Page last updated: 2024-09-03

kelatorphan and substance p

kelatorphan has been researched along with substance p in 3 studies

Compound Research Comparison

Studies
(kelatorphan)
Trials
(kelatorphan)
Recent Studies (post-2010)
(kelatorphan)
Studies
(substance p)
Trials
(substance p)
Recent Studies (post-2010) (substance p)
580117,2892772,010

Protein Interaction Comparison

ProteinTaxonomykelatorphan (IC50)substance p (IC50)
Substance-P receptorRattus norvegicus (Norway rat)0.0005
Substance-K receptorRattus norvegicus (Norway rat)0.2
Substance-K receptorHomo sapiens (human)0.2455
Substance-P receptorHomo sapiens (human)0.0011
Neuromedin-K receptorHomo sapiens (human)0.125
Substance-K receptorMesocricetus auratus (golden hamster)0.148

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19901 (33.33)18.7374
1990's2 (66.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Duggan, AW; Hope, PJ; Lang, CW; Schaible, HG1
Benoliel, JJ; Berthier, JL; Bourgoin, S; Cesselin, F; Hamon, M; Hirsch, M; Mauborgne, A1
Cavero, I; Fardin, V; Floch, A1

Other Studies

3 other study(ies) available for kelatorphan and substance p

ArticleYear
Effect of peptidase inhibition on the pattern of intraspinally released immunoreactive substance P detected with antibody microprobes.
    Brain research, 1992, May-08, Volume: 579, Issue:2

    Topics: Analgesics; Animals; Cats; Decerebrate State; Dipeptides; Electric Stimulation; Enalaprilat; Physical Stimulation; Protease Inhibitors; Spinal Cord; Substance P

1992
Enkephalinase is involved in the degradation of endogenous substance P released from slices of rat substantia nigra.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:2

    Topics: Animals; Captopril; Dipeptides; In Vitro Techniques; Leucine; Male; Metalloendopeptidases; Naloxone; Neprilysin; Oligopeptides; Peptidyl-Dipeptidase A; Potassium; Protease Inhibitors; Rats; Rats, Inbred Strains; Substance P; Substantia Nigra; Thiorphan; Tiopronin

1987
Characterization of NK1 and NK2 tachykinin receptors in guinea-pig and rat bronchopulmonary and vascular systems.
    British journal of pharmacology, 1994, Volume: 111, Issue:3

    Topics: Animals; Binding Sites; Blood Vessels; Bronchi; Dipeptides; Glycopeptides; Guinea Pigs; Lung; Male; Neprilysin; Neurokinin A; Pulmonary Circulation; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Tachykinins; Tritium

1994