ketanserin and altanserin

ketanserin has been researched along with altanserin in 89 studies

Research

Studies (89)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	15 (16.85)	18.2507
2000's	44 (49.44)	29.6817
2010's	28 (31.46)	24.3611
2020's	2 (2.25)	2.80

Authors

Authors	Studies
Chen, Z; Collier, T; Fu, H; Liang, SH; Rong, J; Zhou, J	1
Cantineau, R; Christiaens, L; Guillaume, M; Lemaire, C; Plenevaux, A	1
Baron, JC; Petit Taboué, MC	1
Cantineau, R; Comar, D; Degueldre, C; Guillaume, M; Hermanne, JP; Lemaire, C; Maquet, P; Plenevaux, A; Sadzot, B; Salmon, E	1
Alexoff, D; Ashby, CR; Brodie, JD; Dewey, SL; Ding, YS; King, P; Logan, J; Pappas, N; Smith, GS	1
Biver, F; Forestini, M; Goldman, S; Lotstra, F; Luxen, A; Mendlewicz, J; Monclus, M	1
Brodie, JD; Dewey, SL; Logan, J; Smith, GS	1
Biver, F; Damhaut, P; Goldman, S; Lotstra, F; Mendlewicz, J; Monclus, M; Wikler, D	1
Bormans, G; de Groot, T; Dupont, P; Maes, M; Mortelmans, L; Peuskens, J; Rosier, A; Schiepers, C; Vandenberghe, R; Verbruggen, A	1
Biver, F; Damhaut, P; Dethy, S; Goldman, S; Lotstra, F; Luxen, A; Monclus, M; Wikler, D	1
Biver, F; Damhaut, P; Goldman, S; Lotstra, F; Mendlewicz, J; Wikler, D	1
Ben-Eliezer, D; Cantwell, MN; DeKosky, ST; Greer, P; Kaye, W; Lopresti, B; Mathis, CA; Meltzer, CC; Mintun, MA; Pollock, BG; Price, JC; Reynolds, CF; Smith, G	1
Holt, D; Huang, Y; Lopresti, BJ; Mason, NS; Mathis, CA; Meltzer, CC; Nichols, T; Price, JC; Sashin, D; Simpson, N; Smith, GS; Sweet, RA	1
Baldwin, RM; Charney, DS; Garg, PK; Innis, RB; Soufer, R; Tan, PZ	1
Al-Tikriti, M; Baldwin, RM; Charney, DS; Innis, RB; Khan, N; Roth, B; Tan, PZ; Van Dyck, CH	1
Ben-Eliezer, D; Cantwell, MN; DeKosky, ST; Greer, PJ; Houck, PR; Lopresti, B; Mathis, CA; Meltzer, CC; Mulsant, BH; Price, JC; Reynolds, CF	1
Amici, LA; Baldwin, RM; Charney, DS; Garg, PK; Innis, RB; Ng, CK; Soufer, R; Tan, PZ; van Dyck, CH	1
Amici, LA; Baldwin, RM; Charney, DS; Fu, X; Garg, PK; Innis, RB; Seibyl, JP; Soares, JC; Staley, JK; Tan, PZ; van Dyck, CH	1
Al Tikriti, M; Baldwin, RM; Garg, P; Innis, RB; Klump, H; Ng, C; Ramsby, Q; Soufer, R; Staley, JK; Tan, PZ; Van Dyck, CH	1
Holt, DP; Huang, Y; Lopresti, BJ; Mason, NS; Mathis, CA; Price, JC	1
Gunn, RN; Holt, DP; Huang, Y; Lopresti, BJ; Mason, NS; Mathis, CA; Meltzer, CC; Price, JC; Smith, GS	1
Crossan, PJ; Frank, GK; Kaye, WH; Klump, KL; McConaha, CW; Meltzer, CC; Price, JC; Rhodes, L	1
Coenen, HH; Gaebel, W; Hamacher, K; Herzog, HR; Klimke, A; Larisch, R; Mayoral, F; Müller-Gärtner, HW; Rivas, F; Tosch, M; Vosberg, H	1
Beu, M; Coenen, HH; Estalji, S; Forutan, F; Hamacher, K; Larisch, R; Müller-Gärtner, HW; Nikolaus, S; Vosberg, H	1
Frank, GK; Greer, P; Kaye, WH; McConaha, C; Meltzer, CC; Price, JC; Skovira, K	1
Coenen, HH; Estalji, S; Gaebel, W; Hamacher, K; Henning, U; Hohlfeld, T; Klimke, A; Larisch, R; Müller-Gärtner, HW; Tosch, M; Vosberg, H	1
Epperson, CN; Fujita, M; Garg, PK; Hou, Y; Innis, RB; Kugaya, A; Seibyl, JP; Staley, JK; van Dyck, CH; Zoghbi, S	1
Adams, KH; Hasselbalch, SG; Haugbøl, S; Holm, S; Knudsen, GM; Madsen, J; Pinborg, LH; Svarer, C	1
Berga, SL; Cidis Meltzer, C; Drevets, WC; Greer, PJ; Moses-Kolko, EL; Smith, G	1
Huang, Y; Mintun, MA; Moerlein, SM; Sheline, YI; Snyder, AZ; Vlassenko, AG	1
Adams, KH; Holm, S; Knudsen, GM; Liptrot, M; Lonsdale, MN; Martiny, L; Olsen, NV; Pinborg, LH; Svarer, C	1
Adams, KH; Frøkjaer, V; Hasselbalch, SG; Haugbøl, S; Holm, S; Knudsen, GM; Madsen, K; Martiny, L; Paulson, OB; Pinborg, LH; Svarer, C	1
Bailer, UF; Barbarich, NC; Brooks-Achenbach, S; Frank, GK; Henry, SE; Kaye, WH; Mathis, CA; McConaha, CW; Meltzer, CC; Price, JC; Weissfeld, L	1
Adams, KH; Hasselbalch, SG; Holm, S; Knudsen, GM; Kristiansen, H; Paulson, OB; Pinborg, LH; Yndgaard, S	1
Barch, DM; Mintun, MA; Moerlein, SM; Sheline, YI; Snyder, AZ; Wilkins, C	1
Berga, SL; Butters, M; Drevets, WC; Greer, P; Meltzer, CC; Moses-Kolko, EL; Smith, G	1
Frøkjaer, VG; Hasselbalch, SG; Haugbøl, S; Holm, S; Knudsen, GM; Madsen, K; Paulson, OB; Pinborg, LH; Svarer, C	1
Adams, KH; Bolwig, TG; Hansen, ES; Hasselbalch, SG; Holm, S; Knudsen, GM; Pinborg, LH; Svarer, C	1
Bente, K; Boy, C; Fulton, R; Herzog, H; Hurlemann, R; Pietrzyk, U; Rota Kops, E; Stangier, I; Tellmann, L	1
Bauer, A; Boy, C; Coenen, HH; Falkai, P; Herzog, H; Hurlemann, R; Maier, W; Meyer, PT; Scherk, H; Vogeley, K; Wagner, M; Zilles, K	1
Elfving, B; Gillings, N; Knudsen, GM; Kristiansen, H; Pinborg, LH; Plenge, P	1
Coenen, HH; Hamacher, K	1
Bolwig, TG; Hansen, ES; Haugbøl, S; Knudsen, GM; Nielsen, FA; Pinborg, LH; Regeur, L; Skovgaard, LT; Svarer, C	1
Arfan, HM; Dyrby, TB; Frøkjaer, VM; Haugbøl, S; Knudsen, GM; Madsen, J; Pinborg, LH; Svarer, C	1
Bailer, UF; Becker, CR; Frank, GK; Henry, SE; Hoge, J; Kaye, WH; Mathis, CA; McConaha, CW; Meltzer, CC; Price, JC; Thornton, L; Wagner, A; Ziolko, SK	1
Fabio, A; Frank, GK; Kaye, WH; Meltzer, CC; Price, JC; Soloff, PH	1
Bauer, A; Elmenhorst, D; Herzog, H; Hurlemann, R; Matusch, A; Rota Kops, E; Winz, OH; Zilles, K	1
Adams, KH; Frokjaer, VG; Hasselbalch, SG; Haugbol, S; Holm, S; Knudsen, GM; Mortensen, EL; Nielsen, FA; Paulson, OB; Pinborg, LH; Svarer, C	1
Bauer, A; Berning, J; Elmenhorst, D; Hurlemann, R; Kolsch, H; Kuhn, KU; Maier, W; Matusch, A; Wagner, M; Winz, O; Zilles, K	1
Debus, F; Herth, MM; Knudsen, GM; Lüddens, H; Palner, M; Piel, M; Rösch, F	1
Baaré, W; Erritzoe, D; Frokjaer, VG; Glenthoj, BY; Haugbol, S; Knudsen, GM; Kristiansen, KT; Lublin, H; Madsen, J; Pinborg, L; Rasmussen, H; Svarer, C	1
Arfan, H; Frokjaer, VG; Haugbol, S; Hjelmborg, JV; Holm, S; Knudsen, GM; Kyvik, KO; Paulson, OB; Pinborg, LH; Svarer, C	1
Baaré, W; Hasselbalch, SG; Haugbøl, S; Holm, S; Knudsen, GM; Marner, L	1
Budtz-Joergensen, E; Christensen, R; Frokjaer, VG; Kehlet, H; Knudsen, GM; Kupers, R; Naert, A	1
Bauer, A; Hurlemann, R; Maier, W; Matusch, A; Reich, H; Schlaepfer, TE; Shah, NJ; Zilles, K	1
Ametamey, SM; Cservenyak, T; Hasler, F; Krasikova, RN; Kuznetsova, OF; Quednow, BB; Vollenweider, FX; Westera, G	1
Bauer, A; Eggert, KM; Elmenhorst, D; Höglinger, GU; Hurlemann, R; Matusch, A; Oertel, WH; Stamelou, M; Zilles, K	1
Erritzoe, D; Frokjaer, VG; Knudsen, GM; Madsen, J; Paulson, OB	1
Baldwin, RM; Estok, KM; Macavoy, MG; Mitsis, EM; Santhosh, L; Staley, JK; Tamagnan, GD; van Dyck, CH; Vogel, RS	1
Diksic, M; Evans, AC; Kovacevic, M; Massarweh, G; Rosa-Neto, P; Schirrmacher, R	1
Becker, C; Mason, NS; Meltzer, CC; Price, JC; Soloff, PH	1
Arfan, H; Baaré, W; Erritzoe, D; Frokjaer, VG; Holst, KK; Jernigan, TL; Kessing, LV; Knudsen, GM; Madsen, J; Mortensen, EL; Vinberg, M	1
Aggernaes, B; Andersen, R; Baaré, W; Ebdrup, BH; Erritzoe, D; Glenthoj, B; Kalbitzer, J; Knudsen, GM; Lublin, H; Madsen, J; Oranje, B; Pinborg, LH; Rasmussen, H; Svarer, C	1
Erritzoe, D; Frokjaer, VG; Holst, K; Kalbitzer, J; Knudsen, G; Licht, CL; Madsen, J; Nielsen, FA; Svarer, C	1
Erritzoe, D; Frokjaer, VG; Holst, K; Juul, A; Knudsen, GM; Madsen, J; Nielsen, FA; Paulson, OB; Svarer, C	1
Baaré, WF; Frokjaer, VG; Hasselbalch, SG; Kalbitzer, J; Knudsen, GM; Lehel, S; Madsen, K; Marner, L	1
Aggernaes, B; Baaré, WF; Ebdrup, BH; Erritzoe, D; Glenthoj, B; Kalbitzer, J; Knudsen, GM; Lublin, H; Oranje, B; Pinborg, LH; Rasmussen, H; Svarer, C	1
Herth, MM; Knudsen, GM; Kramer, V; Palner, M; Rösch, F; Santini, MA	1
Aznar, S; Baaré, W; Erritzoe, D; Haugbol, S; Klein, AB; Knudsen, GM; Madsen, J; Trajkovska, V	1
Nagatani, H; Nakata, Y; Oshima, T; Saitoh, Y; Urano, A; Yokota, M	1
Christoffersen, M; Erritzoe, D; Frokjaer, VG; Holst, KK; Jernigan, TL; Johansen, SS; Knudsen, GM; Madsen, J; Ramsøy, T; Rasmussen, PM; Svarer, C	1
Grandt, R; Hautzel, H; Herzog, H; Müller, HW	1
Aigbirhio, FI; Baron, JC; Caprioli, D; Dalley, JW; Ferrari, V; Fryer, TD; Hong, YT; Riss, PJ; Sawiak, SJ; Sitnikov, S; Williamson, D	1
Buck, A; Burger, C; Dörig, N; Hasler, F; Quednow, BB; Rentsch, KM; Schubiger, PA; Treyer, V; Vollenweider, FX; Westera, G; Wyss, MT	1
Collier, L; Dudczak, R; Karanikas, G; Lanzenberger, R; Mitterhauser, M; Richter, S; Ungersboeck, J; Wadsak, W	1
da Cunha-Bang, S; Frokjaer, VG; Holst, K; Jensen, PS; Knudsen, GM; Licht, CL; Mortensen, EL; Stenbæk, DS	1
Callado, LF; González-Maeso, J; Meana, JJ; Moreno, JL; Muguruza, C; Umali, A	1
Bauer, A; Elmenhorst, D; Kroll, T; Matusch, A	1
Dyssegaard, A; Ettrup, A; Gillings, N; Hansen, HD; Herth, MM; Knudsen, GM; Ratner, C	1
Bauer, A; Beer, S; Elmenhorst, D; Kroll, T; Matusch, A; Wedekind, F; Weisshaupt, A	1
Cano, A; Gómez-Vallejo, V; Llop, J; Martín, A; Padró, D; Plaza, S; Szczupak, B	1
Bauer, A; Beer, S; Celik, AA; Elmenhorst, D; Kroll, T; Matusch, A; Wedekind, F; Weisshaupt, A	1
Becker, C; Chiappetta, L; Mason, NS; Price, JC; Soloff, PH	1
Ebdrup, BH; Glenthøj, B; Knudsen, GM; Oranje, B; Pinborg, LH; Rasmussen, H	1
Almdal, T; Baaré, WF; Fisher, PM; Haahr, ME; Hansen, DL; Hojgaard, L; Holst, JJ; Knudsen, GM; Madsen, J; Madsen, K; Stenbæk, DS; Svarer, C	1
Beliveau, V; da Cunha-Bang, S; Dyssegaard, A; Ettrup, A; Ganz, M; Gillings, N; Jørgensen, LM; Knudsen, GM; Lehel, S; McMahon, B; Møller, K; Svarer, C	1
Anhøj, S; Frokjaer, VG; Glenthøj, B; Hilker, RW; Knudsen, GM; Madsen, J; Oranje, B; Pinborg, LH; Rasmussen, H	1
Bosmans, T; De Vos, F; Dobbeleir, A; Dockx, R; Pauwelyn, G; Peremans, K; Polis, I; Vanhove, C; Verhoeven, J; Vlerick, L	1
Higuchi, M; Ikoma, Y; Kawamura, K; Maeda, J; Nishino, A; Obata, T; Suhara, T; Takuwa, H; Zhang, MR	1

Reviews

1 review(s) available for ketanserin and altanserin

Article	Year
Positron Emission Tomography (PET) Imaging Tracers for Serotonin Receptors. Journal of medicinal chemistry, 2022, 08-25, Volume: 65, Issue:16 Topics: Brain; Humans; Ligands; Positron-Emission Tomography; Radiopharmaceuticals; Receptors, Serotonin	2022

Trials

11 trial(s) available for ketanserin and altanserin

Article	Year
Serotonin 5HT2 receptor imaging in the human brain using positron emission tomography and a new radioligand, [18F]altanserin: results in young normal controls. Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1995, Volume: 15, Issue:5 Topics: Adult; Brain; Chromatography, High Pressure Liquid; Fluorine Radioisotopes; Humans; Ketanserin; Receptors, Serotonin; Reference Values; Time Factors; Tissue Distribution; Tomography, Emission-Computed	1995
Sex difference in 5HT2 receptor in the living human brain. Neuroscience letters, 1996, Feb-02, Volume: 204, Issue:1-2 Topics: Adult; Brain Chemistry; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Middle Aged; Receptors, Serotonin; Sex Characteristics; Tomography, Emission-Computed	1996
Equilibrium modeling of 5-HT(2A) receptors with [18F]deuteroaltanserin and PET: feasibility of a constant infusion paradigm. Nuclear medicine and biology, 2000, Volume: 27, Issue:8 Topics: Adolescent; Adult; Algorithms; Brain; Deuterium; Fluorine Radioisotopes; Humans; Image Processing, Computer-Assisted; Infusions, Intravenous; Ketanserin; Male; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Tomography, Emission-Computed	2000
Influence of synaptic serotonin level on [18F]altanserin binding to 5HT2 receptors in man. Behavioural brain research, 2003, Feb-17, Volume: 139, Issue:1-2 Topics: Adult; Antidepressive Agents, Tricyclic; Brain; Clomipramine; Depressive Disorder, Major; Drug Interactions; Feasibility Studies; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Middle Aged; Receptors, Serotonin; Recurrence; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tomography, Emission-Computed	2003
Increase in prefrontal cortex serotonin 2A receptors following estrogen treatment in postmenopausal women. The American journal of psychiatry, 2003, Volume: 160, Issue:8 Topics: Administration, Cutaneous; Adult; Aged; Estradiol; Estrogen Replacement Therapy; Female; Fluorine Radioisotopes; Follow-Up Studies; Humans; Ketanserin; Middle Aged; Neuropsychological Tests; Postmenopause; Prefrontal Cortex; Psychomotor Performance; Pyramidal Cells; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Tomography, Emission-Computed; Treatment Outcome	2003
MR-based automatic delineation of volumes of interest in human brain PET images using probability maps. NeuroImage, 2005, Feb-15, Volume: 24, Issue:4 Topics: Aged; Aged, 80 and over; Aging; Algorithms; Atrophy; Brain; Brain Mapping; Cognition Disorders; Female; Humans; Image Processing, Computer-Assisted; Ketanserin; Magnetic Resonance Imaging; Male; Positron-Emission Tomography; Probability Theory; Radiopharmaceuticals; Reproducibility of Results	2005
Patients with obsessive-compulsive disorder have increased 5-HT2A receptor binding in the caudate nuclei. The international journal of neuropsychopharmacology, 2005, Volume: 8, Issue:3 Topics: Adolescent; Adult; Aged; Antidepressive Agents; Brain Mapping; Caudate Nucleus; Female; Fluorine Radioisotopes; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Middle Aged; Obsessive-Compulsive Disorder; Positron-Emission Tomography; Protein Binding; Receptor, Serotonin, 5-HT2A	2005
Acute S-ketamine application does not alter cerebral [18F]altanserin binding: a pilot PET study in humans. Journal of neural transmission (Vienna, Austria : 1996), 2007, Volume: 114, Issue:11 Topics: Adult; Algorithms; Brain; Butanols; Double-Blind Method; Excitatory Amino Acid Antagonists; Heart Rate; Humans; Image Processing, Computer-Assisted; Ketamine; Ketanserin; Male; Pilot Projects; Positron-Emission Tomography; Psychiatric Status Rating Scales	2007
Endogenous plasma estradiol in healthy men is positively correlated with cerebral cortical serotonin 2A receptor binding. Psychoneuroendocrinology, 2010, Volume: 35, Issue:9 Topics: Adult; Aged; Aged, 80 and over; Binding, Competitive; Cerebral Cortex; Estradiol; Fluorine Radioisotopes; Health; Humans; Ketanserin; Male; Middle Aged; Positron-Emission Tomography; Protein Binding; Receptor, Serotonin, 5-HT2A; Young Adult	2010
Serotonin2A receptor blockade and clinical effect in first-episode schizophrenia patients treated with quetiapine. Psychopharmacology, 2011, Volume: 213, Issue:2-3 Topics: Adult; Antipsychotic Agents; Dibenzothiazepines; Dose-Response Relationship, Drug; Female; Follow-Up Studies; Humans; Ketanserin; Longitudinal Studies; Male; Positron-Emission Tomography; Quetiapine Fumarate; Receptor, Serotonin, 5-HT2A; Schizophrenia; Schizophrenic Psychology; Time Factors; Young Adult	2011
Assessment of serotonin release capacity in the human brain using dexfenfluramine challenge and [18F]altanserin positron emission tomography. NeuroImage, 2012, Feb-15, Volume: 59, Issue:4 Topics: Adult; Brain; Dexfenfluramine; Double-Blind Method; Fluorine Radioisotopes; Humans; Ketanserin; Male; Positron-Emission Tomography; Serotonin; Serotonin Receptor Agonists; Young Adult	2012

Other Studies

77 other study(ies) available for ketanserin and altanserin

Article	Year
Fluorine-18-altanserin: a radioligand for the study of serotonin receptors with PET: radiolabeling and in vivo biologic behavior in rats. Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1991, Volume: 32, Issue:12 Topics: Animals; Female; Fluorine Radioisotopes; Isotope Labeling; Ketanserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tissue Distribution; Tomography, Emission-Computed	1991
Estimation of brain 5HT2 receptor binding potential with a single-dose PET paradigm. European journal of nuclear medicine, 1995, Volume: 22, Issue:6 Topics: Brain; Fluorine Radioisotopes; Humans; Ketanserin; Receptors, Serotonin; Tomography, Emission-Computed	1995
Serotonergic modulation of striatal dopamine measured with positron emission tomography (PET) and in vivo microdialysis. The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:1 Pt 2 Topics: Animals; Cerebellum; Citalopram; Corpus Striatum; Dopamine; Dopamine Antagonists; Female; Ketanserin; Microdialysis; Papio; Raclopride; Salicylamides; Serotonin; Tomography, Emission-Computed	1995
Multicompartmental study of fluorine-18 altanserin binding to brain 5HT2 receptors in humans using positron emission tomography. European journal of nuclear medicine, 1994, Volume: 21, Issue:9 Topics: Adult; Brain; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Receptors, Serotonin; Tomography, Emission-Computed	1994
Modulation of central cholinergic activity by GABA and serotonin: PET studies with 11C-benztropine in primates. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1993, Volume: 8, Issue:4 Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Benztropine; Brain; Carbon Radioisotopes; Female; gamma-Aminobutyric Acid; Ketanserin; Papio; Receptors, Cholinergic; Serotonin; Tomography, Emission-Computed; Vigabatrin	1993
Visualisation of loss of 5-HT2A receptors with age in healthy volunteers using [18F]altanserin and positron emission tomographic imaging. Psychiatry research, 1996, Nov-25, Volume: 68, Issue:1 Topics: Adult; Aging; Brain; Brain Mapping; Cerebral Cortex; Dominance, Cerebral; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Tomography, Emission-Computed	1996
In vivo binding of [18F]altanserin to rat brain 5HT2 receptors: a film and electronic autoradiographic study. Nuclear medicine and biology, 1997, Volume: 24, Issue:4 Topics: Animals; Autoradiography; Brain; Fluorine Radioisotopes; Ketanserin; Male; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists	1997
Serotonin 5-HT2 receptor imaging in major depression: focal changes in orbito-insular cortex. The British journal of psychiatry : the journal of mental science, 1997, Volume: 171 Topics: Brain Diseases; Depressive Disorder; Female; Humans; Ketanserin; Male; Middle Aged; Receptors, Serotonin; Serotonin Antagonists; Tomography, Emission-Computed	1997
Reduced binding of [18F]altanserin to serotonin type 2A receptors in aging: persistence of effect after partial volume correction. Brain research, 1998, Nov-30, Volume: 813, Issue:1 Topics: Adolescent; Adult; Aged; Aging; Brain; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Middle Aged; Radioligand Assay; Receptors, Serotonin	1998
Test-retest variability of serotonin 5-HT2A receptor binding measured with positron emission tomography and [18F]altanserin in the human brain. Synapse (New York, N.Y.), 1998, Volume: 30, Issue:4 Topics: Adult; Animals; Brain; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Models, Neurological; Rats; Receptors, Serotonin; Reference Values; Reproducibility of Results; Tomography, Emission-Computed	1998
A complete remote-control system for reliable preparation of [18F]altanserin. Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine, 1999, Volume: 50, Issue:5 Topics: Calibration; Chromatography, High Pressure Liquid; Fluorine Radioisotopes; Isotope Labeling; Ketanserin; Radiopharmaceuticals	1999
Characterization of radioactive metabolites of 5-HT2A receptor PET ligand [18F]altanserin in human and rodent. Nuclear medicine and biology, 1999, Volume: 26, Issue:6 Topics: Animals; Biotransformation; Brain; Female; Fluorine Radioisotopes; Humans; Ketanserin; Ovariectomy; Papio; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Tissue Distribution; Tomography, Emission-Computed	1999
PET imaging of serotonin type 2A receptors in late-life neuropsychiatric disorders. The American journal of psychiatry, 1999, Volume: 156, Issue:12 Topics: Age Factors; Aged; Alzheimer Disease; Brain; Cerebral Cortex; Depressive Disorder; Female; Fluorine Radioisotopes; Gyrus Cinguli; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Prefrontal Cortex; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Tomography, Emission-Computed	1999
PET quantification of 5-HT2A receptors in the human brain: a constant infusion paradigm with [18F]altanserin. Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2000, Volume: 41, Issue:2 Topics: Adult; Brain; Feasibility Studies; Female; Fluorine Radioisotopes; Humans; Image Processing, Computer-Assisted; Infusions, Intravenous; Ketanserin; Linear Models; Male; Receptors, Serotonin; Time Factors; Tomography, Emission-Computed	2000
Comparison of [(18)F]altanserin and [(18)F]deuteroaltanserin for PET imaging of serotonin(2A) receptors in baboon brain: pharmacological studies. Nuclear medicine and biology, 2001, Volume: 28, Issue:3 Topics: Analysis of Variance; Animals; Brain; Deuterium; Female; Fluorine Radioisotopes; Ketanserin; Papio; Radiochemistry; Receptors, Serotonin; Tomography, Emission-Computed	2001
Analyses of [(18)F] altanserin bolus injection PET data. I: consideration of radiolabeled metabolites in baboons. Synapse (New York, N.Y.), 2001, Volume: 41, Issue:1 Topics: Animals; Blood-Brain Barrier; Brain; Fluorine Radioisotopes; Ketanserin; Models, Biological; Papio; Tissue Distribution; Tomography, Emission-Computed	2001
Analyses of [(18)F]altanserin bolus injection PET data. II: consideration of radiolabeled metabolites in humans. Synapse (New York, N.Y.), 2001, Volume: 41, Issue:1 Topics: Adolescent; Adult; Aged; Blood-Brain Barrier; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Middle Aged; Models, Biological; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Tomography, Emission-Computed	2001
Altered serotonin 2A receptor activity in women who have recovered from bulimia nervosa. The American journal of psychiatry, 2001, Volume: 158, Issue:7 Topics: Adolescent; Adult; Age Factors; Age of Onset; Bulimia; Cerebral Cortex; Female; Fluorine Radioisotopes; Frontal Lobe; Humans; Ketanserin; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Tomography, Emission-Computed	2001
Disturbance of serotonin 5HT2 receptors in remitted patients suffering from hereditary depressive disorder. Nuklearmedizin. Nuclear medicine, 2001, Volume: 40, Issue:4 Topics: Adult; Aged; Aging; Brain; Cerebral Cortex; Depressive Disorder; Female; Fluorine Radioisotopes; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Middle Aged; Organ Specificity; Pedigree; Receptors, Serotonin; Reference Values; Regression Analysis; Tomography, Emission-Computed	2001
Distribution of 5HT2A receptors in the human brain: comparison of data in vivo and post mortem. Nuklearmedizin. Nuclear medicine, 2002, Volume: 41, Issue:4 Topics: Adult; Autopsy; Autoradiography; Brain; Female; Fluorine Radioisotopes; Humans; Informed Consent; Ketanserin; Male; Organ Specificity; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reference Values; Regression Analysis; Tomography, Emission-Computed	2002
Reduced 5-HT2A receptor binding after recovery from anorexia nervosa. Biological psychiatry, 2002, Nov-01, Volume: 52, Issue:9 Topics: Adult; Anorexia Nervosa; Binding, Competitive; Brain; Cerebellum; Convalescence; Female; Fluorodeoxyglucose F18; Humans; Ketanserin; Limbic System; Magnetic Resonance Imaging; Neural Pathways; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Tomography, Emission-Computed	2002
Quantification of 5-HT2A receptors in the human brain using [18F]altanserin-PET and the bolus/infusion approach. Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2003, Volume: 23, Issue:8 Topics: Adult; Aged; Brain Chemistry; Cerebellum; Fluorine Radioisotopes; Humans; Injections; Ketanserin; Middle Aged; Radiochemistry; Receptors, Serotonin; Tomography, Emission-Computed	2003
Widespread increases of cortical serotonin type 2A receptor availability after hormone therapy in euthymic postmenopausal women. Fertility and sterility, 2003, Volume: 80, Issue:3 Topics: Administration, Cutaneous; Administration, Oral; Cerebral Cortex; Drug Administration Schedule; Drug Combinations; Estradiol; Estrogen Replacement Therapy; Female; Fluorine Radioisotopes; Humans; Ketanserin; Progesterone; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Tissue Distribution; Tomography, Emission-Computed	2003
Decreased hippocampal 5-HT2A receptor binding in major depressive disorder: in vivo measurement with [18F]altanserin positron emission tomography. Biological psychiatry, 2004, Feb-01, Volume: 55, Issue:3 Topics: Adult; Age Factors; Aged; Aged, 80 and over; Case-Control Studies; Depressive Disorder, Major; Female; Fluorine Radioisotopes; Hippocampus; Humans; Ketanserin; Male; Middle Aged; Receptor, Serotonin, 5-HT2A; Tomography, Emission-Computed	2004
Cluster analysis in kinetic modelling of the brain: a noninvasive alternative to arterial sampling. NeuroImage, 2004, Volume: 21, Issue:2 Topics: Adult; Aged; Blood Flow Velocity; Blood Specimen Collection; Blood-Brain Barrier; Brain; Cerebellum; Cerebral Cortex; Cluster Analysis; Energy Metabolism; Female; Fluorine Radioisotopes; Humans; Image Processing, Computer-Assisted; Imaging, Three-Dimensional; Ketanserin; Kinetics; Male; Mathematical Computing; Middle Aged; Models, Neurological; Models, Statistical; Reference Values; Regional Blood Flow; Reproducibility of Results; Thalamus; Tomography, Emission-Computed	2004
A database of [(18)F]-altanserin binding to 5-HT(2A) receptors in normal volunteers: normative data and relationship to physiological and demographic variables. NeuroImage, 2004, Volume: 21, Issue:3 Topics: Adult; Aged; Aging; Blood Proteins; Body Mass Index; Brain; Databases, Factual; Female; Fluorine Radioisotopes; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Middle Aged; Models, Neurological; Protein Binding; Receptor, Serotonin, 5-HT2A; Reference Values; Serotonin Antagonists; Sex Characteristics; Tomography, Emission-Computed	2004
Altered 5-HT(2A) receptor binding after recovery from bulimia-type anorexia nervosa: relationships to harm avoidance and drive for thinness. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2004, Volume: 29, Issue:6 Topics: Adult; Age Factors; Anorexia Nervosa; Brain; Brain Mapping; Bulimia; Drive; Female; Fluorine Radioisotopes; Harm Reduction; Humans; Ketanserin; Protein Binding; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Thinness; Time Factors; Tomography, Emission-Computed	2004
[18F]altanserin binding to human 5HT2A receptors is unaltered after citalopram and pindolol challenge. Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2004, Volume: 24, Issue:9 Topics: Adrenergic beta-Antagonists; Adult; Brain; Citalopram; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Pindolol; Prolactin; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Tomography, Emission-Computed	2004
Decreased hippocampal 5-HT(2A) receptor binding in older depressed patients using [18F]altanserin positron emission tomography. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2004, Volume: 29, Issue:12 Topics: Aged; Aged, 80 and over; Brain Mapping; Case-Control Studies; Depressive Disorder; Female; Fluorine Radioisotopes; Hippocampus; Humans; Ketanserin; Male; Middle Aged; Positron-Emission Tomography; Protein Binding; Receptor, Serotonin, 5-HT2A	2004
Estradiol effects on the postmenopausal brain. The American journal of psychiatry, 2004, Volume: 161, Issue:11 Topics: Administration, Cutaneous; Brain; Brain Mapping; Estradiol; Estrogen Replacement Therapy; Female; Fluorine Radioisotopes; Humans; Ketanserin; Positron-Emission Tomography; Postmenopause; Receptor, Serotonin, 5-HT2A	2004
Motion artifact reduction on parametric PET images of neuroreceptor binding. Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2005, Volume: 46, Issue:6 Topics: Artifacts; Brain; Fluorine Radioisotopes; Head Movements; Humans; Image Processing, Computer-Assisted; Ketanserin; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A	2005
Decreased prefrontal 5-HT2A receptor binding in subjects at enhanced risk for schizophrenia. Anatomy and embryology, 2005, Volume: 210, Issue:5-6 Topics: Adult; Brain Mapping; Case-Control Studies; Female; Fluorine Radioisotopes; Humans; Image Processing, Computer-Assisted; Ketanserin; Magnetic Resonance Imaging; Male; Pilot Projects; Positron-Emission Tomography; Prefrontal Cortex; Receptor, Serotonin, 5-HT2A; Risk Factors; Schizophrenia	2005
Binding characteristics of the 5-HT2A receptor antagonists altanserin and MDL 100907. Synapse (New York, N.Y.), 2005, Dec-15, Volume: 58, Issue:4 Topics: Animals; Binding, Competitive; Brain; Carbon Radioisotopes; Fluorine Radioisotopes; Fluorobenzenes; Ketanserin; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists	2005
No-carrier-added nucleophilic 18F-labelling in an electrochemical cell exemplified by the routine production of [18F]altanserin. Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine, 2006, Volume: 64, Issue:9 Topics: Chromatography, High Pressure Liquid; Electrochemistry; Fluorine Radioisotopes; Isotope Labeling; Ketanserin	2006
Cerebral 5-HT2A receptor binding is increased in patients with Tourette's syndrome. The international journal of neuropsychopharmacology, 2007, Volume: 10, Issue:2 Topics: Adolescent; Adult; Brain Chemistry; Female; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Middle Aged; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Tics; Tourette Syndrome	2007
Reproducibility of 5-HT2A receptor measurements and sample size estimations with [18F]altanserin PET using a bolus/infusion approach. European journal of nuclear medicine and molecular imaging, 2007, Volume: 34, Issue:6 Topics: Adolescent; Adult; Aged; Brain; Fluorine Radioisotopes; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Middle Aged; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Reproducibility of Results; Research Design	2007
Exaggerated 5-HT1A but normal 5-HT2A receptor activity in individuals ill with anorexia nervosa. Biological psychiatry, 2007, May-01, Volume: 61, Issue:9 Topics: Adult; Anorexia Nervosa; Cerebrovascular Circulation; Data Interpretation, Statistical; Female; Humans; Ketanserin; Magnetic Resonance Imaging; Oxygen Radioisotopes; Piperazines; Positron-Emission Tomography; Pyridines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists	2007
5HT2A receptor binding is increased in borderline personality disorder. Biological psychiatry, 2007, Sep-15, Volume: 62, Issue:6 Topics: Adult; Aggression; Borderline Personality Disorder; Brain; Child; Child Abuse; Depression; Female; Fluorodeoxyglucose F18; Frontal Lobe; Hippocampus; Humans; Impulsive Behavior; Ketanserin; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Risk Factors; Suicide	2007
Frontolimbic serotonin 2A receptor binding in healthy subjects is associated with personality risk factors for affective disorder. Biological psychiatry, 2008, Mar-15, Volume: 63, Issue:6 Topics: Adolescent; Adult; Aged; Biomarkers; Character; Depressive Disorder, Major; Dominance, Cerebral; Female; Fluorine Radioisotopes; Frontal Lobe; Gyrus Cinguli; Humans; Image Processing, Computer-Assisted; Ketanserin; Limbic System; Magnetic Resonance Imaging; Male; Middle Aged; Neurotic Disorders; Personality Inventory; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Reference Values; Risk Factors; Statistics as Topic; Temporal Lobe	2008
5-HT2A receptor density is decreased in the at-risk mental state. Psychopharmacology, 2008, Volume: 195, Issue:4 Topics: Adult; Brain; Brain Mapping; Cerebral Cortex; Dominance, Cerebral; Early Diagnosis; Female; Fluorine Radioisotopes; Genetic Markers; Genetic Predisposition to Disease; Genotype; Humans; Ketanserin; Male; Positron-Emission Tomography; Psychiatric Status Rating Scales; Receptor, Serotonin, 5-HT2A; Schizophrenia; Schizotypal Personality Disorder	2008
Total synthesis and evaluation of [18F]MHMZ. Bioorganic & medicinal chemistry letters, 2008, Feb-15, Volume: 18, Issue:4 Topics: Animals; Binding, Competitive; Brain; Fluorine Radioisotopes; Fluorobenzenes; Isotope Labeling; Ketanserin; Kinetics; Piperidines; Radioligand Assay; Radionuclide Imaging; Radiopharmaceuticals; Rats; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists	2008
Cortical and subcortical 5-HT2A receptor binding in neuroleptic-naive first-episode schizophrenic patients. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2008, Volume: 33, Issue:10 Topics: Adult; Antipsychotic Agents; Binding, Competitive; Brain; Brain Chemistry; Brain Mapping; Caudate Nucleus; Cerebral Cortex; Female; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin; Serotonin Antagonists; Young Adult	2008
The 5-HT2A receptor binding pattern in the human brain is strongly genetically determined. NeuroImage, 2008, Apr-15, Volume: 40, Issue:3 Topics: Adult; Analysis of Variance; Brain; Brain Chemistry; Humans; Isotope Labeling; Ketanserin; Magnetic Resonance Imaging; Male; Middle Aged; Radionuclide Imaging; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Twins, Dizygotic; Twins, Monozygotic	2008
Longitudinal assessment of cerebral 5-HT2A receptors in healthy elderly volunteers: an [18F]-altanserin PET study. European journal of nuclear medicine and molecular imaging, 2009, Volume: 36, Issue:2 Topics: Aged; Cerebrum; Female; Fluorine Radioisotopes; Health; Humans; Ketanserin; Longitudinal Studies; Male; Middle Aged; Observer Variation; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Reproducibility of Results	2009
A PET [18F]altanserin study of 5-HT2A receptor binding in the human brain and responses to painful heat stimulation. NeuroImage, 2009, Feb-01, Volume: 44, Issue:3 Topics: Adult; Binding Sites; Brain; Female; Fluorine Radioisotopes; Hot Temperature; Humans; Ketanserin; Male; Pain; Pain Threshold; Positron-Emission Tomography; Protein Binding; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Tissue Distribution	2009
Reduced 5-HT(2A) receptor signaling following selective bilateral amygdala damage. Social cognitive and affective neuroscience, 2009, Volume: 4, Issue:1 Topics: Adult; Amygdala; Fluorine Radioisotopes; Humans; Image Processing, Computer-Assisted; Ketanserin; Lipoid Proteinosis of Urbach and Wiethe; Magnetic Resonance Imaging; Male; Neuropsychological Tests; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Serotonin; Synaptic Transmission	2009
GMP-compliant radiosynthesis of [18F]altanserin and human plasma metabolite studies. Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine, 2009, Volume: 67, Issue:4 Topics: Chromatography, High Pressure Liquid; Fluorine Radioisotopes; Humans; Ketanserin; Positron-Emission Tomography; Quality Control	2009
Nigrostriatal upregulation of 5-HT2A receptors correlates with motor dysfunction in progressive supranuclear palsy. Movement disorders : official journal of the Movement Disorder Society, 2009, Jun-15, Volume: 24, Issue:8 Topics: Aged; Brain Mapping; Corpus Striatum; Female; Fluorine Radioisotopes; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Middle Aged; Movement Disorders; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Statistics as Topic; Substantia Nigra; Supranuclear Palsy, Progressive; Up-Regulation	2009
Gender and the use of hormonal contraception in women are not associated with cerebral cortical 5-HT 2A receptor binding. Neuroscience, 2009, Oct-06, Volume: 163, Issue:2 Topics: Adolescent; Adult; Aged; Cerebral Cortex; Contraceptives, Oral, Hormonal; Female; Humans; Ketanserin; Linear Models; Magnetic Resonance Imaging; Male; Middle Aged; Personality; Personality Assessment; Positron-Emission Tomography; Protein Binding; Receptor, Serotonin, 5-HT2A; Sex Characteristics; Young Adult	2009
Regional distribution and behavioral correlates of 5-HT(2A) receptors in Alzheimer's disease with [(18)F]deuteroaltanserin and PET. Psychiatry research, 2009, Sep-30, Volume: 173, Issue:3 Topics: Aged; Aged, 80 and over; Alzheimer Disease; Analysis of Variance; Brain; Brain Mapping; Brief Psychiatric Rating Scale; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Middle Aged; Positron-Emission Tomography; Protein Binding; Receptor, Serotonin, 5-HT2A	2009
Time-efficient and convenient synthesis of [(18)F]altanserin for human PET imaging by a new work-up procedure. Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine, 2009, Volume: 67, Issue:11 Topics: Animals; Brain; Fluorine Radioisotopes; Humans; Isotope Labeling; Ketanserin; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Time Factors	2009
Gender, personality, and serotonin-2A receptor binding in healthy subjects. Psychiatry research, 2010, Jan-30, Volume: 181, Issue:1 Topics: Adolescent; Adult; Aggression; Brain; Brain Mapping; Female; Health Status; Humans; Impulsive Behavior; Ketanserin; Male; Middle Aged; Personality; Personality Tests; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Sex Characteristics; Temperament; Young Adult	2010
Familial risk for mood disorder and the personality risk factor, neuroticism, interact in their association with frontolimbic serotonin 2A receptor binding. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2010, Volume: 35, Issue:5 Topics: Adult; Family; Female; Frontal Lobe; Genetic Predisposition to Disease; Humans; Ketanserin; Limbic System; Male; Middle Aged; Mood Disorders; Personality; Personality Tests; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Risk Factors; Sex Factors; Surveys and Questionnaires; Twins; Young Adult	2010
Decreased frontal serotonin2A receptor binding in antipsychotic-naive patients with first-episode schizophrenia. Archives of general psychiatry, 2010, Volume: 67, Issue:1 Topics: Adult; Antipsychotic Agents; Brain; Case-Control Studies; Female; Fluorine Radioisotopes; Frontal Lobe; Humans; Ketanserin; Male; Neuropsychological Tests; Radionuclide Imaging; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin	2010
A nonlinear relationship between cerebral serotonin transporter and 5-HT(2A) receptor binding: an in vivo molecular imaging study in humans. The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Mar-03, Volume: 30, Issue:9 Topics: Adult; Aged; Aged, 80 and over; Benzylamines; Binding, Competitive; Brain Chemistry; Brain Mapping; Cerebral Cortex; Computer Simulation; Female; Humans; Ketanserin; Male; Middle Aged; Positron-Emission Tomography; Radioisotopes; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Plasma Membrane Transport Proteins; Synaptic Transmission; Young Adult	2010
Loss of serotonin 2A receptors exceeds loss of serotonergic projections in early Alzheimer's disease: a combined [11C]DASB and [18F]altanserin-PET study. Neurobiology of aging, 2012, Volume: 33, Issue:3 Topics: Aged; Aged, 80 and over; Alzheimer Disease; Benzylamines; Carbon Radioisotopes; Cerebral Cortex; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Neural Pathways; Positron-Emission Tomography; Raphe Nuclei; Receptor, Serotonin, 5-HT2A; Serotonergic Neurons	2012
Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode. Chemical biology & drug design, 2010, Volume: 76, Issue:4 Topics: Binding, Competitive; Combinatorial Chemistry Techniques; Fluorobenzenes; Hydrophobic and Hydrophilic Interactions; Ketanserin; Ligands; Phenols; Piperidines; Protein Binding; Pyridines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists	2010
Cerebral 5-HT2A receptor and serotonin transporter binding in humans are not affected by the val66met BDNF polymorphism status or blood BDNF levels. Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2010, Volume: 30, Issue:11 Topics: Adolescent; Adult; Aged; Aged, 80 and over; Alleles; Benzylamines; Brain; Brain-Derived Neurotrophic Factor; Cohort Studies; Female; Fluorine Radioisotopes; Genotype; Heterozygote; Humans; Ketanserin; Magnetic Resonance Imaging; Male; Methionine; Middle Aged; Neocortex; Polymorphism, Genetic; Polymorphism, Single Nucleotide; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Reference Values; Serotonin; Serotonin Plasma Membrane Transport Proteins; Valine; Young Adult	2010
Blockade of 5-HT(2A) and/or 5-HT(2C) receptors modulates sevoflurane-induced immobility. Journal of anesthesia, 2011, Volume: 25, Issue:2 Topics: Anesthetics, Inhalation; Animals; Immobilization; Indoles; Ketanserin; Male; Methyl Ethers; Pyridines; Rats; Rats, Wistar; Serotonin 5-HT2 Receptor Antagonists; Sevoflurane	2011
In vivo imaging of cerebral serotonin transporter and serotonin(2A) receptor binding in 3,4-methylenedioxymethamphetamine (MDMA or "ecstasy") and hallucinogen users. Archives of general psychiatry, 2011, Volume: 68, Issue:6 Topics: Adult; Amphetamine-Related Disorders; Aniline Compounds; Brain; Case-Control Studies; Cross-Sectional Studies; Female; Fluorine Radioisotopes; Hallucinogens; Humans; Ketanserin; Male; N-Methyl-3,4-methylenedioxyamphetamine; Positron-Emission Tomography; Protein Binding; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Serotonin Plasma Membrane Transport Proteins; Sulfides	2011
Cognition-induced modulation of serotonin in the orbitofrontal cortex: a controlled cross-over PET study of a delayed match-to-sample task using the 5-HT2a receptor antagonist [18F]altanserin. NeuroImage, 2011, Oct-01, Volume: 58, Issue:3 Topics: Brain Mapping; Cognition; Cross-Over Studies; Fluorine Radioisotopes; Frontal Lobe; Humans; Ketanserin; Male; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin 5-HT2 Receptor Antagonists	2011
Validation and quantification of [18F]altanserin binding in the rat brain using blood input and reference tissue modeling. Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2011, Volume: 31, Issue:12 Topics: Animals; Brain; Cerebellum; Cerebrovascular Circulation; Chromatography, High Pressure Liquid; Fluorine Radioisotopes; Ketanserin; Models, Biological; Positron-Emission Tomography; Protein Binding; Quality Control; Radiopharmaceuticals; Rats; Receptor, Serotonin, 5-HT2A; Reference Standards	2011
Radiolabeling of [18F]altanserin - a microfluidic approach. Nuclear medicine and biology, 2012, Volume: 39, Issue:7 Topics: Fluorine Radioisotopes; Isotope Labeling; Ketanserin; Microfluidic Analytical Techniques; Radiochemistry; Temperature	2012
Trait aggression and trait impulsivity are not related to frontal cortex 5-HT2A receptor binding in healthy individuals. Psychiatry research, 2013, May-30, Volume: 212, Issue:2 Topics: Adult; Age Factors; Aged; Aged, 80 and over; Aggression; Female; Fluorodeoxyglucose F18; Frontal Lobe; Hormones; Humans; Impulsive Behavior; Ketanserin; Male; Middle Aged; Personality; Personality Inventory; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Statistics, Nonparametric; Young Adult	2013
Dysregulated 5-HT(2A) receptor binding in postmortem frontal cortex of schizophrenic subjects. European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2013, Volume: 23, Issue:8 Topics: Amphetamines; Animals; Antipsychotic Agents; Diagnostic and Statistical Manual of Mental Disorders; Frontal Lobe; Humans; Ketanserin; Mice; Mice, Knockout; Nerve Tissue Proteins; Neurons; Prefrontal Cortex; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin Antagonists; Serotonin Receptor Agonists; Suicide; Up-Regulation	2013
Sleep deprivation increases cerebral serotonin 2A receptor binding in humans. Sleep, 2012, Dec-01, Volume: 35, Issue:12 Topics: Adult; Brain; Case-Control Studies; Electroencephalography; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Middle Aged; Positron-Emission Tomography; Psychomotor Performance; Receptor, Serotonin, 5-HT2A; Sleep Deprivation; Time Factors	2012
Direct comparison of [(18) F]MH.MZ and [(18) F] altanserin for 5-HT2A receptor imaging with PET. Synapse (New York, N.Y.), 2013, Volume: 67, Issue:6 Topics: Animals; Brain; Fluorine Radioisotopes; Fluorobenzenes; Ketanserin; Piperidines; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Swine; Tissue Distribution; Tritium	2013
Suitability of [18F]altanserin and PET to determine 5-HT2A receptor availability in the rat brain: in vivo and in vitro validation of invasive and non-invasive kinetic models. Molecular imaging and biology, 2013, Volume: 15, Issue:4 Topics: Animals; Brain; Cerebral Arteries; Fluorine Radioisotopes; Ketanserin; Kinetics; Male; Models, Biological; Positron-Emission Tomography; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Regression Analysis; Time Factors; Tissue Distribution	2013
PET imaging of serotoninergic neurotransmission with [(11)C]DASB and [(18)F]altanserin after focal cerebral ischemia in rats. Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2013, Volume: 33, Issue:12 Topics: Animals; Benzylamines; Brain; Brain Ischemia; Carbon Radioisotopes; Contrast Media; Fluorine Radioisotopes; Infarction, Middle Cerebral Artery; Ketanserin; Positron-Emission Tomography; Rats; Serotonin; Serotonin Plasma Membrane Transport Proteins; Synaptic Transmission	2013
[¹⁸F]Altanserin and small animal PET: impact of multidrug efflux transporters on ligand brain uptake and subsequent quantification of 5-HT₂A receptor densities in the rat brain. Nuclear medicine and biology, 2014, Volume: 41, Issue:1 Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Blood-Brain Barrier; Brain; Cyclosporine; Fluorine Radioisotopes; Ketanserin; Ligands; Positron-Emission Tomography; Protein Transport; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A	2014
Effects of serotonin-2A receptor binding and gender on personality traits and suicidal behavior in borderline personality disorder. Psychiatry research, 2014, Jun-30, Volume: 222, Issue:3 Topics: Adult; Aggression; Borderline Personality Disorder; Contrast Media; Depression; Female; Fluorodeoxyglucose F18; Humans; Impulsive Behavior; Ketanserin; Male; Personality; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Sex Factors; Suicidal Ideation; Suicide, Attempted; Temperament	2014
Neocortical serotonin2A receptor binding predicts quetiapine associated weight gain in antipsychotic-naive first-episode schizophrenia patients. The international journal of neuropsychopharmacology, 2014, Volume: 17, Issue:11 Topics: Adult; Antipsychotic Agents; Body Mass Index; Dibenzothiazepines; Female; Follow-Up Studies; Humans; Imaging, Three-Dimensional; Ketanserin; Male; Neocortex; Positron-Emission Tomography; Predictive Value of Tests; Protein Binding; Quetiapine Fumarate; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin Antagonists; Weight Gain; Young Adult	2014
Central 5-HT neurotransmission modulates weight loss following gastric bypass surgery in obese individuals. The Journal of neuroscience : the official journal of the Society for Neuroscience, 2015, Apr-08, Volume: 35, Issue:14 Topics: Adult; Body Mass Index; Brain; Brain Mapping; Case-Control Studies; Denmark; Female; Gastric Bypass; Glucagon-Like Peptide 1; Humans; Ketanserin; Male; Middle Aged; Obesity; Protein Binding; Radionuclide Imaging; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Time Factors; Treatment Outcome; Weight Loss	2015
Serotonin 2A receptor agonist binding in the human brain with [(11)C]Cimbi-36: Test-retest reproducibility and head-to-head comparison with the antagonist [(18)F]altanserin. NeuroImage, 2016, Apr-15, Volume: 130 Topics: Benzylamines; Brain; Carbon Radioisotopes; Female; Fluorine Radioisotopes; Humans; Ketanserin; Male; Neuroimaging; Phenethylamines; Positron-Emission Tomography; Radiopharmaceuticals; Reproducibility of Results; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Young Adult	2016
Low frontal serotonin 2A receptor binding is a state marker for schizophrenia? European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2016, Volume: 26, Issue:7 Topics: Adolescent; Adult; Antipsychotic Agents; Female; Fluorine Radioisotopes; Frontal Lobe; Humans; Ketanserin; Male; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Schizophrenia; Twins, Monozygotic; Young Adult	2016
Kinetic analysis of [ BMC veterinary research, 2019, Nov-21, Volume: 15, Issue:1 Topics: Animals; Brain; Dogs; Female; Fluorine Radioisotopes; Ketanserin; Models, Biological; Positron-Emission Tomography; Serotonin Antagonists	2019
Measurement of changes in endogenous serotonin level by positron emission tomography with [ Annals of nuclear medicine, 2021, Volume: 35, Issue:8 Topics: Animals; Brain; Ketanserin; Male; Mice; Positron-Emission Tomography; Serotonin	2021