ketanserin has been researched along with colforsin in 8 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (37.50) | 18.2507 |
2000's | 4 (50.00) | 29.6817 |
2010's | 1 (12.50) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM | 1 |
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
Bansse, MT; Stam, NJ; van Huizen, F | 1 |
Colpaert, FC; Pauwels, PJ | 1 |
Chapman, K; Diorio, J; Francis, D; Meaney, MJ; Seckl, JR; Weaver, S; Yau, J | 1 |
Carson, MJ; Hu, JL; Matli, JR; Sutcliffe, JG; Thomas, EA | 1 |
Cutz, E; Farragher, SM; Fu, XW; Pan, J; Wang, D; Wong, V | 1 |
Saifullah, AS; Tomioka, K | 1 |
1 review(s) available for ketanserin and colforsin
Article | Year |
---|---|
The role of receptor binding in drug discovery.
Topics: Animals; Drug Design; Humans; Receptors, Drug | 1993 |
7 other study(ies) available for ketanserin and colforsin
Article | Year |
---|---|
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
Agonist-induced down-regulation of human 5-HT1A and 5-HT2 receptors in Swiss 3T3 cells.
Topics: 3T3 Cells; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Colforsin; Cyclic AMP; Down-Regulation; Humans; Hydrolysis; Ketanserin; Kinetics; Mice; Mice, Inbred Strains; Pertussis Toxin; Phosphatidylinositols; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Virulence Factors, Bordetella | 1993 |
Selective antagonism of human 5-HT1D and 5-HT1B receptor-mediated responses in stably transfected C6-glial cells by ketanserin and GR 127,935.
Topics: Animals; Cell Line; Colforsin; Cyclic AMP; Drug Interactions; Humans; Ketanserin; Neuroglia; Oxadiazoles; Piperazines; Rats; Serotonin Antagonists; Transfection | 1996 |
Postnatal handling increases the expression of cAMP-inducible transcription factors in the rat hippocampus: the effects of thyroid hormones and serotonin.
Topics: Adenylyl Cyclases; Animals; Antithyroid Agents; Blotting, Western; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; DNA-Binding Proteins; Early Growth Response Protein 1; Gene Expression Regulation, Enzymologic; Handling, Psychological; Hippocampus; Immediate-Early Proteins; Ketanserin; Male; Neuronal Plasticity; Neurons; Phosphorylation; Propylthiouracil; Rats; Rats, Long-Evans; RNA, Messenger; Serotonin; Serotonin Antagonists; Thyroid Hormones; Transcription Factor AP-2; Transcription Factors; Tritium | 2000 |
Pertussis toxin treatment prevents 5-HT(5a) receptor-mediated inhibition of cyclic AMP accumulation in rat C6 glioma cells.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Gene Expression; Glioma; GTP-Binding Protein alpha Subunits, Gi-Go; Ketanserin; Neurons; Pertussis Toxin; Protein Structure, Tertiary; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella | 2000 |
Neuroepithelial bodies in mammalian lung express functional serotonin type 3 receptor.
Topics: Aminopyridines; Animals; Calcium; Chemoreceptor Cells; Colforsin; Cricetinae; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Situ Hybridization; Indoles; Ion Channel Gating; Ketanserin; Lung; Mammals; Membrane Potentials; Mesocricetus; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Piperazines; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Respiratory Mucosa; RNA, Messenger; Serotonin; Serotonin Antagonists; Tropisetron | 2001 |
5-HT(7)-like receptors mediate serotonergic modulation of photo-responsiveness of the medulla bilateral neurons in the cricket, Gryllus bimaculatus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Clozapine; Colforsin; Dose-Response Relationship, Drug; Electrophysiology; Gryllidae; Ketanserin; Light; Neurons; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Visual Pathways | 2003 |