ketanserin and colforsin

ketanserin has been researched along with colforsin in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (37.50)18.2507
2000's4 (50.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Bansse, MT; Stam, NJ; van Huizen, F1
Colpaert, FC; Pauwels, PJ1
Chapman, K; Diorio, J; Francis, D; Meaney, MJ; Seckl, JR; Weaver, S; Yau, J1
Carson, MJ; Hu, JL; Matli, JR; Sutcliffe, JG; Thomas, EA1
Cutz, E; Farragher, SM; Fu, XW; Pan, J; Wang, D; Wong, V1
Saifullah, AS; Tomioka, K1

Reviews

1 review(s) available for ketanserin and colforsin

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993

Other Studies

7 other study(ies) available for ketanserin and colforsin

ArticleYear
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Agonist-induced down-regulation of human 5-HT1A and 5-HT2 receptors in Swiss 3T3 cells.
    Neuroreport, 1993, Sep-30, Volume: 4, Issue:12

    Topics: 3T3 Cells; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Colforsin; Cyclic AMP; Down-Regulation; Humans; Hydrolysis; Ketanserin; Kinetics; Mice; Mice, Inbred Strains; Pertussis Toxin; Phosphatidylinositols; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Virulence Factors, Bordetella

1993
Selective antagonism of human 5-HT1D and 5-HT1B receptor-mediated responses in stably transfected C6-glial cells by ketanserin and GR 127,935.
    European journal of pharmacology, 1996, Apr-04, Volume: 300, Issue:1-2

    Topics: Animals; Cell Line; Colforsin; Cyclic AMP; Drug Interactions; Humans; Ketanserin; Neuroglia; Oxadiazoles; Piperazines; Rats; Serotonin Antagonists; Transfection

1996
Postnatal handling increases the expression of cAMP-inducible transcription factors in the rat hippocampus: the effects of thyroid hormones and serotonin.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, May-15, Volume: 20, Issue:10

    Topics: Adenylyl Cyclases; Animals; Antithyroid Agents; Blotting, Western; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; DNA-Binding Proteins; Early Growth Response Protein 1; Gene Expression Regulation, Enzymologic; Handling, Psychological; Hippocampus; Immediate-Early Proteins; Ketanserin; Male; Neuronal Plasticity; Neurons; Phosphorylation; Propylthiouracil; Rats; Rats, Long-Evans; RNA, Messenger; Serotonin; Serotonin Antagonists; Thyroid Hormones; Transcription Factor AP-2; Transcription Factors; Tritium

2000
Pertussis toxin treatment prevents 5-HT(5a) receptor-mediated inhibition of cyclic AMP accumulation in rat C6 glioma cells.
    Journal of neuroscience research, 2000, Jul-01, Volume: 61, Issue:1

    Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Gene Expression; Glioma; GTP-Binding Protein alpha Subunits, Gi-Go; Ketanserin; Neurons; Pertussis Toxin; Protein Structure, Tertiary; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella

2000
Neuroepithelial bodies in mammalian lung express functional serotonin type 3 receptor.
    American journal of physiology. Lung cellular and molecular physiology, 2001, Volume: 281, Issue:4

    Topics: Aminopyridines; Animals; Calcium; Chemoreceptor Cells; Colforsin; Cricetinae; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Situ Hybridization; Indoles; Ion Channel Gating; Ketanserin; Lung; Mammals; Membrane Potentials; Mesocricetus; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Piperazines; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Respiratory Mucosa; RNA, Messenger; Serotonin; Serotonin Antagonists; Tropisetron

2001
5-HT(7)-like receptors mediate serotonergic modulation of photo-responsiveness of the medulla bilateral neurons in the cricket, Gryllus bimaculatus.
    Zoological science, 2003, Volume: 20, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Clozapine; Colforsin; Dose-Response Relationship, Drug; Electrophysiology; Gryllidae; Ketanserin; Light; Neurons; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Visual Pathways

2003