ketanserin and cinanserin

ketanserin has been researched along with cinanserin in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-199010 (58.82)18.7374
1990's4 (23.53)18.2507
2000's3 (17.65)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA; Herrick-Davis, K; Lyon, RA; Seggel, MR; Soine, WH; Titeler, M1
Glennon, RA1
Baldessarini, RJ; Booth, RG; Charifson, PS; Kula, NS; McPhail, AT; Myers, AM; Owens, CE; Wyrick, SD1
Neuman, RS; Zebrowska, G1
Koss, MC1
Ramage, AG1
Closse, A; Davies, H; Hoyer, D; Palacios, JM; Pazos, A; Vos, P1
Barrett, JE; Brady, LS1
Pranzatelli, MR; Snodgrass, SR1
Geyer, MA; Tapson, GS1
Hole, DR; Hunter, AJ; Wilson, CA1
Frost, JJ; Hartig, PR; Scheffel, U; Wagner, HN1
Battaglia, G; Borgundvaag, B; Shannon, M; Titeler, M1
Antonaccio, MJ; Dzwonczyk, S; Grover, GJ; Normandin, DE; Sargent, CA1
DiNardo, LA; Ehlen, JC; Glass, JD1
Pulido, M; Wilson, C1
Gebhard, MM; Martin, E; Peter, C; Schmidt, H; Secchi, A; Walther, A1

Reviews

1 review(s) available for ketanserin and cinanserin

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987

Other Studies

16 other study(ies) available for ketanserin and cinanserin

ArticleYear
[125I]-1-(2,5-dimethoxy-4-iodophenyl)-2-amino-propane: an iodinated radioligand that specifically labels the agonist high-affinity state of 5-HT2 serotonin receptors.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:1

    Topics: Amphetamines; Indicators and Reagents; Iodine Radioisotopes; Kinetics; Radioligand Assay; Receptors, Serotonin

1988
Conformational analysis, pharmacophore identification, and comparative molecular field analysis of ligands for the neuromodulatory sigma 3 receptor.
    Journal of medicinal chemistry, 1994, Nov-25, Volume: 37, Issue:24

    Topics: Animals; Ligands; Models, Molecular; Molecular Conformation; Receptors, sigma; Rodentia; Structure-Activity Relationship; Tetrahydronaphthalenes

1994
Serotonin (5-HT2) receptor mediated enhancement of cortical unit activity.
    Canadian journal of physiology and pharmacology, 1992, Volume: 70, Issue:12

    Topics: Animals; Cerebral Cortex; Cinanserin; Cyproheptadine; Iontophoresis; Ketanserin; Male; Microelectrodes; Neurons; Pain; Physical Stimulation; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1992
Mechanism of ketanserin-induced sympatho-inhibition.
    European journal of pharmacology, 1991, Mar-05, Volume: 194, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Animals; Biogenic Monoamines; Cats; Central Nervous System; Cinanserin; Electric Stimulation; Female; Galvanic Skin Response; Hypothalamus, Posterior; Ketanserin; Male; Sympathetic Nervous System; Synapses

1991
Are drugs that act both on serotonin receptors and alpha 1-adrenoceptors more potent hypotensive agents than those that act only on alpha 1-adrenoceptors?
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Cats; Cinanserin; Ergolines; Ketanserin; Male; Metergoline; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes

1988
[3H]ketanserin labels 5-HT2 receptors and alpha 1-adrenoceptors in human and pig brain membranes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Cinanserin; In Vitro Techniques; Ketanserin; Kinetics; Male; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Species Specificity; Swine; Tetralones

1987
Effects of serotonin receptor agonists and antagonists on schedule-controlled behavior of squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Cinanserin; Conditioning, Operant; Cyproheptadine; Electroshock; Female; Ketanserin; Male; Metergoline; Methysergide; Piperazines; Piperidines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri

1985
Antimyoclonic properties of S2 serotonin receptor antagonists in the rat.
    Neuropharmacology, 1986, Volume: 25, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Brain Chemistry; Butyrophenones; Cinanserin; Ketanserin; Male; Myoclonus; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1986
Habituation of tactile startle is altered by drugs acting on serotonin-2 receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1988, Volume: 1, Issue:2

    Topics: Animals; Cinanserin; Cyproheptadine; Habituation, Psychophysiologic; Ketanserin; Male; Piperidines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reference Values; Reflex, Startle; Ritanserin; Serotonin; Serotonin Antagonists; Touch

1988
Studies into the dual effects of serotonergic pharmacological agents on female sexual behaviour in the rat: preliminary evidence that endogenous 5HT is stimulatory.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:1

    Topics: 5-Hydroxytryptophan; Adrenalectomy; Alanine; Animals; Castration; Cinanserin; Female; Ketanserin; Metergoline; Methysergide; Mianserin; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal; Zimeldine

1985
In vivo binding of 125I-LSD to serotonin 5-HT2 receptors in mouse brain.
    Life sciences, 1985, Aug-19, Volume: 37, Issue:7

    Topics: Animals; Binding, Competitive; Brain; Cinanserin; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Mice; Piperidines; Receptors, Serotonin; Spiperone; Time Factors; Tissue Distribution

1985
Alpha 1 adrenergic receptors in the porcine pituitary neurointermediate lobe: detection with [3H]ketanserin.
    Journal of receptor research, 1984, Volume: 4, Issue:7

    Topics: Animals; Binding, Competitive; Brain; Cinanserin; In Vitro Techniques; Ketanserin; Kinetics; Piperidines; Pituitary Gland; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Swine

1984
Protective effect of serotonin (5-HT2) receptor antagonists in ischemic rat hearts.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:4

    Topics: Animals; Cinanserin; Disease Models, Animal; Ergolines; Heart; Hemodynamics; Ketanserin; L-Lactate Dehydrogenase; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardial Ischemia; Myocardial Reperfusion Injury; Myocardium; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Serotonin Antagonists

1993
Dorsal raphe nuclear stimulation of SCN serotonin release and circadian phase-resetting.
    Brain research, 2000, Mar-24, Volume: 859, Issue:2

    Topics: Animals; Cinanserin; Circadian Rhythm; Cricetinae; Electric Stimulation; Ketanserin; Male; Mesocricetus; Neural Pathways; Piperazines; Raphe Nuclei; Ritanserin; Serotonin; Serotonin Antagonists; Suprachiasmatic Nucleus

2000
Effects of serotonergic agents on the transport response in rats.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:3

    Topics: Age Factors; Analysis of Variance; Animals; Cinanserin; Female; Growth; Ketanserin; Metergoline; Motor Activity; Quipazine; Rats; Rats, Sprague-Dawley; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2000
Selective serotonin receptor antagonism and leukocyte-independent plasma extravasation during endotoxemia.
    Microvascular research, 2002, Volume: 63, Issue:1

    Topics: Animals; Binding Sites; Cinanserin; Endothelium, Vascular; Endotoxemia; Extravasation of Diagnostic and Therapeutic Materials; Ketanserin; Leukocytes; Methysergide; Microcirculation; Protein Binding; Rats; Receptors, Serotonin; Serotonin Antagonists; Time Factors

2002