ketanserin and bemesetron

ketanserin has been researched along with bemesetron in 52 studies

Research

Studies (52)

TimeframeStudies, this research(%)All Research%
pre-199013 (25.00)18.7374
1990's19 (36.54)18.2507
2000's11 (21.15)29.6817
2010's9 (17.31)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO1
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X1
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG1
Colau, D; Dolusić, E; Frédérick, R; Larrieu, P; Masereel, B; Moineaux, L; Pilotte, L; Pochet, L; Stroobant, V; Van den Eynde, B; Wouters, J1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L1
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E1
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E1
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A1
Miletic, V; Tan, H1
Barrett, JE; Grant, KA1
Giordano, J1
Cervoni, P; Lai, FM; Tanikella, T1
Danzebrink, RM; Gebhart, GF1
Gaw, AJ; Humphrey, PP; Wadsworth, RM1
Jarrott, B; Louis, WJ; Verberne, AJ; Widdop, RE1
Anderson, EG; Todorovic, SM1
Adler-Graschinsky, E; Butta, NV; Elgoyhen, AB1
Feniuk, W; Humphrey, PP; Perren, MJ1
Chalmers, JP; Mills, EH; Minson, JB1
Heiligers, J; Mylecharane, EJ; Saxena, PR1
Gilbert, MJ; Newberry, NR1
Heiligers, J; Mylecharane, EJ; Saxena, PR; Tio, R1
Kilbinger, H; Pfeuffer-Friederich, I1
Birrell, GJ; Dutia, MB; Grubb, BD; Iggo, A; McQueen, DS1
Newberry, NR; Priestley, T1
Choquet, D; Korn, H1
Davies, M; Roberts, MH; Wilkinson, LS1
Andreini, R; Del Bianco, PL; Franchi, G; Panconesi, A; Sicuteri, F1
Kirby, GC; McQueen, DS1
Walcourt-Ambakederemo, A; Winlow, W1
Grant, KA; Hellevuo, K; Tabakoff, B1
Ageel, AM; Alhaider, AA; Ginawi, OT1
Lacosta, S; Roberts, DC1
Gibbs, J; Greenberg, D; Poeschla, B; Simansky, KJ; Smith, GP1
Horisaka, K; Kimura, I; Sugimoto, Y; Takeuchi, N; Watanabe, Y; Yamada, J1
Hayashi, T; Kagaya, A; Kugaya, A; Motohashi, N; Okamoto, Y; Shinno, H; Takebayashi, M; Uchitomi, Y; Yamaji, T; Yamawaki, S1
Albert, AP; Brooks, PA; Spyer, KM1
Cottrell, GA; Green, KA; Lambert, JJ1
Bodelsson, G; Bodelsson, M; Karlsson, C; Stjernquist, M1
Li, Y; Matsuda, H; Yamahara, J; Yoshikawa, M1
Goto, T; Ochi, T1
Naylor, RJ; Tuladhar, BR; Womack, MD1
English, KB; He, L; Tuckett, RP1
Kopczyńska, B; Szereda-Przestaszewska, M1
Asgari, K; Body, S; Bradshaw, CM; Fone, KC; Rickard, JF; Szabadi, E; Zhang, Z2
Kajos, M; Kankaanpää, A; Meririnne, E; Seppälä, T1
Jaworek, J; Konturek, SJ; Leja-Szpak, A; Nawrot-Porąbka, K; Reiter, RJ; Szklarczyk, J1
Go, D; Kim, SK; Lee, JH; Li, DX; Min, BI; Quan, FS; Yoon, H1
Bonior, J; Goralska, M; Jastrzebska, M; Jaworek, J; Leja-Szpak, A; Link-Lenczowski, P; Nawrot-Porabka, K; Pierzchalski, P1

Other Studies

52 other study(ies) available for ketanserin and bemesetron

ArticleYear
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
    Journal of medicinal chemistry, 2005, Nov-03, Volume: 48, Issue:22

    Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles

2005
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
    Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship

2008
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
    Journal of medicinal chemistry, 2008, Nov-27, Volume: 51, Issue:22

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship

2008
Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators.
    Journal of medicinal chemistry, 2011, Aug-11, Volume: 54, Issue:15

    Topics: Animals; Antineoplastic Agents; Biological Availability; Cell Line; Drug Design; Enzyme Inhibitors; Humans; Immunologic Factors; Indoles; Kinetics; Mice; Neoplasms; Structure-Activity Relationship; Tryptophan Oxygenase

2011
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2013
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
    Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

    Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
    Bioorganic & medicinal chemistry, 2016, Apr-15, Volume: 24, Issue:8

    Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine

2016
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
    Bioorganic & medicinal chemistry, 2017, 01-15, Volume: 25, Issue:2

    Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship

2017
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 101, Issue:2

    Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1992
Diverse actions of 5-hydroxytryptamine on frog spinal dorsal horn neurons in vitro.
    Neuroscience, 1992, Volume: 49, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dioxanes; Electric Stimulation; Evoked Potentials; Female; In Vitro Techniques; Ketanserin; Kinetics; Male; Membrane Potentials; Methysergide; Mianserin; Neurons; Rana pipiens; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Synapses; Tetrodotoxin; Tropanes

1992
Blockade of the discriminative stimulus effects of ethanol with 5-HT3 receptor antagonists.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Columbidae; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Ethanol; Haloperidol; Indoles; Ketanserin; Male; Serotonin Antagonists; Tropanes; Tropisetron

1991
Analgesic profile of centrally administered 2-methylserotonin against acute pain in rats.
    European journal of pharmacology, 1991, Jun-25, Volume: 199, Issue:2

    Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Mianserin; Motor Activity; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Respiration; Serotonin; Serotonin Antagonists; Tropanes

1991
Characterization of serotonin receptors in isolated rat intramyocardial coronary artery.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:1

    Topics: Animals; Coronary Vessels; Dinoprost; Endothelium; Ketanserin; Kinetics; Male; Muscle Contraction; Muscle, Smooth, Vascular; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes

1991
Evidence that spinal 5-HT1, 5-HT2 and 5-HT3 receptor subtypes modulate responses to noxious colorectal distension in the rat.
    Brain research, 1991, Jan-04, Volume: 538, Issue:1

    Topics: Amidines; Animals; Blood Pressure; Colon; Indoles; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Muscles; Pressure; Rats; Rats, Inbred Strains; Receptors, Serotonin; Rectum; Reflex; Serotonin Antagonists; Spinal Cord; Tropanes; Tropisetron

1991
Pharmacological characterisation of postjunctional 5-HT receptors in cerebral arteries from the sheep.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Animals; Basilar Artery; Cerebral Arteries; Indoles; Ketanserin; Norepinephrine; Receptors, Serotonin; Serotonin; Sheep; Sulfonamides; Sumatriptan; Tropanes; Vasoconstriction

1990
The effect of ketanserin on cardiovascular reflexes in conscious normotensive and spontaneously hypertensive rats.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: Animals; Atropine; Biguanides; Blood Pressure; Cardiovascular System; Dose-Response Relationship, Drug; Electric Stimulation; Female; Heart Rate; Hypoglycemic Agents; Ketanserin; Nitroprusside; Pressoreceptors; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Reflex; Tropanes; Vagus Nerve

1990
Pharmacological characterization of 5-hydroxytryptamine2 and 5-hydroxytryptamine3 receptors in rat dorsal root ganglion cells.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Indoles; Ketanserin; Male; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropanes; Tropisetron

1990
Different receptor subtypes mediate the dual presynaptic effects of 5-hydroxytryptamine on peripheral sympathetic neurones.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cats; Cyproheptadine; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Ketanserin; Male; Membranes; Metoclopramide; Neurons; Norepinephrine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes; Tropanes

1989
The selective carotid arterial vasoconstrictor action of GR43175 in anaesthetized dogs.
    British journal of pharmacology, 1989, Volume: 96, Issue:1

    Topics: Animals; Barbital; Carotid Arteries; Dogs; Female; Hemodynamics; Indoles; Ketanserin; Male; Methiothepin; Phentolamine; Serotonin Antagonists; Sulfonamides; Sumatriptan; Tropanes; Vasoconstrictor Agents

1989
The effect of intrathecal serotonergic antagonists on the pressor response to stimulation of the brainstem in the rat.
    Clinical and experimental hypertension. Part A, Theory and practice, 1989, Volume: 11, Issue:2

    Topics: Animals; Blood Pressure; Electric Stimulation; Glutamates; Indoles; Injections, Spinal; Ketanserin; Medulla Oblongata; Methysergide; Microinjections; Rats; Rats, Inbred WKY; Receptors, Serotonin; Spinal Cord; Tropanes; Tropisetron

1989
Analysis of the heart rate effects of 5-hydroxytryptamine in the cat; mediation of tachycardia by 5-HT1-like receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 330, Issue:2

    Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Isoproterenol; Ketanserin; Male; Methysergide; Piperidines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tropanes; Vagus Nerve

1985
A 5-HT1-like receptor mediates a sympathetic ganglionic hyperpolarization.
    European journal of pharmacology, 1987, Dec-15, Volume: 144, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ganglia, Sympathetic; In Vitro Techniques; Ketanserin; Membrane Potentials; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Tropanes

1987
Excitatory 5-hydroxytryptamine receptors in the cat urinary bladder are of the M- and 5-HT2-type.
    Journal of autonomic pharmacology, 1985, Volume: 5, Issue:2

    Topics: Animals; Atropine; Cats; Cyproheptadine; Dimethylphenylpiperazinium Iodide; Drug Interactions; Female; Guanethidine; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Urinary Bladder

1985
Two types of receptors for 5-hydroxytryptamine on the cholinergic nerves of the guinea-pig myenteric plexus.
    British journal of pharmacology, 1985, Volume: 85, Issue:2

    Topics: Acetylcholine; Animals; Binding, Competitive; Cocaine; Electric Stimulation; Female; Guinea Pigs; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Myenteric Plexus; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes

1985
A study of 5-HT-receptors associated with afferent nerves located in normal and inflamed rat ankle joints.
    Agents and actions, 1988, Volume: 25, Issue:3-4

    Topics: Action Potentials; Animals; Ankle Joint; Arthritis; Ketanserin; Neurons, Afferent; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes

1988
A 5-HT1-like receptor mediates a pertussis toxin-sensitive inhibition of rat ventromedial hypothalamic neurones in vitro.
    British journal of pharmacology, 1988, Volume: 95, Issue:1

    Topics: Animals; In Vitro Techniques; Ketanserin; Male; Neurons; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Ventromedial Hypothalamic Nucleus; Virulence Factors, Bordetella

1988
Dual effects of serotonin on a voltage-gated conductance in lymphocytes.
    Proceedings of the National Academy of Sciences of the United States of America, 1988, Volume: 85, Issue:12

    Topics: Abelson murine leukemia virus; Animals; B-Lymphocytes; Cell Line, Transformed; Electric Conductivity; Indoles; Ketanserin; Membrane Potentials; Metergoline; Methiothepin; Mice; Potassium; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1988
Evidence for depressant 5-HT1-like receptors on rat brainstem neurones.
    British journal of pharmacology, 1988, Volume: 94, Issue:2

    Topics: Animals; Brain Stem; Ketanserin; Male; Membrane Potentials; Metergoline; Methysergide; Neurons; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tropanes

1988
In vivo characterization of serotonin receptors on hand vein.
    Pharmacological research communications, 1988, Volume: 20, Issue:5

    Topics: Adolescent; Adult; Female; Hand; Humans; Ketanserin; Male; Muscle, Smooth, Vascular; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Tropanes; Vasoconstriction

1988
Effects of the antagonists MDL 72222 and ketanserin on responses of cat carotid body chemoreceptors to 5-hydroxytryptamine.
    British journal of pharmacology, 1984, Volume: 83, Issue:1

    Topics: Action Potentials; Animals; Carotid Body; Cats; Chemoreceptor Cells; Domperidone; Dopamine; Electrophysiology; Female; Hypoxia; Ketanserin; Male; Piperidines; Serotonin; Serotonin Antagonists; Tropanes

1984
5-HT receptors on identified Lymnaea neurones in culture: pharmacological characterization of 5-HT3 receptors.
    General pharmacology, 1995, Volume: 26, Issue:3

    Topics: Animals; Biguanides; Cells, Cultured; Ketanserin; Lymnaea; Neurons; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes

1995
The 5-HT3 antagonist MDL-72222 exacerbates ethanol withdrawal seizures in mice.
    Alcoholism, clinical and experimental research, 1994, Volume: 18, Issue:2

    Topics: Alcohol Withdrawal Delirium; Animals; Dose-Response Relationship, Drug; Electroencephalography; Evoked Potentials; Ketanserin; Male; Mice; Mice, Inbred C57BL; Postural Balance; Receptors, Serotonin; Seizures; Serotonin Antagonists; Stimulation, Chemical; Tropanes

1994
The quipazine- and TFMPP-increased conditioned avoidance response in rats: role of 5HT1C/5-HT2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: Animals; Avoidance Learning; Conditioning, Operant; Ketanserin; Male; Mianserin; Nadolol; Pindolol; Piperazines; Prazosin; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tropanes

1993
MDL 72222, ketanserin, and methysergide pretreatments fail to alter breaking points on a progressive ratio schedule reinforced by intravenous cocaine.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:1

    Topics: Animals; Cocaine; Conditioning, Operant; Injections, Intravenous; Ketanserin; Male; Methysergide; Rats; Rats, Wistar; Reinforcement Schedule; Self Administration; Serotonin Antagonists; Tropanes

1993
Cholecystokinin-induced satiety depends on activation of 5-HT1C receptors.
    The American journal of physiology, 1993, Volume: 264, Issue:1 Pt 2

    Topics: Animals; Eating; Ketanserin; Male; Mianserin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Satiation; Serotonin Antagonists; Sincalide; Tropanes

1993
Peripherally administered serotonin induces hyperglucagonemia in mice.
    Life sciences, 1993, Volume: 52, Issue:23

    Topics: Animals; Glucagon; Indoles; Injections, Intraperitoneal; Ketanserin; Male; Methysergide; Mice; Mice, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Tropisetron

1993
Cyclic GMP generation mediated by 5-HT-2 receptors via nitric oxide-dependent pathway and its effect on the desensitization of 5-HT-2 receptors in C6 glioma cells.
    Journal of neural transmission. General section, 1995, Volume: 100, Issue:1

    Topics: Animals; Arginine; Calcium; Chelating Agents; Cyclic GMP; Dopamine Antagonists; Edetic Acid; Egtazic Acid; Glioma; Haloperidol; Ketanserin; Nitric Oxide; omega-N-Methylarginine; Rats; Receptors, Serotonin; Risperidone; Serotonin Antagonists; Tropanes; Tumor Cells, Cultured

1995
The effect of 5-HT and selective 5-HT receptor agonists and antagonists on rat dorsal vagal preganglionic neurones in vitro.
    British journal of pharmacology, 1996, Volume: 119, Issue:3

    Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Ergolines; Female; In Vitro Techniques; Indoles; Ketanserin; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium Channels; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Tropanes; Vagus Nerve

1996
Ligand-gated ion channels opened by 5-HT in molluscan neurones.
    British journal of pharmacology, 1996, Volume: 119, Issue:3

    Topics: Animals; Calcium; Convulsants; Dose-Response Relationship, Drug; Electrophysiology; GTP-Binding Proteins; Helix, Snails; Ion Channel Gating; Ion Channels; Ketanserin; Neurons; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Strychnine; Tropanes

1996
Characterization of 5-hydroxytryptamine receptors mediating circular smooth muscle contraction in the human umbilical artery.
    Gynecologic and obstetric investigation, 1999, Volume: 47, Issue:2

    Topics: Adolescent; Adult; Female; Humans; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth; Pregnancy; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tropanes; Umbilical Arteries

1999
Acceleration of gastrointestinal transit by momordin Ic in mice: possible involvement of 5-hydroxytryptamine, 5-HT(2) receptors and prostaglandins.
    European journal of pharmacology, 2000, Mar-24, Volume: 392, Issue:1-2

    Topics: Animals; Fenclonine; Gastrointestinal Motility; Indomethacin; Ketanserin; Male; Mice; Oleanolic Acid; Prostaglandins; Receptors, Serotonin; Serotonin; Tropanes

2000
The antinociceptive effect induced by FR140423 is mediated through spinal 5-HT2A and 5-HT3 receptors.
    European journal of pharmacology, 2000, Dec-08, Volume: 409, Issue:2

    Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Methysergide; Mice; Pain; Pain Measurement; Piperazines; Pyrazoles; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Sulfoxides; Tropanes

2000
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
5-HT2 and 3 receptor antagonists suppress the response of rat type I slowly adapting mechanoreceptor: an in vitro study.
    Brain research, 2003, Apr-18, Volume: 969, Issue:1-2

    Topics: Action Potentials; Adaptation, Physiological; Animals; Female; Free Radical Scavengers; Ketanserin; Male; Mechanoreceptors; Organ Culture Techniques; Physical Stimulation; Rats; Rats, Sprague-Dawley; Ritanserin; Serotonin; Serotonin Antagonists; Skin; Tropanes

2003
5HT2 and 5HT3 receptors' contribution to modeling of post-serotonin respiratory pattern in cats.
    Life sciences, 2004, Sep-24, Volume: 75, Issue:19

    Topics: Animals; Apnea; Blood Pressure; Bradycardia; Cats; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Ketanserin; Larynx; Male; Phrenic Nerve; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT3; Respiratory Mechanics; Serotonin; Serotonin Antagonists; Tidal Volume; Tropanes

2004
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on the discrimination of durations: evidence for the involvement of 5-HT2A but not 5-HT3 receptors.
    Behavioural pharmacology, 2005, Volume: 16, Issue:1

    Topics: Animals; Biguanides; Discrimination Learning; Discrimination, Psychological; Female; Ketanserin; Quipazine; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes

2005
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on temporal differentiation: evidence for the involvement of 5-HT2A but not 5-HT3 receptors in interval timing behaviour.
    Psychopharmacology, 2005, Volume: 181, Issue:2

    Topics: Animals; Biguanides; Conditioning, Operant; Dose-Response Relationship, Drug; Female; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Psychometrics; Quipazine; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Task Performance and Analysis; Time Perception; Tropanes

2005
Rewarding properties of 1-benzylpiperazine, a new drug of abuse, in rats.
    Basic & clinical pharmacology & toxicology, 2006, Volume: 98, Issue:4

    Topics: Animals; Behavior, Animal; Benzazepines; Conditioning, Psychological; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ketanserin; Male; Piperidines; Psychotropic Drugs; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT3; Reward; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Substance-Related Disorders; Tropanes

2006
Luminal melatonin stimulates pancreatic enzyme secretion via activation of serotonin-dependent nerves.
    Pharmacological reports : PR, 2013, Volume: 65, Issue:2

    Topics: Amylases; Animals; Dose-Response Relationship, Drug; Duodenum; Ketanserin; Melatonin; Pancreas; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Serotonin; Serotonin Antagonists; Time Factors; Tropanes; Tryptophan; Vagus Nerve

2013
Serotonergic mechanism of the relieving effect of bee venom acupuncture on oxaliplatin-induced neuropathic cold allodynia in rats.
    BMC complementary and alternative medicine, 2014, Dec-06, Volume: 14

    Topics: Acupuncture Analgesia; Acupuncture Points; Animals; Apitherapy; Bee Venoms; Cold Temperature; Fenclonine; Hyperalgesia; Ketanserin; Male; Neuralgia; Organoplatinum Compounds; Oxaliplatin; Peripheral Nervous System Diseases; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin 5-HT3 Receptor Agonists; Serotonin Antagonists; Spinal Cord; Tropanes

2014
Kynuramines induce overexpression of heat shock proteins in pancreatic cancer cells via 5-hydroxytryptamine and MT1/MT2 receptors.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2015, Volume: 66, Issue:5

    Topics: Cell Line, Tumor; Heat-Shock Proteins; Humans; Ketanserin; Kynuramine; Melatonin; Pancreatic Neoplasms; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Serotonin; Tropanes; Tryptamines; Tryptophan

2015