ketanserin has been researched along with ly 53857 in 38 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 12 (31.58) | 18.7374 |
1990's | 22 (57.89) | 18.2507 |
2000's | 4 (10.53) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Baez, M; Kursar, JD; Lucaites, VL; Nelson, DL; Sasso, DA; Wainscott, DB | 1 |
Innocent, O; Olufemi, A | 1 |
Jacobs, M; McRee, C; Meyer, DC | 1 |
Jørgensen, H; Knigge, U; Warberg, J | 2 |
Cohen, ML; Cushing, DJ | 1 |
Forrest, CR; Morris, SF; Pang, CY; Sheffield, WD; Zhong, A | 1 |
Buckner, CK; Dea, D; Krell, RD; Liberati, N | 1 |
Anderson, HV; Benedict, CR; Buja, LM; Golino, P; McNatt, J; Murphree, SS; Willerson, JT; Yao, SK | 1 |
Cohen, ML; Mann, JJ; McBride, PA; Nimchinsky, E | 1 |
Ashby, CR; Jiang, LH; Kasser, RJ; Wang, RY | 1 |
Coote, JH; Lewis, DI | 1 |
Docherty, JR; Warnock, P | 1 |
Cohen, ML; Kurz, KD; Schenck, KW | 1 |
Ramage, AG | 2 |
Mistry, A; Voogt, JL | 1 |
Docherty, JR | 1 |
Pan, JT; Teo, KL | 1 |
Gala, RR; Pan, JT | 1 |
Schechter, LE; Simansky, KJ | 1 |
Harris, LT; McCall, RB | 2 |
Brunken, WJ; Daw, NW | 1 |
Antonaccio, MJ; Dzwonczyk, S; Grover, GJ; Normandin, DE; Sargent, CA | 1 |
Chiu, C; Pang, CY; Xu, N; Zhong, A | 1 |
Dykstra, LA; Lin, YP; Powell, KR | 1 |
Elliott, P; Wallis, DI | 1 |
Albert, AP; Brooks, PA; Spyer, KM | 1 |
Baez, M; Johnson, MP; Lucaites, VL; Nelson, DL; Wainscott, DB | 1 |
Chung, JH; Chung, SM; Lee, JY; Lee, MY | 1 |
Sugimoto, Y; Yamada, J; Yoshikawa, T | 1 |
Harvey, JA; Hood, H; Romano, AG; Welsh, SE | 1 |
Yan, QS | 1 |
Inoue, K; Ohkura, M; Sugimoto, Y; Yamada, J | 1 |
Sugimoto, Y; Yamada, J | 1 |
Fink, GD; Li, MW; Ni, W; Thakali, K; Watts, SW | 1 |
38 other study(ies) available for ketanserin and ly 53857
Article | Year |
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Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.
Topics: Adrenergic alpha-Antagonists; Benzofurans; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Imidazoles; Radioligand Assay; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Yohimbine | 1998 |
Receptors mediating the actions of 5-hydroxytryptamine on the isolated retractor muscle of the penis preparations from Archachatina marginata (Swainson).
Topics: Animals; Ergolines; Indoles; Ketanserin; Lysergic Acid Diethylamide; Muscle Contraction; Muscles; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Snails; Tropisetron | 1992 |
Role of 5-hydroxytryptamine receptors on luteinizing-hormone-releasing hormone release in the ovariectomized, estradiol-treated rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Estradiol; Female; Gonadotropin-Releasing Hormone; Hypothalamus, Middle; Ketanserin; Ovariectomy; Pindolol; Preoptic Area; Quipazine; Radioimmunoassay; Rats; Receptors, Serotonin; Serotonin Antagonists; Suprachiasmatic Nucleus; Tetrahydronaphthalenes | 1992 |
Involvement of 5-HT1, 5-HT2, and 5-HT3 receptors in the mediation of the prolactin response to serotonin and 5-hydroxytryptophan.
Topics: 5-Hydroxytryptophan; Animals; Dose-Response Relationship, Drug; Ergolines; Fluoxetine; Imidazoles; Indoles; Ketanserin; Male; Methysergide; Ondansetron; Prolactin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron | 1992 |
Effect of serotonin 5-HT1, 5-HT2, and 5-HT3 receptor antagonists on the prolactin response to restraint and ether stress.
Topics: Animals; Ergolines; Ether; Indoles; Ketanserin; Male; Methysergide; Ondansetron; Prolactin; Rats; Rats, Wistar; Restraint, Physical; Serotonin Antagonists; Stress, Physiological; Tropisetron | 1992 |
Comparison of the serotonin receptors that mediate smooth muscle contraction in canine and porcine coronary artery.
Topics: Animals; Coronary Vessels; Dogs; Ergolines; Jugular Veins; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Receptors, Serotonin; Serotonin Antagonists; Species Specificity; Swine | 1992 |
Augmentation of acute random pattern skin flap viability in the pig.
Topics: Animals; Dose-Response Relationship, Drug; Ergolines; Graft Survival; Ischemia; Ketanserin; Regional Blood Flow; Serotonin Antagonists; Skin; Surgical Flaps; Swine | 1992 |
Guinea pig pulmonary responses to serotonin (5-HT) and related agonists.
Topics: Animals; Ergolines; Guinea Pigs; Ketanserin; Lung; Mianserin; Respiratory Function Tests; Serotonin | 1991 |
Frequency and severity of cyclic flow alternations and platelet aggregation predict the severity of neointimal proliferation following experimental coronary stenosis and endothelial injury.
Topics: Animals; Blood Pressure; Cell Division; Coronary Disease; Coronary Vessels; Dogs; Endothelium, Vascular; Ergolines; Ketanserin; Muscle, Smooth, Vascular; Platelet Aggregation; Serotonin Antagonists | 1991 |
Inhibition of serotonin-amplified human platelet aggregation by ketanserin, ritanserin, and the ergoline 5HT2 receptor antagonists-LY53857, sergolexole, and LY237733.
Topics: Adult; Ergolines; Female; Humans; Ketanserin; Lysergic Acid; Male; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Electrophysiological characterization of 5-hydroxytryptamine2 receptors in the rat medial prefrontal cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ergolines; Frontal Lobe; Ketanserin; Magnesium; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Sodium Glutamate; Tetrahydronaphthalenes | 1990 |
The influence of 5-hydroxytryptamine agonists and antagonists on identified sympathetic preganglionic neurones in the rat, in vivo.
Topics: Anesthesia; Animals; Electric Stimulation; Ergolines; Ganglia, Sympathetic; Homocysteine; Indoles; Iontophoresis; Ketanserin; Male; Neurons; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron | 1990 |
Effects of antagonists of 5-hydroxytryptamine on blood pressure in the anesthetised spontaneously hypertensive rat.
Topics: Animals; Blood Pressure; Consciousness; Ergolines; Ketanserin; Male; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists | 1987 |
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Ergolines; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pyrimidinones; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone | 1988 |
Are drugs that act both on serotonin receptors and alpha 1-adrenoceptors more potent hypotensive agents than those that act only on alpha 1-adrenoceptors?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Cats; Cinanserin; Ergolines; Ketanserin; Male; Metergoline; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes | 1988 |
Role of serotonin in nocturnal and diurnal surges of prolactin in the pregnant rat.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Circadian Rhythm; Dopamine; Ergolines; Female; Fenclonine; Hydroxyindoleacetic Acid; Hypothalamus; Ketanserin; Pregnancy; Pregnancy, Animal; Prolactin; Rats; Rats, Inbred Strains; Serotonin | 1989 |
An investigation of the effects of intravenous injection of the 5-hydroxytryptamine 2 receptor antagonists ketanserin and LY 53857 on blood pressure in anesthetized spontaneously hypertensive rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Blood Pressure; Ergolines; Heart Rate; Hypertension; Ketanserin; Male; Prazosin; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Xylazine | 1989 |
Fentanyl stimulates prolactin release through mu-opiate receptors, but not the serotonergic system.
Topics: Animals; Dose-Response Relationship, Drug; Ergolines; Female; Fenclonine; Fentanyl; Ketanserin; Prolactin; Rats; Receptors, Opioid; Serotonin; Serotonin Antagonists | 1989 |
The serotonin 5-HT2 receptor system, but not the alpha 1-adrenergic receptor system, is involved in the estrogen-induced afternoon prolactin surge in the rat.
Topics: Animals; Circadian Rhythm; Ergolines; Estradiol; Estrogens; Female; Ketanserin; Ovariectomy; Prazosin; Prolactin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists | 1988 |
The effects of ketanserin, methysergide and LY 53857 on sympathetic nerve activity.
Topics: Anesthesia; Animals; Blood Pressure; Cats; Ergolines; Heart Rate; Hemodynamics; Ketanserin; Lactates; Lactic Acid; Male; Methysergide; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Sympathetic Nervous System | 1985 |
1-(2,5-Dimethoxy-4-iodophenyl)-2-aminopropane (DOI) exerts an anorexic action that is blocked by 5-HT2 antagonists in rats.
Topics: Amidines; Amphetamines; Animals; Appetite Depressants; Diet; Eating; Ergolines; Ketanserin; Male; Rats; Rats, Inbred Strains; Serotonin Antagonists | 1988 |
5-HT2 receptor agonists increase spontaneous sympathetic nerve discharge.
Topics: Amphetamines; Animals; Blood Pressure; Cats; Ergolines; Heart Rate; Ketanserin; Neurons; Receptors, Serotonin; Serotonin Antagonists; Sympathetic Nervous System | 1988 |
Characterization of the central sympathoinhibitory action of ketanserin.
Topics: Animals; Blood Pressure; Cats; Clonidine; Electrophysiology; Ergolines; Heart Rate; Ketanserin; Prazosin; Sympathetic Nervous System | 1987 |
5-HT2 antagonists reduce ON responses in the rabbit retina.
Topics: Animals; Butyrophenones; Ergolines; Evoked Potentials, Visual; Ketanserin; Photic Stimulation; Rabbits; Retina; Retinal Ganglion Cells; Serotonin Antagonists | 1986 |
Protective effect of serotonin (5-HT2) receptor antagonists in ischemic rat hearts.
Topics: Animals; Cinanserin; Disease Models, Animal; Ergolines; Heart; Hemodynamics; Ketanserin; L-Lactate Dehydrogenase; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardial Ischemia; Myocardial Reperfusion Injury; Myocardium; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Serotonin Antagonists | 1993 |
Pharmacologic intervention of skin vasospasm and ischemic necrosis in pigs.
Topics: Adrenergic alpha-Antagonists; Animals; Arginine; Dose-Response Relationship, Drug; Ergolines; In Vitro Techniques; Ischemia; Ketanserin; Necrosis; omega-N-Methylarginine; Prostaglandin H2; Prostaglandins H; Regional Blood Flow; Serotonin; Serotonin Antagonists; Skin; Surgical Flaps; Swine; Thromboxane A2; Vasoconstriction | 1993 |
Antinociceptive effects of the kappa opioid, U50,488: lack of modulation by 5-HT2 antagonists.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Ergolines; Ketanserin; Male; Piperidines; Pyrrolidines; Receptors, Opioid, kappa; Saimiri; Serotonin Antagonists | 1993 |
Glutamatergic and non-glutamatergic responses evoked in neonatal rat lumbar motoneurons on stimulation of the lateroventral spinal cord surface.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Bicuculline; Citalopram; Cocaine; Desipramine; Electric Stimulation; Ergolines; Evoked Potentials; Excitatory Amino Acid Antagonists; In Vitro Techniques; Ketanserin; Membrane Potentials; Motor Neurons; Quinoxalines; Rats; Rats, Wistar; Receptors, Glutamate; Serotonin Antagonists; Spinal Cord; Strychnine; Synapses | 1993 |
The effect of 5-HT and selective 5-HT receptor agonists and antagonists on rat dorsal vagal preganglionic neurones in vitro.
Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Ergolines; Female; In Vitro Techniques; Indoles; Ketanserin; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium Channels; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Tropanes; Vagus Nerve | 1996 |
Mutations of transmembrane IV and V serines indicate that all tryptamines do not bind to the rat 5-HT2A receptor in the same manner.
Topics: Amino Acid Sequence; Amino Acid Substitution; Amphetamines; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Ergolines; Ketanserin; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Protein Structure, Secondary; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Recombinant Proteins; Serine; Serotonin; Serotonin Antagonists; Tryptamines | 1997 |
Chemically induced platelet lysis causes vasoconstriction by release of serotonin.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Aorta, Thoracic; Blood Platelets; Bridged Bicyclo Compounds, Heterocyclic; Endothelium, Vascular; Ergolines; Fatty Acids, Unsaturated; Hemostatics; Hydrazines; In Vitro Techniques; Ketanserin; L-Lactate Dehydrogenase; Male; Platelet Aggregation Inhibitors; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Thromboxane A2; Vasoconstriction; Vasoconstrictor Agents; Vitamin K | 1998 |
p-Chloroamphetamine, a serotonin-releasing drug, elicited in rats a hyperglycemia mediated by the 5-HT1A and 5-HT2B/2C receptors.
Topics: 4-Aminobenzoic Acid; Adrenal Medulla; Adrenalectomy; Aminopyridines; Animals; Blood Glucose; Dose-Response Relationship, Drug; Ergolines; Fenclonine; Hyperglycemia; Indoles; Ketanserin; Male; Methysergide; p-Chloroamphetamine; para-Aminobenzoates; Piperazines; Propranolol; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Ritanserin; Serotonin; Serotonin Agents; Serotonin Antagonists; Tropisetron | 1998 |
Effect of 5-HT2 receptor antagonists on a cranial nerve reflex in the rabbit: evidence for inverse agonism.
Topics: Animals; Cranial Nerves; Ergolines; Female; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Piperidines; Rabbits; Receptors, Serotonin; Reflex; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 1999 |
Activation of 5-HT2A/2C receptors within the nucleus accumbens increases local dopaminergic transmission.
Topics: Amphetamines; Animals; Dopamine; Ergolines; Ketanserin; Kinetics; Male; Microdialysis; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium Channel Blockers; Synaptic Transmission; Tetrodotoxin | 2000 |
Involvement of the 5-HT(2) receptor in hyperthermia induced by p-chloroamphetamine, a serotonin-releasing drug in mice.
Topics: Animals; Body Temperature Regulation; Dose-Response Relationship, Drug; Ergolines; Fever; Indoles; Ketanserin; Male; Mice; Motor Activity; p-Chloroamphetamine; Pyridines; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists | 2000 |
Effects of 5-HT(2) receptor antagonists on the anti-immobility effects of imipramine in the forced swimming test with mice.
Topics: Animals; Antidepressive Agents, Tricyclic; Dose-Response Relationship, Drug; Ergolines; Imipramine; Indoles; Ketanserin; Male; Mice; Motor Activity; Pyridines; Receptors, Serotonin; Serotonin Antagonists; Swimming | 2001 |
The fenfluramine metabolite (+)-norfenfluramine is vasoactive.
Topics: Animals; Aorta; Blood Pressure; Ergolines; Fenfluramine; In Vitro Techniques; Ketanserin; Male; Norfenfluramine; Prazosin; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Adrenergic, alpha; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Sympathectomy; Sympathetic Nervous System; Vasoconstriction | 2004 |