Page last updated: 2024-08-21

isoxazoles and mefloquine

isoxazoles has been researched along with mefloquine in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Franzblau, SG; Kozikowski, AP; Mao, J; Wan, B; Wang, Y1
Franzblau, SG; Huang, Q; Kozikowski, AP; Mao, J; Pieroni, M; van Breemen, RB; Wan, B; Wang, Y; Yuan, H1
Franzblau, SG; He, R; Mao, J; Pak, D; Wan, B; Wang, Y; Yuan, H1

Other Studies

3 other study(ies) available for isoxazoles and mefloquine

ArticleYear
HTS, chemical hybridization, and drug design identify a chemically unique antituberculosis agent-coupling serendipity and rational approaches to drug discovery.
    ChemMedChem, 2007, Volume: 2, Issue:6

    Topics: Animals; Antitubercular Agents; Cell Line; Chlorocebus aethiops; Drug Delivery Systems; Drug Design; Isoxazoles; Leucine; Mefloquine; Mice; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Small Molecule Libraries; Vero Cells

2007
From serendipity to rational antituberculosis drug discovery of mefloquine-isoxazole carboxylic acid esters.
    Journal of medicinal chemistry, 2009, Nov-26, Volume: 52, Issue:22

    Topics: Animals; Antitubercular Agents; Chlorocebus aethiops; Drug Discovery; Esters; Female; Humans; Isoxazoles; Mefloquine; Mice; Microbial Sensitivity Tests; Microsomes, Liver; Mycobacterium tuberculosis; Vero Cells

2009
Synthesis and antituberculosis activity of novel mefloquine-isoxazole carboxylic esters as prodrugs.
    Bioorganic & medicinal chemistry letters, 2010, Feb-01, Volume: 20, Issue:3

    Topics: Antitubercular Agents; Carboxylic Acids; Esters; Humans; Isoxazoles; Mefloquine; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Prodrugs

2010