Page last updated: 2024-09-03

kelatorphan and actinonin

kelatorphan has been researched along with actinonin in 2 studies

Compound Research Comparison

Studies
(kelatorphan)
Trials
(kelatorphan)
Recent Studies (post-2010)
(kelatorphan)
Studies
(actinonin)
Trials
(actinonin)
Recent Studies (post-2010) (actinonin)
5801166057

Protein Interaction Comparison

ProteinTaxonomykelatorphan (IC50)actinonin (IC50)
Urokinase-type plasminogen activatorHomo sapiens (human)0.14
Interstitial collagenaseHomo sapiens (human)1.1
NeprilysinOryctolagus cuniculus (rabbit)8.2
72 kDa type IV collagenaseHomo sapiens (human)3
Stromelysin-1Homo sapiens (human)6
NeprilysinHomo sapiens (human)6.7
Aminopeptidase NHomo sapiens (human)0.4
Peptide deformylaseStaphylococcus aureus subsp. aureus Mu500.005
Peptide deformylaseStaphylococcus aureus0.02
Peptide deformylase 1A, chloroplastic/mitochondrialArabidopsis thaliana (thale cress)0.027
Peptide deformylase, mitochondrialHomo sapiens (human)0.5622
Peptide deformylase Escherichia coli0.052

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19901 (50.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bihovsky, R; Erhardt, PW; Levinson, BL; Loewi, RC; Polokoff, MA1
Aoyagi, T; Hachisu, M; Hiranuma, T; Murata, S; Shibazaki, Y; Umezawa, H; Uotani, K1

Other Studies

2 other study(ies) available for kelatorphan and actinonin

ArticleYear
Hydroxamic acids as potent inhibitors of endothelin-converting enzyme from human bronchiolar smooth muscle.
    Journal of medicinal chemistry, 1995, Jun-09, Volume: 38, Issue:12

    Topics: Aspartic Acid Endopeptidases; Bronchi; Cells, Cultured; Endothelin-Converting Enzymes; Humans; Hydroxamic Acids; Metalloendopeptidases; Muscle, Smooth

1995
Composite effects of actinonin when inhibiting enkephalin-degrading enzymes.
    European journal of pharmacology, 1987, May-07, Volume: 137, Issue:1

    Topics: Aminopeptidases; Analgesia; Angiotensin-Converting Enzyme Inhibitors; Animals; Brain; CD13 Antigens; Dipeptides; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Endopeptidases; Enkephalin, Methionine; Guinea Pigs; Hydroxamic Acids; Leucine; Male; Neprilysin; Protease Inhibitors

1987