Page last updated: 2024-09-03

kelatorphan and phosphoramidon

kelatorphan has been researched along with phosphoramidon in 5 studies

Compound Research Comparison

Studies
(kelatorphan)
Trials
(kelatorphan)
Recent Studies (post-2010)
(kelatorphan)
Studies
(phosphoramidon)
Trials
(phosphoramidon)
Recent Studies (post-2010) (phosphoramidon)
58017811233

Protein Interaction Comparison

ProteinTaxonomykelatorphan (IC50)phosphoramidon (IC50)
ThermolysinBacillus thermoproteolyticus0.033
NeprilysinRattus norvegicus (Norway rat)0.0578
NeprilysinOryctolagus cuniculus (rabbit)0.0028
NeprilysinHomo sapiens (human)0.0405
Angiotensin-converting enzyme Homo sapiens (human)0.615
Endothelin-converting enzyme 1Homo sapiens (human)1.0695
P2Y purinoceptor 12Homo sapiens (human)0.017

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19901 (20.00)18.7374
1990's3 (60.00)18.2507
2000's0 (0.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bihovsky, R; Erhardt, PW; Levinson, BL; Loewi, RC; Polokoff, MA1
Devi, LA; FourniƩ-Zaluski, MC; Gagnidze, K; Orng, SV; Ouimet, T; Poras, H; Roques, BP1
Arock, M; Devillier, P; Gros, C; Guillosson, JJ; Schwartz, JC1
Cavero, I; Fardin, V; Floch, A1
Kojima, T; Matsumura, Y; Morimoto, S; Murakami, A; Murata, S; Takada, K; Takaoka, M; Tsukahara, Y1

Other Studies

5 other study(ies) available for kelatorphan and phosphoramidon

ArticleYear
Hydroxamic acids as potent inhibitors of endothelin-converting enzyme from human bronchiolar smooth muscle.
    Journal of medicinal chemistry, 1995, Jun-09, Volume: 38, Issue:12

    Topics: Aspartic Acid Endopeptidases; Bronchi; Cells, Cultured; Endothelin-Converting Enzymes; Humans; Hydroxamic Acids; Metalloendopeptidases; Muscle, Smooth

1995
Identification of an endothelin-converting enzyme-2-specific fluorigenic substrate and development of an in vitro and ex vivo enzymatic assay.
    The Journal of biological chemistry, 2010, Nov-05, Volume: 285, Issue:45

    Topics: Animals; Aspartic Acid Endopeptidases; Endothelin-Converting Enzymes; Endothelins; Enzyme Assays; Enzyme Inhibitors; Fluorescent Dyes; Gene Expression Regulation, Enzymologic; Humans; Metalloendopeptidases; Mice; Organ Specificity; Peptide Library; Peptides; Substrate Specificity

2010
Characterisation of enkephalinase (EC 3.4.24.11) activity on various leukemic cells expressing the common acute lymphocytic leukemia antigen (CALLA).
    FEBS letters, 1989, May-08, Volume: 248, Issue:1-2

    Topics: Antigens, Differentiation; Antigens, Neoplasm; Bone Marrow; Cell Division; Cell Line; Cell Membrane; Dipeptides; Glycopeptides; Humans; In Vitro Techniques; Neprilysin; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Thiorphan; Tumor Cells, Cultured

1989
Characterization of NK1 and NK2 tachykinin receptors in guinea-pig and rat bronchopulmonary and vascular systems.
    British journal of pharmacology, 1994, Volume: 111, Issue:3

    Topics: Animals; Binding Sites; Blood Vessels; Bronchi; Dipeptides; Glycopeptides; Guinea Pigs; Lung; Male; Neprilysin; Neurokinin A; Pulmonary Circulation; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Tachykinins; Tritium

1994
Effects of phosphoramidon on endothelin-1 and big endothelin-1 production in human aortic endothelial cells.
    Biological & pharmaceutical bulletin, 1995, Volume: 18, Issue:3

    Topics: Analgesics; Aorta; Aspartic Acid Endopeptidases; Cell Membrane; Cells, Cultured; Dipeptides; Endothelin-1; Endothelin-Converting Enzymes; Endothelins; Endothelium, Vascular; Glycopeptides; Humans; Metalloendopeptidases; Protein Precursors; RNA, Messenger; Sensitivity and Specificity; Stimulation, Chemical

1995