ketanserin and clonidine

ketanserin has been researched along with clonidine in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-199016 (50.00)18.7374
1990's10 (31.25)18.2507
2000's3 (9.38)29.6817
2010's2 (6.25)24.3611
2020's1 (3.13)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Chen, Y; Feng, F; He, S; Li, Q; Liao, Q; Liu, W; Liu, Y; Lu, W; Sun, H; Xing, S; Xiong, B; Yang, H1
Celuch, SM; Enero, MA; Ramirez, AJ1
Hansson, E; Nilsson, M; Rönnbäck, L1
Mustafa, AA1
Kinami, J; Maruyama, K; Nagatomo, T; Sugita, Y; Sugiyama, E; Takada, Y; Tsuchihashi, H1
Bortone, F; Ceriani, R; Moruzzi, P; Ruju, P; Salvi, L; Solinas, C; Susini, G1
Alling, C; Hansson, E; Simonsson, P1
Coffman, JD; Cohen, RA1
Brunello, N; Galimberti, R; Racagni, G; Riva, M; Rovescalli, AC1
Nagatomo, T; Tsuchihashi, H1
Gallager, D; Goldman-Rakic, PS; Rakic, P1
Baldwin, JJ; Clineschmidt, BV; Huff, JR; Lotti, VJ; Pettibone, DJ; Randall, WC; Vacca, J; Young, SD1
Hong, M; Jenner, P; Marsden, CD; Roots, EJ1
Kawasaki, H; Takasaki, K1
Cheng, JT; Lee, JM; Lin, MT1
Doğan, N; Ilhan, M; Kayaalp, SO; Tuncer, M1
Harris, LT; McCall, RB1
Matsumoto, M; Minami, M; Saito, H; Togashi, H; Yoshioka, M1
Beubler, E; Bukhave, K; Rask-Madsen, J1
Timmermans, PB; Van Brummelen, P; Van Zwieten, PA1
Opie, LH1
McCall, RB; Schuette, MR1
Genkova-Papazova, M; Lazarova-Bakarova, M; Petkov, VD1
Lidow, MS; Rakic, P1
Banache, M; Bonnet, F; Joris, J; Lamy, M; Sessler, DI1
Matsumoto, K; Mizowaki, M; Murakami, Y; Thongpraditchote, S; Watanabe, H1
Eberhart, LH; Kranke, P; Roewer, N; Tramèr, MR1

Reviews

2 review(s) available for ketanserin and clonidine

ArticleYear
Role of alpha adrenoceptors in hypertension and in antihypertensive drug treatment.
    The American journal of medicine, 1984, Oct-05, Volume: 77, Issue:4A

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Calcium Channel Blockers; Clonidine; Guanfacine; Guanidines; Humans; Hypertension; Ketanserin; Methyldopa; Muscle, Smooth, Vascular; Phenylacetates; Piperazines; Piperidines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Vascular Resistance

1984
Pharmacological treatment of postoperative shivering: a quantitative systematic review of randomized controlled trials.
    Anesthesia and analgesia, 2002, Volume: 94, Issue:2

    Topics: Adrenergic alpha-Agonists; Analgesics, Opioid; Clonidine; Humans; Ketanserin; Lidocaine; Meperidine; Postoperative Complications; Randomized Controlled Trials as Topic; Shivering

2002

Trials

1 trial(s) available for ketanserin and clonidine

ArticleYear
Clonidine and ketanserin both are effective treatment for postanesthetic shivering.
    Anesthesiology, 1993, Volume: 79, Issue:3

    Topics: Adult; Anesthesia Recovery Period; Anesthesia, General; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Humans; Ketanserin; Male; Middle Aged; Shivering; Surgical Procedures, Operative

1993

Other Studies

29 other study(ies) available for ketanserin and clonidine

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Discovery and Biological Evaluation of a Novel Highly Potent Selective Butyrylcholinsterase Inhibitor.
    Journal of medicinal chemistry, 2020, 09-10, Volume: 63, Issue:17

    Topics: Aminoquinolines; Animals; Benzimidazoles; Butyrylcholinesterase; Cell Line, Tumor; Cholinesterase Inhibitors; Drug Discovery; Drug Evaluation, Preclinical; Female; Humans; Male; Mice, Inbred ICR; Microsomes, Liver; Molecular Docking Simulation; Molecular Dynamics Simulation; Neuroprotective Agents; Protein Binding; Small Molecule Libraries

2020
Activation of 5-HT2 receptors inhibits the evoked release of [3H]noradrenaline in the rat spinal cord.
    General pharmacology, 1992, Volume: 23, Issue:6

    Topics: Amphetamines; Animals; Clonidine; Electric Stimulation; Female; Hallucinogens; In Vitro Techniques; Ketanserin; Norepinephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Serotonin Receptor Agonists; Spinal Cord; Yohimbine

1992
Receptor-coupled uptake of valproate in rat astroglial primary cultures.
    Neuroscience letters, 1992, Feb-17, Volume: 136, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Astrocytes; Biological Transport; Cells, Cultured; Cerebral Cortex; Clonidine; Drug Interactions; Glutamates; Glutamic Acid; Isoproterenol; Kainic Acid; Ketanserin; Phenylephrine; Prazosin; Quinoxalines; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Serotonin; Valproic Acid; Yohimbine

1992
Rapid desensitization of central beta-adrenoceptors in rat after subacute treatment with imipramine and calcium entry blockers.
    Neuropharmacology, 1991, Volume: 30, Issue:8

    Topics: 1-Propanol; Animals; Calcium Channel Blockers; Clonidine; Diltiazem; DOM 2,5-Dimethoxy-4-Methylamphetamine; Drinking Behavior; Fenclonine; Imipramine; Isoproterenol; Ketanserin; Nicardipine; Nifedipine; Oxidopamine; Rats; Receptors, Adrenergic, beta; Verapamil

1991
MCI-9042: high affinity for serotonergic receptors as assessed by radioligand binding assay.
    Journal of pharmacobio-dynamics, 1991, Volume: 14, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Brain Chemistry; Clonidine; Hippocampus; In Vitro Techniques; Ketanserin; Kinetics; Platelet Aggregation Inhibitors; Prazosin; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Muscarinic; Receptors, Serotonin; Succinates

1991
[Effectiveness and hemodynamic effects of clonidine, meperidine, taurine, ketanserin in the therapy of post-anesthesia shivering in patients undergoing ECC in moderate hypothermia].
    Minerva anestesiologica, 1991, Volume: 57, Issue:9

    Topics: Anesthesia Recovery Period; Clonidine; Extracorporeal Circulation; Hemodynamics; Humans; Hypothermia, Induced; Ketanserin; Meperidine; Prospective Studies; Shivering; Taurine

1991
Interactions between cyclic AMP and inositol phosphate transduction systems in astrocytes in primary culture.
    Neuropharmacology, 1990, Volume: 29, Issue:6

    Topics: Adenylyl Cyclases; Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Clonidine; Cyclic AMP; Inositol Phosphates; Isoproterenol; Ketanserin; Norepinephrine; Phenylephrine; Rats; Rats, Inbred Strains; Serotonin; Signal Transduction

1990
Alpha-adrenergic and serotonergic mechanisms in the human digit.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: Adult; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Fingers; Humans; Ketanserin; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Reflex; Regional Blood Flow; Serotonin; Sympathetic Nervous System; Vascular Resistance; Vasoconstriction; Yohimbine

1988
Age-related changes in rat serotonergic and adrenergic systems and in receptor responsiveness to subchronic desipramine treatment.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:3

    Topics: Aging; Animals; Brain; Clonidine; Desipramine; Dihydroalprenolol; Hydroxyindoleacetic Acid; Imipramine; Ketanserin; Kinetics; Male; Paroxetine; Piperidines; Prazosin; Proteins; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Serotonin; Serotonin; Time Factors

1988
Alpha-blocking potencies of antihypertensive agents (prazosin, terazosin, bunazosin, SGB-1534 and ketanserin) having with quinazoline or quinazolinedione as assessed by radioligand binding assay methods in rat brain.
    Journal of pharmacobio-dynamics, 1989, Volume: 12, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Brain; Cell Membrane; Clonidine; Dihydroalprenolol; Ketanserin; Male; Prazosin; Quinazolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1989
Quantitative autoradiography of major neurotransmitter receptors in the monkey striate and extrastriate cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1988, Volume: 8, Issue:10

    Topics: Animals; Autoradiography; Cerebral Cortex; Clonidine; Female; Flunitrazepam; Ketanserin; Macaca mulatta; Male; Muscimol; Pindolol; Prazosin; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Neurotransmitter; Serotonin; Spiperone; Visual Cortex

1988
Pharmacological profile of a new potent and specific alpha 2-adrenoceptor antagonist, L-657,743.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 336, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Binding, Competitive; Blood Platelets; Cattle; Cerebral Cortex; Clonidine; Humans; In Vitro Techniques; Ketanserin; Male; Prazosin; Quinolizines; Radioligand Assay; Rats; Rats, Inbred Strains; Serotonin; Spiperone; Vas Deferens

1987
The effect of long-term treatment with amine-depleting drugs or chlorpromazine on alpha-adrenoreceptors and 5-HT2 receptors in the brain of the rat.
    Neuropharmacology, 1988, Volume: 27, Issue:5

    Topics: Animals; Binding, Competitive; Biogenic Amines; Brain; Chlorpromazine; Clonidine; In Vitro Techniques; Ketanserin; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Reserpine; Tetrabenazine

1988
Central alpha-2 adrenoceptor-mediated hypertensive response to clonidine in conscious, normotensive rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:3

    Topics: Animals; Azepines; Blood Pressure; Brain; Cimetidine; Clonidine; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Male; Methoxamine; Oxidopamine; Piperidines; Prazosin; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1986
Changes in central serotoninergic transmission affect clonidine analgesia in monkeys.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:5

    Topics: 5-Hydroxytryptophan; 5,7-Dihydroxytryptamine; Analgesics; Animals; Clonidine; Fenclonine; Injections, Intraventricular; Ketanserin; Macaca; Male; Microinjections; Nociceptors; Periaqueductal Gray; Raphe Nuclei; Serotonin; Synaptic Transmission

1987
Serotonin-induced contraction of canine saphenous vein: mediation by 5-HT1 receptors.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 274, Issue:2

    Topics: Animals; Clonidine; Dogs; Drug Interactions; Emetics; In Vitro Techniques; Ketanserin; Mianserin; Muscle Contraction; Naphthols; Piperidines; Receptors, Serotonin; Saphenous Vein; Serotonin; Yohimbine

1985
Characterization of the central sympathoinhibitory action of ketanserin.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: Animals; Blood Pressure; Cats; Clonidine; Electrophysiology; Ergolines; Heart Rate; Ketanserin; Prazosin; Sympathetic Nervous System

1987
Central sympathoinhibitory action of ketanserin in rats.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:3

    Topics: Animals; Blood Pressure; Brain; Clonidine; Dose-Response Relationship, Drug; Heart; Heart Rate; Ketanserin; Kidney; Male; Pressoreceptors; Rats; Rats, Inbred Strains; Sympathetic Nervous System

1987
Colonic secretion mediated by prostaglandin E2 and 5-hydroxytryptamine may contribute to diarrhea due to morphine withdrawal in the rat.
    Gastroenterology, 1984, Volume: 87, Issue:5

    Topics: Animals; Atropine; Clonidine; Colon; Cyclic AMP; Diarrhea; Dinoprostone; Female; Humans; Indomethacin; Ketanserin; Morphine Dependence; Naloxone; Piperidines; Prostaglandins E; Rats; Rats, Inbred Strains; Serotonin; Substance Withdrawal Syndrome

1984
Principles of therapy for congestive heart failure.
    European heart journal, 1983, Volume: 4 Suppl A

    Topics: Calcium; Calcium Channel Blockers; Calmodulin; Cardiotonic Agents; Clonidine; Cyclic AMP; Cytosol; Digitalis Glycosides; Diuretics; Heart Failure; Humans; Ketanserin; Models, Cardiovascular; Muscle, Smooth, Vascular; Myocardium; Myosins; Piperidines; Receptors, Adrenergic, alpha; Vasodilator Agents

1983
Evidence for an alpha-1 receptor-mediated central sympathoinhibitory action of ketanserin.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 228, Issue:3

    Topics: Animals; Blood Pressure; Brain; Cats; Clonidine; Heart Rate; Ketanserin; Piperidines; Receptors, Adrenergic, alpha; Serotonin Antagonists; Sympathetic Nervous System; Sympatholytics

1984
The 5-HT2 receptor antagonist ketanserine prevents electroconvulsive shock- and clonidine-induced amnesia.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:4

    Topics: Amnesia; Animals; Avoidance Learning; Clonidine; Electroshock; Injections, Intraperitoneal; Ketanserin; Male; Rats; Rats, Wistar; Seizures; Serotonin Antagonists

1994
Distribution and density of monoamine receptors in the primate visual cortex devoid of retinal input from early embryonic stages.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:3 Pt 2

    Topics: Animals; Anophthalmos; Benzazepines; Clonidine; Eye Enucleation; Gene Expression Regulation, Developmental; Gestational Age; Ketanserin; Macaca mulatta; Pindolol; Prazosin; Radioligand Assay; Receptors, Adrenergic; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Spiperone; Visual Cortex; Visual Pathways

1995
alpha2-Adrenoceptor antagonists reverse the 5-HT2 receptor antagonist suppression of head-twitch behavior in mice.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 56, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Drug Evaluation, Preclinical; Fenclonine; Head Movements; Ketanserin; Male; Mice; Mice, Inbred Strains; Norepinephrine; Oxidopamine; Ritanserin; Serotonin; Serotonin Antagonists

1997