Page last updated: 2024-08-21

isoxazoles and sazetidine-a

isoxazoles has been researched along with sazetidine-a in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brunner, D; Caldarone, B; Cavino, K; Eaton, JB; Fedolak, A; Ghavami, A; Kozikowski, AP; Liu, J; Lowe, DA; Lukas, RJ; Ruiz, C; Terry, M; Wang, D; Yu, LF1
Brown, JL; Wonnacott, S1

Other Studies

2 other study(ies) available for isoxazoles and sazetidine-a

ArticleYear
Discovery of isoxazole analogues of sazetidine-A as selective α4β2-nicotinic acetylcholine receptor partial agonists for the treatment of depression.
    Journal of medicinal chemistry, 2011, Oct-27, Volume: 54, Issue:20

    Topics: Animals; Antidepressive Agents; Azetidines; Behavior, Animal; Binding, Competitive; Blood Proteins; Drug Partial Agonism; Humans; In Vitro Techniques; Isoxazoles; Mice; Microsomes, Liver; Nicotinic Agonists; Protein Binding; Pyridines; Rats; Receptors, Neurotransmitter; Receptors, Nicotinic; Structure-Activity Relationship

2011
Sazetidine-A Activates and Desensitizes Native α7 Nicotinic Acetylcholine Receptors.
    Neurochemical research, 2015, Volume: 40, Issue:10

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Azetidines; Benzamides; Bridged Bicyclo Compounds; Calcium; Cell Line, Tumor; Humans; Isoxazoles; Mice; Neurons; Patch-Clamp Techniques; Phenylurea Compounds; Pyridines; Receptors, Nicotinic

2015