Page last updated: 2024-09-04

ivabradine and uk 68798

ivabradine has been researched along with uk 68798 in 2 studies

Compound Research Comparison

Studies
(ivabradine)
Trials
(ivabradine)
Recent Studies (post-2010)
(ivabradine)
Studies
(uk 68798)
Trials
(uk 68798)
Recent Studies (post-2010) (uk 68798)
1,14319783369865199

Protein Interaction Comparison

ProteinTaxonomyivabradine (IC50)uk 68798 (IC50)
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.1455

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Duff, HJ; Gerull, B; Guo, J; Kudaibergenova, M; Lees-Miller, J; Muruve, DA; Noskov, SY; Ol'khovich, M; Perissinotti, L; Perlovich, GL; Sharapova, A1
Gabrielsson, J; Jirstrand, M; Martel, E; Pairet, N; Scheuerer, S; Wallman, M1

Other Studies

2 other study(ies) available for ivabradine and uk 68798

ArticleYear
The Pore-Lipid Interface: Role of Amino-Acid Determinants of Lipophilic Access by Ivabradine to the hERG1 Pore Domain.
    Molecular pharmacology, 2019, Volume: 96, Issue:2

    Topics: Binding Sites; Ether-A-Go-Go Potassium Channels; Humans; Ivabradine; Membrane Lipids; Models, Molecular; Molecular Docking Simulation; Molecular Dynamics Simulation; Mutagenesis, Site-Directed; Phenethylamines; Protein Binding; Protein Structure, Tertiary; Sulfonamides

2019
An Integrative Approach for Improved Assessment of Cardiovascular Safety Data.
    The Journal of pharmacology and experimental therapeutics, 2021, Volume: 377, Issue:2

    Topics: Animals; Biomarkers, Pharmacological; Blood Pressure; Cardiotoxicity; Cardiovascular Agents; Heart Rate; Ivabradine; Male; Phenethylamines; Pyridazines; Rats; Rats, Wistar; Sildenafil Citrate; Sulfonamides

2021