Page last updated: 2024-09-03

kelatorphan and u-50488

kelatorphan has been researched along with u-50488 in 1 studies

Compound Research Comparison

Studies
(kelatorphan)
Trials
(kelatorphan)
Recent Studies (post-2010)
(kelatorphan)
Studies
(u-50488)
Trials
(u-50488)
Recent Studies (post-2010) (u-50488)
58011,6643209

Protein Interaction Comparison

ProteinTaxonomykelatorphan (IC50)u-50488 (IC50)
Delta-type opioid receptorRattus norvegicus (Norway rat)2.15
Kappa-type opioid receptorMus musculus (house mouse)0.0027
Mu-type opioid receptorRattus norvegicus (Norway rat)2.15
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.7171
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.0958
Kappa-type opioid receptorHomo sapiens (human)0.0537

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baghdoyan, HA; Cronin, A; Keifer, JC; Lydic, R1

Other Studies

1 other study(ies) available for kelatorphan and u-50488

ArticleYear
Opioid inhibition of rapid eye movement sleep by a specific mu receptor agonist.
    British journal of anaesthesia, 1995, Volume: 74, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cats; Dipeptides; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Neprilysin; Pyrrolidines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Respiration; Reticular Formation; Sleep, REM; Wakefulness

1995