ketanserin and captopril

ketanserin has been researched along with captopril in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19904 (25.00)18.7374
1990's5 (31.25)18.2507
2000's3 (18.75)29.6817
2010's4 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Coffman, JD1
Barbara, C; Bruzzone, F; Canale, C; Masperone, MA; Provinciali, L; Romeo, M; Terrachini, V; Zanna, C1
Buczko, W; Chabielska, E; Malinowska, B; Pietraszek, MH1
Assogna, G; Ladetto, PE; Lavezzaro, G; Salvetti, A; Stramignoni, D; Valente, M; Zanna, C1
Buczko, W; Malinowska, B1
Lazareth, I1
Meyer, P; Safar, M1
McGoon, MD; Vlietstra, RE1
Glusa, E1

Reviews

2 review(s) available for ketanserin and captopril

ArticleYear
Raynaud's phenomenon. An update.
    Hypertension (Dallas, Tex. : 1979), 1991, Volume: 17, Issue:5

    Topics: Calcium Channel Blockers; Captopril; Humans; Ketanserin; Prostaglandins; Raynaud Disease; Sympatholytics

1991
Vasodilator therapy for primary pulmonary hypertension.
    Mayo Clinic proceedings, 1984, Volume: 59, Issue:10

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Blood Pressure; Calcium Channel Blockers; Captopril; Epoprostenol; Hemodynamics; Humans; Hypertension, Pulmonary; Ketanserin; Piperidines; Serotonin Antagonists; Vascular Resistance; Vasodilator Agents

1984

Trials

3 trial(s) available for ketanserin and captopril

ArticleYear
[Short and medium term evaluation of captopril-ketanserin combination in mild to moderate arterial hypertension].
    La Clinica terapeutica, 1990, Apr-15, Volume: 133, Issue:1

    Topics: Adult; Aged; Captopril; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Randomized Controlled Trials as Topic; Time Factors

1990
Ketanserin and captopril interaction in the treatment of essential hypertensives.
    Cardiovascular drugs and therapy, 1990, Volume: 4 Suppl 1

    Topics: Adult; Aldosterone; Blood Pressure; Body Weight; Captopril; Double-Blind Method; Drug Therapy, Combination; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Potassium; Sodium

1990
Comparison of ketanserin with captopril in older hypertensives. A double-blind randomised trial.
    Drugs, 1988, Volume: 36 Suppl 1

    Topics: Aged; Aged, 80 and over; Captopril; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Humans; Hypertension; Ketanserin; Middle Aged; Multicenter Studies as Topic; Random Allocation

1988

Other Studies

11 other study(ies) available for ketanserin and captopril

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
    Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
The serotonergic mechanisms are not involved in the inhibitory effect of captopril on rat platelet aggregation.
    Haemostasis, 1990, Volume: 20, Issue:1

    Topics: Adenosine Diphosphate; Animals; Blood Platelets; Captopril; Collagen; Ketanserin; Male; Platelet Aggregation; Rats; Rats, Inbred Strains; Serotonin

1990
Influence of captopril on the vasopressor effect of serotonin in pithed rats.
    Pharmacology, 1989, Volume: 38, Issue:5

    Topics: Animals; Arteries; Blood Pressure; Captopril; Decerebrate State; Dose-Response Relationship, Drug; Ketanserin; Male; Rats; Rats, Inbred Strains; Regional Blood Flow; Serotonin; Tail

1989
[Treatment of Raynaud's phenomenon].
    Annales de dermatologie et de venereologie, 1987, Volume: 114, Issue:8

    Topics: Adrenergic alpha-Antagonists; Calcium Channel Blockers; Captopril; Humans; Ketanserin; Prostaglandins; Raynaud Disease

1987
Desulfated hirugen (hirudin 54-65) induces endothelium-dependent relaxation of porcine pulmonary arteries.
    Thrombosis and haemostasis, 1994, Volume: 72, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Amino Acid Sequence; Animals; Arginine; Atropine; Bradykinin; Calcium; Captopril; Cyclic GMP; Dinoprost; Endothelium, Vascular; Hirudins; Histamine; Indomethacin; Ketanserin; Methiothepin; Molecular Sequence Data; Muscle, Smooth, Vascular; Nitric Oxide; Nitroarginine; Peptide Fragments; Phentolamine; Pulmonary Artery; Swine; Vasodilation

1994