ketanserin and granisetron

ketanserin has been researched along with granisetron in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (52.17)18.2507
2000's8 (34.78)29.6817
2010's3 (13.04)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Dalvie, D; Loi, CM; Smith, DA1
Cassuto, J; Jodal, M; Lundgren, O; Sjöqvist, A1
Balestra, B; Candura, SM; Lucchelli, A; Messori, E; Rizzi, CA; Tonini, M1
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI1
Blackshaw, LA; Dent, J; Nisyrios, V1
Dias, JA; Farthing, MJ; Mourad, FH; O'Donnell, LJ; Ogutu, E1
Hansen, MB; Skadhauge, E1
Beubler, E; Hansen, MB; Skadhauge, E; Thørboll, JE1
Hansen, MB; Skadhauge, E; Thorbøll, JE1
Beubler, E; Gamse, R; Schirgi-Degen, A1
Grondahi, ML; Hansen, MB; Jensen, GM; Skadhauge, E1
Donnerer, J; Heinemann, A; Holzer, P; Pabst, MA; Wachter, CH1
Kaibara, M; Mameya, S; Takada, K; Takemura, K; Taniyama, K1
Naylor, RJ; Tuladhar, BR; Womack, MD1
Li, Y; Owyang, C; Zhu, JX; Zhu, XY1
Alloui, A; Bardin, L; Chassaing, C; Courade, JP; Eschalier, A1
Lograno, MD; Romano, MR1
Ge, L; Naylor, RJ; Tuladhar, BR1
Karaki, S; Kuwahara, A; Mitsui, R; Ono, S1
Fazzari, J; Mersov, A; Mothersill, C; Seymour, C; Smith, R1

Other Studies

23 other study(ies) available for ketanserin and granisetron

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Which metabolites circulate?
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:5

    Topics: Humans; Metabolic Clearance Rate; Pharmaceutical Preparations

2013
Actions of serotonin antagonists on cholera-toxin-induced intestinal fluid secretion.
    Acta physiologica Scandinavica, 1992, Volume: 145, Issue:3

    Topics: Animals; Body Fluids; Cholera Toxin; Female; Granisetron; Imidazoles; Indazoles; Intestinal Mucosa; Ketanserin; Lysergic Acid Diethylamide; Male; Methysergide; Ondansetron; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Zimeldine

1992
5-Hydroxytryptamine receptors that facilitate excitatory neuromuscular transmission in the guinea-pig isolated detrusor muscle.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Acetylcholine; Adenosine Triphosphate; Amphetamines; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Granisetron; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Synaptic Transmission; Urinary Bladder

1995
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach

1995
Responses of ferret lower esophageal sphincter to 5-hydroxytryptamine: pathways and receptor subtypes.
    The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 1

    Topics: Animals; Atropine; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Esophagus; Female; Ferrets; Granisetron; Guanethidine; Indoles; Ketanserin; Male; Muscle, Smooth; Receptors, Serotonin; Reference Values; Serotonin; Serotonin Antagonists; Splanchnic Nerves; Time Factors; Vagotomy; Vagus Nerve

1995
Role of 5-hydroxytryptamine in intestinal water and electrolyte movement during gut anaphylaxis.
    Gut, 1995, Volume: 36, Issue:4

    Topics: Anaphylaxis; Animals; Body Water; Electrolytes; Food Hypersensitivity; Granisetron; Immunoglobulin E; Intestinal Absorption; Intestines; Ketanserin; Male; Rats; Rats, Inbred Strains; Serotonin; Time Factors

1995
Ketanserin and granisetron reduce cholera toxin-induced hypersecretion in pig jejunum.
    Scandinavian journal of gastroenterology, 1994, Volume: 29, Issue:10

    Topics: Animals; Animals, Newborn; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cholera Toxin; Diarrhea; Dose-Response Relationship, Drug; Drug Therapy, Combination; Granisetron; Indoles; Intestinal Secretions; Jejunum; Ketanserin; Methysergide; Serotonin Antagonists; Swine; Tropisetron

1994
Effect of indomethacin, renzapride, methysergide, ketanserin, granisetron and citalopram on serotonin-induced fluid accumulation in pig jejunum.
    Physiological research, 1994, Volume: 43, Issue:2

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Citalopram; Dose-Response Relationship, Drug; Granisetron; Indomethacin; Intestinal Absorption; Jejunum; Ketanserin; Methysergide; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Swine

1994
5-Hydroxytryptamine2 and 5-hydroxytryptamine3 receptors mediate serotonin-induced short-circuit current in pig jejunum.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 1994, Volume: 164, Issue:5

    Topics: Animals; Benzamides; Electrophysiology; Female; Granisetron; Jejunum; Ketanserin; Receptors, Serotonin; Serotonin; Swine

1994
Inhibition of 5-hydroxytryptamine- and enterotoxin-induced fluid secretion by 5-HT receptor antagonists in the rat jejunum.
    European journal of pharmacology, 1993, Aug-02, Volume: 248, Issue:2

    Topics: Animals; Bacterial Toxins; Body Fluids; Cholera Toxin; Enterotoxins; Escherichia coli; Escherichia coli Proteins; Female; Granisetron; Indoles; Jejunum; Ketanserin; Ondansetron; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron

1993
Effect of 5-HT2 and 5-HT3 receptor antagonists on cholera toxin-induced fluid hypersecretion in the pig jejunum.
    Zentralblatt fur Veterinarmedizin. Reihe A, 1996, Volume: 43, Issue:9

    Topics: Analysis of Variance; Animals; Cholera Toxin; Dose-Response Relationship, Drug; Granisetron; Indoles; Jejunal Diseases; Jejunum; Ketanserin; Ondansetron; Serotonin Antagonists; Swine; Swine Diseases; Tropisetron

1996
Mediation by 5_hydroxytryptamine of the femoral vasoconstriction induced by acid challenge of the rat gastric mucosa.
    The Journal of physiology, 1998, Jun-01, Volume: 509 ( Pt 2)

    Topics: Animals; Ethanol; Female; Femoral Artery; Gastric Acid; Gastric Mucosa; Granisetron; Hydrochloric Acid; Ketanserin; Methiothepin; Muscle, Smooth, Vascular; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Taurocholic Acid; Vasoconstriction

1998
Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach.
    Japanese journal of pharmacology, 1999, Volume: 79, Issue:1

    Topics: Animals; Atropine; Dioxanes; Enzyme Inhibitors; Female; Gastric Fundus; Granisetron; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscarinic Antagonists; Muscle Relaxation; Muscle Tonus; Nitroarginine; Piperidines; Pyloric Antrum; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Tetrodotoxin

1999
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
Intestinal serotonin acts as a paracrine substance to mediate vagal signal transmission evoked by luminal factors in the rat.
    The Journal of physiology, 2001, Feb-01, Volume: 530, Issue:Pt 3

    Topics: Action Potentials; Afferent Pathways; Anesthetics, Local; Animals; Brain Stem; Cholecystokinin; Duodenum; Granisetron; Intestinal Mucosa; Intestines; Ketanserin; Lidocaine; Male; Muscle, Smooth; Nerve Fibers; Neurons, Afferent; Nodose Ganglion; Rats; Rats, Sprague-Dawley; Serotonin; Vagotomy; Vagus Nerve

2001
5-HT receptor subtypes involved in the spinal antinociceptive effect of acetaminophen in rats.
    European journal of pharmacology, 2001, Nov-30, Volume: 432, Issue:1

    Topics: Acetaminophen; Analgesics; Animals; Ergolines; Granisetron; Injections, Spinal; Ketanserin; Male; Pain Threshold; Penbutolol; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Time Factors; Vocalization, Animal

2001
Pharmacological characterization of the 5-HT1A, 5-HT2 and 5-HT3 receptors in the bovine ciliary muscle.
    European journal of pharmacology, 2003, Mar-07, Volume: 464, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Cattle; Cell Membrane; Ciliary Body; Dose-Response Relationship, Drug; Granisetron; In Vitro Techniques; Ketanserin; Muscle Contraction; Muscle, Smooth; Ondansetron; Radioligand Assay; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium

2003
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides

2003
Propionate modulates spontaneous contractions via enteric nerves and prostaglandin release in the rat distal colon.
    The Japanese journal of physiology, 2005, Volume: 55, Issue:6

    Topics: Acetates; Animals; Atropine; Cholinergic Fibers; Colon, Descending; Cyclooxygenase Inhibitors; Enteric Nervous System; Gastrointestinal Motility; Granisetron; Hexamethonium; Ketanserin; Male; Motor Neurons; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nicotinic Antagonists; Piroxicam; Propionates; Prostaglandins; Rats; Rats, Wistar; Serotonin Antagonists; Tetrodotoxin

2005
Effect of 5-hydroxytryptamine (serotonin) receptor inhibitors on the radiation-induced bystander effect.
    International journal of radiation biology, 2012, Volume: 88, Issue:10

    Topics: Bystander Effect; Calcium; Cell Line; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Granisetron; Humans; Intracellular Space; Ketanserin; Receptors, Serotonin; Serotonin Antagonists

2012