ketanserin and fenfluramine

ketanserin has been researched along with fenfluramine in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19904 (20.00)18.7374
1990's6 (30.00)18.2507
2000's9 (45.00)29.6817
2010's1 (5.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA1
Liebelt, HJ; Menadue, MF; Willoughby, JO1
Hewson, G; Hill, RG; Hughes, J; Leighton, GE1
Glennon, RA; McKenney, JD; Young, R1
Barbieri, C; Bevilacqua, M; Bigatti, G; Diena, A; Guffanti, A; Norbiato, G; Rauhe, WG; Sala, M; Scorza, D1
Goshadrou, F; Pourgholami, MH1
Day, J; Fibiger, HC; Hirano, H1
Grignaschi, G; Samanin, R; Sironi, F1
Delcroix, M; Leeman, M; Maggiorini, M; Naeije, R; Wauthy, P1
Holtzman, SG; Steinfels, GF1
Deis, RP; Hole, D; Jahn, GA; Kalia, V; Wilson, CA1
Cryan, JF; Harkin, A; Kelly, JP; Leonard, BE; Naughton, M1
Piguet, P; Schlichter, R; Stoeckel, ME1
Barrett, RJ; Gresch, PJ; Sanders-Bush, E; Smith, RL1
Cunningham, KA; Filip, M; McCreary, AC1
Grasby, P; Hirani, E; Hume, S; Sharp, T; Sprakes, M1
Fink, GD; Li, MW; Ni, W; Thakali, K; Watts, SW1
Bosker, FJ; Cremers, TI; den Boer, JA; Postema, F; Tiemersma-Wegman, TD; Udo de Haes, JI1
Wee, S; Woolverton, WL1
Arai, Y; Mitazaki, S; Murata, A; Nakagawasai, O; Niijima, F; Ohba, A; Tadano, T; Tan-No, K; Wakui, K1

Other Studies

20 other study(ies) available for ketanserin and fenfluramine

ArticleYear
The 2014 Philip S. Portoghese Medicinal Chemistry Lectureship: The "Phenylalkylaminome" with a Focus on Selected Drugs of Abuse.
    Journal of medicinal chemistry, 2017, 04-13, Volume: 60, Issue:7

    Topics: Animals; Central Nervous System Stimulants; Chemistry, Pharmaceutical; Dopamine; Drug Discovery; Hallucinogens; Humans; Illicit Drugs; Norepinephrine; Phenethylamines; Psychotropic Drugs; Receptors, Serotonin; Serotonin

2017
Activation of 5-HT 1 serotonin receptors in the medial basal hypothalamus stimulates prolactin secretion in the unanaesthetized rat.
    Neuroendocrinology, 1988, Volume: 47, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Fenfluramine; Hypothalamus, Middle; Ketanserin; Male; Metergoline; Prolactin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin

1988
Ketanserin antagonises the anorectic effect of DL-fenfluramine in the rat.
    European journal of pharmacology, 1988, Jan-12, Volume: 145, Issue:2

    Topics: Animals; Anorexia; Fenfluramine; Ketanserin; Male; Prazosin; Rats; Receptors, Adrenergic; Receptors, Serotonin

1988
Discriminative stimulus properties of the serotonin agonist 1-(3-trifluoromethylphenyl)piperazine (TFMPP).
    Life sciences, 1984, Oct-01, Volume: 35, Issue:14

    Topics: Animals; Discrimination Learning; DOM 2,5-Dimethoxy-4-Methylamphetamine; Extinction, Psychological; Fenfluramine; Indoles; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Serotonin

1984
Serotonergic regulation of cortisol secretion in dogs.
    Endocrinology, 1984, Volume: 115, Issue:2

    Topics: Animals; Dogs; Fenfluramine; Hydrocortisone; Ketanserin; Piperidines; Quipazine; Serotonin; Time Factors

1984
Evidence for serotonergic system involvement in the effect of morphine on gastrointestinal motility in the rat.
    General pharmacology, 1995, Volume: 26, Issue:4

    Topics: 5,7-Dihydroxytryptamine; Animals; Central Nervous System; Charcoal; Depression, Chemical; Dose-Response Relationship, Drug; Fenclonine; Fenfluramine; Gastrointestinal Motility; Ketanserin; Male; Morphine; Naloxone; Rats; Serotonin

1995
Serotonergic regulation of acetylcholine release in rat frontal cortex.
    Journal of neurochemistry, 1995, Volume: 65, Issue:3

    Topics: Acetylcholine; Animals; Benzazepines; Dialysis; Fenfluramine; Fluoxetine; Frontal Lobe; Ketanserin; Kinetics; Male; Rats; Rats, Wistar; Serotonin

1995
The 5-HT1B receptor mediates the effect of d-fenfluramine on eating caused by intra-hypothalamic injection of neuropeptide Y.
    European journal of pharmacology, 1995, Feb-14, Volume: 274, Issue:1-3

    Topics: Analysis of Variance; Animals; Antiparkinson Agents; Drug Interactions; Eating; Ergolines; Fenfluramine; Hyperphagia; Hypothalamus; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Male; Metergoline; Neuropeptide Y; Paraventricular Hypothalamic Nucleus; Pindolol; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists

1995
Effects of dexfenfluramine on hypoxic pulmonary vasoconstriction and embolic pulmonary hypertension in dogs.
    American journal of respiratory and critical care medicine, 1995, Volume: 151, Issue:3 Pt 1

    Topics: Animals; Dogs; Fenfluramine; Hypertension, Pulmonary; Hypoxia; Ketanserin; Pulmonary Artery; Pulmonary Embolism; Pulmonary Wedge Pressure; Receptors, Serotonin; Vasoconstriction

1995
Monoamine systems in the discriminative effects of spiradoline, a kappa-opioid agonist.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Analgesics; Animals; Avoidance Learning; Biogenic Monoamines; Discrimination, Psychological; Dopamine Antagonists; Fenfluramine; Fluoxetine; Generalization, Stimulus; Ketanserin; Male; Piperidines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Selective Serotonin Reuptake Inhibitors; Serotonin; Synaptic Transmission

1994
Receptors and neurotransmitters involved in the dual modulation of prolactin release by the serotoninergic system in pregnant and lactating rats.
    Journal of reproduction and fertility, 1999, Volume: 116, Issue:2

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amphetamines; Analysis of Variance; Animals; Brain Chemistry; Dopamine; Female; Fenclonine; Fenfluramine; Gestational Age; Ketanserin; Metoprolol; Norepinephrine; p-Chloroamphetamine; Prazosin; Pregnancy; Pregnancy, Animal; Prolactin; Rats; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction

1999
Characterization of D-fenfluramine-induced hypothermia: evidence for multiple sites of action.
    European journal of pharmacology, 2000, Mar-03, Volume: 390, Issue:3

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Benzofurans; Body Temperature; Cerebral Cortex; Dopamine Antagonists; Dose-Response Relationship, Drug; Fenclonine; Fenfluramine; Haloperidol; Hydroxyindoleacetic Acid; Hypothalamus; Hypothermia; Ketanserin; Male; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Sertraline; Sulpiride; Yohimbine

2000
Synaptically released 5-HT modulates the activity of tonically discharging neuronal populations in the rostral ventral medulla (RVM).
    The European journal of neuroscience, 2000, Volume: 12, Issue:8

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Bicuculline; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fenfluramine; GABA Antagonists; Glycine Agents; Ketanserin; Medulla Oblongata; Neural Inhibition; Neurons; Organ Culture Techniques; Piperazines; Prazosin; Propranolol; Rats; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Strychnine; Synaptic Transmission

2000
Stimulus generalization by fenfluramine in a quipazine-ketanserin drug discrimination is not dependent on indirect serotonin release.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 72, Issue:1-2

    Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Fenfluramine; Ketanserin; Male; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin

2002
Discriminative stimulus properties of (+/-)-fenfluramine: the role of 5-HT2 receptor subtypes.
    Behavioral neuroscience, 2003, Volume: 117, Issue:2

    Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Fenfluramine; Fluorobenzenes; Indoles; Ketanserin; Male; Piperidines; Pyrazines; Pyridines; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Thiophenes

2003
Fenfluramine evokes 5-HT2A receptor-mediated responses but does not displace [11C]MDL 100907: small animal PET and gene expression studies.
    Synapse (New York, N.Y.), 2003, Dec-01, Volume: 50, Issue:3

    Topics: Animals; Carbon Radioisotopes; Cerebellum; Fenfluramine; Fluorobenzenes; Gene Expression; Genes, Immediate-Early; In Situ Hybridization; Ketanserin; Male; Neurons; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Time Factors; Tomography, Emission-Computed

2003
The fenfluramine metabolite (+)-norfenfluramine is vasoactive.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 309, Issue:2

    Topics: Animals; Aorta; Blood Pressure; Ergolines; Fenfluramine; In Vitro Techniques; Ketanserin; Male; Norfenfluramine; Prazosin; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Adrenergic, alpha; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Sympathectomy; Sympathetic Nervous System; Vasoconstriction

2004
Effect of increased serotonin levels on [18F]MPPF binding in rat brain: fenfluramine vs the combination of citalopram and ketanserin.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:9

    Topics: Animals; Autoradiography; Behavior, Animal; Brain; Brain Chemistry; Citalopram; Drug Combinations; Drug Interactions; Fenfluramine; Ketanserin; Male; Microdialysis; Movement; Piperazines; Posture; Protein Binding; Pyridines; Rats; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Time Factors

2005
Self-administration of mixtures of fenfluramine and amphetamine by rhesus monkeys.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 84, Issue:2

    Topics: Animals; Dextroamphetamine; Fenfluramine; Ketanserin; Macaca mulatta; Male; Receptors, Serotonin, 5-HT2; Self Administration

2006
Enhanced head-twitch response to 5-HT-related agonists in thiamine-deficient mice.
    Journal of neural transmission (Vienna, Austria : 1996), 2007, Volume: 114, Issue:8

    Topics: Amphetamines; Animals; Brain; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Tolerance; Fenfluramine; Head Movements; Ketanserin; Korsakoff Syndrome; Male; Mice; Movement Disorders; Raphe Nuclei; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Thiamine; Thiamine Deficiency; Tryptophan Hydroxylase

2007