ketanserin has been researched along with bemesetron in 52 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 13 (25.00) | 18.7374 |
1990's | 19 (36.54) | 18.2507 |
2000's | 11 (21.15) | 29.6817 |
2010's | 9 (17.31) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO | 1 |
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X | 1 |
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG | 1 |
Colau, D; Dolusić, E; Frédérick, R; Larrieu, P; Masereel, B; Moineaux, L; Pilotte, L; Pochet, L; Stroobant, V; Van den Eynde, B; Wouters, J | 1 |
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L | 1 |
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S | 1 |
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L | 1 |
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E | 1 |
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E | 1 |
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A | 1 |
Miletic, V; Tan, H | 1 |
Barrett, JE; Grant, KA | 1 |
Giordano, J | 1 |
Cervoni, P; Lai, FM; Tanikella, T | 1 |
Danzebrink, RM; Gebhart, GF | 1 |
Gaw, AJ; Humphrey, PP; Wadsworth, RM | 1 |
Jarrott, B; Louis, WJ; Verberne, AJ; Widdop, RE | 1 |
Anderson, EG; Todorovic, SM | 1 |
Adler-Graschinsky, E; Butta, NV; Elgoyhen, AB | 1 |
Feniuk, W; Humphrey, PP; Perren, MJ | 1 |
Chalmers, JP; Mills, EH; Minson, JB | 1 |
Heiligers, J; Mylecharane, EJ; Saxena, PR | 1 |
Gilbert, MJ; Newberry, NR | 1 |
Heiligers, J; Mylecharane, EJ; Saxena, PR; Tio, R | 1 |
Kilbinger, H; Pfeuffer-Friederich, I | 1 |
Birrell, GJ; Dutia, MB; Grubb, BD; Iggo, A; McQueen, DS | 1 |
Newberry, NR; Priestley, T | 1 |
Choquet, D; Korn, H | 1 |
Davies, M; Roberts, MH; Wilkinson, LS | 1 |
Andreini, R; Del Bianco, PL; Franchi, G; Panconesi, A; Sicuteri, F | 1 |
Kirby, GC; McQueen, DS | 1 |
Walcourt-Ambakederemo, A; Winlow, W | 1 |
Grant, KA; Hellevuo, K; Tabakoff, B | 1 |
Ageel, AM; Alhaider, AA; Ginawi, OT | 1 |
Lacosta, S; Roberts, DC | 1 |
Gibbs, J; Greenberg, D; Poeschla, B; Simansky, KJ; Smith, GP | 1 |
Horisaka, K; Kimura, I; Sugimoto, Y; Takeuchi, N; Watanabe, Y; Yamada, J | 1 |
Hayashi, T; Kagaya, A; Kugaya, A; Motohashi, N; Okamoto, Y; Shinno, H; Takebayashi, M; Uchitomi, Y; Yamaji, T; Yamawaki, S | 1 |
Albert, AP; Brooks, PA; Spyer, KM | 1 |
Cottrell, GA; Green, KA; Lambert, JJ | 1 |
Bodelsson, G; Bodelsson, M; Karlsson, C; Stjernquist, M | 1 |
Li, Y; Matsuda, H; Yamahara, J; Yoshikawa, M | 1 |
Goto, T; Ochi, T | 1 |
Naylor, RJ; Tuladhar, BR; Womack, MD | 1 |
English, KB; He, L; Tuckett, RP | 1 |
Kopczyńska, B; Szereda-Przestaszewska, M | 1 |
Asgari, K; Body, S; Bradshaw, CM; Fone, KC; Rickard, JF; Szabadi, E; Zhang, Z | 2 |
Kajos, M; Kankaanpää, A; Meririnne, E; Seppälä, T | 1 |
Jaworek, J; Konturek, SJ; Leja-Szpak, A; Nawrot-Porąbka, K; Reiter, RJ; Szklarczyk, J | 1 |
Go, D; Kim, SK; Lee, JH; Li, DX; Min, BI; Quan, FS; Yoon, H | 1 |
Bonior, J; Goralska, M; Jastrzebska, M; Jaworek, J; Leja-Szpak, A; Link-Lenczowski, P; Nawrot-Porabka, K; Pierzchalski, P | 1 |
52 other study(ies) available for ketanserin and bemesetron
Article | Year |
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2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles | 2005 |
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship | 2008 |
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship | 2008 |
Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators.
Topics: Animals; Antineoplastic Agents; Biological Availability; Cell Line; Drug Design; Enzyme Inhibitors; Humans; Immunologic Factors; Indoles; Kinetics; Mice; Neoplasms; Structure-Activity Relationship; Tryptophan Oxygenase | 2011 |
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship | 2013 |
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship | 2013 |
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship | 2013 |
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine | 2016 |
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship | 2017 |
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1992 |
Diverse actions of 5-hydroxytryptamine on frog spinal dorsal horn neurons in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dioxanes; Electric Stimulation; Evoked Potentials; Female; In Vitro Techniques; Ketanserin; Kinetics; Male; Membrane Potentials; Methysergide; Mianserin; Neurons; Rana pipiens; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Synapses; Tetrodotoxin; Tropanes | 1992 |
Blockade of the discriminative stimulus effects of ethanol with 5-HT3 receptor antagonists.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Columbidae; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Ethanol; Haloperidol; Indoles; Ketanserin; Male; Serotonin Antagonists; Tropanes; Tropisetron | 1991 |
Analgesic profile of centrally administered 2-methylserotonin against acute pain in rats.
Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Mianserin; Motor Activity; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Respiration; Serotonin; Serotonin Antagonists; Tropanes | 1991 |
Characterization of serotonin receptors in isolated rat intramyocardial coronary artery.
Topics: Animals; Coronary Vessels; Dinoprost; Endothelium; Ketanserin; Kinetics; Male; Muscle Contraction; Muscle, Smooth, Vascular; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes | 1991 |
Evidence that spinal 5-HT1, 5-HT2 and 5-HT3 receptor subtypes modulate responses to noxious colorectal distension in the rat.
Topics: Amidines; Animals; Blood Pressure; Colon; Indoles; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Muscles; Pressure; Rats; Rats, Inbred Strains; Receptors, Serotonin; Rectum; Reflex; Serotonin Antagonists; Spinal Cord; Tropanes; Tropisetron | 1991 |
Pharmacological characterisation of postjunctional 5-HT receptors in cerebral arteries from the sheep.
Topics: Animals; Basilar Artery; Cerebral Arteries; Indoles; Ketanserin; Norepinephrine; Receptors, Serotonin; Serotonin; Sheep; Sulfonamides; Sumatriptan; Tropanes; Vasoconstriction | 1990 |
The effect of ketanserin on cardiovascular reflexes in conscious normotensive and spontaneously hypertensive rats.
Topics: Animals; Atropine; Biguanides; Blood Pressure; Cardiovascular System; Dose-Response Relationship, Drug; Electric Stimulation; Female; Heart Rate; Hypoglycemic Agents; Ketanserin; Nitroprusside; Pressoreceptors; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Reflex; Tropanes; Vagus Nerve | 1990 |
Pharmacological characterization of 5-hydroxytryptamine2 and 5-hydroxytryptamine3 receptors in rat dorsal root ganglion cells.
Topics: Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Indoles; Ketanserin; Male; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropanes; Tropisetron | 1990 |
Different receptor subtypes mediate the dual presynaptic effects of 5-hydroxytryptamine on peripheral sympathetic neurones.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cats; Cyproheptadine; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Ketanserin; Male; Membranes; Metoclopramide; Neurons; Norepinephrine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes; Tropanes | 1989 |
The selective carotid arterial vasoconstrictor action of GR43175 in anaesthetized dogs.
Topics: Animals; Barbital; Carotid Arteries; Dogs; Female; Hemodynamics; Indoles; Ketanserin; Male; Methiothepin; Phentolamine; Serotonin Antagonists; Sulfonamides; Sumatriptan; Tropanes; Vasoconstrictor Agents | 1989 |
The effect of intrathecal serotonergic antagonists on the pressor response to stimulation of the brainstem in the rat.
Topics: Animals; Blood Pressure; Electric Stimulation; Glutamates; Indoles; Injections, Spinal; Ketanserin; Medulla Oblongata; Methysergide; Microinjections; Rats; Rats, Inbred WKY; Receptors, Serotonin; Spinal Cord; Tropanes; Tropisetron | 1989 |
Analysis of the heart rate effects of 5-hydroxytryptamine in the cat; mediation of tachycardia by 5-HT1-like receptors.
Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Isoproterenol; Ketanserin; Male; Methysergide; Piperidines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tropanes; Vagus Nerve | 1985 |
A 5-HT1-like receptor mediates a sympathetic ganglionic hyperpolarization.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ganglia, Sympathetic; In Vitro Techniques; Ketanserin; Membrane Potentials; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Tropanes | 1987 |
Excitatory 5-hydroxytryptamine receptors in the cat urinary bladder are of the M- and 5-HT2-type.
Topics: Animals; Atropine; Cats; Cyproheptadine; Dimethylphenylpiperazinium Iodide; Drug Interactions; Female; Guanethidine; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Urinary Bladder | 1985 |
Two types of receptors for 5-hydroxytryptamine on the cholinergic nerves of the guinea-pig myenteric plexus.
Topics: Acetylcholine; Animals; Binding, Competitive; Cocaine; Electric Stimulation; Female; Guinea Pigs; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Myenteric Plexus; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes | 1985 |
A study of 5-HT-receptors associated with afferent nerves located in normal and inflamed rat ankle joints.
Topics: Action Potentials; Animals; Ankle Joint; Arthritis; Ketanserin; Neurons, Afferent; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes | 1988 |
A 5-HT1-like receptor mediates a pertussis toxin-sensitive inhibition of rat ventromedial hypothalamic neurones in vitro.
Topics: Animals; In Vitro Techniques; Ketanserin; Male; Neurons; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Ventromedial Hypothalamic Nucleus; Virulence Factors, Bordetella | 1988 |
Dual effects of serotonin on a voltage-gated conductance in lymphocytes.
Topics: Abelson murine leukemia virus; Animals; B-Lymphocytes; Cell Line, Transformed; Electric Conductivity; Indoles; Ketanserin; Membrane Potentials; Metergoline; Methiothepin; Mice; Potassium; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1988 |
Evidence for depressant 5-HT1-like receptors on rat brainstem neurones.
Topics: Animals; Brain Stem; Ketanserin; Male; Membrane Potentials; Metergoline; Methysergide; Neurons; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tropanes | 1988 |
In vivo characterization of serotonin receptors on hand vein.
Topics: Adolescent; Adult; Female; Hand; Humans; Ketanserin; Male; Muscle, Smooth, Vascular; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Tropanes; Vasoconstriction | 1988 |
Effects of the antagonists MDL 72222 and ketanserin on responses of cat carotid body chemoreceptors to 5-hydroxytryptamine.
Topics: Action Potentials; Animals; Carotid Body; Cats; Chemoreceptor Cells; Domperidone; Dopamine; Electrophysiology; Female; Hypoxia; Ketanserin; Male; Piperidines; Serotonin; Serotonin Antagonists; Tropanes | 1984 |
5-HT receptors on identified Lymnaea neurones in culture: pharmacological characterization of 5-HT3 receptors.
Topics: Animals; Biguanides; Cells, Cultured; Ketanserin; Lymnaea; Neurons; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes | 1995 |
The 5-HT3 antagonist MDL-72222 exacerbates ethanol withdrawal seizures in mice.
Topics: Alcohol Withdrawal Delirium; Animals; Dose-Response Relationship, Drug; Electroencephalography; Evoked Potentials; Ketanserin; Male; Mice; Mice, Inbred C57BL; Postural Balance; Receptors, Serotonin; Seizures; Serotonin Antagonists; Stimulation, Chemical; Tropanes | 1994 |
The quipazine- and TFMPP-increased conditioned avoidance response in rats: role of 5HT1C/5-HT2 receptors.
Topics: Animals; Avoidance Learning; Conditioning, Operant; Ketanserin; Male; Mianserin; Nadolol; Pindolol; Piperazines; Prazosin; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tropanes | 1993 |
MDL 72222, ketanserin, and methysergide pretreatments fail to alter breaking points on a progressive ratio schedule reinforced by intravenous cocaine.
Topics: Animals; Cocaine; Conditioning, Operant; Injections, Intravenous; Ketanserin; Male; Methysergide; Rats; Rats, Wistar; Reinforcement Schedule; Self Administration; Serotonin Antagonists; Tropanes | 1993 |
Cholecystokinin-induced satiety depends on activation of 5-HT1C receptors.
Topics: Animals; Eating; Ketanserin; Male; Mianserin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Satiation; Serotonin Antagonists; Sincalide; Tropanes | 1993 |
Peripherally administered serotonin induces hyperglucagonemia in mice.
Topics: Animals; Glucagon; Indoles; Injections, Intraperitoneal; Ketanserin; Male; Methysergide; Mice; Mice, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Tropisetron | 1993 |
Cyclic GMP generation mediated by 5-HT-2 receptors via nitric oxide-dependent pathway and its effect on the desensitization of 5-HT-2 receptors in C6 glioma cells.
Topics: Animals; Arginine; Calcium; Chelating Agents; Cyclic GMP; Dopamine Antagonists; Edetic Acid; Egtazic Acid; Glioma; Haloperidol; Ketanserin; Nitric Oxide; omega-N-Methylarginine; Rats; Receptors, Serotonin; Risperidone; Serotonin Antagonists; Tropanes; Tumor Cells, Cultured | 1995 |
The effect of 5-HT and selective 5-HT receptor agonists and antagonists on rat dorsal vagal preganglionic neurones in vitro.
Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Ergolines; Female; In Vitro Techniques; Indoles; Ketanserin; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium Channels; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Tropanes; Vagus Nerve | 1996 |
Ligand-gated ion channels opened by 5-HT in molluscan neurones.
Topics: Animals; Calcium; Convulsants; Dose-Response Relationship, Drug; Electrophysiology; GTP-Binding Proteins; Helix, Snails; Ion Channel Gating; Ion Channels; Ketanserin; Neurons; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Strychnine; Tropanes | 1996 |
Characterization of 5-hydroxytryptamine receptors mediating circular smooth muscle contraction in the human umbilical artery.
Topics: Adolescent; Adult; Female; Humans; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth; Pregnancy; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tropanes; Umbilical Arteries | 1999 |
Acceleration of gastrointestinal transit by momordin Ic in mice: possible involvement of 5-hydroxytryptamine, 5-HT(2) receptors and prostaglandins.
Topics: Animals; Fenclonine; Gastrointestinal Motility; Indomethacin; Ketanserin; Male; Mice; Oleanolic Acid; Prostaglandins; Receptors, Serotonin; Serotonin; Tropanes | 2000 |
The antinociceptive effect induced by FR140423 is mediated through spinal 5-HT2A and 5-HT3 receptors.
Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Methysergide; Mice; Pain; Pain Measurement; Piperazines; Pyrazoles; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Sulfoxides; Tropanes | 2000 |
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron | 2000 |
5-HT2 and 3 receptor antagonists suppress the response of rat type I slowly adapting mechanoreceptor: an in vitro study.
Topics: Action Potentials; Adaptation, Physiological; Animals; Female; Free Radical Scavengers; Ketanserin; Male; Mechanoreceptors; Organ Culture Techniques; Physical Stimulation; Rats; Rats, Sprague-Dawley; Ritanserin; Serotonin; Serotonin Antagonists; Skin; Tropanes | 2003 |
5HT2 and 5HT3 receptors' contribution to modeling of post-serotonin respiratory pattern in cats.
Topics: Animals; Apnea; Blood Pressure; Bradycardia; Cats; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Ketanserin; Larynx; Male; Phrenic Nerve; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT3; Respiratory Mechanics; Serotonin; Serotonin Antagonists; Tidal Volume; Tropanes | 2004 |
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on the discrimination of durations: evidence for the involvement of 5-HT2A but not 5-HT3 receptors.
Topics: Animals; Biguanides; Discrimination Learning; Discrimination, Psychological; Female; Ketanserin; Quipazine; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes | 2005 |
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on temporal differentiation: evidence for the involvement of 5-HT2A but not 5-HT3 receptors in interval timing behaviour.
Topics: Animals; Biguanides; Conditioning, Operant; Dose-Response Relationship, Drug; Female; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Psychometrics; Quipazine; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Task Performance and Analysis; Time Perception; Tropanes | 2005 |
Rewarding properties of 1-benzylpiperazine, a new drug of abuse, in rats.
Topics: Animals; Behavior, Animal; Benzazepines; Conditioning, Psychological; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ketanserin; Male; Piperidines; Psychotropic Drugs; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT3; Reward; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Substance-Related Disorders; Tropanes | 2006 |
Luminal melatonin stimulates pancreatic enzyme secretion via activation of serotonin-dependent nerves.
Topics: Amylases; Animals; Dose-Response Relationship, Drug; Duodenum; Ketanserin; Melatonin; Pancreas; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Serotonin; Serotonin Antagonists; Time Factors; Tropanes; Tryptophan; Vagus Nerve | 2013 |
Serotonergic mechanism of the relieving effect of bee venom acupuncture on oxaliplatin-induced neuropathic cold allodynia in rats.
Topics: Acupuncture Analgesia; Acupuncture Points; Animals; Apitherapy; Bee Venoms; Cold Temperature; Fenclonine; Hyperalgesia; Ketanserin; Male; Neuralgia; Organoplatinum Compounds; Oxaliplatin; Peripheral Nervous System Diseases; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin 5-HT3 Receptor Agonists; Serotonin Antagonists; Spinal Cord; Tropanes | 2014 |
Kynuramines induce overexpression of heat shock proteins in pancreatic cancer cells via 5-hydroxytryptamine and MT1/MT2 receptors.
Topics: Cell Line, Tumor; Heat-Shock Proteins; Humans; Ketanserin; Kynuramine; Melatonin; Pancreatic Neoplasms; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Serotonin; Tropanes; Tryptamines; Tryptophan | 2015 |