue:3

    Topics: Aminopyridines; Amphetamines; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Ethylamines; Fluorobenzenes; Hallucinogens; Head; Indoles; Ketanserin; Male; Mice; Mice, Inbred Strains; Movement; Piperidines; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Spiro Compounds; Sulfonamides

2010
Antagonism of 5-HT(2A) receptors inhibits the expression of pronociceptive mediator and enhances endogenous opioid mechanism in carrageenan-induced inflammation in rats.
    European journal of pharmacology, 2011, Mar-01, Volume: 654, Issue:1

    Topics: Animals; beta-Endorphin; Calcitonin Gene-Related Peptide; Carrageenan; Ganglia, Spinal; Inflammation; Ketanserin; Male; Pain; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Opioid, mu; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Spinal Cord

2011
Serotonin 2A and 2B receptor-induced phrenic motor facilitation: differential requirement for spinal NADPH oxidase activity.
    Neuroscience, 2011, Mar-31, Volume: 178

    Topics: Acetophenones; Action Potentials; Amphetamines; Animals; Indoles; Injections, Spinal; Ketanserin; Male; NADPH Oxidases; Onium Compounds; Phrenic Nerve; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Thiophenes

2011
Effects of 5-HT(2A) and 5-HT(2C) receptor antagonists on acute and chronic dyskinetic effects induced by haloperidol in rats.
    Behavioural brain research, 2011, Jun-01, Volume: 219, Issue:2

    Topics: Aminopyridines; Animals; Antipsychotic Agents; Brain Chemistry; Catalepsy; Dyskinesia, Drug-Induced; Fluorobenzenes; Gene Expression Regulation; Haloperidol; Immunohistochemistry; In Situ Hybridization; Indoles; Ketanserin; Male; Mouth; Piperidines; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; RNA, Messenger; Serotonin Antagonists

2011
Blockade of 5-HT(2A) and/or 5-HT(2C) receptors modulates sevoflurane-induced immobility.
    Journal of anesthesia, 2011, Volume: 25, Issue:2

    Topics: Anesthetics, Inhalation; Animals; Immobilization; Indoles; Ketanserin; Male; Methyl Ethers; Pyridines; Rats; Rats, Wistar; Serotonin 5-HT2 Receptor Antagonists; Sevoflurane

2011
A spinal mechanism of action for duloxetine in a rat model of painful diabetic neuropathy.
    British journal of pharmacology, 2011, Volume: 164, Issue:1

    Topics: Amphetamines; Animals; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Duloxetine Hydrochloride; Female; Hyperalgesia; Ketanserin; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Thiophenes

2011
Subchronic treatment with fluoxetine and ketanserin increases hippocampal brain-derived neurotrophic factor, β-catenin and antidepressant-like effects.
    British journal of pharmacology, 2012, Volume: 165, Issue:4b

    Topics: Animals; Antidepressive Agents, Second-Generation; Behavior, Animal; beta Catenin; Brain-Derived Neurotrophic Factor; Fluoxetine; Hippocampus; Ketanserin; Male; Rats; Rats, Sprague-Dawley; RNA, Messenger; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT2 Receptor Antagonists; Swimming

2012
p-Hydroxyamphetamine causes prepulse inhibition disruption in mice: contribution of serotonin neurotransmission.
    Behavioural brain research, 2011, Oct-10, Volume: 224, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Acoustic Stimulation; Analysis of Variance; Animals; Autoradiography; Brain; Dose-Response Relationship, Drug; Fenclonine; Fluorobenzenes; Inhibition, Psychological; Ketanserin; Male; Mice; p-Hydroxyamphetamine; Piperidines; Reflex, Startle; Serotonin; Serotonin Agents; Serotonin Plasma Membrane Transport Proteins; Time Factors

2011
Cognition-induced modulation of serotonin in the orbitofrontal cortex: a controlled cross-over PET study of a delayed match-to-sample task using the 5-HT2a receptor antagonist [18F]altanserin.
    NeuroImage, 2011, Oct-01, Volume: 58, Issue:3

    Topics: Brain Mapping; Cognition; Cross-Over Studies; Fluorine Radioisotopes; Frontal Lobe; Humans; Ketanserin; Male; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Antagonists

2011
Pulmonary vascular effects of serotonin and selective serotonin reuptake inhibitors in the late-gestation ovine fetus.
    American journal of physiology. Lung cellular and molecular physiology, 2011, Volume: 301, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Dose-Response Relationship, Drug; Female; Fetus; Fluoxetine; Hemodynamics; Hypertension, Pulmonary; Hysterotomy; Indoles; Ketanserin; Lung; Oxadiazoles; Piperazines; Pregnancy; Pulmonary Artery; Pyridines; Receptors, Serotonin; rho-Associated Kinases; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Sertraline; Sheep; Vascular Resistance

2011
Preservation of serotonin-mediated contractility in adult sheep pulmonary arteries following long-term high-altitude hypoxia.
    High altitude medicine & biology, 2011,Fall, Volume: 12, Issue:3

    Topics: Altitude Sickness; Animals; Benzamides; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Female; In Vitro Techniques; Ketanserin; Microscopy, Confocal; Muscle Contraction; Muscle, Smooth, Vascular; Myography; Nickel; Pulmonary Artery; Pyridines; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Sheep; Sodium-Calcium Exchanger; Spermine; Time Factors; TRPC Cation Channels; TRPM Cation Channels

2011
The role of MAPK and Nrf2 pathways in ketanserin-elicited attenuation of cigarette smoke-induced IL-8 production in human bronchial epithelial cells.
    Toxicological sciences : an official journal of the Society of Toxicology, 2012, Volume: 125, Issue:2

    Topics: Anti-Inflammatory Agents; Antioxidants; Bronchi; Cell Survival; Cells, Cultured; Dose-Response Relationship, Drug; Glutathione; Humans; Interleukin-8; Ketanserin; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; NF-E2-Related Factor 2; Oxidation-Reduction; Oxidative Stress; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Receptor, Serotonin, 5-HT2A; RNA Interference; RNA, Messenger; Serotonin 5-HT2 Receptor Antagonists; Smoke; Smoking; Time Factors; Transfection; Up-Regulation

2012
Antiserotonergic properties of terguride in blood vessels, platelets, and valvular interstitial cells.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenosine Diphosphate; Animals; Aortic Valve; Blood Vessels; Cells, Cultured; Collagen; Coronary Vessels; Dose-Response Relationship, Drug; Heart Valves; Humans; In Vitro Techniques; Inhibitory Concentration 50; Ketanserin; Kinetics; Lisuride; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitral Valve; Phosphorylation; Platelet Aggregation; Pulmonary Artery; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Sus scrofa; Vasoconstriction; Vasodilation

2012
Impulsive action and impulsive choice are mediated by distinct neuropharmacological substrates in rat.
    The international journal of neuropsychopharmacology, 2012, Volume: 15, Issue:10

    Topics: Adrenergic Uptake Inhibitors; Aminopyridines; Animals; Atomoxetine Hydrochloride; Choice Behavior; Dopamine Uptake Inhibitors; Impulsive Behavior; Indoles; Ketanserin; Male; Methylphenidate; Propylamines; Rats; Rats, Long-Evans; Reaction Time; Serotonin 5-HT2 Receptor Antagonists

2012
Ferulic acid exerts antidepressant-like effect in the tail suspension test in mice: evidence for the involvement of the serotonergic system.
    European journal of pharmacology, 2012, Mar-15, Volume: 679, Issue:1-3

    Topics: Animals; Antidepressive Agents; Coumaric Acids; Dose-Response Relationship, Drug; Drug Interactions; Fluoxetine; Immobility Response, Tonic; Ketanserin; Male; Mice; Motor Activity; Paroxetine; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Sertraline

2012
Inhibition of SNL-induced upregulation of CGRP and NPY in the spinal cord and dorsal root ganglia by the 5-HT(2A) receptor antagonist ketanserin in rats.
    Pharmacology, biochemistry, and behavior, 2012, Volume: 101, Issue:3

    Topics: Animals; Calcitonin Gene-Related Peptide; Denervation; Disease Models, Animal; Ganglia, Spinal; Hyperalgesia; Immunohistochemistry; Ketanserin; Male; Neuralgia; Neuronal Plasticity; Neuropeptide Y; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Spinal Cord; Spinal Nerves; Up-Regulation

2012
Functional selectivity in serotonin receptor 2A (5-HT2A) endocytosis, recycling, and phosphorylation.
    Molecular pharmacology, 2013, Volume: 83, Issue:1

    Topics: Amphetamines; Animals; Clozapine; Dopamine; Drug Partial Agonism; Endocytosis; Enzyme Activation; HEK293 Cells; Humans; Ketanserin; Ligands; Phosphorylation; Protein Kinase C; Protein Phosphatase 2; Protein Transport; Rats; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Signal Transduction

2013
Deficits in LTP induction by 5-HT2A receptor antagonist in a mouse model for fragile X syndrome.
    PloS one, 2012, Volume: 7, Issue:10

    Topics: Animals; Blotting, Western; Cells, Cultured; Disease Models, Animal; Fragile X Mental Retardation Protein; Fragile X Syndrome; Gyrus Cinguli; Humans; Ketanserin; Long-Term Potentiation; Male; Mice; Mice, 129 Strain; Mice, Knockout; Patch-Clamp Techniques; Pyrrolidines; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Serotonin 5-HT2 Receptor Antagonists; Synaptic Potentials

2012
Serotonin inhibits apoptosis of pulmonary artery smooth muscle cells through 5-HT2A receptors involved in the pulmonary artery remodeling of pulmonary artery hypertension.
    Experimental lung research, 2013, Volume: 39, Issue:2

    Topics: Animals; Apoptosis; Cell Proliferation; Cells, Cultured; Disease Models, Animal; Familial Primary Pulmonary Hypertension; Humans; Hypertension, Pulmonary; Hypertrophy, Right Ventricular; Ketanserin; Male; MAP Kinase Signaling System; Membrane Potential, Mitochondrial; Muscle, Smooth, Vascular; Protein Serine-Threonine Kinases; Pulmonary Artery; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; Random Allocation; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Antagonists

2013
5-HT2A receptor antagonists inhibit hepatic stellate cell activation and facilitate apoptosis.
    Liver international : official journal of the International Association for the Study of the Liver, 2013, Volume: 33, Issue:4

    Topics: Actins; Animals; Apoptosis; Cell Line; Cell Survival; Collagen Type I; Dose-Response Relationship, Drug; Hepatic Stellate Cells; Humans; Ketanserin; Liver Cirrhosis, Experimental; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptor, Serotonin, 5-HT2A; Ritanserin; RNA, Messenger; Serotonin 5-HT2 Receptor Antagonists; Smad2 Protein; Smad3 Protein; Succinates; Thioacetamide; Time Factors; Transforming Growth Factor beta; Wound Healing

2013
Direct comparison of [(18) F]MH.MZ and [(18) F] altanserin for 5-HT2A receptor imaging with PET.
    Synapse (New York, N.Y.), 2013, Volume: 67, Issue:6

    Topics: Animals; Brain; Fluorine Radioisotopes; Fluorobenzenes; Ketanserin; Piperidines; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Swine; Tissue Distribution; Tritium

2013
Serotonergic mechanisms are necessary for central respiratory chemoresponsiveness in situ.
    Respiratory physiology & neurobiology, 2013, Apr-01, Volume: 186, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Stem; Hypercapnia; Ketanserin; Phrenic Nerve; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Respiratory Mechanics; Serotonergic Neurons; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists

2013
[Involvement of some subtypes of 5-HT2-receptors in affective behavior in female rats].
    Fiziolohichnyi zhurnal (Kiev, Ukraine : 1994), 2012, Volume: 58, Issue:6

    Topics: Animals; Animals, Outbred Strains; Anti-Anxiety Agents; Anxiety; Depression; Estrogens; Estrus; Female; Injections, Intraperitoneal; Ketanserin; Piperazines; Proestrus; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2012
Serotonin contributes to high pulmonary vascular tone in a sheep model of persistent pulmonary hypertension of the newborn.
    American journal of physiology. Lung cellular and molecular physiology, 2013, Jun-15, Volume: 304, Issue:12

    Topics: Adult; Animals; Cells, Cultured; Disease Models, Animal; Endothelial Cells; Familial Primary Pulmonary Hypertension; Fetus; Gene Expression; Humans; Hypertension, Pulmonary; Infant, Newborn; Ketanserin; Lung; Pulmonary Artery; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Sertraline; Sheep, Domestic; Tryptophan Hydroxylase; Vascular Resistance

2013
Serotonin₂A/C receptors mediate the aggressive phenotype of TLX gene knockout mice.
    Behavioural brain research, 2013, Nov-01, Volume: 256

    Topics: Aggression; Animals; Behavior, Animal; Clozapine; Ketanserin; Male; Mice; Mice, Knockout; Motor Activity; Phenotype; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Cytoplasmic and Nuclear; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2013
Hallucinogenic 5-HT2AR agonists LSD and DOI enhance dopamine D2R protomer recognition and signaling of D2-5-HT2A heteroreceptor complexes.
    Biochemical and biophysical research communications, 2014, Jan-03, Volume: 443, Issue:1

    Topics: Amphetamines; Animals; Basal Ganglia; Gene Expression Regulation; Genes, Reporter; Hallucinogens; HEK293 Cells; Humans; Ketanserin; Luciferases; Lysergic Acid Diethylamide; Male; Promoter Regions, Genetic; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2014
Serotonin contracts the rat mesenteric artery by inhibiting 4-aminopyridine-sensitive Kv channels via the 5-HT2A receptor and Src tyrosine kinase.
    Experimental & molecular medicine, 2013, Dec-13, Volume: 45

    Topics: 4-Aminopyridine; Action Potentials; Animals; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Ketanserin; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nifedipine; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Spiperone; src-Family Kinases; Vasoconstriction

2013
The analgesia effect of duloxetine on post-operative pain via intrathecal or intraperitoneal administration.
    Neuroscience letters, 2014, May-07, Volume: 568

    Topics: Adrenergic alpha-2 Receptor Antagonists; Analgesics; Animals; Duloxetine Hydrochloride; Hyperalgesia; Idazoxan; Injections, Intraperitoneal; Injections, Spinal; Ketanserin; Male; Microdialysis; Norepinephrine; Pain, Postoperative; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Spinal Cord; Thiophenes

2014
Serotonin modulates electrosensory processing and behavior via 5-HT2-like receptors.
    Neuroscience, 2014, Jun-20, Volume: 271

    Topics: Action Potentials; Animals; Electric Organ; Electric Stimulation; Gymnotiformes; Ketanserin; Microelectrodes; Motor Activity; Perception; Pyramidal Cells; Receptors, Serotonin; Rhombencephalon; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Tissue Culture Techniques

2014
Citral: a monoterpene with prophylactic and therapeutic anti-nociceptive effects in experimental models of acute and chronic pain.
    European journal of pharmacology, 2014, Aug-05, Volume: 736

    Topics: Acute Pain; Acyclic Monoterpenes; Analgesics; Animals; Capsaicin; Chronic Pain; Excitatory Amino Acids; Formaldehyde; Glutamic Acid; Hyperalgesia; Ischemia; Ketanserin; Male; Mice; Monoterpenes; Neuralgia; Pain, Postoperative; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Stomach Ulcer; Substance P; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha

2014
Ketanserin, a serotonin 2A receptor antagonist, alleviates ischemia-related biliary fibrosis following donation after cardiac death liver transplantation in rats.
    Liver transplantation : official publication of the American Association for the Study of Liver Diseases and the International Liver Transplantation Society, 2014, Volume: 20, Issue:11

    Topics: Animals; Biliary Tract Diseases; Cells, Cultured; Drug Evaluation, Preclinical; Fibroblasts; Fibrosis; Ischemia; Ketanserin; Liver; Liver Transplantation; Male; Postoperative Complications; Rats, Sprague-Dawley; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Signal Transduction; Transforming Growth Factor beta1; Up-Regulation

2014
Effect of 5-HT(2A) receptor antagonists on blood flow in the carotid vessels upon elevation of serotonin level.
    Bulletin of experimental biology and medicine, 2014, Volume: 157, Issue:3

    Topics: Animals; Animals, Outbred Strains; Carotid Arteries; Drug Evaluation, Preclinical; Ketanserin; Male; Rats; Regional Blood Flow; Ritanserin; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Vasoconstriction

2014
Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT₂A receptors, in mice.
    Psychopharmacology, 2015, Volume: 232, Issue:6

    Topics: Amphetamines; Animals; Dose-Response Relationship, Drug; Fluorobenzenes; Hallucinogens; Head Movements; Ketanserin; Male; Mice; Phenethylamines; Piperidines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2015
Serotonin antagonists induce anxiolytic and anxiogenic-like behavior in zebrafish in a receptor-subtype dependent manner.
    Pharmacology, biochemistry, and behavior, 2014, Volume: 126

    Topics: Aminopyridines; Animals; Anti-Anxiety Agents; Anxiety; Benzamides; Ketanserin; Ondansetron; Piperazines; Pyridines; Receptors, Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Zebrafish

2014
Attenuated methamphetamine-induced locomotor sensitization in serotonin transporter knockout mice is restored by serotonin 1B receptor antagonist treatment.
    Behavioural pharmacology, 2015, Volume: 26, Issue:1-2

    Topics: Animals; Behavior, Animal; Benzamides; Central Nervous System Stimulants; Dopamine; Female; Ketanserin; Male; Methamphetamine; Mice; Mice, Inbred C57BL; Mice, Knockout; Microdialysis; Motor Activity; Oxadiazoles; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Plasma Membrane Transport Proteins

2015
Individual Differences in Impulsive Action Reflect Variation in the Cortical Serotonin 5-HT2A Receptor System.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2015, Volume: 40, Issue:8

    Topics: Animals; Choice Behavior; Dimethoxyphenylethylamine; Fluorobenzenes; Head Movements; Immunoprecipitation; Impulsive Behavior; Individuality; Ketanserin; Male; Piperidines; Prefrontal Cortex; Protein Binding; Rats; Rats, Sprague-Dawley; Reaction Time; Receptor, Serotonin, 5-HT2A; Serotonin Agents; Tritium

2015
5-HT2a receptor antagonism reduces burn-induced macromolecular efflux in rats.
    European journal of trauma and emergency surgery : official publication of the European Trauma Society, 2015, Volume: 41, Issue:5

    Topics: Animals; Burns; Edema; Endothelium, Vascular; Hemodynamics; Ketanserin; Leukocytes; Mesentery; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serum Albumin

2015
Effect of Systemic Application of 5-Hydroxytryptamine on Hypoglossal Nerve Discharge in Anesthetized Rats.
    Journal of molecular neuroscience : MN, 2015, Volume: 57, Issue:3

    Topics: Action Potentials; Anesthesia, General; Animals; Carotid Body; Hypoglossal Nerve; Injections, Intravenous; Ketanserin; Long-Term Potentiation; Male; Nerve Tissue Proteins; Nodose Ganglion; Oxidative Stress; Phosphorylation; Protein Isoforms; Protein Kinase C; Protein Processing, Post-Translational; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptor, Serotonin, 5-HT2A; Respiration; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Staurosporine

2015
[Effects of blockade of 5-HT2A receptors in inflammatory site on complete Freund's adjuvant-induced chronic hyperalgesia and neuropeptide Y expression in the spinal dorsal horn in rats].
    Sheng li xue bao : [Acta physiologica Sinica], 2015, Oct-25, Volume: 67, Issue:5

    Topics: Animals; Freund's Adjuvant; Ganglia, Spinal; Hot Temperature; Hyperalgesia; Inflammation; Ketanserin; Neuropeptide Y; Pain; Pain Measurement; Rats; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Spinal Cord Dorsal Horn

2015
Alternative Viewpoint Against Breast Cancer Based on Selective Serotonin Receptors 5HTR3A and 5HTR2A Antagonists that can Mediate Apoptosis in MCF-7 Cell Line.
    Current drug discovery technologies, 2015, Volume: 12, Issue:4

    Topics: Antineoplastic Agents; Apoptosis; Breast Neoplasms; Gene Expression; Humans; Indoles; Ketanserin; MCF-7 Cells; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Tropisetron

2015
Serotonin 2A receptor agonist binding in the human brain with [(11)C]Cimbi-36: Test-retest reproducibility and head-to-head comparison with the antagonist [(18)F]altanserin.
    NeuroImage, 2016, Apr-15, Volume: 130

    Topics: Benzylamines; Brain; Carbon Radioisotopes; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Neuroimaging; Phenethylamines; Positron-Emission Tomography; Radiopharmaceuticals; Reproducibility of Results; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Young Adult

2016
Blockade of 5-HT2A receptors at the site of inflammation inhibits activation of spinal dorsal horn neurons in rats.
    Brain research bulletin, 2016, Volume: 124

    Topics: Animals; Carrageenan; Gene Expression Regulation; Inflammation; Ketanserin; Male; NADH Dehydrogenase; Nitric Oxide Synthase; Posterior Horn Cells; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Spinal Cord

2016
Distinct effect of 5-HT1A and 5-HT2A receptors in the medial nucleus of the amygdala on tonic immobility behavior.
    Brain research, 2016, 07-15, Volume: 1643

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anxiety; Corticomedial Nuclear Complex; Fear; Guinea Pigs; Immobility Response, Tonic; Ketanserin; Male; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2016
Reformulating a Pharmacophore for 5-HT2A Serotonin Receptor Antagonists.
    ACS chemical neuroscience, 2016, 09-21, Volume: 7, Issue:9

    Topics: Animals; Barium; Calcium; G Protein-Coupled Inwardly-Rectifying Potassium Channels; HEK293 Cells; Humans; Hydrophobic and Hydrophilic Interactions; Ketanserin; Membrane Potentials; Mutation; Oocytes; Protein Binding; Receptor, Serotonin, 5-HT2A; Risperidone; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Tritium; Xenopus laevis

2016
Serotonin modifies the spontaneous spiking activity of gracile nucleus neurons in rats: role of 5-HT1A and 5-HT2 receptors.
    Archives italiennes de biologie, 2016, Jun-01, Volume: 154, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Iontophoresis; Ketanserin; Male; Medulla Oblongata; Neurons; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT2; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2016
Dreamlike effects of LSD on waking imagery in humans depend on serotonin 2A receptor activation.
    Psychopharmacology, 2017, Volume: 234, Issue:13

    Topics: Dopamine; Healthy Volunteers; Humans; Ketanserin; Lysergic Acid Diethylamide; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin 5-HT2 Receptor Antagonists

2017
Serotonin 2A Receptor Signaling Underlies LSD-induced Alteration of the Neural Response to Dynamic Changes in Music.
    Cerebral cortex (New York, N.Y. : 1991), 2018, 11-01, Volume: 28, Issue:11

    Topics: Auditory Perception; Brain; Brain Mapping; Double-Blind Method; Emotions; Hallucinogens; Humans; Ketanserin; Lysergic Acid Diethylamide; Magnetic Resonance Imaging; Memory; Music; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists

2018
Effect of 5-HT
    Neuroscience letters, 2018, 11-20, Volume: 687

    Topics: Animals; Ketanserin; Male; Motor Neurons; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Antagonists; Urethane; Urethra; Urinary Bladder; Urination

2018
Serotonin receptors 5-HTR2A and 5-HTR2B are involved in cigarette smoke-induced airway inflammation, mucus hypersecretion and airway remodeling in mice.
    International immunopharmacology, 2020, Volume: 81

    Topics: Airway Remodeling; Animals; Bronchoalveolar Lavage Fluid; Disease Models, Animal; Humans; Injections, Intraperitoneal; Ketanserin; Lung; Male; Mice; Mucus; Nicotiana; Pulmonary Disease, Chronic Obstructive; Pyrimidines; Quercetin; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Respiratory Mucosa; Serotonin 5-HT2 Receptor Antagonists; Smoke; Specific Pathogen-Free Organisms

2020
Ritanserin blocks Ca
    Acta pharmacologica Sinica, 2020, Volume: 41, Issue:9

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arteries; Binding Sites; Calcium Channels, L-Type; Electrophysiological Phenomena; Ketanserin; Male; Molecular Docking Simulation; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Protein Binding; Rats, Wistar; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Vasoconstriction

2020
Hypoxia-induced hypotension elicits adenosine-dependent phrenic long-term facilitation after carotid denervation.
    Experimental neurology, 2020, Volume: 333

    Topics: Adenosine; Animals; Arterial Pressure; Blood Gas Analysis; Carotid Body; Denervation; Hypotension; Hypoxia; Ketanserin; Long-Term Potentiation; Male; Phenylephrine; Phrenic Nerve; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Serotonin 5-HT2 Receptor Antagonists; Spinal Cord

2020
Risperidone and 5-HT2A Receptor Antagonists Attenuate and Reverse Cocaine-Induced Hyperthermia in Rats.
    The international journal of neuropsychopharmacology, 2020, 12-29, Volume: 23, Issue:12

    Topics: Animals; Benzazepines; Cocaine; Disease Models, Animal; Dopamine Antagonists; Dopamine Uptake Inhibitors; Haloperidol; Hyperthermia; Ketanserin; Male; Rats; Rats, Wistar; Risperidone; Ritanserin; Serotonin 5-HT2 Receptor Antagonists

2020
Acute intermittent hypoxia evokes ventilatory long-term facilitation and active expiration in unanesthetized rats.
    Respiratory physiology & neurobiology, 2021, Volume: 294

    Topics: Animals; Disease Models, Animal; Hypoxia; Ketanserin; Male; Pulmonary Ventilation; Rats; Rats, Sprague-Dawley; Respiratory Mechanics; Serotonin 5-HT2 Receptor Antagonists; Tidal Volume

2021
Effects of Ketanserin, M100907 and Olanzapine on hallucinogenic like action induced by 2,5-dimethoxy-4-methylamphetamine.
    Behavioural pharmacology, 2023, 04-01, Volume: 34, Issue:2-3

    Topics: Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Hallucinogens; Ketanserin; Male; Methamphetamine; Mice; Mice, Inbred C57BL; Olanzapine; Receptor, Serotonin, 5-HT2A

2023
Acute psilocybin enhances cognitive flexibility in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2023, Volume: 48, Issue:7

    Topics: Animals; Anxiety; Cognition; Female; Hallucinogens; Ketanserin; Male; Psilocybin; Rats; Serotonin; Serotonin 5-HT2 Receptor Antagonists

2023