Compounds > isoxazoles
Page last updated: 2024-08-21

isoxazoles and epiboxidine

isoxazoles has been researched along with epiboxidine in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (14.29)18.2507
2000's4 (57.14)29.6817
2010's2 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Badio, B; Daly, JW; Garraffo, HM; Padgett, WL; Plummer, CV1
Daly, JW; Federova, I; Fitch, RW; Gupta, T; Kaneko, Y; Pei, XF; Shi, D1
Armstrong, A; Bhonoah, Y; Shanahan, SE1
Clementi, F; Dallanoce, C; De Amici, M; Gotti, C; Magrone, P; Matera, C; Pucci, L; Rizzi, L1
Bazza, P; Clementi, F; Dallanoce, C; De Amici, M; Frydenvang, K; Gotti, C; Grazioso, G; Magrone, P; Riganti, L; Rizzi, L1
Dallanoce, C; De Amici, M; Grazioso, G; Liberti, V; Roda, G1
Clementi, F; Dallanoce, C; De Amici, M; De Micheli, C; Gotti, C; Matera, C; Pucci, L; Rizzi, L1

Other Studies

7 other study(ies) available for isoxazoles and epiboxidine

ArticleYear
Synthesis and nicotinic activity of epiboxidine: an isoxazole analogue of epibatidine.
    European journal of pharmacology, 1997, Feb-26, Volume: 321, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Cerebral Cortex; Ganglia; Isoxazoles; Kinetics; Male; Mice; Nicotine; Nicotinic Agonists; Nociceptors; PC12 Cells; Pyrrolidines; Rats; Receptors, Nicotinic; Tritium

1997
Homoepiboxidines: further potent agonists for nicotinic receptors.
    Bioorganic & medicinal chemistry, 2004, Jan-02, Volume: 12, Issue:1

    Topics: Analgesics; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cell Line, Tumor; Humans; Isoxazoles; Male; Mice; Nicotinic Agonists; PC12 Cells; Protein Binding; Pyridines; Rats; Receptors, Nicotinic

2004
Aza-Prins-pinacol approach to 7-azabicyclo[2.2.1]heptanes: syntheses of (+/-)-epibatidine and (+/-)-epiboxidine.
    The Journal of organic chemistry, 2007, Oct-12, Volume: 72, Issue:21

    Topics: Aza Compounds; Azabicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Heptanes; Isoxazoles; Molecular Structure; Oligopeptides; Pyridines; Stereoisomerism

2007
Epiboxidine and novel-related analogues: a convenient synthetic approach and estimation of their affinity at neuronal nicotinic acetylcholine receptor subtypes.
    Bioorganic & medicinal chemistry letters, 2008, Aug-15, Volume: 18, Issue:16

    Topics: Animals; Binding, Competitive; Catalysis; Cerebral Cortex; Chemistry, Pharmaceutical; Drug Design; Isoxazoles; Kinetics; Ligands; Models, Chemical; Neurons; Rats; Receptors, Nicotinic; Structure-Activity Relationship; Temperature

2008
New analogues of epiboxidine incorporating the 4,5-dihydroisoxazole nucleus: synthesis, binding affinity at neuronal nicotinic acetylcholine receptors, and molecular modeling investigations.
    Chemistry & biodiversity, 2009, Volume: 6, Issue:2

    Topics: Isoxazoles; Kinetics; Models, Molecular; Protein Binding; Receptors, Nicotinic; Structure-Activity Relationship

2009
Determination of acid dissociation constants of compounds active at neuronal nicotinic acetylcholine receptors by means of electrophoretic and potentiometric techniques.
    Analytical sciences : the international journal of the Japan Society for Analytical Chemistry, 2010, Volume: 26, Issue:1

    Topics: Buffers; Drug Industry; Electrophoresis, Capillary; Isoxazoles; Kinetics; Nicotinic Agonists; Potentiometry; Receptors, Nicotinic; Solubility; Solvents

2010
The enantiomers of epiboxidine and of two related analogs: synthesis and estimation of their binding affinity at α4β2 and α7 neuronal nicotinic acetylcholine receptors.
    Chirality, 2012, Volume: 24, Issue:7

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Chemistry Techniques, Synthetic; Isoxazoles; Neurons; Protein Binding; Rats; Receptors, Nicotinic; Stereoisomerism

2012