isoxazoles has been researched along with pyrrolidine in 5 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (20.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 3 (60.00) | 24.3611 |
2020's | 1 (20.00) | 2.80 |
Authors | Studies |
---|---|
Fotsch, C; St Jean, DJ | 1 |
Buriak, J; Fevig, JM; Knabb, RM; Lam, GN; Stouten, PF; Wexler, RR; Wong, PC | 1 |
Chiacchio, U; Corsaro, A; Merino, P; Romeo, G | 1 |
Baumann, U; Brunstein, E; Gainsford, GJ; Ianes, C; Knippschild, U; Krüger, M; Luxenburger, A; Peifer, C; Pichlo, C; Schmidt, D; von Drathen, T | 1 |
Cerqueira, AFR; Guieu, S; Paz, FAA; Snarskis, G; Tomé, AC; Zurauskas, J | 1 |
2 review(s) available for isoxazoles and pyrrolidine
Article | Year |
---|---|
Mitigating heterocycle metabolism in drug discovery.
Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats | 2012 |
Chemical synthesis of heterocyclic-sugar nucleoside analogues.
Topics: Carbohydrates; Dioxolanes; Heterocyclic Compounds; Isoxazoles; Nucleosides; Oxazoles; Pyrrolidines; Sulfhydryl Compounds; Sulfides; Thiazolidines | 2010 |
3 other study(ies) available for isoxazoles and pyrrolidine
Article | Year |
---|---|
Preparation of pyrrolidine and isoxazolidine benzamidines as potent inhibitors of coagulation factor Xa.
Topics: Animals; Benzamidines; Factor Xa Inhibitors; Isoxazoles; Models, Molecular; Pyrrolidines; Rabbits | 1999 |
Design, Synthesis and Biological Evaluation of Isoxazole-Based CK1 Inhibitors Modified with Chiral Pyrrolidine Scaffolds.
Topics: Adenosine Triphosphate; Binding Sites; Casein Kinase Idelta; Crystallography, X-Ray; Drug Design; Enzyme Inhibitors; Humans; Isoxazoles; Ligands; Multiprotein Complexes; Pyrrolidines; Structure-Activity Relationship | 2019 |
Site-Selective Modification of a Porpholactone-Selective Synthesis of 12,13- and 17,18-Dihydroporpholactones.
Topics: Isoxazoles; Lactones; Porphyrins; Pyrrolidines; X-Ray Diffraction | 2020 |