Page last updated: 2024-09-04

ivabradine and ranolazine

ivabradine has been researched along with ranolazine in 26 studies

Compound Research Comparison

Studies
(ivabradine)
Trials
(ivabradine)
Recent Studies (post-2010)
(ivabradine)
Studies
(ranolazine)
Trials
(ranolazine)
Recent Studies (post-2010) (ranolazine)
1,143197833799104498

Protein Interaction Comparison

ProteinTaxonomyivabradine (IC50)ranolazine (IC50)
Sodium channel protein type 5 subunit alphaHomo sapiens (human)6.85
Voltage-gated sodium channel Nav1.5 cardiac isoform Canis lupus familiaris (dog)6.9

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (19.23)29.6817
2010's19 (73.08)24.3611
2020's2 (7.69)2.80

Authors

AuthorsStudies
Cuisiat, F; Le Grand, B; Létienne, R; Mas, A; Pignier, C; Rolland, F; Vacher, B1
Barsness, GW; Yang, EH1
Chaitman, BR; Sano, J1
Arora, R; Jawad, E1
DiMarco, JP; Mason, PK1
Battler, A; Dvir, D1
Köster, R; Meinertz, T1
Carbajal, EV; Deedwania, PC1
Henderson, RA; Timmis, AD1
Athanasiadis, A; Sechtem, U1
De Silva, R; Purcell, H1
Brambilla, G; Dei Cas, L; Della Pina, P; Gavazzoni, M; Gorga, E; Raddino, R; Regazzoni, V1
Crea, F; Di Franco, A; Di Monaco, A; Lamendola, P; Lanza, GA; Nerla, R; Sarullo, FM; Sestito, A; Tarzia, P; Villano, A1
Jacobshagen, C1
Jones, DA; Timmis, A; Wragg, A1
Biscaglia, S; Valgimigli, M1
Batatinha, JA; Belardinelli, L; Bonatti, R; Liu, G; Nearing, BD; Rajamani, S; Silva, AF; Verrier, RL; Zeng, D1
Mittal, SR1
Castriota, F; Cremonesi, A; De Luca, G; Fattori, R; Lupi, A; Marino, PN; Mirabella, F; Parisi, R; Rognoni, A; Secco, GG1
Dixit, D; Kimborowicz, K1
Cacciapuoti, F1
Colombo, A; Fragasso, G; Fumero, A; Giannini, F; Godino, C; Maranta, F; Margonato, A; Oppizzi, M; Slavich, M1
Balla, C; Ferrari, R; Pavasini, R1
Chen, T; Fang, X; Huang, J; Xu, X; Zhao, Q; Zheng, J; Zhu, H2
Tolunay, H1

Reviews

16 review(s) available for ivabradine and ranolazine

ArticleYear
Evolving treatment strategies for chronic refractory angina.
    Expert opinion on pharmacotherapy, 2006, Volume: 7, Issue:3

    Topics: Acetanilides; Angina Pectoris; Arginine; Benzazepines; Cardiovascular Agents; Chronic Disease; Combined Modality Therapy; Counterpulsation; Electric Stimulation Therapy; Humans; Ivabradine; Myocardial Revascularization; Piperazines; Randomized Controlled Trials as Topic; Ranolazine; Spinal Cord

2006
Novel therapeutic approaches to treating chronic angina in the setting of chronic ischemic heart disease.
    Clinical cardiology, 2007, Volume: 30, Issue:2 Suppl 1

    Topics: Acetanilides; Adrenergic beta-Antagonists; Angina Pectoris; Angiotensin-Converting Enzyme Inhibitors; Benzazepines; Calcium Channel Blockers; Chronic Disease; Enzyme Inhibitors; Humans; Ivabradine; Myocardial Ischemia; Nicorandil; Nitro Compounds; Piperazines; Ranolazine; rho-Associated Kinases; Sinoatrial Node; Trimetazidine; Vasodilator Agents

2007
Chronic stable angina pectoris.
    Disease-a-month : DM, 2008, Volume: 54, Issue:9

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetanilides; Angina Pectoris; Antihypertensive Agents; Benzazepines; Bosentan; Chronic Disease; Counterpulsation; Cyclic Nucleotide-Gated Cation Channels; Exercise Test; Heart Murmurs; Humans; Ivabradine; Myocardial Contraction; Myocardial Ischemia; Myocardial Revascularization; Myocardium; Nicorandil; Oxygen Consumption; Perhexiline; Piperazines; Protein Kinase Inhibitors; Ranolazine; Sulfonamides; Trimetazidine; Vasodilator Agents

2008
New pharmacological agents for arrhythmias.
    Circulation. Arrhythmia and electrophysiology, 2009, Volume: 2, Issue:5

    Topics: Acetanilides; Adenosine A1 Receptor Agonists; Amiodarone; Anisoles; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Benzazepines; Benzofurans; Clinical Trials as Topic; Dronedarone; Humans; Ivabradine; Piperazines; Pyrrolidines; Ranolazine

2009
Conventional and novel drug therapeutics to relief myocardial ischemia.
    Cardiovascular drugs and therapy, 2010, Volume: 24, Issue:4

    Topics: Acetanilides; Adrenergic beta-Antagonists; Angina Pectoris; Angiotensin-Converting Enzyme Inhibitors; Aspirin; Benzazepines; Calcium Channel Blockers; Cardiovascular Agents; Cardiovascular System; Coronary Artery Disease; Hemodynamics; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Ivabradine; Nicorandil; Nitrates; Piperazines; Ranolazine

2010
[New agents for the therapy of angina pectoris].
    Der Internist, 2011, Volume: 52, Issue:7

    Topics: Acetanilides; Angina Pectoris; Benzazepines; Coronary Artery Disease; Cyclic Nucleotide-Gated Cation Channels; Double-Blind Method; Drug Approval; Enzyme Inhibitors; Humans; Ivabradine; Nicorandil; Piperazines; Randomized Controlled Trials as Topic; Ranolazine; Vasodilator Agents

2011
Medical therapy versus myocardial revascularization in chronic coronary syndrome and stable angina.
    The American journal of medicine, 2011, Volume: 124, Issue:8

    Topics: Acetanilides; Adrenergic beta-Antagonists; Angina Pectoris; Angiotensin-Converting Enzyme Inhibitors; Benzazepines; Calcium Channel Blockers; Cardiovascular Agents; Coronary Disease; Drug Therapy, Combination; Humans; Hypolipidemic Agents; Ivabradine; Myocardial Revascularization; Nitrates; Piperazines; Ranolazine; Treatment Outcome

2011
[Almanac 2011: Stable coronary artery disease. An editorial overview of selected research that has driven recent advances in clinical cardiology].
    Giornale italiano di cardiologia (2006), 2012, Volume: 13, Issue:4

    Topics: Acetanilides; Angioplasty, Balloon, Coronary; Anti-Arrhythmia Agents; Benzazepines; Biomarkers; Cardiology; Coronary Artery Bypass; Coronary Artery Disease; Drug-Eluting Stents; Enzyme Inhibitors; Evidence-Based Medicine; Humans; Ivabradine; Natriuretic Agents; Natriuretic Peptide, Brain; Piperazines; Randomized Controlled Trials as Topic; Ranolazine; Risk Assessment; Risk Factors; Treatment Outcome

2012
[Late sodium current and calcium overload--pathogenesis and adequate treatment].
    Deutsche medizinische Wochenschrift (1946), 2013, Volume: 138, Issue:16

    Topics: Acetanilides; Adrenergic beta-Antagonists; Angina Pectoris; Atrial Fibrillation; Benzazepines; Calcium; Calcium Channel Blockers; Cardiovascular Agents; Coronary Artery Disease; Electrocardiography; Endothelium, Vascular; Heart Failure, Diastolic; Humans; Hypercalcemia; Ivabradine; Myocardial Ischemia; Nitrates; Piperazines; Ranolazine; Sodium; Sodium Channels; Sodium-Calcium Exchanger

2013
Novel drugs for treating angina.
    BMJ (Clinical research ed.), 2013, Sep-09, Volume: 347

    Topics: Acetanilides; Angina Pectoris; Benzazepines; Enzyme Inhibitors; Heart Rate; Humans; Ivabradine; Nicorandil; Piperazines; Ranolazine; Trimetazidine; Vasodilator Agents

2013
Stable angina pectoris.
    Current atherosclerosis reports, 2014, Volume: 16, Issue:7

    Topics: Acetanilides; Angina, Stable; Benzazepines; Coronary Artery Bypass; Coronary Artery Disease; Coronary Vasospasm; Echocardiography, Stress; Exercise Test; Humans; Ivabradine; Microvessels; Nicorandil; Nitrates; Percutaneous Coronary Intervention; Piperazines; Ranolazine; Smoking Cessation; Vasodilator Agents

2014
Old and New Drugs for Treatment of Stable Angina: New Anti-Anginal Drugs and Coronary Revascularization.
    Cardiovascular & hematological agents in medicinal chemistry, 2015, Volume: 13, Issue:1

    Topics: Angina, Stable; Animals; Benzazepines; Cardiovascular Agents; Humans; Ivabradine; Nicorandil; Percutaneous Coronary Intervention; Ranolazine; Trimetazidine

2015
Pharmacologic management of chronic stable angina.
    JAAPA : official journal of the American Academy of Physician Assistants, 2015, Volume: 28, Issue:6

    Topics: Adrenergic beta-Antagonists; Angina, Stable; Benzazepines; Calcium Channel Blockers; Cardiovascular Agents; Humans; Isosorbide Dinitrate; Ivabradine; Nicorandil; Nitroglycerin; Ranolazine; Sodium Channel Blockers; Vasodilator Agents

2015
Ranolazine and Ivabradine: two different modalities to act against ischemic heart disease.
    Therapeutic advances in cardiovascular disease, 2016, Volume: 10, Issue:2

    Topics: Angina, Stable; Benzazepines; Cardiovascular Agents; Heart Rate; Humans; Ivabradine; Myocardial Ischemia; Oxygen Consumption; Ranolazine

2016
Treatment of Angina: Where Are We?
    Cardiology, 2018, Volume: 140, Issue:1

    Topics: Adrenergic beta-Antagonists; Angina, Stable; Calcium Channel Blockers; Cardiovascular Agents; Chest Pain; Humans; Ivabradine; Nicorandil; Patient Selection; Practice Guidelines as Topic; Ranolazine; Treatment Outcome; Trimetazidine

2018
Effects of the Antianginal Drugs Ranolazine, Nicorandil, and Ivabradine on Coronary Microvascular Function in Patients With Nonobstructive Coronary Artery Disease: A Meta-analysis of Randomized Controlled Trials.
    Clinical therapeutics, 2019, Volume: 41, Issue:10

    Topics: Angina Pectoris; Cardiovascular Agents; Coronary Artery Disease; Humans; Ivabradine; Myocardial Ischemia; Nicorandil; Randomized Controlled Trials as Topic; Ranolazine; Treatment Outcome

2019

Trials

1 trial(s) available for ivabradine and ranolazine

ArticleYear
Effects of ivabradine and ranolazine in patients with microvascular angina pectoris.
    The American journal of cardiology, 2013, Jul-01, Volume: 112, Issue:1

    Topics: Acetanilides; Analysis of Variance; Angina Pectoris; Benzazepines; Chi-Square Distribution; Coronary Angiography; Enzyme Inhibitors; Exercise Test; Female; Humans; Ivabradine; Male; Middle Aged; Piperazines; Placebos; Quality of Life; Ranolazine; Surveys and Questionnaires; Treatment Outcome

2013

Other Studies

9 other study(ies) available for ivabradine and ranolazine

ArticleYear
Sodium late current blockers in ischemia reperfusion: is the bullet magic?
    Journal of medicinal chemistry, 2008, Jul-10, Volume: 51, Issue:13

    Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Female; Guinea Pigs; Humans; Imaging, Three-Dimensional; Male; Models, Molecular; Molecular Structure; Myocardial Ischemia; Rabbits; Rats; Rats, Wistar; Reperfusion; Sodium Channel Blockers; Structure-Activity Relationship

2008
[Update coronary artery disease: important progresses in acute and chronic therapy].
    MMW Fortschritte der Medizin, 2012, Mar-22, Volume: 154, Issue:5

    Topics: Acetanilides; Angina Pectoris; Angioplasty, Balloon, Coronary; Benzazepines; Coronary Artery Disease; Early Medical Intervention; Humans; Ivabradine; Myocardial Infarction; Piperazines; Platelet Aggregation Inhibitors; Practice Guidelines as Topic; Randomized Controlled Trials as Topic; Ranolazine; Survival Rate; Thrombolytic Therapy

2012
Treating stable angina - is there a NICE way towards an international consensus?
    International journal of clinical practice, 2012, Volume: 66, Issue:7

    Topics: Acetanilides; Angina, Stable; Anti-Arrhythmia Agents; Benzazepines; Cardiac Imaging Techniques; Consensus; Humans; International Cooperation; Ivabradine; Myocardial Revascularization; Nicorandil; Piperazines; Practice Guidelines as Topic; Ranolazine; Vasodilator Agents

2012
[New pharmacological approaches to ischemic heart disease].
    Giornale italiano di cardiologia (2006), 2012, Volume: 13, Issue:10 Suppl 2

    Topics: Acetanilides; Benzazepines; Humans; Ivabradine; Myocardial Ischemia; Piperazines; Ranolazine

2012
Combined actions of ivabradine and ranolazine reduce ventricular rate during atrial fibrillation.
    Journal of cardiovascular electrophysiology, 2015, Volume: 26, Issue:3

    Topics: Animals; Atrial Fibrillation; Benzazepines; Cardiovascular Agents; Drug Therapy, Combination; Guinea Pigs; Heart Rate; Ivabradine; Male; Ranolazine; Swine

2015
Slow junctional rhythm, QTc prolongation and transient torsades de-pointes following combined use of Ivabradine, Diltiazem and Ranolazine.
    The Journal of the Association of Physicians of India, 2014, Volume: 62, Issue:5

    Topics: Acetanilides; Aged, 80 and over; Angina, Unstable; Benzazepines; Bradycardia; Diltiazem; Drug Interactions; Drug Substitution; Drug Therapy, Combination; Electrocardiography; Female; Humans; Ivabradine; Long QT Syndrome; Piperazines; Ranolazine; Torsades de Pointes

2014
Long-Term Preservation of Left Ventricular Systolic Function in Patients With Refractory Angina Pectoris and Inducible Myocardial Ischemia on Optimal Medical Therapy.
    The American journal of cardiology, 2016, 05-15, Volume: 117, Issue:10

    Topics: Aged; Angina Pectoris; Benzazepines; Cardiovascular Agents; Echocardiography; Exercise Test; Female; Follow-Up Studies; Humans; Ivabradine; Male; Myocardial Ischemia; Ranolazine; Retrospective Studies; Sodium Channel Blockers; Stroke Volume; Systole; Time Factors; Tomography, Emission-Computed, Single-Photon; Trimetazidine; Vasodilator Agents; Ventricular Function, Left

2016
Does Ranolazine Reduce Pain Perception With Cerebral Effect?
    Clinical therapeutics, 2020, Volume: 42, Issue:2

    Topics: Acetanilides; Coronary Artery Disease; Humans; Ivabradine; Nicorandil; Pain Perception; Randomized Controlled Trials as Topic; Ranolazine

2020
Response to Letter Regarding Article, "Effects of the Antianginal Drugs Ranolazine, Nicorandil and Ivabradine on Coronary Microvascular Function in Patients with Non-obstructive Coronary Artery Disease: A Meta-analysis of Randomized Controlled Trials".
    Clinical therapeutics, 2020, Volume: 42, Issue:2

    Topics: Coronary Artery Disease; Humans; Ivabradine; Nicorandil; Randomized Controlled Trials as Topic; Ranolazine

2020