Page last updated: 2024-09-03

kallidin, des-arg(10)- and bradykinin

kallidin, des-arg(10)- has been researched along with bradykinin in 48 studies

Compound Research Comparison

Studies
(kallidin, des-arg(10)-)
Trials
(kallidin, des-arg(10)-)
Recent Studies (post-2010)
(kallidin, des-arg(10)-)
Studies
(bradykinin)
Trials
(bradykinin)
Recent Studies (post-2010) (bradykinin)
8041714,1953551,520

Protein Interaction Comparison

ProteinTaxonomykallidin, des-arg(10)- (IC50)bradykinin (IC50)
B2 bradykinin receptorHomo sapiens (human)0.0018

Research

Studies (48)

TimeframeStudies, this research(%)All Research%
pre-19901 (2.08)18.7374
1990's16 (33.33)18.2507
2000's24 (50.00)29.6817
2010's6 (12.50)24.3611
2020's1 (2.08)2.80

Authors

AuthorsStudies
Borkowski, JA; Fraher, J; Hess, JF; Macneil, T; Ransom, RW; Stonesifer, GY; Strader, CD1
Borkowski, JA; Derrick, AW; Hess, JF; MacNeil, T1
Austin, CE; Bathon, JM; Chakravarty, S; Faussner, A; Kyle, DJ; Proud, D; Robinson, HE1
Arbuckle, J; Bevan, SJ; Burgess, GM; Davis, C; Docherty, RJ; Jones, C; McIntyre, P; Phillips, E; Webb, M; Yaqoob, M1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
deBlois, D; Drapeau, G; Marceau, F1
Churchill, L; Ward, PE1
Bowery, BJ; Hill, RG; Seabrook, GR1
Bierilo, KK; Borkowski, JA; Derrick, AW; Hess, JF; Linemeyer, DL; MacNeil, T; Menke, JG; Ransom, RW; Schneck, KA; Strader, CD1
Hess, JF; Ransom, RW; Schneck, KA; Stonesifer, GY1
Champion, HC; Del Rio, O; Garrison, EA; Kadowitz, PJ; Santiago, JA; Smith, RE1
Carl, VS; Moore, EE; Moore, FA; Whalley, ET1
Calixto, JB; Vianna, RM1
Calixto, JB; de Campos, RO; Henriques, MG1
Barnes, PJ; Belvisi, MG; Cirino, G; Mitchell, JA; Saunders, MA; Warner, TD1
Criscuoli, M; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Patacchini, R; Tramontana, M1
Beani, L; Bianchi, C; Borea, PA; Bregola, G; Gessi, S; Regoli, D; Simonato, M; Varani, K1
Gobeil, F; Pelletier, S; Perron, MS; Regoli, D; Sirois, P1
Bastian, S; Bonnafous, JC; Loillier, B; Paquet, JL; Pruneau, D; Robert, C1
Polgar, P; Prado, GN; Taylor, L; Yang, X; Zhou, X1
deBlois, D; Horlick, RA1
Borges, DR; Loureiro-Silva, MR; Molina, HM1
Brand, M; Klusch, A; Kurzai, O; Petersen, M; Schmidt, RF; Valdeolmillos, M1
Banik, RK; Gera, L; Kozaki, Y; Mizumura, K; Sato, J1
Bachvarov, DR; Bastien, L; Marceau, F; Sabourin, T1
Chambers, SS; Christiansen, SC; Eddleston, J; Pan, ZK; Woessner, KM; Ye, R; Zuraw, BL1
Chang, RS; Chen, TB; Hess, JF; Hey, PJ; Pettibone, DJ1
Bouthillier, J; Fortin, JP; Marceau, F1
Kohno, S; Mizutani, N; Nabe, T; Sugahara, S; Takenaka, H1
Bhoola, KD; Hoffmann, TF; Kuebler, JF; Messmer, K; Roscher, AA; Schremmer-Danninger, E1
Eisenbarth, H; Petersen, M; Rukwied, R; Schmelz, M1
Imai, C; Kitamura, Y; Okamura, A; Peng, JF; Printz, MP1
Binaschi, A; Mantovani, S; Mazzuferi, M; Rodi, D; Simonato, M1
Argaman, M; Fleisher-Berkovich, S; Levant, A; Levy, E1
Adam, A; Bawolak, MT; Fortin, JP; Marceau, F; Vogel, LK1
Bellucci, F; Cucchi, P; Lazzeri, M; Meini, S; Santicioli, P; Turini, D1
Baltic, S; Bertram, CM; Bhoola, KD; Fogel-Petrovic, M; Foster, PS; Misso, NL; Thompson, PJ1
Daray, FM; Errasti, AE; Falcioni, AG; Gago, JE; Goldschmidt, ED; Nowak, W; Pelorosso, FG; Pugliese, MI; Rothlin, RP1
Bova, MP; Butelman, ER; Chavez, RA; Chen, L; Dreyer, M; Fukuda, JY; Garofalo, AW; Hawkinson, JE; Holcomb, R; Hom, DS; Ko, MC; Liao, A; Malmberg, AB; Ruslim, L; Samant, B; Simmonds, S; Szoke, BG; Wadsworth, A; Zeitz, KP; Zhang, H; Zmolek, W1
Bader, M; Cibrián-Uhalte, E; Costa-Neto, CM; de Picoli Souza, K; Oliveira, L; Oliveira, SM; Pesquero, JB; Santos, EL1
Bloomfield, P; Cruden, NL; Fox, KA; Lang, NN; Ludlam, CA; Newby, DE; Tse, GH1
Florkowska, M; Guevara-Lora, I; Kozik, A1
Mamenko, M; O'Neil, RG; Pochynyuk, O; Zaika, O1
Cruden, NL; Fox, KA; Lang, NN; MacGillivray, TJ; Newby, DE; Uren, NG1
Bovenzi, V; Côté, J; Dubuc, C; Fortier, A; Fortin, D; Gobeil, F; Lepage, M; Müller-Esterl, W; Neugebauer, W; Savard, M; Tremblay, L; Tsanaclis, AM1
Bhoola, KD; Borquez, C; Ehrenfeld, P; Figueroa, CD; Lizama, A; Manso, L; Matus, CE; Naran, A; Pavicic, MF; Poblete, MT; Sarmiento, J1
Guevara-Lora, I; Kozik, A; Niewiarowska-Sendo, A1
Burckhardt, BB; Gangnus, T1

Trials

2 trial(s) available for kallidin, des-arg(10)- and bradykinin

ArticleYear
Vascular B1 kinin receptors in patients with congestive heart failure.
    Journal of cardiovascular pharmacology, 2008, Volume: 52, Issue:5

    Topics: Adult; Aged; Angiotensin-Converting Enzyme Inhibitors; Blood Pressure; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cross-Over Studies; Double-Blind Method; Female; Heart Failure; Humans; Infusions, Intra-Arterial; Kallidin; Middle Aged; Nitroprusside; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Tissue Plasminogen Activator; Vasodilation

2008
Vasomotor and fibrinolytic responses to kinin receptor agonists in the atherosclerotic human lower limb.
    Heart and vessels, 2012, Volume: 27, Issue:2

    Topics: Adult; Aged; Analysis of Variance; Angiotensin-Converting Enzyme Inhibitors; Atherosclerosis; Blood Flow Velocity; Bradykinin; Dose-Response Relationship, Drug; Female; Femoral Artery; Fibrinolysis; Humans; Infusions, Intra-Arterial; Kallidin; Lower Extremity; Male; Middle Aged; Nitroprusside; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Scotland; Tissue Plasminogen Activator; Ultrasonography, Doppler; Ultrasonography, Interventional; Vasodilation; Vasodilator Agents; Vasomotor System

2012

Other Studies

46 other study(ies) available for kallidin, des-arg(10)- and bradykinin

ArticleYear
Differential pharmacology of cloned human and mouse B2 bradykinin receptors.
    Molecular pharmacology, 1994, Volume: 45, Issue:1

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; DNA, Complementary; Humans; Mice; Molecular Sequence Data; Receptors, Bradykinin; Species Specificity

1994
The agonist selectivity of a mouse B1 bradykinin receptor differs from human and rabbit B1 receptors.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Bradykinin; Cattle; Cloning, Molecular; COS Cells; DNA Primers; DNA, Complementary; Humans; Kallidin; Mice; Molecular Sequence Data; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin; Sequence Homology, Amino Acid; Species Specificity; Transfection

1996
Stable expression of the human kinin B1 receptor in Chinese hamster ovary cells. Characterization of ligand binding and effector pathways.
    The Journal of biological chemistry, 1997, Apr-25, Volume: 272, Issue:17

    Topics: Animals; Binding, Competitive; Biological Transport; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; GTP-Binding Proteins; Humans; Inositol Phosphates; Kallidin; Ligands; Oligopeptides; Precipitin Tests; Protein Binding; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Proteins; Signal Transduction; Type C Phospholipases

1997
Molecular characterisation of cloned bradykinin B1 receptors from rat and human.
    European journal of pharmacology, 1999, Jun-25, Volume: 374, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Cell Line; Cloning, Molecular; COS Cells; DNA, Complementary; Female; Gene Expression; Genes; Humans; Kallidin; Molecular Sequence Data; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

1999
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Hypotensive effects of Lys-des-Arg9-bradykinin and metabolically protected agonists of B1 receptors for kinins.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:3

    Topics: Animals; Blood Pressure; Bradykinin; Cardiovascular System; Female; Hypotension; Kallidin; Kinins; Lipopolysaccharides; Male; Prostaglandins; Protease Inhibitors; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter

1991
Conversion of B1 kinin receptor-mediated vascular relaxation to contraction.
    Hypertension (Dallas, Tex. : 1979), 1987, Volume: 9, Issue:6 Pt 2

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Bradykinin; Dose-Response Relationship, Drug; Indomethacin; Kallidin; Male; Pyrazoles; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Vasoconstriction; Vasodilation

1987
Bradykinin receptors in mouse and rat isolated superior cervical ganglia.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Amino Acid Sequence; Animals; Bradykinin; Bradykinin Receptor Antagonists; Electrophysiology; Interleukin-1; Kallidin; Male; Mice; Molecular Sequence Data; Muscarine; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin; Structure-Activity Relationship; Superior Cervical Ganglion

1995
Expression cloning of a human B1 bradykinin receptor.
    The Journal of biological chemistry, 1994, Aug-26, Volume: 269, Issue:34

    Topics: Amino Acid Sequence; Animals; Bradykinin; Cloning, Molecular; DNA, Complementary; Gene Expression Regulation; Humans; Interleukin-1; Kallidin; Molecular Sequence Data; Oocytes; Receptors, Bradykinin; Recombinant Proteins; Sequence Homology, Amino Acid; Xenopus laevis

1994
Bradykinin B1 receptors in rabbit aorta smooth muscle cells in culture.
    European journal of pharmacology, 1994, Feb-15, Volume: 266, Issue:3

    Topics: Animals; Aorta; Binding Sites; Binding, Competitive; Bradykinin; Cells, Cultured; Enzyme Activation; Hydrolysis; Kallidin; Lysophospholipase; Muscle, Smooth, Vascular; Phosphatidylinositols; Rabbits; Receptors, Bradykinin

1994
Analysis of responses to kallidin, DABK, and DAK in feline hindlimb vascular bed.
    The American journal of physiology, 1995, Volume: 269, Issue:6 Pt 2

    Topics: Adamantane; Animals; Arginine; Atropine; Blood Vessels; Bradykinin; Bradykinin Receptor Antagonists; Cats; Female; Hindlimb; Kallidin; Male; Meclofenamic Acid; Morpholines; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Potassium Channels

1995
Involvement of bradykinin B1 and B2 receptors in human PMN elastase release and increase in endothelial cell monolayer permeability.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Amino Acid Chloromethyl Ketones; Bradykinin; Cells, Cultured; Endothelium, Vascular; Humans; In Vitro Techniques; Kallidin; Leukocyte Elastase; Neutrophils; Permeability; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Serine Proteinase Inhibitors

1996
Characterization of the receptor and the mechanisms underlying the inflammatory response induced by des-Arg9-BK in mouse pleurisy.
    British journal of pharmacology, 1998, Volume: 123, Issue:2

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Capillary Permeability; Cell Cycle; Disease Models, Animal; Edema; Inflammation; Kallidin; Kinins; Lipopolysaccharides; Male; Mice; Neuropeptides; Nitric Oxide; Pleura; Pleurisy; Receptors, Bradykinin; Receptors, Tachykinin

1998
Systemic treatment with Mycobacterium bovis bacillus Calmette-Guérin (BCG) potentiates kinin B1 receptor agonist-induced nociception and oedema formation in the formalin test in mice.
    Neuropeptides, 1998, Volume: 32, Issue:5

    Topics: Animals; Bradykinin; Dexamethasone; Dose-Response Relationship, Drug; Drug Synergism; Edema; Formaldehyde; Hindlimb; Indomethacin; Kallidin; Male; Mice; Mycobacterium bovis; Pain; Pain Measurement; Pyrazoles; Receptor, Bradykinin B1; Receptors, Bradykinin

1998
Mechanisms of prostaglandin E2 release by intact cells expressing cyclooxygenase-2: evidence for a 'two-component' model.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Arachidonic Acid; Bradykinin; Calcimycin; Cell Line; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Humans; Inflammation; Interleukin-1; Isoenzymes; Kallidin; Membrane Proteins; Phospholipases A; Phospholipases A2; Prostaglandin-Endoperoxide Synthases; Receptors, Bradykinin

1999
Effect of dexamethasone on cyclophosphamide-induced cystitis in rats: lack of relation with bradykinin B1 receptor-mediated motor responses.
    European journal of pharmacology, 1999, Mar-12, Volume: 369, Issue:1

    Topics: Animals; Anti-Inflammatory Agents; Binding, Competitive; Bradykinin; Carcinogens; Cyclophosphamide; Cystitis; Dexamethasone; Dose-Response Relationship, Drug; Kallidin; Male; Muscle Contraction; Radioligand Assay; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; Tritium; Urinary Bladder

1999
Changes in hippocampal and cortical B1 bradykinin receptor biological activity in two experimental models of epilepsy.
    Neuroscience, 1999, Volume: 92, Issue:3

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Cerebral Cortex; Electric Stimulation; Epilepsy; Glutamic Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Kallidin; Kindling, Neurologic; Male; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin

1999
Involvement of bradykinin B1 and B2 receptors in pulmonary leukocyte accumulation induced by Sephadex beads in guinea pigs.
    European journal of pharmacology, 1999, Jul-02, Volume: 376, Issue:1-2

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Bronchoalveolar Lavage Fluid; Cell Count; Dextrans; Guinea Pigs; Indicators and Reagents; Inflammation; Kallidin; Leukocytes; Lung Diseases; Male; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin

1999
Identification of a key region of kinin B(1) receptor for high affinity binding of peptide antagonists.
    The Journal of biological chemistry, 2000, Mar-03, Volume: 275, Issue:9

    Topics: Amino Acid Sequence; Animals; Binding Sites; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; Humans; Inositol Phosphates; Kallidin; Molecular Sequence Data; Mutation; Peptides; Protein Binding; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Fusion Proteins; Tetrahydroisoquinolines; Transfection

2000
Regulation of inducible bradykinin B1 receptor gene expression through absence of internalization and resensitization.
    Journal of cellular biochemistry, 2000, Jun-06, Volume: 78, Issue:3

    Topics: Arachidonic Acid; Blotting, Northern; Bradykinin; Calcium; Cells, Cultured; DNA Primers; Endocytosis; Fibroblasts; Gene Expression Regulation; Genetic Vectors; Humans; Kallidin; Lung; Phosphatidylinositols; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Transfection

2000
Endotoxin sensitization to kinin B(1) receptor agonist in a non-human primate model: haemodynamic and pro-inflammatory effects.
    British journal of pharmacology, 2001, Volume: 132, Issue:1

    Topics: Animals; Blood Pressure; Body Temperature; Bradykinin; Chlorocebus aethiops; Dose-Response Relationship, Drug; Edema; Endotoxins; Hemodynamics; Inflammation; Kallidin; Lipopolysaccharides; Male; Receptor, Bradykinin B1; Receptors, Bradykinin

2001
Portal hypertensive response to bradykinin in inflamed or cirrhotic rat livers is mediated by B2-type receptors.
    Journal of gastroenterology and hepatology, 2001, Volume: 16, Issue:1

    Topics: Analysis of Variance; Animals; Bradykinin; Carbon Tetrachloride; Hypertension, Portal; Inflammation; Kallidin; Liver Cirrhosis; Male; Rats; Rats, Wistar; Receptors, Bradykinin; Turpentine

2001
No evidence for bradykinin B1 receptors in rat dorsal root ganglion neurons.
    Neuroreport, 2001, Oct-08, Volume: 12, Issue:14

    Topics: Animals; Blotting, Northern; Bradykinin; Calcium; Calcium Signaling; Cells, Cultured; Drug Administration Schedule; Fluorescent Dyes; Fura-2; Ganglia, Spinal; Intracellular Fluid; Kallidin; Male; Neuralgia; Neurons, Afferent; Peripheral Nervous System Diseases; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger

2001
B2 receptor-mediated enhanced bradykinin sensitivity of rat cutaneous C-fiber nociceptors during persistent inflammation.
    Journal of neurophysiology, 2001, Volume: 86, Issue:6

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Electrophysiology; Hot Temperature; In Vitro Techniques; Inflammation; Kallidin; Male; Nerve Fibers; Nociceptors; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B2; Receptors, Bradykinin; Skin; Stimulation, Chemical; Tachyphylaxis

2001
Agonist-induced translocation of the kinin B(1) receptor to caveolae-related rafts.
    Molecular pharmacology, 2002, Volume: 61, Issue:3

    Topics: Animals; Antigens, Human Platelet; Bacterial Proteins; beta-Cyclodextrins; Biological Transport; Bradykinin; Caveolae; Caveolin 1; Caveolins; Cell Fractionation; Cells, Cultured; COS Cells; Cyclodextrins; Endocytosis; Green Fluorescent Proteins; Humans; Kallidin; Luminescent Proteins; Membrane Microdomains; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin; Subcellular Fractions; Transfection; Tritium

2002
Up-regulation of functional kinin B1 receptors in allergic airway inflammation.
    Journal of immunology (Baltimore, Md. : 1950), 2002, Aug-15, Volume: 169, Issue:4

    Topics: Adult; Allergens; Animals; Bradykinin; Case-Control Studies; Enzyme Activation; Epithelial Cells; Humans; In Vitro Techniques; Kallidin; Mitogen-Activated Protein Kinases; Nasal Mucosa; Nasal Provocation Tests; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; RNA, Messenger; Transcription Factor AP-1; Up-Regulation

2002
Molecular and pharmacological diversity of the kinin B1 receptor.
    International immunopharmacology, 2002, Volume: 2, Issue:13-14

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Bradykinin; Chlorocebus aethiops; Cloning, Molecular; Dogs; Gene Frequency; Humans; Kallidin; Macaca mulatta; Molecular Sequence Data; Polymorphism, Single Nucleotide; Rats; Receptor, Bradykinin B1; Receptors, Bradykinin; Recombinant Fusion Proteins; Sequence Alignment; Species Specificity

2002
High agonist-independent clearance of rabbit kinin B1 receptors in cultured cells.
    American journal of physiology. Heart and circulatory physiology, 2003, Volume: 284, Issue:5

    Topics: Animals; Anisomycin; Aorta; Bradykinin; Cells, Cultured; Green Fluorescent Proteins; Humans; Immunoblotting; Indicators and Reagents; Jugular Veins; Kallidin; Kidney; Luminescent Proteins; Muscle Contraction; Muscle, Smooth, Vascular; Protein Synthesis Inhibitors; Rabbits; Radioligand Assay; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Proteins; Tritium

2003
Kinins are involved in the development of allergic nasal hyperresponsiveness in guinea pigs.
    European journal of pharmacology, 2003, Aug-29, Volume: 476, Issue:3

    Topics: Airway Resistance; Allergens; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Disease Models, Animal; Guinea Pigs; Kallidin; Kinins; Leukotriene D4; Male; Nasal Lavage Fluid; Pollen; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Rhinitis, Allergic, Seasonal; Time Factors

2003
Kinin-B1 receptors in ischaemia-induced pancreatitis: functional importance and cellular localisation.
    Biological chemistry, 2003, Volume: 384, Issue:9

    Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cell Adhesion; GPI-Linked Proteins; Kallidin; Leukocytes; Male; Metalloendopeptidases; Pancreatitis; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Reperfusion Injury; Survival Rate; Up-Regulation; Venules

2003
Sensitization to bradykinin B1 and B2 receptor activation in UV-B irradiated human skin.
    Pain, 2004, Volume: 110, Issue:1-2

    Topics: Adult; Analysis of Variance; Bradykinin; Dose-Response Relationship, Drug; Erythema; Female; Humans; Kallidin; Laser-Doppler Flowmetry; Male; Microdialysis; Pain; Pain Measurement; Proteins; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Regional Blood Flow; Skin; Time Factors; Ultraviolet Rays

2004
Interleukin-1beta enhanced action of kinins on extracellular matrix of spontaneous hypertensive rat cardiac fibroblasts.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2005, Volume: 27, Issue:1

    Topics: Animals; Bradykinin; Cells, Cultured; Collagenases; Drug Synergism; Enzyme Precursors; Extracellular Matrix; Fibroblasts; Gelatinases; Gene Expression; Hypertension; Interleukin-1; Kallidin; Matrix Metalloproteinase 9; Metalloendopeptidases; Myocardium; Procollagen; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptor, Bradykinin B1; Receptor, Bradykinin B2; RNA, Messenger; Tissue Inhibitor of Metalloproteinase-1; Tissue Inhibitor of Metalloproteinase-2

2005
Induction of B1 bradykinin receptors in the kindled hippocampus increases extracellular glutamate levels: a microdialysis study.
    Neuroscience, 2005, Volume: 135, Issue:3

    Topics: Animals; Behavior, Animal; Bradykinin; Electroencephalography; Extracellular Space; Glutamic Acid; Hippocampus; Kallidin; Kindling, Neurologic; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1

2005
Kinins and neuroinflammation: dual effect on prostaglandin synthesis.
    European journal of pharmacology, 2006, Sep-28, Volume: 546, Issue:1-3

    Topics: Animals; Animals, Newborn; Bradykinin; Cells, Cultured; Dinoprostone; Dose-Response Relationship, Drug; Encephalitis; Kallidin; Kinins; Lipopolysaccharides; Neuroglia; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2

2006
The bradykinin B2 receptor antagonist icatibant (Hoe 140) blocks aminopeptidase N at micromolar concentrations: off-target alterations of signaling mediated by the bradykinin B1 and angiotensin receptors.
    European journal of pharmacology, 2006, Dec-03, Volume: 551, Issue:1-3

    Topics: Angiotensin II; Angiotensin III; Aniline Compounds; Animals; Aorta; Bradykinin; Bradykinin B2 Receptor Antagonists; CD13 Antigens; Dose-Response Relationship, Drug; In Vitro Techniques; Kallidin; Kinetics; Protease Inhibitors; Quinolines; Rabbits; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Angiotensin; Recombinant Proteins; Signal Transduction; Vasoconstriction; Vasoconstrictor Agents

2006
Characterization of kinin receptors in human cultured detrusor smooth muscle cells.
    British journal of pharmacology, 2007, Volume: 150, Issue:2

    Topics: Bradykinin; Bradykinin B1 Receptor Antagonists; Cells, Cultured; Dinoprostone; Humans; Inositol Phosphates; Interleukin-1beta; Kallidin; Male; Middle Aged; Muscle, Smooth; Ornithine; Radioligand Assay; Receptor, Bradykinin B1; Sulfonamides; Transforming Growth Factor alpha; Urinary Bladder

2007
Expression of kinin B1 and B2 receptors in immature, monocyte-derived dendritic cells and bradykinin-mediated increase in intracellular Ca2+ and cell migration.
    Journal of leukocyte biology, 2007, Volume: 81, Issue:6

    Topics: Bradykinin; Calcium; Cell Differentiation; Cell Movement; Cells, Cultured; Dendritic Cells; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Interleukin-4; Intracellular Fluid; Kallidin; Monocytes; Receptor, Bradykinin B1; Receptor, Bradykinin B2

2007
Functional evidence of des-Arg10-kallidin enzymatic inactivating pathway in isolated human umbilical vein.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Bradykinin; Captopril; CD13 Antigens; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Female; Glycopeptides; Humans; In Vitro Techniques; Kallidin; Metalloproteases; Neprilysin; Peptides; Protease Inhibitors; Receptor, Bradykinin B1; Umbilical Veins; Vasoconstriction

2007
Pharmacological, pharmacokinetic, and primate analgesic efficacy profile of the novel bradykinin B1 Receptor antagonist ELN441958.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 322, Issue:2

    Topics: Analgesics; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bradykinin; Bradykinin B1 Receptor Antagonists; Calcium; Carrageenan; Cell Line; Cell Membrane Permeability; Fibroblasts; Humans; Hyperalgesia; Kallidin; Macaca mulatta; Mice; Mice, Knockout; Microsomes, Liver; Molecular Structure; Naltrexone; Naproxen; Narcotic Antagonists; Rats; Receptor, Bradykinin B1; Species Specificity; Spiro Compounds; Transfection

2007
Essential role of TM V and VI for binding the C-terminal sequences of Des-Arg-kinins.
    International immunopharmacology, 2008, Volume: 8, Issue:2

    Topics: Amino Acid Sequence; Animals; Bradykinin; CHO Cells; Cricetinae; Cricetulus; HeLa Cells; Humans; Kallidin; Molecular Sequence Data; Protein Structure, Tertiary; Rats; Receptor, Bradykinin B1

2008
Bradykinin-related peptides up-regulate the expression of kinin B1 and B2 receptor genes in human promonocytic cell line U937.
    Acta biochimica Polonica, 2009, Volume: 56, Issue:3

    Topics: Bradykinin; Cell Differentiation; Gene Expression; Humans; Immunohistochemistry; Kallidin; Peptides; Phorbol Esters; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Tretinoin; U937 Cells; Up-Regulation

2009
Bradykinin acutely inhibits activity of the epithelial Na+ channel in mammalian aldosterone-sensitive distal nephron.
    American journal of physiology. Renal physiology, 2011, Volume: 300, Issue:5

    Topics: Absorption; Aldosterone; Animals; Biosensing Techniques; Bradykinin; Caffeine; Cyclic AMP; Dose-Response Relationship, Drug; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Estrenes; GTP-Binding Protein alpha Subunits, Gq-G11; Hydrolysis; Ion Channel Gating; Kallidin; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Natriuresis; Nephrons; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phosphodiesterase Inhibitors; Pyrrolidinones; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Signal Transduction; Sodium; Sodium Channel Blockers; Thapsigargin; Thionucleotides; Tissue Culture Techniques; Type C Phospholipases

2011
Induction of selective blood-tumor barrier permeability and macromolecular transport by a biostable kinin B1 receptor agonist in a glioma rat model.
    PloS one, 2012, Volume: 7, Issue:5

    Topics: Adult; Aged; Animals; Biological Transport; Bradykinin; Brain Neoplasms; Capillary Permeability; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Glioma; Humans; Kallidin; Male; Middle Aged; Permeability; Rats; Rats, Inbred F344; Receptor, Bradykinin B1

2012
Bioregulation of kallikrein-related peptidases 6, 10 and 11 by the kinin B₁ receptor in breast cancer cells.
    Anticancer research, 2014, Volume: 34, Issue:12

    Topics: Bradykinin; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Down-Regulation; Female; Humans; Kallidin; Kallikreins; Kininogens; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; MCF-7 Cells; Neoplasm Invasiveness; Receptor, Bradykinin B1; RNA Interference; RNA, Small Interfering; Serine Endopeptidases; Tissue Kallikreins; Up-Regulation

2014
Kinin Peptides Enhance Inflammatory and Oxidative Responses Promoting Apoptosis in a Parkinson's Disease Cellular Model.
    Mediators of inflammation, 2016, Volume: 2016

    Topics: 1-Methyl-4-phenylpyridinium; Apoptosis; Bradykinin; Cell Differentiation; Cell Line, Tumor; Cell Survival; Cytokines; Humans; Kallidin; Kinins; Oxidative Stress; Parkinson Disease; Reactive Oxygen Species

2016
Targeted LC-MS/MS platform for the comprehensive determination of peptides in the kallikrein-kinin system.
    Analytical and bioanalytical chemistry, 2021, Volume: 413, Issue:11

    Topics: Bradykinin; Chromatography, Liquid; COVID-19; Humans; Kallidin; Kallikrein-Kinin System; Limit of Detection; Peptide Fragments; Tandem Mass Spectrometry

2021