isradipine and caffeine

isradipine has been researched along with caffeine in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19902 (12.50)18.7374
1990's5 (31.25)18.2507
2000's4 (25.00)29.6817
2010's5 (31.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Coronado, R; el-Hayek, R; Hogan, K; Parness, J; Valdivia, HH1
Dacquet, C; Martin, C; Mironneau, C; Mironneau, J1
Dacquet, C; Mironneau, C; Mironneau, J1
Duprat, AM; Gualandris-Parisot, L; Leclerc, C; Moreau, M1
Damiani, E; Larsson, L; Margreth, A1
Bkaily, G; D'Orléans-Juste, P; Economos, D; Jaalouk, D; Jacques, D; Naik, R; Pothier, P1
Aardal, S; Helle, KB; Lillestłl, IK1
Armstrong, RB; Hamilton, SL; Ingalls, CP; Warren, GL; Zhang, JZ1
Boehm, S; Geier, P; Gupta, KD; Kubista, H; Lagler, M; Rubi, L; Schandl, U; Spies, D1

Reviews

1 review(s) available for isradipine and caffeine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

15 other study(ies) available for isradipine and caffeine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Dantrolene and azumolene inhibit [3H]PN200-110 binding to porcine skeletal muscle dihydropyridine receptors.
    Biochemical and biophysical research communications, 1992, Sep-16, Volume: 187, Issue:2

    Topics: Animals; Caffeine; Calcium Channels; Dantrolene; Dihydropyridines; Imidazoles; Isradipine; Malignant Hyperthermia; Muscle Relaxants, Central; Muscles; Oxazoles; Receptors, Cholinergic; Receptors, Nicotinic; Ryanodine; Ryanodine Receptor Calcium Release Channel; Sarcoplasmic Reticulum; Swine; Tritium

1992
Caffeine-induced inhibition of calcium channel current in cultured smooth cells from pregnant rat myometrium.
    British journal of pharmacology, 1989, Volume: 98, Issue:2

    Topics: Animals; Binding, Competitive; Caffeine; Calcium Channels; Electrophysiology; Female; In Vitro Techniques; Isradipine; Kinetics; Muscle, Smooth; Myometrium; Pregnancy; Pyridines; Rats; Sarcolemma

1989
Effects of calcium entry blockers on calcium-dependent contractions of rat portal vein.
    British journal of pharmacology, 1987, Volume: 92, Issue:1

    Topics: Animals; Caffeine; Calcium; Calcium Channel Blockers; Diltiazem; In Vitro Techniques; Isradipine; Muscle Contraction; Muscle, Smooth, Vascular; Oxadiazoles; Portal Vein; Potassium; Rats; Rats, Inbred Strains

1987
Increased internal Ca2+ mediates neural induction in the amphibian embryo.
    Proceedings of the National Academy of Sciences of the United States of America, 1994, Dec-20, Volume: 91, Issue:26

    Topics: Alkaloids; Animals; Caffeine; Calcium; Calcium Channels; Cells, Cultured; Concanavalin A; Ectoderm; Embryonic Induction; In Vitro Techniques; Ion Channel Gating; Isradipine; Nervous System; Nimodipine; Pleurodeles; Protein Kinase C; Ryanodine; Staurosporine; Tetradecanoylphorbol Acetate

1994
Age-related abnormalities in regulation of the ryanodine receptor in rat fast-twitch muscle.
    Cell calcium, 1996, Volume: 19, Issue:1

    Topics: Aging; Animals; Antibiotics, Antineoplastic; Binding Sites; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium-Calmodulin-Dependent Protein Kinases; Calcium-Transporting ATPases; Calmodulin; Calmodulin-Binding Proteins; Dose-Response Relationship, Drug; Doxorubicin; Isradipine; Kinetics; Male; Membrane Proteins; Muscle Fibers, Fast-Twitch; Muscle Proteins; Muscle, Skeletal; Phosphodiesterase Inhibitors; Rats; Rats, Wistar; Ryanodine Receptor Calcium Release Channel; Sensitivity and Specificity; Tritium

1996
Endothelin-1 and insulin activate the steady-state voltage dependent R-type Ca2+ channel in aortic smooth muscle cells via a pertussis toxin and cholera toxin sensitive G-protein.
    Molecular and cellular biochemistry, 1998, Volume: 183, Issue:1-2

    Topics: Animals; Aorta; Caffeine; Calcium Channels; Cholera Toxin; Endothelin-1; GTP-Binding Proteins; Indoles; Insulin; Ion Transport; Isradipine; Maleimides; Muscle, Smooth, Vascular; Nifedipine; Pertussis Toxin; Protein Kinase C; Rabbits; Ryanodine; Virulence Factors, Bordetella

1998
Relaxing effects of cyclic GMP and cyclic AMP-enhancing agents on the long-lasting contraction to endothelin-1 in the porcine coronary artery.
    Scandinavian journal of clinical and laboratory investigation, 1998, Volume: 58, Issue:8

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Atrial Natriuretic Factor; Caffeine; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Colforsin; Coronary Vessels; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Endothelin-1; In Vitro Techniques; Isradipine; Milrinone; Muscle, Smooth, Vascular; Papaverine; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Purinones; Pyrrolidinones; Rolipram; Swine; Vasoactive Intestinal Peptide; Vasoconstriction; Vasodilation; Verapamil; Vinca Alkaloids

1998
Dihydropyridine and ryanodine receptor binding after eccentric contractions in mouse skeletal muscle.
    Journal of applied physiology (Bethesda, Md. : 1985), 2004, Volume: 96, Issue:5

    Topics: Animals; Binding Sites; Caffeine; Calcium Channels, L-Type; Female; Isometric Contraction; Isradipine; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Skeletal; Ryanodine Receptor Calcium Release Channel; Tarsus, Animal; Torque; Wounds and Injuries

2004
Raised activity of L-type calcium channels renders neurons prone to form paroxysmal depolarization shifts.
    Neuromolecular medicine, 2013, Volume: 15, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Anthracenes; Caffeine; Calcium Channels, L-Type; Calcium Signaling; Cells, Cultured; Dimethyl Sulfoxide; Epilepsy; Excitatory Postsynaptic Potentials; Hippocampus; Hydrogen Peroxide; Isradipine; Magnesium; Neurons; Oxidative Stress; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley

2013