ketanserin and alfentanil

ketanserin has been researched along with alfentanil in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19902 (25.00)18.7374
1990's1 (12.50)18.2507
2000's2 (25.00)29.6817
2010's3 (37.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Arroyo, JL; Carrasco, MS; De Castro, J; Esteban, J; Sanchez, G1
Cline, EJ; Koob, GF; Smith, NT; Weinger, MB1
Chen, DY; Koob, GF; Lau, C; Lin, T; Smith, NT; Weinger, MB1

Other Studies

8 other study(ies) available for ketanserin and alfentanil

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
[Endocrine and metabolic changes induced in surgery by the combination of ketanserin and alfentanyl].
    Agressologie: revue internationale de physio-biologie et de pharmacologie appliquees aux effets de l'agression, 1985, Volume: 26, Issue:7

    Topics: Abdomen; Adolescent; Adult; Aged; Alfentanil; Analgesics, Opioid; Drug Therapy, Combination; Female; Fentanyl; Humans; Intraoperative Complications; Ketanserin; Male; Middle Aged; Piperidines; Premedication; Serotonin Antagonists; Stress, Physiological

1985
Ketanserin pretreatment reverses alfentanil-induced muscle rigidity.
    Anesthesiology, 1987, Volume: 67, Issue:3

    Topics: Adjuvants, Anesthesia; Alfentanil; Animals; Fentanyl; Ketanserin; Male; Muscle Rigidity; Preanesthetic Medication; Rats

1987
A role for CNS alpha-2 adrenergic receptors in opiate-induced muscle rigidity in the rat.
    Brain research, 1995, Jan-09, Volume: 669, Issue:1

    Topics: Adrenergic alpha-Agonists; Alfentanil; Animals; Electromyography; Hindlimb; Imidazoles; Ketanserin; Male; Medetomidine; Muscle Rigidity; Naloxone; Narcotics; Quaternary Ammonium Compounds; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2

1995