kallidin, des-arg(10)- has been researched along with bradykinin in 48 studies
Studies (kallidin, des-arg(10)-) | Trials (kallidin, des-arg(10)-) | Recent Studies (post-2010) (kallidin, des-arg(10)-) | Studies (bradykinin) | Trials (bradykinin) | Recent Studies (post-2010) (bradykinin) |
---|---|---|---|---|---|
80 | 4 | 17 | 14,195 | 355 | 1,520 |
Protein | Taxonomy | kallidin, des-arg(10)- (IC50) | bradykinin (IC50) |
---|---|---|---|
B2 bradykinin receptor | Homo sapiens (human) | 0.0018 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (2.08) | 18.7374 |
1990's | 16 (33.33) | 18.2507 |
2000's | 24 (50.00) | 29.6817 |
2010's | 6 (12.50) | 24.3611 |
2020's | 1 (2.08) | 2.80 |
Authors | Studies |
---|---|
Borkowski, JA; Fraher, J; Hess, JF; Macneil, T; Ransom, RW; Stonesifer, GY; Strader, CD | 1 |
Borkowski, JA; Derrick, AW; Hess, JF; MacNeil, T | 1 |
Austin, CE; Bathon, JM; Chakravarty, S; Faussner, A; Kyle, DJ; Proud, D; Robinson, HE | 1 |
Arbuckle, J; Bevan, SJ; Burgess, GM; Davis, C; Docherty, RJ; Jones, C; McIntyre, P; Phillips, E; Webb, M; Yaqoob, M | 1 |
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L | 1 |
deBlois, D; Drapeau, G; Marceau, F | 1 |
Churchill, L; Ward, PE | 1 |
Bowery, BJ; Hill, RG; Seabrook, GR | 1 |
Bierilo, KK; Borkowski, JA; Derrick, AW; Hess, JF; Linemeyer, DL; MacNeil, T; Menke, JG; Ransom, RW; Schneck, KA; Strader, CD | 1 |
Hess, JF; Ransom, RW; Schneck, KA; Stonesifer, GY | 1 |
Champion, HC; Del Rio, O; Garrison, EA; Kadowitz, PJ; Santiago, JA; Smith, RE | 1 |
Carl, VS; Moore, EE; Moore, FA; Whalley, ET | 1 |
Calixto, JB; Vianna, RM | 1 |
Calixto, JB; de Campos, RO; Henriques, MG | 1 |
Barnes, PJ; Belvisi, MG; Cirino, G; Mitchell, JA; Saunders, MA; Warner, TD | 1 |
Criscuoli, M; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Patacchini, R; Tramontana, M | 1 |
Beani, L; Bianchi, C; Borea, PA; Bregola, G; Gessi, S; Regoli, D; Simonato, M; Varani, K | 1 |
Gobeil, F; Pelletier, S; Perron, MS; Regoli, D; Sirois, P | 1 |
Bastian, S; Bonnafous, JC; Loillier, B; Paquet, JL; Pruneau, D; Robert, C | 1 |
Polgar, P; Prado, GN; Taylor, L; Yang, X; Zhou, X | 1 |
deBlois, D; Horlick, RA | 1 |
Borges, DR; Loureiro-Silva, MR; Molina, HM | 1 |
Brand, M; Klusch, A; Kurzai, O; Petersen, M; Schmidt, RF; Valdeolmillos, M | 1 |
Banik, RK; Gera, L; Kozaki, Y; Mizumura, K; Sato, J | 1 |
Bachvarov, DR; Bastien, L; Marceau, F; Sabourin, T | 1 |
Chambers, SS; Christiansen, SC; Eddleston, J; Pan, ZK; Woessner, KM; Ye, R; Zuraw, BL | 1 |
Chang, RS; Chen, TB; Hess, JF; Hey, PJ; Pettibone, DJ | 1 |
Bouthillier, J; Fortin, JP; Marceau, F | 1 |
Kohno, S; Mizutani, N; Nabe, T; Sugahara, S; Takenaka, H | 1 |
Bhoola, KD; Hoffmann, TF; Kuebler, JF; Messmer, K; Roscher, AA; Schremmer-Danninger, E | 1 |
Eisenbarth, H; Petersen, M; Rukwied, R; Schmelz, M | 1 |
Imai, C; Kitamura, Y; Okamura, A; Peng, JF; Printz, MP | 1 |
Binaschi, A; Mantovani, S; Mazzuferi, M; Rodi, D; Simonato, M | 1 |
Argaman, M; Fleisher-Berkovich, S; Levant, A; Levy, E | 1 |
Adam, A; Bawolak, MT; Fortin, JP; Marceau, F; Vogel, LK | 1 |
Bellucci, F; Cucchi, P; Lazzeri, M; Meini, S; Santicioli, P; Turini, D | 1 |
Baltic, S; Bertram, CM; Bhoola, KD; Fogel-Petrovic, M; Foster, PS; Misso, NL; Thompson, PJ | 1 |
Daray, FM; Errasti, AE; Falcioni, AG; Gago, JE; Goldschmidt, ED; Nowak, W; Pelorosso, FG; Pugliese, MI; Rothlin, RP | 1 |
Bova, MP; Butelman, ER; Chavez, RA; Chen, L; Dreyer, M; Fukuda, JY; Garofalo, AW; Hawkinson, JE; Holcomb, R; Hom, DS; Ko, MC; Liao, A; Malmberg, AB; Ruslim, L; Samant, B; Simmonds, S; Szoke, BG; Wadsworth, A; Zeitz, KP; Zhang, H; Zmolek, W | 1 |
Bader, M; Cibrián-Uhalte, E; Costa-Neto, CM; de Picoli Souza, K; Oliveira, L; Oliveira, SM; Pesquero, JB; Santos, EL | 1 |
Bloomfield, P; Cruden, NL; Fox, KA; Lang, NN; Ludlam, CA; Newby, DE; Tse, GH | 1 |
Florkowska, M; Guevara-Lora, I; Kozik, A | 1 |
Mamenko, M; O'Neil, RG; Pochynyuk, O; Zaika, O | 1 |
Cruden, NL; Fox, KA; Lang, NN; MacGillivray, TJ; Newby, DE; Uren, NG | 1 |
Bovenzi, V; Côté, J; Dubuc, C; Fortier, A; Fortin, D; Gobeil, F; Lepage, M; Müller-Esterl, W; Neugebauer, W; Savard, M; Tremblay, L; Tsanaclis, AM | 1 |
Bhoola, KD; Borquez, C; Ehrenfeld, P; Figueroa, CD; Lizama, A; Manso, L; Matus, CE; Naran, A; Pavicic, MF; Poblete, MT; Sarmiento, J | 1 |
Guevara-Lora, I; Kozik, A; Niewiarowska-Sendo, A | 1 |
Burckhardt, BB; Gangnus, T | 1 |
2 trial(s) available for kallidin, des-arg(10)- and bradykinin
Article | Year |
---|---|
Vascular B1 kinin receptors in patients with congestive heart failure.
Topics: Adult; Aged; Angiotensin-Converting Enzyme Inhibitors; Blood Pressure; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cross-Over Studies; Double-Blind Method; Female; Heart Failure; Humans; Infusions, Intra-Arterial; Kallidin; Middle Aged; Nitroprusside; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Tissue Plasminogen Activator; Vasodilation | 2008 |
Vasomotor and fibrinolytic responses to kinin receptor agonists in the atherosclerotic human lower limb.
Topics: Adult; Aged; Analysis of Variance; Angiotensin-Converting Enzyme Inhibitors; Atherosclerosis; Blood Flow Velocity; Bradykinin; Dose-Response Relationship, Drug; Female; Femoral Artery; Fibrinolysis; Humans; Infusions, Intra-Arterial; Kallidin; Lower Extremity; Male; Middle Aged; Nitroprusside; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Scotland; Tissue Plasminogen Activator; Ultrasonography, Doppler; Ultrasonography, Interventional; Vasodilation; Vasodilator Agents; Vasomotor System | 2012 |
46 other study(ies) available for kallidin, des-arg(10)- and bradykinin
Article | Year |
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Differential pharmacology of cloned human and mouse B2 bradykinin receptors.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; DNA, Complementary; Humans; Mice; Molecular Sequence Data; Receptors, Bradykinin; Species Specificity | 1994 |
The agonist selectivity of a mouse B1 bradykinin receptor differs from human and rabbit B1 receptors.
Topics: Amino Acid Sequence; Animals; Base Sequence; Bradykinin; Cattle; Cloning, Molecular; COS Cells; DNA Primers; DNA, Complementary; Humans; Kallidin; Mice; Molecular Sequence Data; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin; Sequence Homology, Amino Acid; Species Specificity; Transfection | 1996 |
Stable expression of the human kinin B1 receptor in Chinese hamster ovary cells. Characterization of ligand binding and effector pathways.
Topics: Animals; Binding, Competitive; Biological Transport; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; GTP-Binding Proteins; Humans; Inositol Phosphates; Kallidin; Ligands; Oligopeptides; Precipitin Tests; Protein Binding; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Proteins; Signal Transduction; Type C Phospholipases | 1997 |
Molecular characterisation of cloned bradykinin B1 receptors from rat and human.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Cell Line; Cloning, Molecular; COS Cells; DNA, Complementary; Female; Gene Expression; Genes; Humans; Kallidin; Molecular Sequence Data; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Tissue Distribution; Tritium | 1999 |
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship | 2013 |
Hypotensive effects of Lys-des-Arg9-bradykinin and metabolically protected agonists of B1 receptors for kinins.
Topics: Animals; Blood Pressure; Bradykinin; Cardiovascular System; Female; Hypotension; Kallidin; Kinins; Lipopolysaccharides; Male; Prostaglandins; Protease Inhibitors; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter | 1991 |
Conversion of B1 kinin receptor-mediated vascular relaxation to contraction.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Bradykinin; Dose-Response Relationship, Drug; Indomethacin; Kallidin; Male; Pyrazoles; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Vasoconstriction; Vasodilation | 1987 |
Bradykinin receptors in mouse and rat isolated superior cervical ganglia.
Topics: Amino Acid Sequence; Animals; Bradykinin; Bradykinin Receptor Antagonists; Electrophysiology; Interleukin-1; Kallidin; Male; Mice; Molecular Sequence Data; Muscarine; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin; Structure-Activity Relationship; Superior Cervical Ganglion | 1995 |
Expression cloning of a human B1 bradykinin receptor.
Topics: Amino Acid Sequence; Animals; Bradykinin; Cloning, Molecular; DNA, Complementary; Gene Expression Regulation; Humans; Interleukin-1; Kallidin; Molecular Sequence Data; Oocytes; Receptors, Bradykinin; Recombinant Proteins; Sequence Homology, Amino Acid; Xenopus laevis | 1994 |
Bradykinin B1 receptors in rabbit aorta smooth muscle cells in culture.
Topics: Animals; Aorta; Binding Sites; Binding, Competitive; Bradykinin; Cells, Cultured; Enzyme Activation; Hydrolysis; Kallidin; Lysophospholipase; Muscle, Smooth, Vascular; Phosphatidylinositols; Rabbits; Receptors, Bradykinin | 1994 |
Analysis of responses to kallidin, DABK, and DAK in feline hindlimb vascular bed.
Topics: Adamantane; Animals; Arginine; Atropine; Blood Vessels; Bradykinin; Bradykinin Receptor Antagonists; Cats; Female; Hindlimb; Kallidin; Male; Meclofenamic Acid; Morpholines; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Potassium Channels | 1995 |
Involvement of bradykinin B1 and B2 receptors in human PMN elastase release and increase in endothelial cell monolayer permeability.
Topics: Amino Acid Chloromethyl Ketones; Bradykinin; Cells, Cultured; Endothelium, Vascular; Humans; In Vitro Techniques; Kallidin; Leukocyte Elastase; Neutrophils; Permeability; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Serine Proteinase Inhibitors | 1996 |
Characterization of the receptor and the mechanisms underlying the inflammatory response induced by des-Arg9-BK in mouse pleurisy.
Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Capillary Permeability; Cell Cycle; Disease Models, Animal; Edema; Inflammation; Kallidin; Kinins; Lipopolysaccharides; Male; Mice; Neuropeptides; Nitric Oxide; Pleura; Pleurisy; Receptors, Bradykinin; Receptors, Tachykinin | 1998 |
Systemic treatment with Mycobacterium bovis bacillus Calmette-Guérin (BCG) potentiates kinin B1 receptor agonist-induced nociception and oedema formation in the formalin test in mice.
Topics: Animals; Bradykinin; Dexamethasone; Dose-Response Relationship, Drug; Drug Synergism; Edema; Formaldehyde; Hindlimb; Indomethacin; Kallidin; Male; Mice; Mycobacterium bovis; Pain; Pain Measurement; Pyrazoles; Receptor, Bradykinin B1; Receptors, Bradykinin | 1998 |
Mechanisms of prostaglandin E2 release by intact cells expressing cyclooxygenase-2: evidence for a 'two-component' model.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Arachidonic Acid; Bradykinin; Calcimycin; Cell Line; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Humans; Inflammation; Interleukin-1; Isoenzymes; Kallidin; Membrane Proteins; Phospholipases A; Phospholipases A2; Prostaglandin-Endoperoxide Synthases; Receptors, Bradykinin | 1999 |
Effect of dexamethasone on cyclophosphamide-induced cystitis in rats: lack of relation with bradykinin B1 receptor-mediated motor responses.
Topics: Animals; Anti-Inflammatory Agents; Binding, Competitive; Bradykinin; Carcinogens; Cyclophosphamide; Cystitis; Dexamethasone; Dose-Response Relationship, Drug; Kallidin; Male; Muscle Contraction; Radioligand Assay; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; Tritium; Urinary Bladder | 1999 |
Changes in hippocampal and cortical B1 bradykinin receptor biological activity in two experimental models of epilepsy.
Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Cerebral Cortex; Electric Stimulation; Epilepsy; Glutamic Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Kallidin; Kindling, Neurologic; Male; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin | 1999 |
Involvement of bradykinin B1 and B2 receptors in pulmonary leukocyte accumulation induced by Sephadex beads in guinea pigs.
Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Bronchoalveolar Lavage Fluid; Cell Count; Dextrans; Guinea Pigs; Indicators and Reagents; Inflammation; Kallidin; Leukocytes; Lung Diseases; Male; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin | 1999 |
Identification of a key region of kinin B(1) receptor for high affinity binding of peptide antagonists.
Topics: Amino Acid Sequence; Animals; Binding Sites; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; Humans; Inositol Phosphates; Kallidin; Molecular Sequence Data; Mutation; Peptides; Protein Binding; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Fusion Proteins; Tetrahydroisoquinolines; Transfection | 2000 |
Regulation of inducible bradykinin B1 receptor gene expression through absence of internalization and resensitization.
Topics: Arachidonic Acid; Blotting, Northern; Bradykinin; Calcium; Cells, Cultured; DNA Primers; Endocytosis; Fibroblasts; Gene Expression Regulation; Genetic Vectors; Humans; Kallidin; Lung; Phosphatidylinositols; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Transfection | 2000 |
Endotoxin sensitization to kinin B(1) receptor agonist in a non-human primate model: haemodynamic and pro-inflammatory effects.
Topics: Animals; Blood Pressure; Body Temperature; Bradykinin; Chlorocebus aethiops; Dose-Response Relationship, Drug; Edema; Endotoxins; Hemodynamics; Inflammation; Kallidin; Lipopolysaccharides; Male; Receptor, Bradykinin B1; Receptors, Bradykinin | 2001 |
Portal hypertensive response to bradykinin in inflamed or cirrhotic rat livers is mediated by B2-type receptors.
Topics: Analysis of Variance; Animals; Bradykinin; Carbon Tetrachloride; Hypertension, Portal; Inflammation; Kallidin; Liver Cirrhosis; Male; Rats; Rats, Wistar; Receptors, Bradykinin; Turpentine | 2001 |
No evidence for bradykinin B1 receptors in rat dorsal root ganglion neurons.
Topics: Animals; Blotting, Northern; Bradykinin; Calcium; Calcium Signaling; Cells, Cultured; Drug Administration Schedule; Fluorescent Dyes; Fura-2; Ganglia, Spinal; Intracellular Fluid; Kallidin; Male; Neuralgia; Neurons, Afferent; Peripheral Nervous System Diseases; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger | 2001 |
B2 receptor-mediated enhanced bradykinin sensitivity of rat cutaneous C-fiber nociceptors during persistent inflammation.
Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Electrophysiology; Hot Temperature; In Vitro Techniques; Inflammation; Kallidin; Male; Nerve Fibers; Nociceptors; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B2; Receptors, Bradykinin; Skin; Stimulation, Chemical; Tachyphylaxis | 2001 |
Agonist-induced translocation of the kinin B(1) receptor to caveolae-related rafts.
Topics: Animals; Antigens, Human Platelet; Bacterial Proteins; beta-Cyclodextrins; Biological Transport; Bradykinin; Caveolae; Caveolin 1; Caveolins; Cell Fractionation; Cells, Cultured; COS Cells; Cyclodextrins; Endocytosis; Green Fluorescent Proteins; Humans; Kallidin; Luminescent Proteins; Membrane Microdomains; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin; Subcellular Fractions; Transfection; Tritium | 2002 |
Up-regulation of functional kinin B1 receptors in allergic airway inflammation.
Topics: Adult; Allergens; Animals; Bradykinin; Case-Control Studies; Enzyme Activation; Epithelial Cells; Humans; In Vitro Techniques; Kallidin; Mitogen-Activated Protein Kinases; Nasal Mucosa; Nasal Provocation Tests; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; RNA, Messenger; Transcription Factor AP-1; Up-Regulation | 2002 |
Molecular and pharmacological diversity of the kinin B1 receptor.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Bradykinin; Chlorocebus aethiops; Cloning, Molecular; Dogs; Gene Frequency; Humans; Kallidin; Macaca mulatta; Molecular Sequence Data; Polymorphism, Single Nucleotide; Rats; Receptor, Bradykinin B1; Receptors, Bradykinin; Recombinant Fusion Proteins; Sequence Alignment; Species Specificity | 2002 |
High agonist-independent clearance of rabbit kinin B1 receptors in cultured cells.
Topics: Animals; Anisomycin; Aorta; Bradykinin; Cells, Cultured; Green Fluorescent Proteins; Humans; Immunoblotting; Indicators and Reagents; Jugular Veins; Kallidin; Kidney; Luminescent Proteins; Muscle Contraction; Muscle, Smooth, Vascular; Protein Synthesis Inhibitors; Rabbits; Radioligand Assay; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Proteins; Tritium | 2003 |
Kinins are involved in the development of allergic nasal hyperresponsiveness in guinea pigs.
Topics: Airway Resistance; Allergens; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Disease Models, Animal; Guinea Pigs; Kallidin; Kinins; Leukotriene D4; Male; Nasal Lavage Fluid; Pollen; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Rhinitis, Allergic, Seasonal; Time Factors | 2003 |
Kinin-B1 receptors in ischaemia-induced pancreatitis: functional importance and cellular localisation.
Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cell Adhesion; GPI-Linked Proteins; Kallidin; Leukocytes; Male; Metalloendopeptidases; Pancreatitis; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Reperfusion Injury; Survival Rate; Up-Regulation; Venules | 2003 |
Sensitization to bradykinin B1 and B2 receptor activation in UV-B irradiated human skin.
Topics: Adult; Analysis of Variance; Bradykinin; Dose-Response Relationship, Drug; Erythema; Female; Humans; Kallidin; Laser-Doppler Flowmetry; Male; Microdialysis; Pain; Pain Measurement; Proteins; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Skin; Time Factors; Ultraviolet Rays | 2004 |
Interleukin-1beta enhanced action of kinins on extracellular matrix of spontaneous hypertensive rat cardiac fibroblasts.
Topics: Animals; Bradykinin; Cells, Cultured; Collagenases; Drug Synergism; Enzyme Precursors; Extracellular Matrix; Fibroblasts; Gelatinases; Gene Expression; Hypertension; Interleukin-1; Kallidin; Matrix Metalloproteinase 9; Metalloendopeptidases; Myocardium; Procollagen; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptor, Bradykinin B1; Receptor, Bradykinin B2; RNA, Messenger; Tissue Inhibitor of Metalloproteinase-1; Tissue Inhibitor of Metalloproteinase-2 | 2005 |
Induction of B1 bradykinin receptors in the kindled hippocampus increases extracellular glutamate levels: a microdialysis study.
Topics: Animals; Behavior, Animal; Bradykinin; Electroencephalography; Extracellular Space; Glutamic Acid; Hippocampus; Kallidin; Kindling, Neurologic; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1 | 2005 |
Kinins and neuroinflammation: dual effect on prostaglandin synthesis.
Topics: Animals; Animals, Newborn; Bradykinin; Cells, Cultured; Dinoprostone; Dose-Response Relationship, Drug; Encephalitis; Kallidin; Kinins; Lipopolysaccharides; Neuroglia; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2 | 2006 |
The bradykinin B2 receptor antagonist icatibant (Hoe 140) blocks aminopeptidase N at micromolar concentrations: off-target alterations of signaling mediated by the bradykinin B1 and angiotensin receptors.
Topics: Angiotensin II; Angiotensin III; Aniline Compounds; Animals; Aorta; Bradykinin; Bradykinin B2 Receptor Antagonists; CD13 Antigens; Dose-Response Relationship, Drug; In Vitro Techniques; Kallidin; Kinetics; Protease Inhibitors; Quinolines; Rabbits; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Angiotensin; Recombinant Proteins; Signal Transduction; Vasoconstriction; Vasoconstrictor Agents | 2006 |
Characterization of kinin receptors in human cultured detrusor smooth muscle cells.
Topics: Bradykinin; Bradykinin B1 Receptor Antagonists; Cells, Cultured; Dinoprostone; Humans; Inositol Phosphates; Interleukin-1beta; Kallidin; Male; Middle Aged; Muscle, Smooth; Ornithine; Radioligand Assay; Receptor, Bradykinin B1; Sulfonamides; Transforming Growth Factor alpha; Urinary Bladder | 2007 |
Expression of kinin B1 and B2 receptors in immature, monocyte-derived dendritic cells and bradykinin-mediated increase in intracellular Ca2+ and cell migration.
Topics: Bradykinin; Calcium; Cell Differentiation; Cell Movement; Cells, Cultured; Dendritic Cells; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Interleukin-4; Intracellular Fluid; Kallidin; Monocytes; Receptor, Bradykinin B1; Receptor, Bradykinin B2 | 2007 |
Functional evidence of des-Arg10-kallidin enzymatic inactivating pathway in isolated human umbilical vein.
Topics: Angiotensin-Converting Enzyme Inhibitors; Bradykinin; Captopril; CD13 Antigens; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Female; Glycopeptides; Humans; In Vitro Techniques; Kallidin; Metalloproteases; Neprilysin; Peptides; Protease Inhibitors; Receptor, Bradykinin B1; Umbilical Veins; Vasoconstriction | 2007 |
Pharmacological, pharmacokinetic, and primate analgesic efficacy profile of the novel bradykinin B1 Receptor antagonist ELN441958.
Topics: Analgesics; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bradykinin; Bradykinin B1 Receptor Antagonists; Calcium; Carrageenan; Cell Line; Cell Membrane Permeability; Fibroblasts; Humans; Hyperalgesia; Kallidin; Macaca mulatta; Mice; Mice, Knockout; Microsomes, Liver; Molecular Structure; Naltrexone; Naproxen; Narcotic Antagonists; Rats; Receptor, Bradykinin B1; Species Specificity; Spiro Compounds; Transfection | 2007 |
Essential role of TM V and VI for binding the C-terminal sequences of Des-Arg-kinins.
Topics: Amino Acid Sequence; Animals; Bradykinin; CHO Cells; Cricetinae; Cricetulus; HeLa Cells; Humans; Kallidin; Molecular Sequence Data; Protein Structure, Tertiary; Rats; Receptor, Bradykinin B1 | 2008 |
Bradykinin-related peptides up-regulate the expression of kinin B1 and B2 receptor genes in human promonocytic cell line U937.
Topics: Bradykinin; Cell Differentiation; Gene Expression; Humans; Immunohistochemistry; Kallidin; Peptides; Phorbol Esters; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Tretinoin; U937 Cells; Up-Regulation | 2009 |
Bradykinin acutely inhibits activity of the epithelial Na+ channel in mammalian aldosterone-sensitive distal nephron.
Topics: Absorption; Aldosterone; Animals; Biosensing Techniques; Bradykinin; Caffeine; Cyclic AMP; Dose-Response Relationship, Drug; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Estrenes; GTP-Binding Protein alpha Subunits, Gq-G11; Hydrolysis; Ion Channel Gating; Kallidin; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Natriuresis; Nephrons; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phosphodiesterase Inhibitors; Pyrrolidinones; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Signal Transduction; Sodium; Sodium Channel Blockers; Thapsigargin; Thionucleotides; Tissue Culture Techniques; Type C Phospholipases | 2011 |
Induction of selective blood-tumor barrier permeability and macromolecular transport by a biostable kinin B1 receptor agonist in a glioma rat model.
Topics: Adult; Aged; Animals; Biological Transport; Bradykinin; Brain Neoplasms; Capillary Permeability; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Glioma; Humans; Kallidin; Male; Middle Aged; Permeability; Rats; Rats, Inbred F344; Receptor, Bradykinin B1 | 2012 |
Bioregulation of kallikrein-related peptidases 6, 10 and 11 by the kinin B₁ receptor in breast cancer cells.
Topics: Bradykinin; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Down-Regulation; Female; Humans; Kallidin; Kallikreins; Kininogens; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; MCF-7 Cells; Neoplasm Invasiveness; Receptor, Bradykinin B1; RNA Interference; RNA, Small Interfering; Serine Endopeptidases; Tissue Kallikreins; Up-Regulation | 2014 |
Kinin Peptides Enhance Inflammatory and Oxidative Responses Promoting Apoptosis in a Parkinson's Disease Cellular Model.
Topics: 1-Methyl-4-phenylpyridinium; Apoptosis; Bradykinin; Cell Differentiation; Cell Line, Tumor; Cell Survival; Cytokines; Humans; Kallidin; Kinins; Oxidative Stress; Parkinson Disease; Reactive Oxygen Species | 2016 |
Targeted LC-MS/MS platform for the comprehensive determination of peptides in the kallikrein-kinin system.
Topics: Bradykinin; Chromatography, Liquid; COVID-19; Humans; Kallidin; Kallikrein-Kinin System; Limit of Detection; Peptide Fragments; Tandem Mass Spectrometry | 2021 |