Page last updated: 2024-09-03

kallidin, des-arg(10)- and kallidin

kallidin, des-arg(10)- has been researched along with kallidin in 77 studies

Compound Research Comparison

Studies
(kallidin, des-arg(10)-)
Trials
(kallidin, des-arg(10)-)
Recent Studies (post-2010)
(kallidin, des-arg(10)-)
Studies
(kallidin)
Trials
(kallidin)
Recent Studies (post-2010) (kallidin)
804175341224

Research

Studies (77)

TimeframeStudies, this research(%)All Research%
pre-19901 (1.30)18.7374
1990's24 (31.17)18.2507
2000's36 (46.75)29.6817
2010's15 (19.48)24.3611
2020's1 (1.30)2.80

Authors

AuthorsStudies
Borkowski, JA; Fraher, J; Hess, JF; Macneil, T; Ransom, RW; Stonesifer, GY; Strader, CD1
Borkowski, JA; Derrick, AW; Hess, JF; MacNeil, T1
Austin, CE; Bathon, JM; Chakravarty, S; Faussner, A; Kyle, DJ; Proud, D; Robinson, HE1
Bastian, S; Loillier, B; Paquet, JL; Pruneau, D1
Arbuckle, J; Bevan, SJ; Burgess, GM; Davis, C; Docherty, RJ; Jones, C; McIntyre, P; Phillips, E; Webb, M; Yaqoob, M1
deBlois, D; Drapeau, G; Marceau, F1
Churchill, L; Ward, PE1
Bowery, BJ; Hill, RG; Seabrook, GR1
Bodinier, MC; Chapelain, B; Coussy, L; Galizzi, JP; Giraud, S; Jean, T; Ly, SM; Neliat, G1
Bierilo, KK; Borkowski, JA; Derrick, AW; Hess, JF; Linemeyer, DL; MacNeil, T; Menke, JG; Ransom, RW; Schneck, KA; Strader, CD1
Hess, JF; Ransom, RW; Schneck, KA; Stonesifer, GY1
Champion, HC; Del Rio, O; Garrison, EA; Kadowitz, PJ; Santiago, JA; Smith, RE1
Allogho, SN; Gobeil, F; Neugebauer, W; Nguyen-Le, XK; Pheng, LH; Regoli, D1
Gais, P; Heinz-Erian, P; Offner, A; Roscher, AA; Schremmer-Danninger, E; Siebeck, M1
Carl, VS; Moore, EE; Moore, FA; Whalley, ET1
Eich-Rathfelder, S; Fautz, M; Fritz, H; Hohenbleicher, F; Siebeck, M; Whalley, ET1
Calixto, JB; Vianna, RM1
Barascud, Y; Bascands, JL; Bataillé, E; Gauthier, F; Girolami, JP; Hirtz, C; Marin Castaño, ME; Pecher, C; Pesquero, JB; Schanstra, JP1
Calixto, JB; de Campos, RO; Henriques, MG1
Proud, D; Reynolds, CJ; Togias, A1
Barnes, PJ; Belvisi, MG; Cirino, G; Mitchell, JA; Saunders, MA; Warner, TD1
Criscuoli, M; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Patacchini, R; Tramontana, M1
Dobashi, K; Fukabori, Y; Hisada, T; Horie, T; Iizuka, K; Ishizuka, T; Iwamae, S; Mori, M; Shimizu, Y; Tsukagoshi, H1
Beani, L; Bianchi, C; Borea, PA; Bregola, G; Gessi, S; Regoli, D; Simonato, M; Varani, K1
Gobeil, F; Pelletier, S; Perron, MS; Regoli, D; Sirois, P1
Bastian, S; Bonnafous, JC; Loillier, B; Paquet, JL; Pruneau, D; Robert, C1
Goldstein, RH; Ricupero, DA; Rishikof, DC; Romero, JR1
Polgar, P; Prado, GN; Taylor, L; Yang, X; Zhou, X1
deBlois, D; Horlick, RA1
Herbert, JM; Laplace, MC; Prabonnaud, V; Salel, V; Savi, P; Schaeffer, P1
Borges, DR; Loureiro-Silva, MR; Molina, HM1
Codd, EE; Lovenberg, TW; Wang, HY; Zhang, SP1
Anderson, KD; Leeb-Lundberg, LM; Phagoo, SB; Reddi, K; Warburton, D1
Davis, A; Fox, A; Ganju, P; Núñez, X; Patel, S1
Brand, M; Klusch, A; Kurzai, O; Petersen, M; Schmidt, RF; Valdeolmillos, M1
Banik, RK; Gera, L; Kozaki, Y; Mizumura, K; Sato, J1
Bachvarov, DR; Bastien, L; Marceau, F; Sabourin, T1
Chambers, SS; Christiansen, SC; Eddleston, J; Pan, ZK; Woessner, KM; Ye, R; Zuraw, BL1
Chang, RS; Chen, TB; Hess, JF; Hey, PJ; Pettibone, DJ1
Bouthillier, J; Fortin, JP; Marceau, F1
Adam, A; Fortin, JP; Gobeil, F; Marceau, F; Regoli, D1
Kohno, S; Mizutani, N; Nabe, T; Sugahara, S; Takenaka, H1
Bhoola, KD; Hoffmann, TF; Kuebler, JF; Messmer, K; Roscher, AA; Schremmer-Danninger, E1
Eisenbarth, H; Petersen, M; Rukwied, R; Schmelz, M1
Bock, MG; Chang, RS; Dean, DC; Freidinger, RM; Harrell, CM; Hess, JF; Hey, PJ; Jones, AN; Kunapuli, P; Markowitz, MK; Miller, PJ; Murphy, KL; O'Malley, SS; Pettibone, DJ; Raab, CE; Ransom, RW; Reiss, DR; Su, DS; Wallace, MA1
Cruden, NL; Fox, KA; Ludlam, CA; Megson, I; Newby, DE; Tse, GH1
Bicho, MD; Conlin, PR; Lança, V; Ricupero, DA; Rivera, A; Romero, JR1
Brodsky, PT; Pelorosso, FG; Rothlin, RP; Zold, CL1
Imai, C; Kitamura, Y; Okamura, A; Peng, JF; Printz, MP1
Binaschi, A; Mantovani, S; Mazzuferi, M; Rodi, D; Simonato, M1
Brovkovych, V; Deddish, PA; Erdös, EG; Ignjatovic, T; Skidgel, RA; Stanisavljevic, S; Zhang, K1
Argaman, M; Fleisher-Berkovich, S; Levant, A; Levy, E1
Adam, A; Bawolak, MT; Fortin, JP; Marceau, F; Vogel, LK1
Bellucci, F; Cucchi, P; Lazzeri, M; Meini, S; Santicioli, P; Turini, D1
Baltic, S; Bertram, CM; Bhoola, KD; Fogel-Petrovic, M; Foster, PS; Misso, NL; Thompson, PJ1
Daray, FM; Errasti, AE; Falcioni, AG; Gago, JE; Goldschmidt, ED; Nowak, W; Pelorosso, FG; Pugliese, MI; Rothlin, RP1
Bova, MP; Butelman, ER; Chavez, RA; Chen, L; Dreyer, M; Fukuda, JY; Garofalo, AW; Hawkinson, JE; Holcomb, R; Hom, DS; Ko, MC; Liao, A; Malmberg, AB; Ruslim, L; Samant, B; Simmonds, S; Szoke, BG; Wadsworth, A; Zeitz, KP; Zhang, H; Zmolek, W1
Allcock, BK; Gerovac, TA; McChesney, SL; Miranpuri, GS; Park, SW; Rajpal, S; Resnick, DK; Tilghman, JI; Turner, NA1
Bader, M; Cibrián-Uhalte, E; Costa-Neto, CM; de Picoli Souza, K; Oliveira, L; Oliveira, SM; Pesquero, JB; Santos, EL1
Bloomfield, P; Cruden, NL; Fox, KA; Lang, NN; Ludlam, CA; Newby, DE; Tse, GH1
Florkowska, M; Guevara-Lora, I; Kozik, A1
Mamenko, M; O'Neil, RG; Pochynyuk, O; Zaika, O1
Cruden, NL; Fox, KA; Lang, NN; MacGillivray, TJ; Newby, DE; Uren, NG1
Avalos, Y; Ayala, P; Boza, P; Catalán, M; Contreras, A; Copaja, M; Díaz-Araya, G; Lavandero, S; Olmedo, I; Smolic, C; Velarde, V; Vivar, R1
Bovenzi, V; Côté, J; Dubuc, C; Fortier, A; Fortin, D; Gobeil, F; Lepage, M; Müller-Esterl, W; Neugebauer, W; Savard, M; Tremblay, L; Tsanaclis, AM1
Leeb-Lundberg, LM; Sandén, C1
Bhoola, KD; Burgos, RA; Ehrenfeld, P; Figueroa, CD; Gonzalez, CB; Hidalgo, MA; Matus, CE; Pavicic, F; Sarmiento, J1
Bhoola, KD; Borquez, C; Ehrenfeld, P; Figueroa, CD; Lizama, A; Manso, L; Matus, CE; Naran, A; Pavicic, MF; Poblete, MT; Sarmiento, J1
Andrade, Y; Bhoola, KD; Colivoro, P; Ehrenfeld, P; Figueroa, CD; Gonzalez, CB; Lizama, AJ; Matus, CE; Sarmiento, J1
Amouroux, G; Bénard, F; Colpo, N; Hundal-Jabal, N; Jenni, S; Lau, J; Lin, KS; Liu, Z; Pan, J; Zhang, Z1
Amouroux, G; Bénard, F; Colpo, N; Hundal-Jabal, N; Jenni, S; Lin, KS; Liu, Z; Pan, J; Zhang, C; Zhang, Z1
Concha, M; Ehrenfeld, P; Figueroa, CD; Matus, CE; Mejia, AJ; Pavicic, F1
Armesto, AR; Errasti, AE; Feás, AA; Kilstein, Y; Nowak, W; Pelorosso, FG; Rothlin, RP1
Bhoola, KD; Burgos, RA; Concha, M; Ehrenfeld, P; Figueroa, CD; González, CB; Matus, CE; Pavicic, F1
Guevara-Lora, I; Kozik, A; Niewiarowska-Sendo, A1
An, S; Jiang, C; Lu, Y; Sun, T; Wang, F; Zhang, Y; Zhu, J1
Burckhardt, BB; Gangnus, T1

Trials

4 trial(s) available for kallidin, des-arg(10)- and kallidin

ArticleYear
Airway neural responses to kinins: tachyphylaxis and role of receptor subtypes.
    American journal of respiratory and critical care medicine, 1999, Volume: 159, Issue:2

    Topics: Asthma; Bronchi; Bronchial Provocation Tests; Bronchoconstriction; Capillary Permeability; Cross-Over Studies; Double-Blind Method; Female; Follow-Up Studies; Humans; Inflammation; Kallidin; Kinins; Male; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Reflex; Rhinitis, Allergic, Perennial; Tachyphylaxis

1999
B1 kinin receptor does not contribute to vascular tone or tissue plasminogen activator release in the peripheral circulation of patients with heart failure.
    Arteriosclerosis, thrombosis, and vascular biology, 2005, Volume: 25, Issue:4

    Topics: Adolescent; Aged; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Bradykinin B1 Receptor Antagonists; Cross-Over Studies; Enalapril; Female; Fibrinolysis; Forearm; Heart Failure; Humans; In Vitro Techniques; Kallidin; Losartan; Male; Middle Aged; Plasminogen Activator Inhibitor 1; Pregnancy; Receptor, Bradykinin B1; Regional Blood Flow; Tissue Plasminogen Activator; Umbilical Veins; Vasoconstriction

2005
Vascular B1 kinin receptors in patients with congestive heart failure.
    Journal of cardiovascular pharmacology, 2008, Volume: 52, Issue:5

    Topics: Adult; Aged; Angiotensin-Converting Enzyme Inhibitors; Blood Pressure; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cross-Over Studies; Double-Blind Method; Female; Heart Failure; Humans; Infusions, Intra-Arterial; Kallidin; Middle Aged; Nitroprusside; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Tissue Plasminogen Activator; Vasodilation

2008
Vasomotor and fibrinolytic responses to kinin receptor agonists in the atherosclerotic human lower limb.
    Heart and vessels, 2012, Volume: 27, Issue:2

    Topics: Adult; Aged; Analysis of Variance; Angiotensin-Converting Enzyme Inhibitors; Atherosclerosis; Blood Flow Velocity; Bradykinin; Dose-Response Relationship, Drug; Female; Femoral Artery; Fibrinolysis; Humans; Infusions, Intra-Arterial; Kallidin; Lower Extremity; Male; Middle Aged; Nitroprusside; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Scotland; Tissue Plasminogen Activator; Ultrasonography, Doppler; Ultrasonography, Interventional; Vasodilation; Vasodilator Agents; Vasomotor System

2012

Other Studies

73 other study(ies) available for kallidin, des-arg(10)- and kallidin

ArticleYear
Differential pharmacology of cloned human and mouse B2 bradykinin receptors.
    Molecular pharmacology, 1994, Volume: 45, Issue:1

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; DNA, Complementary; Humans; Mice; Molecular Sequence Data; Receptors, Bradykinin; Species Specificity

1994
The agonist selectivity of a mouse B1 bradykinin receptor differs from human and rabbit B1 receptors.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Bradykinin; Cattle; Cloning, Molecular; COS Cells; DNA Primers; DNA, Complementary; Humans; Kallidin; Mice; Molecular Sequence Data; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin; Sequence Homology, Amino Acid; Species Specificity; Transfection

1996
Stable expression of the human kinin B1 receptor in Chinese hamster ovary cells. Characterization of ligand binding and effector pathways.
    The Journal of biological chemistry, 1997, Apr-25, Volume: 272, Issue:17

    Topics: Animals; Binding, Competitive; Biological Transport; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; GTP-Binding Proteins; Humans; Inositol Phosphates; Kallidin; Ligands; Oligopeptides; Precipitin Tests; Protein Binding; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Proteins; Signal Transduction; Type C Phospholipases

1997
Stable expression of human kinin B1 receptor in 293 cells: pharmacological and functional characterization.
    British journal of pharmacology, 1997, Volume: 122, Issue:2

    Topics: Calcium; Cell Line; Enzyme Activation; Humans; Kallidin; Receptor, Bradykinin B1; Receptors, Bradykinin; Transfection; Type C Phospholipases

1997
Molecular characterisation of cloned bradykinin B1 receptors from rat and human.
    European journal of pharmacology, 1999, Jun-25, Volume: 374, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Cell Line; Cloning, Molecular; COS Cells; DNA, Complementary; Female; Gene Expression; Genes; Humans; Kallidin; Molecular Sequence Data; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

1999
Hypotensive effects of Lys-des-Arg9-bradykinin and metabolically protected agonists of B1 receptors for kinins.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:3

    Topics: Animals; Blood Pressure; Bradykinin; Cardiovascular System; Female; Hypotension; Kallidin; Kinins; Lipopolysaccharides; Male; Prostaglandins; Protease Inhibitors; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter

1991
Conversion of B1 kinin receptor-mediated vascular relaxation to contraction.
    Hypertension (Dallas, Tex. : 1979), 1987, Volume: 9, Issue:6 Pt 2

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Bradykinin; Dose-Response Relationship, Drug; Indomethacin; Kallidin; Male; Pyrazoles; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Vasoconstriction; Vasodilation

1987
Bradykinin receptors in mouse and rat isolated superior cervical ganglia.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Amino Acid Sequence; Animals; Bradykinin; Bradykinin Receptor Antagonists; Electrophysiology; Interleukin-1; Kallidin; Male; Mice; Molecular Sequence Data; Muscarine; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin; Structure-Activity Relationship; Superior Cervical Ganglion

1995
Up-regulation of [3H]-des-Arg10-kallidin binding to the bradykinin B1 receptor by interleukin-1 beta in isolated smooth muscle cells: correlation with B1 agonist-induced PGI2 production.
    British journal of pharmacology, 1994, Volume: 113, Issue:2

    Topics: Animals; Bradykinin Receptor Antagonists; Epoprostenol; In Vitro Techniques; Interleukin-1; Kallidin; Lipopolysaccharides; Mesenteric Arteries; Muscle, Smooth, Vascular; Nitric Oxide; Rabbits; Receptors, Bradykinin; Signal Transduction; Up-Regulation

1994
Expression cloning of a human B1 bradykinin receptor.
    The Journal of biological chemistry, 1994, Aug-26, Volume: 269, Issue:34

    Topics: Amino Acid Sequence; Animals; Bradykinin; Cloning, Molecular; DNA, Complementary; Gene Expression Regulation; Humans; Interleukin-1; Kallidin; Molecular Sequence Data; Oocytes; Receptors, Bradykinin; Recombinant Proteins; Sequence Homology, Amino Acid; Xenopus laevis

1994
Bradykinin B1 receptors in rabbit aorta smooth muscle cells in culture.
    European journal of pharmacology, 1994, Feb-15, Volume: 266, Issue:3

    Topics: Animals; Aorta; Binding Sites; Binding, Competitive; Bradykinin; Cells, Cultured; Enzyme Activation; Hydrolysis; Kallidin; Lysophospholipase; Muscle, Smooth, Vascular; Phosphatidylinositols; Rabbits; Receptors, Bradykinin

1994
Analysis of responses to kallidin, DABK, and DAK in feline hindlimb vascular bed.
    The American journal of physiology, 1995, Volume: 269, Issue:6 Pt 2

    Topics: Adamantane; Animals; Arginine; Atropine; Blood Vessels; Bradykinin; Bradykinin Receptor Antagonists; Cats; Female; Hindlimb; Kallidin; Male; Meclofenamic Acid; Morpholines; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Potassium Channels

1995
Kinin B1 and B2 receptors in the mouse.
    Canadian journal of physiology and pharmacology, 1995, Volume: 73, Issue:12

    Topics: Animals; Bradykinin Receptor Antagonists; Kallidin; Mice; Mice, Inbred C57BL; Receptors, Bradykinin; Stomach; Urinary Bladder

1995
Autoradiographic visualization of B1 bradykinin receptors in porcine vascular tissues in the presence or absence of inflammation.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Animals; Aorta, Thoracic; Autoradiography; Blood Vessels; Inflammation; Kallidin; Lipopolysaccharides; Pulmonary Artery; Receptor, Bradykinin B1; Receptors, Bradykinin; Sepsis; Swine

1996
Involvement of bradykinin B1 and B2 receptors in human PMN elastase release and increase in endothelial cell monolayer permeability.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Amino Acid Chloromethyl Ketones; Bradykinin; Cells, Cultured; Endothelium, Vascular; Humans; In Vitro Techniques; Kallidin; Leukocyte Elastase; Neutrophils; Permeability; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Serine Proteinase Inhibitors

1996
Tachyphylaxis of the B1 kinin receptor in porcine endotoxin shock.
    Immunopharmacology, 1997, Volume: 36, Issue:2-3

    Topics: Animals; Blood Pressure; Bradykinin Receptor Antagonists; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Infusions, Intravenous; Injections, Intra-Arterial; Kallidin; Lipopolysaccharides; Receptor, Bradykinin B1; Receptors, Bradykinin; Shock, Septic; Swine; Tachyphylaxis; Up-Regulation

1997
Characterization of the receptor and the mechanisms underlying the inflammatory response induced by des-Arg9-BK in mouse pleurisy.
    British journal of pharmacology, 1998, Volume: 123, Issue:2

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Capillary Permeability; Cell Cycle; Disease Models, Animal; Edema; Inflammation; Kallidin; Kinins; Lipopolysaccharides; Male; Mice; Neuropeptides; Nitric Oxide; Pleura; Pleurisy; Receptors, Bradykinin; Receptors, Tachykinin

1998
The B1-agonist [des-Arg10]-kallidin activates transcription factor NF-kappaB and induces homologous upregulation of the bradykinin B1-receptor in cultured human lung fibroblasts.
    The Journal of clinical investigation, 1998, May-15, Volume: 101, Issue:10

    Topics: Amino Acid Sequence; Cell Line; Cholera Toxin; DNA-Binding Proteins; Fibroblasts; Humans; Inflammation; Interleukin-1; Kallidin; Lung; Molecular Sequence Data; NF-kappa B; Proline; Pyrrolidines; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Thiocarbamates; Transcriptional Activation; Up-Regulation; Virulence Factors, Bordetella

1998
Systemic treatment with Mycobacterium bovis bacillus Calmette-Guérin (BCG) potentiates kinin B1 receptor agonist-induced nociception and oedema formation in the formalin test in mice.
    Neuropeptides, 1998, Volume: 32, Issue:5

    Topics: Animals; Bradykinin; Dexamethasone; Dose-Response Relationship, Drug; Drug Synergism; Edema; Formaldehyde; Hindlimb; Indomethacin; Kallidin; Male; Mice; Mycobacterium bovis; Pain; Pain Measurement; Pyrazoles; Receptor, Bradykinin B1; Receptors, Bradykinin

1998
Mechanisms of prostaglandin E2 release by intact cells expressing cyclooxygenase-2: evidence for a 'two-component' model.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Arachidonic Acid; Bradykinin; Calcimycin; Cell Line; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Humans; Inflammation; Interleukin-1; Isoenzymes; Kallidin; Membrane Proteins; Phospholipases A; Phospholipases A2; Prostaglandin-Endoperoxide Synthases; Receptors, Bradykinin

1999
Effect of dexamethasone on cyclophosphamide-induced cystitis in rats: lack of relation with bradykinin B1 receptor-mediated motor responses.
    European journal of pharmacology, 1999, Mar-12, Volume: 369, Issue:1

    Topics: Animals; Anti-Inflammatory Agents; Binding, Competitive; Bradykinin; Carcinogens; Cyclophosphamide; Cystitis; Dexamethasone; Dose-Response Relationship, Drug; Kallidin; Male; Muscle Contraction; Radioligand Assay; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; Tritium; Urinary Bladder

1999
Regulation by interleukin-1beta of gene expression of bradykinin B1 receptor in MH-S murine alveolar macrophage cell line.
    Biochemical and biophysical research communications, 1999, Jun-07, Volume: 259, Issue:2

    Topics: Animals; Calcium; Cell Line; Gene Expression Regulation; Interleukin-1; Kallidin; Macrophages, Alveolar; Male; Mice; Mice, Inbred BALB C; Protein Binding; Receptor, Bradykinin B1; Receptors, Bradykinin; Recombinant Proteins; RNA, Messenger; Time Factors; Tumor Necrosis Factor-alpha

1999
Changes in hippocampal and cortical B1 bradykinin receptor biological activity in two experimental models of epilepsy.
    Neuroscience, 1999, Volume: 92, Issue:3

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Cerebral Cortex; Electric Stimulation; Epilepsy; Glutamic Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Kallidin; Kindling, Neurologic; Male; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin

1999
Involvement of bradykinin B1 and B2 receptors in pulmonary leukocyte accumulation induced by Sephadex beads in guinea pigs.
    European journal of pharmacology, 1999, Jul-02, Volume: 376, Issue:1-2

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Bronchoalveolar Lavage Fluid; Cell Count; Dextrans; Guinea Pigs; Indicators and Reagents; Inflammation; Kallidin; Leukocytes; Lung Diseases; Male; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin

1999
Identification of a key region of kinin B(1) receptor for high affinity binding of peptide antagonists.
    The Journal of biological chemistry, 2000, Mar-03, Volume: 275, Issue:9

    Topics: Amino Acid Sequence; Animals; Binding Sites; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; Humans; Inositol Phosphates; Kallidin; Molecular Sequence Data; Mutation; Peptides; Protein Binding; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Fusion Proteins; Tetrahydroisoquinolines; Transfection

2000
Des-Arg(10)-kallidin engagement of the B1 receptor stimulates type I collagen synthesis via stabilization of connective tissue growth factor mRNA.
    The Journal of biological chemistry, 2000, Apr-28, Volume: 275, Issue:17

    Topics: Blotting, Northern; Calcium; Cell Line; Collagen; Connective Tissue Growth Factor; Cycloheximide; Cytosol; Fibroblasts; Growth Substances; Humans; Immediate-Early Proteins; Intercellular Signaling Peptides and Proteins; Kallidin; Luciferases; Lung; Protein Binding; Protein Synthesis Inhibitors; Receptor, Bradykinin B2; Receptors, Bradykinin; RNA, Messenger; Tetradecanoylphorbol Acetate; Time Factors; Transforming Growth Factor beta

2000
Regulation of inducible bradykinin B1 receptor gene expression through absence of internalization and resensitization.
    Journal of cellular biochemistry, 2000, Jun-06, Volume: 78, Issue:3

    Topics: Arachidonic Acid; Blotting, Northern; Bradykinin; Calcium; Cells, Cultured; DNA Primers; Endocytosis; Fibroblasts; Gene Expression Regulation; Genetic Vectors; Humans; Kallidin; Lung; Phosphatidylinositols; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Transfection

2000
Endotoxin sensitization to kinin B(1) receptor agonist in a non-human primate model: haemodynamic and pro-inflammatory effects.
    British journal of pharmacology, 2001, Volume: 132, Issue:1

    Topics: Animals; Blood Pressure; Body Temperature; Bradykinin; Chlorocebus aethiops; Dose-Response Relationship, Drug; Edema; Endotoxins; Hemodynamics; Inflammation; Kallidin; Lipopolysaccharides; Male; Receptor, Bradykinin B1; Receptors, Bradykinin

2001
Detection of bradykinin B1 receptors in rat aortic smooth muscle cells.
    Biochemical pharmacology, 2001, Feb-01, Volume: 61, Issue:3

    Topics: Animals; Aorta; In Vitro Techniques; Kallidin; Male; Muscle, Smooth, Vascular; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Tritium

2001
Portal hypertensive response to bradykinin in inflamed or cirrhotic rat livers is mediated by B2-type receptors.
    Journal of gastroenterology and hepatology, 2001, Volume: 16, Issue:1

    Topics: Analysis of Variance; Animals; Bradykinin; Carbon Tetrachloride; Hypertension, Portal; Inflammation; Kallidin; Liver Cirrhosis; Male; Rats; Rats, Wistar; Receptors, Bradykinin; Turpentine

2001
Functional studies of bradykinin receptors in Chinese hamster ovary cells stably expressing the human B2 bradykinin receptor.
    International immunopharmacology, 2001, Volume: 1, Issue:5

    Topics: Animals; Bradykinin Receptor Antagonists; Calcium Signaling; Cell Membrane; CHO Cells; Cricetinae; Gene Expression; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Kallidin; Kinetics; Ligands; Oligopeptides; Receptor, Bradykinin B2; Receptors, Bradykinin; Signal Transduction

2001
Bradykinin B1 receptor up-regulation by interleukin-1beta and B1 agonist occurs through independent and synergistic intracellular signaling mechanisms in human lung fibroblasts.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:1

    Topics: Cells, Cultured; Drug Synergism; Enzyme Inhibitors; Epithelial Cells; Fibroblasts; Genistein; Humans; Interleukin-1; Kallidin; Lung; Mitogen-Activated Protein Kinase Kinases; NF-kappa B; Protein-Tyrosine Kinases; Receptor, Bradykinin B1; Receptors, Bradykinin; Signal Transduction; Up-Regulation

2001
p38 stress-activated protein kinase inhibitor reverses bradykinin B(1) receptor-mediated component of inflammatory hyperalgesia.
    European journal of pharmacology, 2001, Jun-15, Volume: 421, Issue:3

    Topics: Animals; Cell Line; Cyclooxygenase 2; Cytokines; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hindlimb; Humans; Hyperalgesia; Imidazoles; Inflammation; Interleukin-1; Isoenzymes; Kallidin; Male; Membrane Proteins; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Prostaglandin-Endoperoxide Synthases; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptors, Bradykinin; Tumor Necrosis Factor-alpha

2001
No evidence for bradykinin B1 receptors in rat dorsal root ganglion neurons.
    Neuroreport, 2001, Oct-08, Volume: 12, Issue:14

    Topics: Animals; Blotting, Northern; Bradykinin; Calcium; Calcium Signaling; Cells, Cultured; Drug Administration Schedule; Fluorescent Dyes; Fura-2; Ganglia, Spinal; Intracellular Fluid; Kallidin; Male; Neuralgia; Neurons, Afferent; Peripheral Nervous System Diseases; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger

2001
B2 receptor-mediated enhanced bradykinin sensitivity of rat cutaneous C-fiber nociceptors during persistent inflammation.
    Journal of neurophysiology, 2001, Volume: 86, Issue:6

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Electrophysiology; Hot Temperature; In Vitro Techniques; Inflammation; Kallidin; Male; Nerve Fibers; Nociceptors; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B2; Receptors, Bradykinin; Skin; Stimulation, Chemical; Tachyphylaxis

2001
Agonist-induced translocation of the kinin B(1) receptor to caveolae-related rafts.
    Molecular pharmacology, 2002, Volume: 61, Issue:3

    Topics: Animals; Antigens, Human Platelet; Bacterial Proteins; beta-Cyclodextrins; Biological Transport; Bradykinin; Caveolae; Caveolin 1; Caveolins; Cell Fractionation; Cells, Cultured; COS Cells; Cyclodextrins; Endocytosis; Green Fluorescent Proteins; Humans; Kallidin; Luminescent Proteins; Membrane Microdomains; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin; Subcellular Fractions; Transfection; Tritium

2002
Up-regulation of functional kinin B1 receptors in allergic airway inflammation.
    Journal of immunology (Baltimore, Md. : 1950), 2002, Aug-15, Volume: 169, Issue:4

    Topics: Adult; Allergens; Animals; Bradykinin; Case-Control Studies; Enzyme Activation; Epithelial Cells; Humans; In Vitro Techniques; Kallidin; Mitogen-Activated Protein Kinases; Nasal Mucosa; Nasal Provocation Tests; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; RNA, Messenger; Transcription Factor AP-1; Up-Regulation

2002
Molecular and pharmacological diversity of the kinin B1 receptor.
    International immunopharmacology, 2002, Volume: 2, Issue:13-14

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Bradykinin; Chlorocebus aethiops; Cloning, Molecular; Dogs; Gene Frequency; Humans; Kallidin; Macaca mulatta; Molecular Sequence Data; Polymorphism, Single Nucleotide; Rats; Receptor, Bradykinin B1; Receptors, Bradykinin; Recombinant Fusion Proteins; Sequence Alignment; Species Specificity

2002
High agonist-independent clearance of rabbit kinin B1 receptors in cultured cells.
    American journal of physiology. Heart and circulatory physiology, 2003, Volume: 284, Issue:5

    Topics: Animals; Anisomycin; Aorta; Bradykinin; Cells, Cultured; Green Fluorescent Proteins; Humans; Immunoblotting; Indicators and Reagents; Jugular Veins; Kallidin; Kidney; Luminescent Proteins; Muscle Contraction; Muscle, Smooth, Vascular; Protein Synthesis Inhibitors; Rabbits; Radioligand Assay; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Proteins; Tritium

2003
Do angiotensin-converting enzyme inhibitors directly stimulate the kinin B1 receptor?
    American journal of physiology. Heart and circulatory physiology, 2003, Volume: 285, Issue:1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Aorta, Thoracic; Arachidonic Acid; Bacterial Proteins; Cell Line; Enalaprilat; Humans; In Vitro Techniques; Kallidin; Luminescent Proteins; Mice; Mice, Inbred C57BL; Microscopy, Confocal; Mitogen-Activated Protein Kinases; Muscle Contraction; Muscle, Smooth, Vascular; Phospholipases A; Phosphorylation; Receptor, Bradykinin B1; Receptors, Bradykinin; Subcellular Fractions; Translocation, Genetic; Umbilical Veins

2003
Kinins are involved in the development of allergic nasal hyperresponsiveness in guinea pigs.
    European journal of pharmacology, 2003, Aug-29, Volume: 476, Issue:3

    Topics: Airway Resistance; Allergens; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Disease Models, Animal; Guinea Pigs; Kallidin; Kinins; Leukotriene D4; Male; Nasal Lavage Fluid; Pollen; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Rhinitis, Allergic, Seasonal; Time Factors

2003
Kinin-B1 receptors in ischaemia-induced pancreatitis: functional importance and cellular localisation.
    Biological chemistry, 2003, Volume: 384, Issue:9

    Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cell Adhesion; GPI-Linked Proteins; Kallidin; Leukocytes; Male; Metalloendopeptidases; Pancreatitis; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Reperfusion Injury; Survival Rate; Up-Regulation; Venules

2003
Sensitization to bradykinin B1 and B2 receptor activation in UV-B irradiated human skin.
    Pain, 2004, Volume: 110, Issue:1-2

    Topics: Adult; Analysis of Variance; Bradykinin; Dose-Response Relationship, Drug; Erythema; Female; Humans; Kallidin; Laser-Doppler Flowmetry; Male; Microdialysis; Pain; Pain Measurement; Proteins; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Skin; Time Factors; Ultraviolet Rays

2004
Pharmacological characterization and radioligand binding properties of a high-affinity, nonpeptide, bradykinin B1 receptor antagonist.
    European journal of pharmacology, 2004, Sep-19, Volume: 499, Issue:1-2

    Topics: Animals; Aorta, Thoracic; Binding, Competitive; Blood Pressure; Bradykinin B1 Receptor Antagonists; CHO Cells; Cricetinae; Cricetulus; Dogs; Dose-Response Relationship, Drug; Humans; Imidazoles; In Vitro Techniques; Kallidin; Lipopolysaccharides; Male; Quinoxalines; Rabbits; Radioligand Assay; Rats; Receptor, Bradykinin B1; Transfection; Tritium; Vasoconstriction

2004
Na+/Ca2+ exchanger activity modulates connective tissue growth factor mRNA expression in transforming growth factor beta1- and Des-Arg10-kallidin-stimulated myofibroblasts.
    The Journal of biological chemistry, 2005, Apr-15, Volume: 280, Issue:15

    Topics: Blotting, Northern; Calcium; Cell Line; Cell Membrane; Cells, Cultured; Collagen; Connective Tissue Growth Factor; Cytosol; Fibroblasts; Humans; Immediate-Early Proteins; Intercellular Signaling Peptides and Proteins; Kallidin; Luciferases; Microcirculation; Myocardium; Osteoblasts; Phenotype; Phosphorylation; Protein Binding; Reverse Transcriptase Polymerase Chain Reaction; RNA; RNA, Messenger; Signal Transduction; Sodium-Calcium Exchanger; Tetradecanoylphorbol Acetate; Thiourea; Time Factors; Transforming Growth Factor beta; Transforming Growth Factor beta1

2005
Potentiation of des-Arg9-kallidin-induced vasoconstrictor responses by metallopeptidase inhibition in isolated human umbilical artery.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 313, Issue:3

    Topics: Captopril; CD13 Antigens; Drug Synergism; Humans; In Vitro Techniques; Kallidin; Neprilysin; Protease Inhibitors; Receptor, Bradykinin B1; Umbilical Arteries; Vasoconstriction

2005
Interleukin-1beta enhanced action of kinins on extracellular matrix of spontaneous hypertensive rat cardiac fibroblasts.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2005, Volume: 27, Issue:1

    Topics: Animals; Bradykinin; Cells, Cultured; Collagenases; Drug Synergism; Enzyme Precursors; Extracellular Matrix; Fibroblasts; Gelatinases; Gene Expression; Hypertension; Interleukin-1; Kallidin; Matrix Metalloproteinase 9; Metalloendopeptidases; Myocardium; Procollagen; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptor, Bradykinin B1; Receptor, Bradykinin B2; RNA, Messenger; Tissue Inhibitor of Metalloproteinase-1; Tissue Inhibitor of Metalloproteinase-2

2005
Induction of B1 bradykinin receptors in the kindled hippocampus increases extracellular glutamate levels: a microdialysis study.
    Neuroscience, 2005, Volume: 135, Issue:3

    Topics: Animals; Behavior, Animal; Bradykinin; Electroencephalography; Extracellular Space; Glutamic Acid; Hippocampus; Kallidin; Kindling, Neurologic; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1

2005
Angiotensin I-converting enzyme inhibitors block protein kinase C epsilon by activating bradykinin B1 receptors in human endothelial cells.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 316, Issue:3

    Topics: Amino Acid Sequence; Angiotensin-Converting Enzyme Inhibitors; Cells, Cultured; Endothelial Cells; Humans; Kallidin; Molecular Sequence Data; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Protein Kinase C-epsilon; Receptor, Bradykinin B1

2006
Kinins and neuroinflammation: dual effect on prostaglandin synthesis.
    European journal of pharmacology, 2006, Sep-28, Volume: 546, Issue:1-3

    Topics: Animals; Animals, Newborn; Bradykinin; Cells, Cultured; Dinoprostone; Dose-Response Relationship, Drug; Encephalitis; Kallidin; Kinins; Lipopolysaccharides; Neuroglia; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2

2006
The bradykinin B2 receptor antagonist icatibant (Hoe 140) blocks aminopeptidase N at micromolar concentrations: off-target alterations of signaling mediated by the bradykinin B1 and angiotensin receptors.
    European journal of pharmacology, 2006, Dec-03, Volume: 551, Issue:1-3

    Topics: Angiotensin II; Angiotensin III; Aniline Compounds; Animals; Aorta; Bradykinin; Bradykinin B2 Receptor Antagonists; CD13 Antigens; Dose-Response Relationship, Drug; In Vitro Techniques; Kallidin; Kinetics; Protease Inhibitors; Quinolines; Rabbits; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Angiotensin; Recombinant Proteins; Signal Transduction; Vasoconstriction; Vasoconstrictor Agents

2006
Characterization of kinin receptors in human cultured detrusor smooth muscle cells.
    British journal of pharmacology, 2007, Volume: 150, Issue:2

    Topics: Bradykinin; Bradykinin B1 Receptor Antagonists; Cells, Cultured; Dinoprostone; Humans; Inositol Phosphates; Interleukin-1beta; Kallidin; Male; Middle Aged; Muscle, Smooth; Ornithine; Radioligand Assay; Receptor, Bradykinin B1; Sulfonamides; Transforming Growth Factor alpha; Urinary Bladder

2007
Expression of kinin B1 and B2 receptors in immature, monocyte-derived dendritic cells and bradykinin-mediated increase in intracellular Ca2+ and cell migration.
    Journal of leukocyte biology, 2007, Volume: 81, Issue:6

    Topics: Bradykinin; Calcium; Cell Differentiation; Cell Movement; Cells, Cultured; Dendritic Cells; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Interleukin-4; Intracellular Fluid; Kallidin; Monocytes; Receptor, Bradykinin B1; Receptor, Bradykinin B2

2007
Functional evidence of des-Arg10-kallidin enzymatic inactivating pathway in isolated human umbilical vein.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Bradykinin; Captopril; CD13 Antigens; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Female; Glycopeptides; Humans; In Vitro Techniques; Kallidin; Metalloproteases; Neprilysin; Peptides; Protease Inhibitors; Receptor, Bradykinin B1; Umbilical Veins; Vasoconstriction

2007
Pharmacological, pharmacokinetic, and primate analgesic efficacy profile of the novel bradykinin B1 Receptor antagonist ELN441958.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 322, Issue:2

    Topics: Analgesics; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bradykinin; Bradykinin B1 Receptor Antagonists; Calcium; Carrageenan; Cell Line; Cell Membrane Permeability; Fibroblasts; Humans; Hyperalgesia; Kallidin; Macaca mulatta; Mice; Mice, Knockout; Microsomes, Liver; Molecular Structure; Naltrexone; Naproxen; Narcotic Antagonists; Rats; Receptor, Bradykinin B1; Species Specificity; Spiro Compounds; Transfection

2007
Antihyperalgesic effects of vanilloid-1 and bradykinin-1 receptor antagonists following spinal cord injury in rats.
    Journal of neurosurgery. Spine, 2007, Volume: 6, Issue:5

    Topics: Acrylamides; Animals; Bradykinin Receptor Antagonists; Bridged Bicyclo Compounds, Heterocyclic; Hyperalgesia; Kallidin; Male; Rats; Rats, Sprague-Dawley; Spinal Cord Injuries; TRPV Cation Channels

2007
Essential role of TM V and VI for binding the C-terminal sequences of Des-Arg-kinins.
    International immunopharmacology, 2008, Volume: 8, Issue:2

    Topics: Amino Acid Sequence; Animals; Bradykinin; CHO Cells; Cricetinae; Cricetulus; HeLa Cells; Humans; Kallidin; Molecular Sequence Data; Protein Structure, Tertiary; Rats; Receptor, Bradykinin B1

2008
Bradykinin-related peptides up-regulate the expression of kinin B1 and B2 receptor genes in human promonocytic cell line U937.
    Acta biochimica Polonica, 2009, Volume: 56, Issue:3

    Topics: Bradykinin; Cell Differentiation; Gene Expression; Humans; Immunohistochemistry; Kallidin; Peptides; Phorbol Esters; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Tretinoin; U937 Cells; Up-Regulation

2009
Bradykinin acutely inhibits activity of the epithelial Na+ channel in mammalian aldosterone-sensitive distal nephron.
    American journal of physiology. Renal physiology, 2011, Volume: 300, Issue:5

    Topics: Absorption; Aldosterone; Animals; Biosensing Techniques; Bradykinin; Caffeine; Cyclic AMP; Dose-Response Relationship, Drug; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Estrenes; GTP-Binding Protein alpha Subunits, Gq-G11; Hydrolysis; Ion Channel Gating; Kallidin; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Natriuresis; Nephrons; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phosphodiesterase Inhibitors; Pyrrolidinones; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Signal Transduction; Sodium; Sodium Channel Blockers; Thapsigargin; Thionucleotides; Tissue Culture Techniques; Type C Phospholipases

2011
Differential regulation of collagen secretion by kinin receptors in cardiac fibroblast and myofibroblast.
    Toxicology and applied pharmacology, 2012, Jun-15, Volume: 261, Issue:3

    Topics: Animals; Binding, Competitive; Blotting, Western; Calcium; Calcium Signaling; Collagen; Cyclooxygenase Inhibitors; Fibroblasts; Immunohistochemistry; Kallidin; Kinins; Myocardium; Myofibroblasts; Nitric Oxide Synthase; Prostaglandin-Endoperoxide Synthases; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Signal Transduction

2012
Induction of selective blood-tumor barrier permeability and macromolecular transport by a biostable kinin B1 receptor agonist in a glioma rat model.
    PloS one, 2012, Volume: 7, Issue:5

    Topics: Adult; Aged; Animals; Biological Transport; Bradykinin; Brain Neoplasms; Capillary Permeability; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Glioma; Humans; Kallidin; Male; Middle Aged; Permeability; Rats; Rats, Inbred F344; Receptor, Bradykinin B1

2012
Kinin B1 receptor homo-oligomerization is required for receptor trafficking to the cell surface.
    International immunopharmacology, 2013, Volume: 15, Issue:1

    Topics: Cell Membrane; Endoplasmic Reticulum; HEK293 Cells; Humans; Kallidin; Protein Transport; Receptor, Bradykinin B1

2013
Kinin B1 receptor regulates interactions between neutrophils and endothelial cells by modulating the levels of Mac-1, LFA-1 and intercellular adhesion molecule-1.
    Innate immunity, 2015, Volume: 21, Issue:3

    Topics: Cell Adhesion; Cell Communication; Cell Movement; Cells, Cultured; Cycloheximide; Endothelial Cells; Humans; Inflammation; Intercellular Adhesion Molecule-1; Kallidin; Lymphocyte Function-Associated Antigen-1; Macrophage-1 Antigen; Neutrophils; Receptor, Bradykinin B1; RNA, Small Interfering

2015
Bioregulation of kallikrein-related peptidases 6, 10 and 11 by the kinin B₁ receptor in breast cancer cells.
    Anticancer research, 2014, Volume: 34, Issue:12

    Topics: Bradykinin; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Down-Regulation; Female; Humans; Kallidin; Kallikreins; Kininogens; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; MCF-7 Cells; Neoplasm Invasiveness; Receptor, Bradykinin B1; RNA Interference; RNA, Small Interfering; Serine Endopeptidases; Tissue Kallikreins; Up-Regulation

2014
Expression and bioregulation of the kallikrein-related peptidases family in the human neutrophil.
    Innate immunity, 2015, Volume: 21, Issue:6

    Topics: Adult; Cell Line; Female; Gene Expression Regulation; Humans; Kallidin; Male; Middle Aged; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Proteolysis; Receptor, Bradykinin B1; RNA, Messenger; Tissue Kallikreins; Young Adult

2015
Comparative studies of three 68Ga-labeled [Des-Arg10]kallidin derivatives for imaging bradykinin B1 receptor expression with PET.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2015, Volume: 56, Issue:4

    Topics: Animals; CHO Cells; Contrast Media; Cricetinae; Cricetulus; Gallium Radioisotopes; HEK293 Cells; Humans; Kallidin; Male; Mice; Mice, SCID; Neoplasm Transplantation; Peptides; Positron-Emission Tomography; Receptor, Bradykinin B1; Tomography, X-Ray Computed

2015
Imaging Bradykinin B1 Receptor with 68Ga-Labeled [des-Arg10]Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake.
    Molecular pharmaceutics, 2015, Aug-03, Volume: 12, Issue:8

    Topics: Animals; Contrast Media; Gallium Radioisotopes; HEK293 Cells; Humans; Image Processing, Computer-Assisted; Kallidin; Male; Mice; Mice, Inbred BALB C; Mice, Inbred NOD; Mice, Knockout; Mice, SCID; Neoplasms; Peptide Fragments; Positron-Emission Tomography; Radiopharmaceuticals; Receptor, Bradykinin B1; Receptors, Interleukin-2; Tissue Distribution; Tomography, X-Ray Computed

2015
Intracellular signaling pathways involved in the release of IL-4 and VEGF from human keratinocytes by activation of kinin B1 receptor: functional relevance to angiogenesis.
    Archives of dermatological research, 2015, Volume: 307, Issue:9

    Topics: Angiogenic Proteins; Cell Line; Cell Movement; Cell Proliferation; Culture Media, Conditioned; Endothelial Cells; Enzyme Activation; Humans; Interleukin-4; JNK Mitogen-Activated Protein Kinases; Kallidin; Keratinocytes; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; Neovascularization, Physiologic; Phosphorylation; Proto-Oncogene Proteins c-jun; Receptor, Bradykinin B1; RNA Interference; RNA, Small Interfering; Signal Transduction; Skin; Spheroids, Cellular; Vascular Endothelial Growth Factor A

2015
Involvement of Extracellular Signal-Regulated Kinase 5 in Kinin B1 Receptor Upregulation in Isolated Human Umbilical Veins.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 357, Issue:1

    Topics: Dose-Response Relationship, Drug; Female; Humans; Janus Kinases; Kallidin; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 7; Muscle Contraction; Muscle, Smooth, Vascular; p38 Mitogen-Activated Protein Kinases; Pregnancy; Receptor, Bradykinin B1; RNA, Messenger; Serotonin; Umbilical Veins; Up-Regulation

2016
Activation of the human keratinocyte B1 bradykinin receptor induces expression and secretion of metalloproteases 2 and 9 by transactivation of epidermal growth factor receptor.
    Experimental dermatology, 2016, Volume: 25, Issue:9

    Topics: ADAM17 Protein; Animals; Cell Line; ErbB Receptors; Kallidin; Keratinocytes; Male; MAP Kinase Signaling System; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; Mice, Inbred C57BL; Proto-Oncogene Proteins c-akt; Receptor, Bradykinin B1; src-Family Kinases; Transcriptional Activation; Wound Healing

2016
Kinin Peptides Enhance Inflammatory and Oxidative Responses Promoting Apoptosis in a Parkinson's Disease Cellular Model.
    Mediators of inflammation, 2016, Volume: 2016

    Topics: 1-Methyl-4-phenylpyridinium; Apoptosis; Bradykinin; Cell Differentiation; Cell Line, Tumor; Cell Survival; Cytokines; Humans; Kallidin; Kinins; Oxidative Stress; Parkinson Disease; Reactive Oxygen Species

2016
ATP/pH Dual Responsive Nanoparticle with d-[des-Arg
    Small (Weinheim an der Bergstrasse, Germany), 2017, Volume: 13, Issue:3

    Topics: Adenosine Triphosphate; Animals; Antineoplastic Agents; Cell Line, Tumor; Doxorubicin; Drug Delivery Systems; Drug Liberation; Endocytosis; Female; Hydrogen-Ion Concentration; Kallidin; Male; Mammary Neoplasms, Animal; Mice, Nude; Nanoparticles; Polymers; Rats, Sprague-Dawley; Tissue Distribution; Treatment Outcome; Tumor Burden; Xenograft Model Antitumor Assays

2017
Targeted LC-MS/MS platform for the comprehensive determination of peptides in the kallikrein-kinin system.
    Analytical and bioanalytical chemistry, 2021, Volume: 413, Issue:11

    Topics: Bradykinin; Chromatography, Liquid; COVID-19; Humans; Kallidin; Kallikrein-Kinin System; Limit of Detection; Peptide Fragments; Tandem Mass Spectrometry

2021