kelatorphan has been researched along with sulpiride in 1 studies
Studies (kelatorphan) | Trials (kelatorphan) | Recent Studies (post-2010) (kelatorphan) | Studies (sulpiride) | Trials (sulpiride) | Recent Studies (post-2010) (sulpiride) |
---|---|---|---|---|---|
58 | 0 | 1 | 4,152 | 427 | 635 |
Protein | Taxonomy | kelatorphan (IC50) | sulpiride (IC50) |
---|---|---|---|
Carbonic anhydrase 1 | Homo sapiens (human) | 1.2 | |
Carbonic anhydrase 2 | Homo sapiens (human) | 0.04 | |
Alpha-2A adrenergic receptor | Homo sapiens (human) | 2.019 | |
D(2) dopamine receptor | Homo sapiens (human) | 0.0858 | |
D(3) dopamine receptor | Homo sapiens (human) | 0.2651 | |
D(2) dopamine receptor | Rattus norvegicus (Norway rat) | 0.2215 | |
Carbonic anhydrase 4 | Bos taurus (cattle) | 0.62 | |
D(2) dopamine receptor | Canis lupus familiaris (dog) | 0.2 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Daugé, V; Feger, J; Maldonado, R; Roques, BP | 1 |
1 other study(ies) available for kelatorphan and sulpiride
Article | Year |
---|---|
Chronic blockade of D2 but not D1 dopamine receptors facilitates behavioural responses to endogenous enkephalins, protected by kelatorphan, administered in the accumbens in rats.
Topics: Animals; Behavior, Animal; Benzazepines; Dipeptides; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalins; Haloperidol; Injections; Male; Motor Activity; Narcotic Antagonists; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Opioid; Receptors, Opioid, delta; Sulpiride | 1990 |