Page last updated: 2024-08-21

isoxazoles and bicuculline

isoxazoles has been researched along with bicuculline in 103 studies

Research

Studies (103)

TimeframeStudies, this research(%)All Research%
pre-199060 (58.25)18.7374
1990's18 (17.48)18.2507
2000's14 (13.59)29.6817
2010's11 (10.68)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gale, KN; Guidotti, A1
Gallager, DW; Tallman, JF; Thomas, JW1
Mohler, H; Okada, T1
Curtis, DR; Johnston, GA; Krogsgaard-Larsen, P; Lodge, D1
Snodgrass, SR1
Polc, P1
Braestrup, C; Falch, E; Krogsgaard-Larsen, P; Nielsen, M1
Andrews, PR; Johnston, GA1
Boissier, JR; Dumont, C; Oberlander, C1
Arnt, J; Scheel-Krüger, J1
Leach, MJ; Wilson, JA1
Andre, JM; Boulanger, T; Durant, F; Hoffmann, R; Rognan, D; Vercauteren, DP; Wermuth, CG1
Johnston, GA1
Bonaventure, N; Jardon, B; Kim, MS; Yücel, H1
Ebbesson, SO; Erdö, SL; Hofmann, MH; Malz, CR; Meyer, DL1
Bapna, JS; Ramaswamy, S; Srinivasan, D1
Agmo, A; Gutiérrez, M; Guzmán, M; Pruneda, R1
Bergen, HT; Hejtmancik, JF; Pfaff, DW1
Fromm, GH; Mukawa, J; Nakata, M1
Heinricher, MM; Kaplan, HJ1
Falch, E; Kristiansen, U; Krogsgaard-Larsen, P; Lambert, JD1
Hicks, TP; Kaneko, T1
Amenta, F; Erdö, SL; Mione, MC; Wolff, JR1
Agmo, A; Paredes, R; Soria, P1
Bapna, JS; Ramaswamy, S; Suthakaran, C1
Graeff, FG; Milani, H1
Fujimoto, M; Guidotti, A; Hanbauer, I; Kataoka, Y1
Pooler, GW; Steward, EG1
Mehta, AK; Ticku, MK1
Byberg, JR; Curtis, DR; Falch, E; Gynther, BD; Hjeds, H; Krogsgaard-Larsen, P; Labouta, IM1
Alho, H; Fujimoto, M; Geffard, M; Guidotti, A; Hanbauer, I; Kataoka, Y; Kelly, GD1
Bagri, A; Di Scala, G; Sandner, G1
Iversen, LL; Wong, EH1
Agmo, A; Paredes, R1
Agmo, A; Giordano, M1
Curtis, DR; Falch, E; Krogsgaard-Larsen, P; Nielsen, L1
Depaulis, A; Vergnes, M3
Brandao, ML; Di Scala, G; Karli, P; Schmitt, P1
Bristow, DR; Watling, KJ1
Allan, AM; Harris, RA1
Belhage, B; Meier, E; Schousboe, A1
Apud, JA; Masotto, C; Racagni, G1
Chweh, AY; Swinyard, EA; Wolf, HH1
Lindgren, S1
DaSilva, AM; Gatti, PJ; Gillis, RA1
Gillis, RA; Hamosh, P; Hartley, B; Quest, JA; Taveira da Silva, AM1
Drower, EJ; Hammond, DL1
Zarkovsky, AM1
Borsini, F; Evangelista, S; Meli, A1
Sawynok, J1
Karobath, M; Supavilai, P1
Benson, DI; Klepner, CA; Squires, RF1
Carmona, E; Gomes, C; Trolin, G1
Cavagnini, F; Grandison, L; Guidotti, A; Invitti, SC; Schmid, R1
Blavet, N; Clostre, F; DeFeudis, FV1
Dias Souza, J; Gillis, RA; Quest, JA; Williford, DJ1
Dutton, GR; Freedman, EG; Pearce, BR1
Breese, GR; Frye, GD1
Blavet, N; DeFeudis, FV1
Curtis, DR; Falch, E; Krogsgaard-Larsen, P; Leah, JD; Peet, MJ1
Maksay, G; Ticku, MK1
Bloch, R; Bousquet, P; Feldman, J; Schwartz, J1
Di Scala, G; Karli, P; Schmitt, P1
Baumeister, AA; Frye, GD1
DeFeudis, FV; Grognet, A; Hertz, F1
Mueller, AL; Schwartzkroin, PA; Taube, JS1
Coward, DM1
Cheney, DL; McGill, W; Murray, TF1
Alger, BE; Nicoll, RA1
Aghajanian, GK; Gellman, RL1
Abdulla, FA; Calaminici, MR; Gray, JA; Raevsky, VV; Sinden, JD; Stephenson, JD1
Liske, S; Morris, ME1
Kim, HY; Olsen, RW; Sapp, DW; Tobin, AJ1
Matsutani, S; Yamamoto, N1
Bedingfield, JB; Calder, LD; Karler, R; Thai, DK1
Agmo, A; Contreras, JL; Paredes, RG1
Lerma, J; López-García, JC; Rodríguez-Moreno, A1
Kulinskii, VI; Mikhel'son, GV1
Ebert, B; Fjalland, B; Hansen, SL; Kristiansen, U1
Brünig, I; Fritschy, JM; Studler, B1
Platt, B; White, AM1
Frosini, M; Sgaragli, G; Valoti, M1
Hansen, SL; Sánchez, C; Sperling, BB1
Gong, QH; Shen, H; Smith, SS; Yuan, M1
Goldstein, PA; Harrison, NL; Jia, F; Pignataro, L; Schofield, CM; Yue, M1
Jia, H; Qu, CL; Tang, JS1
Park, JB; Skalska, S; Son, S; Stern, JE1
Hutson, PH; McDonald, LM; Sheppard, WF; Sohal, B; Staveley, SM; Tattersall, FD1
Anderson, NJ; Cremers, TI; Ebert, B; Fahey, JM; Rasmussen, S; Sánchez, C; Vogel, V1
Balfour, DJ; Belelli, D; Brown, VJ; Chandra, D; Foister, N; Herd, MB; Homanics, GE; Lambert, JJ; Peden, DR1
Belcastro, V; Calabresi, P; Costa, C; Ientile, R; Luchetti, E; Picconi, B; Pisani, F; Siliquini, S; Tantucci, M; Tozzi, A1
Avoli, M; Dzakpasu, R; Gonzalez-Sulser, A; Motamedi, GK; Vicini, S; Wang, J1
Bonin, RP; De Koninck, Y; Eng, DG; Labrakakis, C; Orser, BA; Whissell, PD1
Dretchen, KL; Gillis, RA; Herman, MA; Sahibzada, N; Vicini, S1
Charbonnet, M; Gold, MS; Lee, KY1
Kalappa, BI; Uteshev, VV1
Jeon, BH; Jeong, JA; Jo, JY; Kim, HW; Kim, YJ; Lee, GS; Lee, JU; Pandit, S; Park, JB; Song, JG1
Bondy, B; Cui, N; Jiang, C; Jin, X; Johnson, CM; Oginsky, MF; Wu, Y; Zhang, S; Zhong, W1
Bohnsack, JP; Carlson, SL; Morrow, AL; Patel, V1
Johnston, GAR1
Browning, KN; McMenamin, CA; Travagli, RA1

Reviews

3 review(s) available for isoxazoles and bicuculline

ArticleYear
GABAA agonists as targets for drug development.
    Clinical and experimental pharmacology & physiology, 1992, Volume: 19, Issue:1

    Topics: Acetates; Acrylates; Amines; Analgesics; Anthelmintics; Anticonvulsants; Bicuculline; Computer Simulation; Cyclohexanecarboxylic Acids; Cyclopentanes; Drug Design; Gabapentin; gamma-Aminobutyric Acid; Isoxazoles; Molecular Conformation; Molecular Weight; Receptors, GABA-A

1992
Molecular pharmacology of the GABA receptors and GABA agonists.
    Advances in biochemical psychopharmacology, 1983, Volume: 37

    Topics: Animals; Bicuculline; gamma-Aminobutyric Acid; Humans; Isoxazoles; Molecular Conformation; Muscimol; Neurons; Receptors, Cell Surface; Receptors, GABA-A; Stereoisomerism; Synapses

1983
GABA Australis, some reflections on the history of GABA receptor research in Australia.
    Pharmacological research, 2017, Volume: 116

    Topics: Animals; Australia; Baclofen; Bicuculline; Cyclic AMP; Humans; Isoxazoles; Muscimol; Receptors, GABA

2017

Other Studies

100 other study(ies) available for isoxazoles and bicuculline

ArticleYear
GABA-mediated control of rat neostriatal tyrosine hydroxylase revealed by intranigral muscimol.
    Nature, 1976, Oct-21, Volume: 263, Issue:5579

    Topics: Aminobutyrates; Animals; Bicuculline; Caudate Nucleus; Corpus Striatum; Dopamine; Enzyme Activation; gamma-Aminobutyric Acid; Haloperidol; Isoxazoles; Kinetics; Neural Pathways; Olfactory Bulb; Oxazoles; Pimozide; Pteridines; Quaternary Ammonium Compounds; Rats; Substantia Nigra; Tyrosine 3-Monooxygenase

1976
GABAergic modulation of benzodiazepine binding site sensitivity.
    Nature, 1978, Jul-27, Volume: 274, Issue:5669

    Topics: Amanita; Aminobutyrates; Animals; Bicuculline; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Ligands; Neurotransmitter Agents; Rats; Receptors, Drug; Receptors, Neurotransmitter

1978
GABA receptor binding with 3H (+) bicuculline-methiodide in rat CNS.
    Nature, 1977, May-05, Volume: 267, Issue:5606

    Topics: Aminobutyrates; Animals; Bicuculline; Binding, Competitive; Brain; Cell Membrane; Cerebellum; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isoquinolines; Isoxazoles; Kinetics; Rats; Receptors, Neurotransmitter; Stereoisomerism; Taurine

1977
A new class of GABA agonist.
    Nature, 1977, Jul-07, Volume: 268, Issue:5615

    Topics: Action Potentials; Aminobutyrates; Animals; Bicuculline; Biological Transport; Cats; gamma-Aminobutyric Acid; Interneurons; Isonicotinic Acids; Isoxazoles; Molecular Conformation; Neural Inhibition; Oxazoles; Receptors, Neurotransmitter; Spinal Cord; Structure-Activity Relationship; Synaptic Transmission

1977
Use of 3H-muscimol for GABA receptor studies.
    Nature, 1978, Jun-01, Volume: 273, Issue:5661

    Topics: Aminobutyrates; Animals; Bicuculline; Binding, Competitive; Brain; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Oxazoles; Potassium; Rats; Receptors, Neurotransmitter; Stereoisomerism; Synaptosomes

1978
Effects of GABA-mimetic agents on the cat spinal cord.
    Progress in neuro-psychopharmacology, 1979, Volume: 3, Issue:4

    Topics: Animals; Bicuculline; Cats; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Ibotenic Acid; Isonicotinic Acids; Isoxazoles; Male; Muscimol; Neurons, Afferent; Spinal Cord

1979
Partial agonists for brain GABA/benzodiazepine receptor complex.
    Nature, 1979, Jul-26, Volume: 280, Issue:5720

    Topics: Animals; Benzodiazepines; Bicuculline; Brain; Crotonates; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, Drug; Sulfonic Acids

1979
Conformational analysis of muscimol, a GABA agonist.
    Journal of theoretical biology, 1979, Aug-07, Volume: 79, Issue:3

    Topics: Bicuculline; Binding Sites; gamma-Aminobutyric Acid; Isoxazoles; Models, Molecular; Molecular Conformation; Muscimol; Oxazoles; Quantum Theory

1979
Rotational behaviour after unilateral intranigral injection of muscimol in rats.
    European journal of pharmacology, 1977, Jun-15, Volume: 43, Issue:4

    Topics: Aminobutyrates; Animals; Basidiomycota; Behavior; Bicuculline; gamma-Aminobutyric Acid; Humans; Injections; Isoxazoles; Male; Oxazoles; Picrotoxin; Rats; Stereotyped Behavior; Substantia Nigra; Time Factors

1977
GABA in the ventral tegmental area: differential regional effects on locomotion, aggression and food intake after microinjection of GABA agonists and antagonists.
    Life sciences, 1979, Oct-08, Volume: 25, Issue:15

    Topics: Aggression; Animals; Apomorphine; Behavior, Animal; Bicuculline; Carbachol; Cerebral Cortex; Dopamine; Feeding Behavior; gamma-Aminobutyric Acid; Haloperidol; Humans; Isoxazoles; Male; Methyltyrosines; Morphine; Motor Activity; Muscimol; Picrotoxin; Rats; Reserpine

1979
GABA receptor binding with 3H-muscimol in calf cerebellum.
    European journal of pharmacology, 1978, Apr-01, Volume: 48, Issue:3

    Topics: Aminobutyrates; Animals; Bicuculline; Cattle; Cerebellum; gamma-Aminobutyric Acid; In Vitro Techniques; Isoxazoles; Kinetics; Oxazoles; Receptors, Drug

1978
Structure and molecular modeling of GABAA receptor antagonists.
    Journal of medicinal chemistry, 1992, May-29, Volume: 35, Issue:11

    Topics: Alkaloids; Androstanes; Azasteroids; Azepines; Bicuculline; Crystallization; Dibenzazepines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Heterocyclic Compounds, 4 or More Rings; Heterocyclic Compounds, Bridged-Ring; Isoxazoles; Lactones; Models, Molecular; Molecular Conformation; Molecular Structure; Piperidines; Pyridazines; Receptors, GABA-A; Structure-Activity Relationship; Tubocurarine; X-Ray Diffraction

1992
Pharmacological study of the chicken's monocular optokinetic nystagmus: effects of GABAergic agonist and antagonists.
    Vision research, 1992, Volume: 32, Issue:4

    Topics: Animals; Bicuculline; Chickens; Electroretinography; Eye Movements; Injections; Isoxazoles; Nystagmus, Optokinetic; Picrotoxin; Receptors, GABA-A; Retina; Vision, Monocular; Visual Pathways

1992
Changes in ligand binding to GABAA receptor sites in pacific salmon (Oncorhynchus) brain during spawning migration and "aging".
    Journal fur Hirnforschung, 1992, Volume: 33, Issue:4-5

    Topics: Aging; Aminobutyrates; Analgesics; Animals; Baclofen; Bicuculline; Binding, Competitive; Brain; Female; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Ligands; Male; Muscimol; Receptors, GABA-A; Salmon; Sexual Behavior, Animal

1992
Inhibition of tetrahydroisoxazolo-pyridin-3-ol and muscimol and its mechanism on gastrointestinal transit in mice.
    European journal of pharmacology, 1992, Sep-22, Volume: 220, Issue:2-3

    Topics: Animals; Bicuculline; Dose-Response Relationship, Drug; Drug Interactions; Gastrointestinal Transit; Isoxazoles; Male; Mice; Muscimol; Phentolamine; Propranolol; Yohimbine

1992
GABAergic drugs and conflict behavior in the rat: lack of similarities with the actions of benzodiazepines.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:3

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Behavior, Animal; Benzodiazepines; Bicuculline; Brain; Conflict, Psychological; Drug Interactions; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Nicotinic Acids; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission

1991
Effects of gamma-aminobutyric acid receptor agonists and antagonist on LHRH-synthesizing neurons as detected by immunocytochemistry and in situ hybridization.
    Experimental brain research, 1991, Volume: 87, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Female; GABA-A Receptor Antagonists; Gene Expression Regulation; Gonadotropin-Releasing Hormone; Immunohistochemistry; Isoxazoles; Neurons; Nucleic Acid Hybridization; Ovariectomy; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; RNA Probes; RNA, Messenger

1991
Why are most GABA agonists not effective antiepileptic drugs?
    The Japanese journal of psychiatry and neurology, 1991, Volume: 45, Issue:2

    Topics: Animals; Anticonvulsants; Bicuculline; Cats; Electroencephalography; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Muscimol; Receptors, GABA-A; Synaptic Transmission; Trigeminal Nucleus, Spinal

1991
GABA-mediated inhibition in rostral ventromedial medulla: role in nociceptive modulation in the lightly anesthetized rat.
    Pain, 1991, Volume: 47, Issue:1

    Topics: Analgesics; Anesthesia; Animals; Bicuculline; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Medulla Oblongata; Microinjections; Nociceptors; Pyridazines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Receptors, Glycine; Receptors, Neurotransmitter

1991
Electrophysiological studies of the GABAA receptor ligand, 4-PIOL, on cultured hippocampal neurones.
    British journal of pharmacology, 1991, Volume: 104, Issue:1

    Topics: Animals; Bicuculline; Cells, Cultured; Female; Hippocampus; Isonicotinic Acids; Isoxazoles; Membrane Potentials; Neurons; Piperidines; Pregnancy; Rats; Receptors, GABA-A; Spinal Cord

1991
GABA(B)-related activity involved in synaptic processing of somatosensory information in S1 cortex of the anaesthetized cat.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Anesthesia; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrodes; Female; gamma-Aminobutyric Acid; Iontophoresis; Isoxazoles; Male; Muscimol; Neurons; Physical Stimulation; Somatosensory Cortex; Synapses

1990
Binding of [3H]-muscimol to GABAA sites in the guinea-pig urinary bladder: biochemical assay and autoradiography.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: Animals; Autoradiography; Bicuculline; Binding, Competitive; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Isoxazoles; Muscimol; Receptors, GABA-A; Tritium; Urinary Bladder

1989
GABAergic drugs and lordosis behavior in the female rat.
    Hormones and behavior, 1989, Volume: 23, Issue:3

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Estradiol; Female; gamma-Aminobutyric Acid; Isoxazoles; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal; Taurine

1989
Role of GABAergic system in prolactin analgesia.
    Clinical and experimental pharmacology & physiology, 1989, Volume: 16, Issue:11

    Topics: Analgesics; Animals; Bicuculline; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Morphine; Prolactin

1989
GABA-benzodiazepine modulation of aversion in the medial hypothalamus of the rat.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:1

    Topics: Animals; Avoidance Learning; Bicuculline; Dose-Response Relationship, Drug; Electric Stimulation; Electrodes, Implanted; Flumazenil; Hypothalamus, Middle; Isoxazoles; Male; Microinjections; Midazolam; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Effect of gamma-aminobutyric acidA receptor agonists and antagonists on the release of enkephalin-containing peptides from dog adrenal gland.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:1

    Topics: Adrenal Medulla; Analgesics; Animals; Bicuculline; Catecholamines; Dogs; Electric Stimulation; Enkephalins; Female; Isoxazoles; Oxazoles; Receptors, GABA-A; Splanchnic Nerves

1987
Structural factors governing agonist and antagonist activity in the GABAA system.
    Biochemical pharmacology, 1988, Mar-01, Volume: 37, Issue:5

    Topics: Bicuculline; gamma-Aminobutyric Acid; Isoxazoles; Models, Molecular; Receptors, GABA-A; Structure-Activity Relationship

1988
Interactions of pentobarbital and phenobarbital with GABAergic drugs against chemoconvulsants in rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Convulsants; Diazepam; Drug Interactions; Isoxazoles; Male; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Strychnine

1988
Synthesis and biological activity of a GABAA agonist which has no effect on benzodiazepine binding and of structurally related glycine antagonists.
    Drug design and delivery, 1987, Volume: 1, Issue:4

    Topics: Animals; Bicuculline; Brain Chemistry; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Isoxazoles; Oxazoles; Piperidines; Pyrrolidines; Rats; Receptors, GABA-A; Synaptic Membranes

1987
Intrinsic gamma aminobutyric acid receptors modulate the release of catecholamine from canine adrenal gland in situ.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: Adrenal Medulla; Animals; Baclofen; Bicuculline; Chromaffin Granules; Dogs; Electric Stimulation; Epinephrine; Female; Hexamethonium; Hexamethonium Compounds; Histocytochemistry; Isoxazoles; Muscimol; Naloxone; Norepinephrine; Receptors, GABA-A; Splanchnic Nerves

1986
Effects of unilateral microinjections of GABAergic drugs into the inferior colliculus on auditory evoked potentials and on audiogenic seizure susceptibility.
    Experimental neurology, 1989, Volume: 104, Issue:1

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Bicuculline; Evoked Potentials, Auditory; Functional Laterality; gamma-Aminobutyric Acid; Inferior Colliculi; Isoxazoles; Male; Microinjections; Oxazoles; Rats; Rats, Inbred Strains; Reference Values; Seizures

1989
Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Androstanes; Animals; Azasteroids; Bicuculline; Cell Membrane; Cerebral Cortex; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isonicotinic Acids; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, GABA-A; Taurine

1985
GABAergic drugs and sexual behaviour in the male rat.
    European journal of pharmacology, 1985, Jun-19, Volume: 112, Issue:3

    Topics: 4-Aminobutyrate Transaminase; Alkynes; Aminocaproates; Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal

1985
The locomotor-reducing effects of GABAergic drugs do not depend on the GABAA receptor.
    Psychopharmacology, 1985, Volume: 87, Issue:1

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Isoxazoles; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taurine

1985
GABA agonists. Resolution, absolute stereochemistry, and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:11

    Topics: Animals; Bicuculline; Brain; Cats; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Molecular Conformation; Muscimol; Neurons; Oxazolidinones; Piperidines; Rats; Receptors, GABA-A; Spinal Cord; Stereoisomerism; Structure-Activity Relationship; Synaptic Membranes

1985
Elicitation of conspecific attack or defense in the male rat by intraventricular injection of a GABA agonist or antagonist.
    Physiology & behavior, 1985, Volume: 35, Issue:3

    Topics: Aggression; Animals; Bicuculline; Brain; gamma-Aminobutyric Acid; Injections, Intraventricular; Isoxazoles; Male; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission

1985
Behavioral effects of microinjections of SR 95103, a new GABA-A antagonist, into the medial hypothalamus or the mesencephalic central gray.
    European journal of pharmacology, 1985, Nov-05, Volume: 117, Issue:2

    Topics: Animals; Behavior, Animal; Bicuculline; Escape Reaction; Hypothalamus, Middle; Isoxazoles; Male; Mesencephalon; Microinjections; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Superior Colliculi

1985
GABAB receptor-mediated enhancement of vasoactive intestinal peptide-stimulated cyclic AMP production in slices of rat cerebral cortex.
    Journal of neurochemistry, 1986, Volume: 46, Issue:6

    Topics: Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Bicuculline; Cerebral Cortex; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; gamma-Aminobutyric Acid; Isoxazoles; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vasoactive Intestinal Peptide

1986
gamma-Aminobutyric acid agonists and antagonists alter chloride flux across brain membranes.
    Molecular pharmacology, 1986, Volume: 29, Issue:5

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Animals; Baclofen; Bicuculline; Brain; Cell Membrane; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Liver; Male; Mice; Mice, Inbred DBA; Muscimol; Picrotoxin; Receptors, GABA-A; Sodium; Sulfates; Taurine; Temperature

1986
GABA-agonists induce the formation of low-affinity GABA-receptors on cultured cerebellar granule cells via preexisting high affinity GABA receptors.
    Neurochemical research, 1986, Volume: 11, Issue:4

    Topics: Animals; Bicuculline; Cells, Cultured; Cerebellum; Intracellular Membranes; Isoxazoles; Kinetics; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
Effect of THIP and SL 76002, two clinically experimented GABA-mimetic compounds, on anterior pituitary GABA receptors and prolactin secretion in the rat.
    Life sciences, 1987, Mar-02, Volume: 40, Issue:9

    Topics: Animals; Anticonvulsants; Bicuculline; Binding, Competitive; Female; gamma-Aminobutyric Acid; Haloperidol; Isoxazoles; Kinetics; Male; Muscimol; Ovariectomy; Oxazoles; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Hypnotic action of pentobarbital in mice: a possible mechanism.
    Experimental neurology, 1987, Volume: 97, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Isoxazoles; Male; Mice; Oxazoles; Pentobarbital; Receptors, GABA-A; Reflex; Sleep

1987
Effects of GABAergic drugs on the GABA turnover in the substantia nigra and the corpus striatum of the rat.
    Journal of neural transmission, 1987, Volume: 69, Issue:1-2

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Corpus Striatum; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1987
Cardiorespiratory effects produced by injecting drugs that affect GABA receptors into nuclei associated with the ventral surface of the medulla.
    Neuropharmacology, 1987, Volume: 26, Issue:5

    Topics: Animals; Bicuculline; Brain Mapping; Cardiovascular Physiological Phenomena; Cats; Female; gamma-Aminobutyric Acid; Isoxazoles; Male; Medulla Oblongata; Muscimol; Respiration; Synaptic Transmission

1987
Respiratory depressant effects of GABA alpha- and beta-receptor agonists in the cat.
    Journal of applied physiology (Bethesda, Md. : 1985), 1987, Volume: 62, Issue:6

    Topics: Animals; Baclofen; Bicuculline; Cats; Female; Heart; Injections, Intravenous; Injections, Intraventricular; Isoxazoles; Male; Oxazoles; Receptors, GABA-A; Respiration

1987
GABAergic modulation of nociceptive threshold: effects of THIP and bicuculline microinjected in the ventral medulla of the rat.
    Brain research, 1988, May-31, Volume: 450, Issue:1-2

    Topics: Animals; Bicuculline; gamma-Aminobutyric Acid; Isoxazoles; Male; Medulla Oblongata; Microinjections; Oxazoles; Pain; Raphe Nuclei; Rats; Rats, Inbred Strains; Reaction Time; Sensory Thresholds

1988
Bicuculline-sensitive and insensitive effects of THIP on the binding of [3H]flunitrazepam.
    Neuropharmacology, 1987, Volume: 26, Issue:7A

    Topics: Animals; Bicuculline; Brain; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Isoxazoles; Male; Osmolar Concentration; Oxazoles; Rats; Rats, Inbred Strains; Sodium Chloride; Tritium

1987
Effect of GABAergic drugs in the behavioral 'despair' test in rats.
    European journal of pharmacology, 1986, Feb-18, Volume: 121, Issue:2

    Topics: Acetates; Aminooxyacetic Acid; Animals; Baclofen; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Muscimol; Oxazoles; Picrotoxin; Rats

1986
GABAergic mechanisms in antinociception.
    Progress in neuro-psychopharmacology & biological psychiatry, 1984, Volume: 8, Issue:4-6

    Topics: Alkynes; Aminocaproates; Aminooxyacetic Acid; Analgesics; Animals; Baclofen; Bicuculline; Central Nervous System; gamma-Aminobutyric Acid; Isoxazoles; Mice; Muscimol; Pain; Rats; Stereoisomerism; Substance P; Synaptic Transmission; Vigabatrin

1984
Involvement of central GABAergic receptors in the control over offensive and defensive behaviours in the rat.
    Progress in clinical and biological research, 1984, Volume: 167

    Topics: Aggression; Animals; Bicuculline; Electroshock; Humans; Injections, Intraventricular; Isoxazoles; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Action of pyrazolopyridines as modulators of [3H]flunitrazepam binding to the gaba/benzodiazepine receptor complex of the cerebellum.
    European journal of pharmacology, 1981, Mar-12, Volume: 70, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Bicuculline; Binding Sites; Cerebellum; Chlorides; Etazolate; Flunitrazepam; Isoxazoles; Male; Muscimol; Nicotinic Acids; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium

1981
Multiple benzodiazepine receptor complexes: some benzodiazepine recognition sites are coupled to GABA receptors and ionophores.
    Advances in biochemical psychopharmacology, 1980, Volume: 21

    Topics: Animals; Anions; Benzodiazepines; Bicuculline; Brain; Buffers; Flunitrazepam; gamma-Aminobutyric Acid; Haplorhini; Hot Temperature; Ionophores; Isonicotinic Acids; Isoxazoles; Macromolecular Substances; Papio; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter

1980
Role of GABA-ergic receptors for the synthesis of GABA in different compartments of the rat cerebellum.
    Acta physiologica Scandinavica, 1981, Volume: 112, Issue:1

    Topics: Aminooxyacetic Acid; Animals; Bicuculline; Cerebellum; gamma-Aminobutyric Acid; Isoxazoles; Male; Rats; Receptors, Cell Surface; Receptors, GABA-A

1981
gamma-Aminobutyric acid- and benzodiazepine-binding sites in human anterior pituitary tissue.
    The Journal of clinical endocrinology and metabolism, 1982, Volume: 54, Issue:3

    Topics: Adult; Aged; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Humans; Isonicotinic Acids; Isoxazoles; Middle Aged; Muscimol; Pituitary Gland, Anterior; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A

1982
Orally administered THIP inhibits food intake in the rat.
    Behavioral and neural biology, 1982, Volume: 34, Issue:1

    Topics: Administration, Oral; Animals; Bicuculline; Dose-Response Relationship, Drug; Eating; Isoxazoles; Male; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1982
Central cardiovascular effects produced by the GABA receptor agonist drug, THIP.
    Neuropharmacology, 1982, Volume: 21, Issue:6

    Topics: Animals; Autonomic Nervous System; Bicuculline; Blood Pressure; Brain; Cats; Dose-Response Relationship, Drug; Female; Heart; Heart Rate; Injections, Intraventricular; Isoxazoles; Male; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A

1982
Autoreceptors modify the evoked release of [3H]GABA from cerebellar neurons in dissociated cell culture.
    European journal of pharmacology, 1982, Aug-27, Volume: 82, Issue:3-4

    Topics: Animals; Bicuculline; Cells, Cultured; Cerebellum; Fluspirilene; gamma-Aminobutyric Acid; Isoxazoles; Muscimol; Neurons; Potassium; Rats; Receptors, Cell Surface; Receptors, GABA-A

1982
GABAergic modulation of ethanol-induced motor impairment.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 223, Issue:3

    Topics: 4-Aminobutyrate Transaminase; Alkynes; Aminobutyrates; Aminocaproates; Animals; Bicuculline; Brain; Ethanol; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Skills; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1982
Further characterization of the anorexic action of orally-administered THIP, a GABA-analogue, in the rat.
    Physiology & behavior, 1982, Volume: 29, Issue:5

    Topics: Administration, Oral; Animals; Bicuculline; Eating; gamma-Aminobutyric Acid; Isoxazoles; Male; Oxazoles; Pentylenetetrazole; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Strychnine

1982
Diazotization and thiocyanate differentiate agonists from antagonists for the high- and low-affinity receptors of gamma-aminobutyric acid.
    Journal of neurochemistry, 1984, Volume: 43, Issue:1

    Topics: Androstanes; Animals; Azasteroids; Benzenesulfonates; Bicuculline; Cerebral Cortex; Diazonium Compounds; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Sulfanilic Acids; Thiocyanates; Tubocurarine

1984
Pharmacological analysis of the central cardiovascular effects of four GABA analogues.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 325, Issue:4

    Topics: Animals; Atropine; Bicuculline; Blood Pressure; Brain; GABA Antagonists; gamma-Aminobutyric Acid; Heart Rate; Isonicotinic Acids; Isoxazoles; Kainic Acid; Muscimol; Pyrones; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1984
Flight induced by infusion of bicuculline methiodide into periventricular structures.
    Brain research, 1984, Sep-10, Volume: 309, Issue:2

    Topics: Animals; Bicuculline; Brain Mapping; Escape Reaction; gamma-Aminobutyric Acid; Hypothalamic Area, Lateral; Hypothalamus, Middle; Isoxazoles; Male; Motor Activity; Periaqueductal Gray; Rats; Rats, Inbred Strains

1984
Self-injurious behavior in rats produced by intranigral microinjection of GABA agonists.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Brain; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Male; Microinjections; Muscimol; Rats; Rats, Inbred Strains; Self Mutilation; Stress, Physiological; Substantia Nigra

1984
Comparison of the analgesic actions of THIP and morphine.
    General pharmacology, 1983, Volume: 14, Issue:6

    Topics: Analgesics; Animals; Atropine; Benzoquinones; Bicuculline; Hypnotics and Sedatives; Isoxazoles; Male; Mice; Morphine; Naloxone; Oxazoles; Quinones; Reaction Time

1983
Induction of mouse-killing in the rat by intraventricular injection of a GABA-agonist.
    Physiology & behavior, 1983, Volume: 30, Issue:3

    Topics: Aggression; Animals; Arousal; Bicuculline; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Humans; Injections, Intraventricular; Isoxazoles; Male; Motor Activity; Oxazoles; Rats; Rats, Inbred Strains; Reaction Time

1983
Development of hyperpolarizing inhibitory postsynaptic potentials and hyperpolarizing response to gamma-aminobutyric acid in rabbit hippocampus studied in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1984, Volume: 4, Issue:3

    Topics: Action Potentials; Aging; Animals; Animals, Newborn; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isoxazoles; Membrane Potentials; Neurons; Rabbits; Synapses

1984
Nigral actions of GABA agonists are enhanced by chronic fluphenazine and differentiated by concomitant flurazepam.
    Psychopharmacology, 1982, Volume: 76, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Female; Fluphenazine; Flurazepam; gamma-Aminobutyric Acid; Humans; Isoxazoles; Muscimol; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substantia Nigra

1982
A comparison of the analgesic activities of 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol (THIP) and 6-chloro-2[1-piperazinyl]pyrazine (MK 212).
    European journal of pharmacology, 1983, Jun-03, Volume: 90, Issue:2-3

    Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Drug Synergism; Drug Tolerance; Isoxazoles; Male; Mice; Morphine; Oxazoles; Pyrazines; Time Factors

1983
Pharmacological evidence for two kinds of GABA receptor on rat hippocampal pyramidal cells studied in vitro.
    The Journal of physiology, 1982, Volume: 328

    Topics: Animals; Bicuculline; Dendrites; Diazepam; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isoxazoles; Membrane Potentials; Penicillins; Pentobarbital; Pyramidal Tracts; Rats; Receptors, Drug

1982
Serotonin2 receptor-mediated excitation of interneurons in piriform cortex: antagonism by atypical antipsychotic drugs.
    Neuroscience, 1994, Volume: 58, Issue:3

    Topics: Action Potentials; Animals; Antipsychotic Agents; Bicuculline; Cerebral Cortex; Chlorpromazine; Clozapine; Electrophysiology; gamma-Aminobutyric Acid; Haloperidol; In Vitro Techniques; Interneurons; Isoxazoles; Male; Membrane Potentials; Piperidines; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Risperidone; Serotonin Antagonists

1994
An iontophoretic study of the effects of alpha-amino-hydroxy-5-methyl-4-isoxazole propionic acid lesions of the nucleus basalis magnocellularis on cholinergic and GABAergic influences on frontal cortex neurones of rats.
    Experimental brain research, 1994, Volume: 98, Issue:3

    Topics: Acetylcholine; Animals; Bicuculline; Carbachol; Frontal Lobe; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Iontophoresis; Isoxazoles; Male; Medulla Oblongata; Neurons; Parasympathetic Nervous System; Propionates; Rats; Rats, Sprague-Dawley

1994
Extrasynaptic effects of GABA (gamma-aminobutyric acid) agonists on myelinated axons of peripheral nerve.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:4

    Topics: Action Potentials; Animals; Axons; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Isoxazoles; Motor Neurons; Nerve Fibers, Myelinated; Peripheral Nerves; Rana catesbeiana; Ranidae; Sciatic Nerve; Spinal Nerve Roots; Synapses

1994
GABA alters GABAA receptor mRNAs and increases ligand binding.
    Journal of neurochemistry, 1993, Volume: 61, Issue:6

    Topics: Animals; Anticonvulsants; Base Sequence; Bicuculline; Cells, Cultured; Cerebellum; DNA Primers; gamma-Aminobutyric Acid; Gene Expression; Isoxazoles; Macromolecular Substances; Molecular Sequence Data; Muscimol; Neurons; Polymerase Chain Reaction; Rats; Receptors, GABA-A; RNA, Messenger

1993
Neuronal regulation of astrocyte morphology in vitro is mediated by GABAergic signaling.
    Glia, 1997, Volume: 20, Issue:1

    Topics: Animals; Animals, Newborn; Astrocytes; Baclofen; Bicuculline; Cell Adhesion; Cells, Cultured; Coculture Techniques; GABA Agonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Isoxazoles; Muscimol; Neurons; Rats; Rats, Wistar; Signal Transduction; Sodium Channel Blockers; Tetrodotoxin; Time Factors

1997
The role of dopamine and GABA in the frontal cortex of mice in modulating a motor-stimulant effect of amphetamine and cocaine.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:1

    Topics: Amphetamine; Animals; Bicuculline; Cocaine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Frontal Lobe; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Models, Neurological; Motor Activity; Stereotyped Behavior; Sulpiride

1998
GABAergic drugs and sexual behaviour in the rabbit: evidence for species-specific effects.
    Journal of psychopharmacology (Oxford, England), 1998, Volume: 12, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Copulation; Dose-Response Relationship, Drug; Escape Reaction; GABA Agents; Isoxazoles; Male; Picrotoxin; Rabbits; Rats; Sexual Behavior, Animal; Species Specificity; Structure-Activity Relationship

1998
Two populations of kainate receptors with separate signaling mechanisms in hippocampal interneurons.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, Feb-01, Volume: 97, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Bicuculline; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Indoles; Interneurons; Isoxazoles; Kainic Acid; Lidocaine; Maleimides; Naphthalenes; Nerve Tissue Proteins; Patch-Clamp Techniques; Propionates; Protein Kinase C; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Kainic Acid; Receptors, Presynaptic; Signal Transduction; Staurosporine; Virulence Factors, Bordetella

2000
Additivity and independence of neuroprotective effects of GABAA and GABAB receptor agonists in complete global cerebral ischemia.
    Bulletin of experimental biology and medicine, 2000, Volume: 130, Issue:8

    Topics: Animals; Baclofen; Bicuculline; Brain Ischemia; Drug Interactions; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Isoxazoles; Male; Mice; Mice, Inbred CBA; Muscimol; Neuroprotective Agents; Picrotoxin

2000
Effects of GABA(A) receptor partial agonists in primary cultures of cerebellar granule neurons and cerebral cortical neurons reflect different receptor subunit compositions.
    British journal of pharmacology, 2001, Volume: 133, Issue:4

    Topics: Animals; Bicuculline; Cells, Cultured; Cerebellum; Cerebral Cortex; Electrophysiology; GABA Agonists; GABA-A Receptor Agonists; Isonicotinic Acids; Isoxazoles; Mice; Neurons; Oocytes; Patch-Clamp Techniques; Piperidines; Pyridazines; Receptors, GABA-A; Xenopus laevis

2001
GABAergic and glutamatergic terminals differentially influence the organization of GABAergic synapses in rat cerebellar granule cells in vitro.
    Neuroscience, 2002, Volume: 114, Issue:1

    Topics: Age Factors; Animals; Animals, Newborn; Bicuculline; Carrier Proteins; Cell Differentiation; Cells, Cultured; Cerebellar Cortex; Fluorescent Antibody Technique; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Glutamic Acid; Isoxazoles; Membrane Proteins; Membrane Transport Proteins; Muscimol; Presynaptic Terminals; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes; Synaptic Transmission; Vesicular Glutamate Transport Protein 1; Vesicular Transport Proteins

2002
Gamma-aminobutyric acid-induced calcium signalling in rat superior collicular neurones.
    Neuroscience letters, 2002, Dec-13, Volume: 334, Issue:2

    Topics: Animals; Bicuculline; Calcium; Cells, Cultured; Cytarabine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Immunohistochemistry; Isoxazoles; Neurons; Phosphinic Acids; Pyridines; Rats; Receptors, GABA; Superior Colliculi

2002
Changes in rectal temperature and ECoG spectral power of sensorimotor cortex elicited in conscious rabbits by i.c.v. injection of GABA, GABA(A) and GABA(B) agonists and antagonists.
    British journal of pharmacology, 2004, Volume: 141, Issue:1

    Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Body Temperature Regulation; Electroencephalography; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Isoxazoles; Lateral Ventricles; Male; Muscimol; Nipecotic Acids; Preoptic Area; Rabbits; Receptors, GABA-A; Receptors, GABA-B; Rectum; Somatosensory Cortex

2004
Anticonvulsant and antiepileptogenic effects of GABAA receptor ligands in pentylenetetrazole-kindled mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2004, Volume: 28, Issue:1

    Topics: Animals; Anticonvulsants; Bicuculline; Convulsants; Dehydroepiandrosterone Sulfate; Diazepam; Dose-Response Relationship, Drug; Epilepsy; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; Isoxazoles; Kindling, Neurologic; Ligands; Mice; Pentylenetetrazole; Pregnanediones; Receptors, GABA-A

2004
Short-term steroid treatment increases delta GABAA receptor subunit expression in rat CA1 hippocampus: pharmacological and behavioral effects.
    Neuropharmacology, 2005, Volume: 49, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Bicuculline; Blotting, Western; Cell Separation; Electrophysiology; Estradiol; Female; GABA Agonists; GABA Antagonists; Hippocampus; Homeostasis; In Vitro Techniques; Isoxazoles; Lanthanum; Lorazepam; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pregnanolone; Rats; Rats, Long-Evans; Receptors, GABA-A; Steroids

2005
An extrasynaptic GABAA receptor mediates tonic inhibition in thalamic VB neurons.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: Action Potentials; Animals; Animals, Newborn; Azides; Benzodiazepines; Bicuculline; Blotting, Western; Cells, Cultured; Chlorides; Dose-Response Relationship, Drug; Electric Stimulation; GABA Agonists; GABA Antagonists; Humans; Immunohistochemistry; Immunoprecipitation; In Vitro Techniques; Indoles; Isoxazoles; Membrane Potentials; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Patch-Clamp Techniques; Prokaryotic Initiation Factors; Protein Subunits; Pyridines; Receptors, GABA-A; Synapses; Synaptophysin; Transfection; Ventral Thalamic Nuclei; Zinc Compounds; Zolpidem

2005
Involvement of GABAergic modulation of antinociception induced by morphine microinjected into the ventrolateral orbital cortex.
    Brain research, 2006, Feb-16, Volume: 1073-1074

    Topics: Analysis of Variance; Animals; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; Drug Interactions; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Microinjections; Morphine; Muscimol; Narcotics; Neurons; Nociceptors; Pain Measurement; Picrotoxin; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Reaction Time

2006
Dual GABAA receptor-mediated inhibition in rat presympathetic paraventricular nucleus neurons.
    The Journal of physiology, 2007, Jul-15, Volume: 582, Issue:Pt 2

    Topics: Animals; Bicuculline; Electrophysiology; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Isoxazoles; Male; Medulla Oblongata; Neural Inhibition; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Synapses

2007
Discriminative stimulus effects of tiagabine and related GABAergic drugs in rats.
    Psychopharmacology, 2008, Volume: 197, Issue:4

    Topics: Administration, Oral; Amines; Animals; Anticonvulsants; Azabicyclo Compounds; Baclofen; Benzodiazepines; Bicuculline; Brain; Cyclohexanecarboxylic Acids; Discrimination Learning; Dose-Response Relationship, Drug; GABA Agents; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; Gabapentin; gamma-Aminobutyric Acid; Generalization, Stimulus; Hypnotics and Sedatives; Injections, Intraperitoneal; Isoxazoles; Male; Nipecotic Acids; Piperazines; Pyridines; Rats; Thiophenes; Tiagabine; Zolpidem

2008
Gaboxadol -- a different hypnotic profile with no tolerance to sleep EEG and sedative effects after repeated daily dosing.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 90, Issue:1

    Topics: Anesthetics; Animals; Bicuculline; Central Nervous System; Dose-Response Relationship, Drug; Down-Regulation; Drug Tolerance; Electrodes, Implanted; Electroencephalography; GABA Antagonists; Hypnotics and Sedatives; Isoxazoles; Male; Postural Balance; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sleep

2008
Inhibition of thalamic excitability by 4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridine-3-ol: a selective role for delta-GABA(A) receptors.
    The European journal of neuroscience, 2009, Volume: 29, Issue:6

    Topics: Analysis of Variance; Animals; Animals, Newborn; Bicuculline; Dose-Response Relationship, Drug; Electric Stimulation; Female; GABA Agonists; GABA Antagonists; Glycine Agents; In Vitro Techniques; Isoxazoles; Locomotion; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Neural Inhibition; Patch-Clamp Techniques; Receptors, GABA-A; Strychnine; Thalamus; Time Factors

2009
Electrophysiological actions of zonisamide on striatal neurons: Selective neuroprotection against complex I mitochondrial dysfunction.
    Experimental neurology, 2010, Volume: 221, Issue:1

    Topics: Action Potentials; Animals; Antioxidants; Bicuculline; Corpus Striatum; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; GABA Antagonists; Glucose; Glutamic Acid; In Vitro Techniques; Isoxazoles; Male; Neurons; Nitro Compounds; Propionates; Rats; Rats, Wistar; Rotenone; Uncoupling Agents; Zonisamide

2010
The 4-aminopyridine in vitro epilepsy model analyzed with a perforated multi-electrode array.
    Neuropharmacology, 2011, Volume: 60, Issue:7-8

    Topics: 4-Aminopyridine; Animals; Anticonvulsants; Bicuculline; CA3 Region, Hippocampal; Disease Models, Animal; Electrodes; Epilepsy; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isoxazoles; Mice; Mice, Inbred C57BL; Microarray Analysis; Motion Pictures; Piperazines; Potassium Channel Blockers; Quinoxalines; Receptors, N-Methyl-D-Aspartate; Software; Somatosensory Cortex

2011
Pharmacological enhancement of δ-subunit-containing GABA(A) receptors that generate a tonic inhibitory conductance in spinal neurons attenuates acute nociception in mice.
    Pain, 2011, Volume: 152, Issue:6

    Topics: Action Potentials; Analgesics; Anesthetics; Animals; Bicuculline; Desoxycorticosterone; Dose-Response Relationship, Drug; Electric Stimulation; Formaldehyde; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hindlimb Suspension; In Vitro Techniques; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neural Inhibition; Pain Measurement; Psychomotor Performance; Receptors, GABA-A; Sensory Receptor Cells; Spinal Cord

2011
Tonic GABAA receptor conductance in medial subnucleus of the tractus solitarius neurons is inhibited by activation of μ-opioid receptors.
    Journal of neurophysiology, 2012, Volume: 107, Issue:3

    Topics: Analgesics, Opioid; Animals; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Opioid, mu; Sodium Channel Blockers; Solitary Nucleus; Tetrodotoxin

2012
Upregulation of high-affinity GABA(A) receptors in cultured rat dorsal root ganglion neurons.
    Neuroscience, 2012, Apr-19, Volume: 208

    Topics: Animals; Bicuculline; Blotting, Western; Cells, Cultured; Crotonates; Electrophysiological Phenomena; GABA Agonists; GABA Antagonists; Ganglia, Spinal; Isoxazoles; Male; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Real-Time Polymerase Chain Reaction; Receptors, GABA-A; Time Factors; Up-Regulation

2012
The dual effect of PNU-120596 on α7 nicotinic acetylcholine receptor channels.
    European journal of pharmacology, 2013, Oct-15, Volume: 718, Issue:1-3

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Bicuculline; Choline; Drug Synergism; Female; In Vitro Techniques; Ion Channel Gating; Isoxazoles; Male; Phenylurea Compounds; Rats; Rats, Sprague-Dawley

2013
Attenuated benzodiazepine-sensitive tonic GABAA currents of supraoptic magnocellular neuroendocrine cells in 24-h water-deprived rats.
    Journal of neuroendocrinology, 2014, Volume: 26, Issue:1

    Topics: Animals; Bicuculline; Diazepam; GABA Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Imidazoles; Inhibitory Postsynaptic Potentials; Isoxazoles; Male; Neuroendocrine Cells; Propofol; Protein Subunits; Rats; Receptors, GABA-A; Supraoptic Nucleus; Water Deprivation

2014
Methyl CpG Binding Protein 2 Gene Disruption Augments Tonic Currents of γ-Aminobutyric Acid Receptors in Locus Coeruleus Neurons: IMPACT ON NEURONAL EXCITABILITY AND BREATHING.
    The Journal of biological chemistry, 2015, Jul-24, Volume: 290, Issue:30

    Topics: Animals; Bicuculline; GABA Agonists; GABAergic Neurons; Humans; Isoxazoles; Locus Coeruleus; Methyl-CpG-Binding Protein 2; Mice; Mice, Transgenic; Receptors, GABA; Receptors, GABA-A; Respiration; Rett Syndrome; Single-Cell Analysis; Synapses

2015
Regulation of Extrasynaptic GABAA α4 Receptors by Ethanol-Induced Protein Kinase A, but Not Protein Kinase C Activation in Cultured Rat Cerebral Cortical Neurons.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 356, Issue:1

    Topics: Animals; Bicuculline; Cells, Cultured; Cerebral Cortex; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Activators; Ethanol; Female; GABA Antagonists; Isoxazoles; Male; Neurons; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses

2016
Perinatal high fat diet increases inhibition of dorsal motor nucleus of the vagus neurons regulating gastric functions.
    Neurogastroenterology and motility, 2018, Volume: 30, Issue:1

    Topics: Animals; Bicuculline; Brain Stem; Diet, High-Fat; GABA Agonists; GABA Antagonists; Gastrointestinal Motility; Isoxazoles; Male; Neural Inhibition; Neurons; Pyridazines; Rats, Sprague-Dawley; Vagus Nerve

2018