Page last updated: 2024-08-21

isoxazoles and baclofen

isoxazoles has been researched along with baclofen in 79 studies

Research

Studies (79)

TimeframeStudies, this research(%)All Research%
pre-199045 (56.96)18.7374
1990's22 (27.85)18.2507
2000's9 (11.39)29.6817
2010's3 (3.80)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Waddington, JL1
Guidotti, A; Kurosawa, A; Naik, SR1
Agnati, L; Fuxe, K; Hökfelt, T; Johansson, O; Ljungdahl, A; Perez de la Mora, M1
Amit, Z; Robidoux, J; Smith, BR1
Ebbesson, SO; Erdö, SL; Hofmann, MH; Malz, CR; Meyer, DL1
Barolet, AW; Morris, ME1
Agmo, A; Gutiérrez, M; Guzmán, M; Pruneda, R1
Bergen, HT; Hejtmancik, JF; Pfaff, DW1
Boelen, MK; Chubb, IW; Dowton, M; Morgan, IG; Wellard, J1
Catt, KJ; Stojilković, SS; Virmani, MA1
Balcar, VJ; Dreher, B1
Michler, A1
Hicks, TP; Kaneko, T1
Agmo, A; Paredes, R; Soria, P1
Erdö, SL; Michler, A1
Karlsson, G; Olpe, HR1
Aarslew-Jensen, M; Diemer, NH; Krogsgaard-Larsen, P; Nielsen, EO; Schousboe, A1
Thalmann, RH2
Mehta, AK; Ticku, MK1
Bitran, D; Leipheimer, RE; McQuade, DB; Miller, SA; Sachs, BD1
Bond, A; Neal, H1
Alho, H; Fujimoto, M; Geffard, M; Guidotti, A; Hanbauer, I; Kataoka, Y; Kelly, GD1
Borsini, F; Giuliani, S; Meli, A2
Karobath, M; Supavilai, P1
Costa, LG; Enna, SJ; Pelley, K; Setler, P; Vaught, JL1
Gianutsos, G; Suzdak, PD2
Agmo, A; Paredes, R1
Agmo, A; Giordano, M1
Hösli, E; Hösli, L; Krogsgaard-Larsen, P1
Bristow, DR; Watling, KJ1
Chweh, AY; Swinyard, EA; Ulloque, RA1
Allan, AM; Harris, RA1
Audi, EA; Graeff, FG1
Chweh, AY; Swinyard, EA; Wolf, HH1
Lindgren, S1
Zharkovskaia, TA; Zharkovskiĭ, AM1
Gillis, RA; Hamosh, P; Hartley, B; Quest, JA; Taveira da Silva, AM1
Pelley, KA; Vaught, JL1
Borsini, F; Evangelista, S; Meli, A1
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K1
Enna, SJ; Zorn, SH1
Beart, PM; Lloyd, KG; Scatton, B1
Sawynok, J1
Meldrum, B1
Maksay, G; Ticku, MK1
Depaulis, A; Marescaux, C; Micheletti, G; Rumbach, L; Vergnes, M; Warter, JM1
Baumeister, AA; Frye, GD1
Drower, EJ; Hammond, DL1
Di Scala, G; Karli, P; Schmitt, P1
Coward, DM1
Buescher, HH; Hill, RC; Maurer, R; Roemer, D1
Clark, WG; Menon, MK; Vivonia, C1
Damgaard, I; Elster, L; Kardos, J; Krogsgaard-Larsen, P; Schousboe, A1
Liske, S; Morris, ME1
Batini, C; Billard, JM; Vigot, R1
Alger, BE; Kirov, SA; Lenz, RA; Martin, LA; Morishita, W; Pitler, TA1
Matsutani, S; Yamamoto, N1
Kulinskiĭ, VI; Mikhel'son, GV2
Eriksson, B; Magnusson, AK; Tham, R1
Agmo, A; Contreras, JL; Paredes, RG1
Ghanipoor, N; Parvini, S; Rezayat, M; Zarrindast, MR1
Broadbent, J; Harless, WE1
Parvini, S; Pirali, M; Rezayat, M; Tabarrai, E; Zarrindast, MR1
Asnis, N; Barros, HM; Gomez, R; Tannhauser, SL1
Firestone, LL; Hammond, DL; Homanics, GE; Ugarte, SD1
Allikmets, L; Matto, V; Pruus, K; Rudissaar, R; Skrebuhhova-Malmros, T1
de Almeida, OM; de Mello, FG; de Mello, MC; Gardino, PF; Hokoç, JN; Loureiro dos Santos, NE; Yamasaki, EN1
Frosini, M; Sgaragli, G; Valoti, M1
Abílio, VC; Araujo, NP; Castro, JP; Faria, RR; Frussa-Filho, R; Fukushiro, DF; Medrano, WA; Peixoto, MF; Silva, RH; Zanier-Gomes, PH1
Collingridge, GL; Isaac, JT; Lauri, SE; Maingret, F; Mulle, C; Segerstråle, M; Taira, T; Vesikansa, A1
Boehm, SL; Goldfarb, KJ; Linsenbardt, DN; Moore, EM; Serio, KM; Stepanovska, S1
Hutson, PH; McDonald, LM; Sheppard, WF; Sohal, B; Staveley, SM; Tattersall, FD1
Ang, D; De Santis, A; Pauwels, A; Scarpellini, E; Tack, J; Vanuytsel, T1
Johnston, GAR1
Alabed, S; Bergman, H; Latifeh, Y; Mohammad, HA1

Reviews

3 review(s) available for isoxazoles and baclofen

ArticleYear
Management of refractory typical GERD symptoms.
    Nature reviews. Gastroenterology & hepatology, 2016, Volume: 13, Issue:5

    Topics: Alginates; Algorithms; Antacids; Baclofen; Chronic Disease; Esophagoscopy; Gastroesophageal Reflux; Gastrointestinal Agents; Gastroscopy; Humans; Isoxazoles; Muscle Relaxants, Central; Neurotransmitter Agents; Phosphinic Acids; Propylamines; Triazoles

2016
GABA Australis, some reflections on the history of GABA receptor research in Australia.
    Pharmacological research, 2017, Volume: 116

    Topics: Animals; Australia; Baclofen; Bicuculline; Cyclic AMP; Humans; Isoxazoles; Muscimol; Receptors, GABA

2017
Gamma-aminobutyric acid agonists for antipsychotic-induced tardive dyskinesia.
    The Cochrane database of systematic reviews, 2018, 04-17, Volume: 4

    Topics: Antipsychotic Agents; Baclofen; Dyskinesia, Drug-Induced; GABA Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Placebos; Randomized Controlled Trials as Topic; Valproic Acid

2018

Other Studies

76 other study(ies) available for isoxazoles and baclofen

ArticleYear
GABA-like properties of flurazepam and baclofen suggested by rotational behaviour following unilateral intranigral injection: a comparison with the GABA agonist muscimol [proceedings].
    British journal of pharmacology, 1977, Volume: 60, Issue:2

    Topics: Aminobutyrates; Animals; Anti-Anxiety Agents; Baclofen; Behavior; Flurazepam; gamma-Aminobutyric Acid; Humans; Injections; Isoxazoles; Male; Oxazoles; Rats; Stereotyped Behavior; Substantia Nigra

1977
Possible role of gamma aminobutyric acid (GABA) in the regulation of cAMP system in rat anterior pituitary.
    Psychoneuroendocrinology, 1977, Volume: 2, Issue:3

    Topics: Aminobutyrates; Animals; Baclofen; Cyclic AMP; Diazepam; gamma-Aminobutyric Acid; Hypothalamus; Isoniazid; Isoxazoles; Male; Nipecotic Acids; Pargyline; Picrotoxin; Pituitary Gland, Anterior; Protein Kinases; Rats; Reserpine

1977
Regulation of the mesocortical dopamine neurons.
    Advances in biochemical psychopharmacology, 1977, Volume: 16

    Topics: 4-Butyrolactone; Acetylcholine; Aminooxyacetic Acid; Baclofen; Cerebral Cortex; Dopamine; gamma-Aminobutyric Acid; Isoxazoles; Neurons; Pimozide; Pyrrolidinones; Sulpiride

1977
GABAergic involvement in the acquisition of voluntary ethanol intake in laboratory rats.
    Alcohol and alcoholism (Oxford, Oxfordshire), 1992, Volume: 27, Issue:3

    Topics: Alcohol Drinking; Animals; Baclofen; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Isoxazoles; Male; Rats; Receptors, GABA-A

1992
Changes in ligand binding to GABAA receptor sites in pacific salmon (Oncorhynchus) brain during spawning migration and "aging".
    Journal fur Hirnforschung, 1992, Volume: 33, Issue:4-5

    Topics: Aging; Aminobutyrates; Analgesics; Animals; Baclofen; Bicuculline; Binding, Competitive; Brain; Female; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Ligands; Male; Muscimol; Receptors, GABA-A; Salmon; Sexual Behavior, Animal

1992
Changes in extracellular K+ evoked by GABA, THIP and baclofen in the guinea-pig hippocampal slice.
    Experimental brain research, 1991, Volume: 84, Issue:3

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Electrodes; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Isoxazoles; Nipecotic Acids; Potassium; Proline; Receptors, GABA-A; Temperature

1991
GABAergic drugs and conflict behavior in the rat: lack of similarities with the actions of benzodiazepines.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:3

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Behavior, Animal; Benzodiazepines; Bicuculline; Brain; Conflict, Psychological; Drug Interactions; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Nicotinic Acids; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission

1991
Effects of gamma-aminobutyric acid receptor agonists and antagonist on LHRH-synthesizing neurons as detected by immunocytochemistry and in situ hybridization.
    Experimental brain research, 1991, Volume: 87, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Female; GABA-A Receptor Antagonists; Gene Expression Regulation; Gonadotropin-Releasing Hormone; Immunohistochemistry; Isoxazoles; Neurons; Nucleic Acid Hybridization; Ovariectomy; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; RNA Probes; RNA, Messenger

1991
Glycinergic control of [Leu5]enkephalin levels in chicken retina.
    Brain research, 1991, Aug-23, Volume: 557, Issue:1-2

    Topics: Animals; Baclofen; Chickens; Enkephalin, Leucine; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Isoxazoles; Muscimol; Neurotransmitter Agents; Picrotoxin; Radioimmunoassay; Retina; Strychnine

1991
Stimulation of luteinizing hormone release by gamma-aminobutyric acid (GABA) agonists: mediation by GABAA-type receptors and activation of chloride and voltage-sensitive calcium channels.
    Endocrinology, 1990, Volume: 126, Issue:5

    Topics: Amino Acid Sequence; Animals; Baclofen; Calcium Channels; Cells, Cultured; Chloride Channels; Chlorides; Female; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Isoxazoles; Luteinizing Hormone; Membrane Proteins; Molecular Sequence Data; Muscimol; Nifedipine; Pituitary Gland, Anterior; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Neurochemical correlates of gamma-aminobutyrate (GABA) inhibition in cat visual cortex.
    Life sciences, 1990, Volume: 47, Issue:15

    Topics: Animals; Baclofen; Calcium; Cats; Cell Membrane; Female; GABA Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Neurons; Potassium; Pyridazines; Receptors, GABA-A; Visual Cortex

1990
Involvement of GABA receptors in the regulation of neurite growth in cultured embryonic chick tectum.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1990, Volume: 8, Issue:4

    Topics: Animals; Axons; Baclofen; Cells, Cultured; Chick Embryo; Culture Media; gamma-Aminobutyric Acid; Isoxazoles; Ligands; Muscimol; Receptors, GABA-A; Superior Colliculi

1990
GABA(B)-related activity involved in synaptic processing of somatosensory information in S1 cortex of the anaesthetized cat.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Anesthesia; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrodes; Female; gamma-Aminobutyric Acid; Iontophoresis; Isoxazoles; Male; Muscimol; Neurons; Physical Stimulation; Somatosensory Cortex; Synapses

1990
GABAergic drugs and lordosis behavior in the female rat.
    Hormones and behavior, 1989, Volume: 23, Issue:3

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Estradiol; Female; gamma-Aminobutyric Acid; Isoxazoles; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal; Taurine

1989
Stimulation by phaclofen of inositol 1,4,5-triphosphate production in cultured neurons from chick tectum.
    European journal of pharmacology, 1989, Aug-29, Volume: 167, Issue:3

    Topics: Animals; Baclofen; Chick Embryo; gamma-Aminobutyric Acid; Inosine Nucleotides; Inosine Triphosphate; Isoxazoles; Neurons; Receptors, GABA-A; Superior Colliculi

1989
Late inhibitory postsynaptic potentials in rat prefrontal cortex may be mediated by GABAB receptors.
    Experientia, 1989, Feb-15, Volume: 45, Issue:2

    Topics: Animals; Baclofen; Electric Conductivity; Electric Stimulation; Evoked Potentials; Frontal Lobe; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Isoxazoles; Male; Membrane Potentials; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synapses

1989
Baclofen-induced, calcium-dependent stimulation of in vivo release of D-[3H]aspartate from rat hippocampus monitored by intracerebral microdialysis.
    Neurochemical research, 1989, Volume: 14, Issue:4

    Topics: Animals; Aspartic Acid; Baclofen; Calcium; GABA Antagonists; Hippocampus; Ischemic Attack, Transient; Isoxazoles; Male; Potassium; Rats; Rats, Inbred Strains

1989
Pertussis toxin blocks a late inhibitory postsynaptic potential in hippocampal CA3 neurons.
    Neuroscience letters, 1987, Nov-10, Volume: 82, Issue:1

    Topics: Action Potentials; Adenylate Cyclase Toxin; Animals; Baclofen; Hippocampus; In Vitro Techniques; Isoxazoles; Neural Conduction; Neural Inhibition; Pertussis Toxin; Rats; Receptors, GABA-A; Virulence Factors, Bordetella

1987
Interactions of pentobarbital and phenobarbital with GABAergic drugs against chemoconvulsants in rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Convulsants; Diazepam; Drug Interactions; Isoxazoles; Male; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Strychnine

1988
Inhibition of sexual reflexes by lumbosacral injection of a GABAB agonist in the male rat.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:3

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Injections, Spinal; Isoxazoles; Lumbosacral Region; Male; Penile Erection; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal; Spinal Cord

1988
Quantitative electrocortical changes in the rat induced by phencyclidine and other stimulants.
    Neuropharmacology, 1985, Volume: 24, Issue:4

    Topics: Animals; Apomorphine; Baclofen; Cerebral Cortex; Chlordiazepoxide; Chlorpromazine; Dextroamphetamine; Dioxolanes; Electroencephalography; Isoquinolines; Isoxazoles; Male; Muscimol; Phencyclidine; Rats; Rats, Inbred Strains

1985
Intrinsic gamma aminobutyric acid receptors modulate the release of catecholamine from canine adrenal gland in situ.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: Adrenal Medulla; Animals; Baclofen; Bicuculline; Chromaffin Granules; Dogs; Electric Stimulation; Epinephrine; Female; Hexamethonium; Hexamethonium Compounds; Histocytochemistry; Isoxazoles; Muscimol; Naloxone; Norepinephrine; Receptors, GABA-A; Splanchnic Nerves

1986
Functional evidence for altered activity of GABAergic receptors following chronic desipramine treatment in rats.
    The Journal of pharmacy and pharmacology, 1986, Volume: 38, Issue:12

    Topics: Analgesics; Animals; Baclofen; Desipramine; Isoxazoles; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
Modulation of acetylcholine release from rat striatal slices by the GABA/benzodiazepine receptor complex.
    Life sciences, 1985, Feb-04, Volume: 36, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Baclofen; Benzodiazepinones; Clonazepam; Corpus Striatum; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Haloperidol; In Vitro Techniques; Isoxazoles; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
A comparison of the antinociceptive responses to the GABA-receptor agonists THIP and baclofen.
    Neuropharmacology, 1985, Volume: 24, Issue:3

    Topics: Analgesics; Animals; Baclofen; Dose-Response Relationship, Drug; Drug Tolerance; Isoxazoles; Male; Mice; Oxazoles; Postural Balance; Receptors, GABA-A

1985
Parallel changes in the sensitivity of gamma-aminobutyric acid and noradrenergic receptors following chronic administration of antidepressant and GABAergic drugs. A possible role in affective disorders.
    Neuropharmacology, 1985, Volume: 24, Issue:3

    Topics: Animals; Anticonvulsants; Antidepressive Agents; Baclofen; Cerebral Cortex; Dihydroalprenolol; gamma-Aminobutyric Acid; Hippocampus; Humans; Imipramine; Isoxazoles; Kinetics; Male; Mice; Mood Disorders; Nomifensine; Receptors, Adrenergic; Receptors, GABA-A

1985
GABAergic drugs and sexual behaviour in the male rat.
    European journal of pharmacology, 1985, Jun-19, Volume: 112, Issue:3

    Topics: 4-Aminobutyrate Transaminase; Alkynes; Aminocaproates; Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal

1985
GABAergic effects of reserpine following chronic treatment.
    Psychopharmacology, 1985, Volume: 87, Issue:2

    Topics: Animals; Baclofen; Binding, Competitive; Cerebral Cortex; Dihydroalprenolol; gamma-Aminobutyric Acid; Hippocampus; Imipramine; Isoxazoles; Male; Mice; Receptors, GABA-A; Reserpine

1985
The locomotor-reducing effects of GABAergic drugs do not depend on the GABAA receptor.
    Psychopharmacology, 1985, Volume: 87, Issue:1

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Isoxazoles; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taurine

1985
Autoradiographic localization of binding sites for the gamma-aminobutyric acid analogues 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol (THIP)isoguvacine and baclofen on cultured neurons of rat cerebellum and spinal cord.
    Neuroscience letters, 1985, Oct-24, Volume: 61, Issue:1-2

    Topics: Animals; Animals, Newborn; Autoradiography; Baclofen; Binding Sites; Cells, Cultured; Cerebellum; Fetus; Isonicotinic Acids; Isoxazoles; Oxazoles; Rats; Receptors, GABA-A; Spinal Cord

1985
GABAB receptor-mediated enhancement of vasoactive intestinal peptide-stimulated cyclic AMP production in slices of rat cerebral cortex.
    Journal of neurochemistry, 1986, Volume: 46, Issue:6

    Topics: Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Bicuculline; Cerebral Cortex; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; gamma-Aminobutyric Acid; Isoxazoles; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vasoactive Intestinal Peptide

1986
Effects of gamma-aminobutyric acid (GABA) receptor agonists on the neurotoxicity and anticonvulsant activity of barbiturates in mice.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Anticonvulsants; Baclofen; Barbiturates; Dose-Response Relationship, Drug; Drug Synergism; Electroshock; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Nervous System; Oxazoles; Receptors, GABA-A; Seizures

1986
gamma-Aminobutyric acid agonists and antagonists alter chloride flux across brain membranes.
    Molecular pharmacology, 1986, Volume: 29, Issue:5

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Animals; Baclofen; Bicuculline; Brain; Cell Membrane; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Liver; Male; Mice; Mice, Inbred DBA; Muscimol; Picrotoxin; Receptors, GABA-A; Sodium; Sulfates; Taurine; Temperature

1986
GABAA receptors in the midbrain central grey mediate the antiaversive action of GABA.
    European journal of pharmacology, 1987, Mar-17, Volume: 135, Issue:2

    Topics: Animals; Avoidance Learning; Baclofen; Electrodes, Implanted; gamma-Aminobutyric Acid; Isoxazoles; Male; Mesencephalon; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Hypnotic action of pentobarbital in mice: a possible mechanism.
    Experimental neurology, 1987, Volume: 97, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Isoxazoles; Male; Mice; Oxazoles; Pentobarbital; Receptors, GABA-A; Reflex; Sleep

1987
Effects of GABAergic drugs on the GABA turnover in the substantia nigra and the corpus striatum of the rat.
    Journal of neural transmission, 1987, Volume: 69, Issue:1-2

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Corpus Striatum; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1987
[Antiabstinent action of fenibut and baclofen on a model of abstinence induced by the benzodiazepine receptor antagonist CGS 8216 in rats receiving diazepam].
    Biulleten' eksperimental'noi biologii i meditsiny, 1987, Volume: 103, Issue:6

    Topics: Animals; Baclofen; Behavior, Animal; Diazepam; Drug Evaluation, Preclinical; gamma-Aminobutyric Acid; Isoxazoles; Male; Pyrazoles; Rats; Receptors, GABA-A; Substance Withdrawal Syndrome; Tranquilizing Agents

1987
Respiratory depressant effects of GABA alpha- and beta-receptor agonists in the cat.
    Journal of applied physiology (Bethesda, Md. : 1985), 1987, Volume: 62, Issue:6

    Topics: Animals; Baclofen; Bicuculline; Cats; Female; Heart; Injections, Intravenous; Injections, Intraventricular; Isoxazoles; Male; Oxazoles; Receptors, GABA-A; Respiration

1987
Evidence that guanosine triphosphate (GTP)-binding proteins control a synaptic response in brain: effect of pertussis toxin and GTP gamma S on the late inhibitory postsynaptic potential of hippocampal CA3 neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1988, Volume: 8, Issue:12

    Topics: Adenylate Cyclase Toxin; Animals; Baclofen; Brain; Electric Conductivity; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Isoxazoles; Membrane Potentials; Neural Inhibition; Neurons; Pertussis Toxin; Rats; Synapses; Thionucleotides; Time Factors; Virulence Factors, Bordetella

1988
Functional responses to baclofen and 4,5,6,7-tetrahydroisoxazolo (5,4-c) pyridin-3-ol (THIP) in rats repeatedly treated with desipramine.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:1

    Topics: Analgesics; Animals; Baclofen; Behavior, Animal; Body Temperature; Desipramine; Isoxazoles; Male; Oxazoles; Rats; Rats, Inbred Strains

1988
An antinociceptive profile of kojic amine: an analogue of gamma-aminobutyric acid (GABA).
    Neuropharmacology, 1987, Volume: 26, Issue:4

    Topics: Animals; Atropine; Atropine Derivatives; Baclofen; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Morphine; Motor Activity; Pain; Pyrans; Pyrones

1987
Effect of GABAergic drugs in the behavioral 'despair' test in rats.
    European journal of pharmacology, 1986, Feb-18, Volume: 121, Issue:2

    Topics: Acetates; Aminooxyacetic Acid; Animals; Baclofen; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Muscimol; Oxazoles; Picrotoxin; Rats

1986
Effects of GABA-mimetic drugs on turnover of histamine in the mouse brain.
    Japanese journal of pharmacology, 1986, Volume: 41, Issue:3

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Brain; Brain Chemistry; gamma-Aminobutyric Acid; Histamine; Isoxazoles; Male; Methylhistamines; Methylhistidines; Mice; Muscimol

1986
The effect of mouse spinal cord transection on the antinociceptive response to the gamma-aminobutyric acid agonists THIP (4,5,6,7-tetrahydroisoxazolo [5,4-c]pyridine-3-ol) and baclofen.
    Brain research, 1985, Jul-15, Volume: 338, Issue:2

    Topics: Analgesics; Animals; Baclofen; Central Nervous System; Clonidine; Cordotomy; Isoxazoles; Male; Mice; Morphine; Oxazoles; Oxotremorine

1985
Subchronic administration of GABAergic agonists elevates [3H]GABA binding and produces tolerance in striatal dopamine catabolism.
    Brain research, 1985, May-27, Volume: 335, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Alkynes; Aminocaproates; Aminooxyacetic Acid; Animals; Baclofen; Corpus Striatum; Dopamine; gamma-Aminobutyric Acid; Isoxazoles; Male; Pyrones; Rats; Rats, Inbred Strains; Vigabatrin

1985
GABAergic mechanisms in antinociception.
    Progress in neuro-psychopharmacology & biological psychiatry, 1984, Volume: 8, Issue:4-6

    Topics: Alkynes; Aminocaproates; Aminooxyacetic Acid; Analgesics; Animals; Baclofen; Bicuculline; Central Nervous System; gamma-Aminobutyric Acid; Isoxazoles; Mice; Muscimol; Pain; Rats; Stereoisomerism; Substance P; Synaptic Transmission; Vigabatrin

1984
GABAergic agents as anticonvulsants in baboons with photosensitive epilepsy.
    Neuroscience letters, 1984, Jun-29, Volume: 47, Issue:3

    Topics: Aminocaproates; Animals; Anticonvulsants; Baclofen; Carbolines; Cerebral Cortex; Dose-Response Relationship, Drug; Epilepsies, Myoclonic; gamma-Aminobutyric Acid; Isoxazoles; Muscimol; Papio; Photic Stimulation; Receptors, Cell Surface; Receptors, GABA-A; Taurine; Vigabatrin

1984
Pretreatment with GABA and modulatory ligands enhances GABA receptor binding.
    European journal of pharmacology, 1984, Sep-03, Volume: 104, Issue:1-2

    Topics: Animals; Baclofen; Binding Sites; Cerebral Cortex; Drug Interactions; gamma-Aminobutyric Acid; In Vitro Techniques; Isoxazoles; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes

1984
Enhancement of spike and wave discharges by GABAmimetic drugs in rats with spontaneous petit-mal-like epilepsy.
    Neuroscience letters, 1984, Jan-27, Volume: 44, Issue:1

    Topics: Action Potentials; Aminocaproates; Animals; Baclofen; Epilepsy, Absence; gamma-Aminobutyric Acid; Isoxazoles; Muscimol; Rats; Vigabatrin

1984
Self-injurious behavior in rats produced by intranigral microinjection of GABA agonists.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Brain; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Male; Microinjections; Muscimol; Rats; Rats, Inbred Strains; Self Mutilation; Stress, Physiological; Substantia Nigra

1984
Effects of intrathecally administered THIP, baclofen and muscimol on nociceptive threshold.
    European journal of pharmacology, 1984, Aug-03, Volume: 103, Issue:1-2

    Topics: Animals; Baclofen; Injections, Spinal; Isoxazoles; Male; Muscimol; Muscle Hypotonia; Nociceptors; Oxazoles; Rats; Rats, Inbred Strains; Reaction Time; Sensory Thresholds

1984
Unilateral injection of GABA agonists in the superior colliculus: asymmetry to tactile stimulation.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:2

    Topics: Analgesics; Animals; Baclofen; Functional Laterality; gamma-Aminobutyric Acid; Isoxazoles; Motor Activity; Muscimol; Oxazoles; Physical Stimulation; Rats; Rats, Inbred Strains; Superior Colliculi; Touch

1983
Nigral actions of GABA agonists are enhanced by chronic fluphenazine and differentiated by concomitant flurazepam.
    Psychopharmacology, 1982, Volume: 76, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Female; Fluphenazine; Flurazepam; gamma-Aminobutyric Acid; Humans; Isoxazoles; Muscimol; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substantia Nigra

1982
Analgesic properties of the GABA-mimetic THIP.
    European journal of pharmacology, 1981, Jan-16, Volume: 69, Issue:2

    Topics: Analgesics; Animals; Arthritis, Experimental; Baclofen; Electric Stimulation; Isoxazoles; Macaca mulatta; Mice; Morphine; Muscimol; Oxazoles; Reaction Time

1981
Interaction between phencyclidine (PCP) and GABA-ergic drugs: clinical implications.
    Pharmacology, biochemistry, and behavior, 1980, Volume: 12, Issue:1

    Topics: Aminooxyacetic Acid; Anesthesia; Animals; Baclofen; Dextroamphetamine; Diazepam; Drug Interactions; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Motor Activity; Muscimol; Pain; Phencyclidine; Reflex

1980
Role of GABAB receptors in intracellular Ca2+ homeostasis and possible interaction between GABAA and GABAB receptors in regulation of transmitter release in cerebellar granule neurons.
    Journal of neuroscience research, 1994, Dec-15, Volume: 39, Issue:6

    Topics: Animals; Aspartic Acid; Baclofen; Calcium; Calcium Radioisotopes; Cells, Cultured; Cerebellum; GABA Agonists; GTP-Binding Proteins; Homeostasis; Isonicotinic Acids; Isoxazoles; Mice; Neurons; Neurotransmitter Agents; Pertussis Toxin; Receptors, GABA-A; Receptors, GABA-B; Virulence Factors, Bordetella

1994
Extrasynaptic effects of GABA (gamma-aminobutyric acid) agonists on myelinated axons of peripheral nerve.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:4

    Topics: Action Potentials; Animals; Axons; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Isoxazoles; Motor Neurons; Nerve Fibers, Myelinated; Peripheral Nerves; Rana catesbeiana; Ranidae; Sciatic Nerve; Spinal Nerve Roots; Synapses

1994
GABA, THIP and baclofen inhibition of Purkinje cells and cerebellar nuclei neurons.
    Neuroscience research, 1993, Volume: 16, Issue:1

    Topics: Animals; Baclofen; Cerebellar Nuclei; Dose-Response Relationship, Drug; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Neural Inhibition; Neurons; Purkinje Cells; Rats; Rats, Sprague-Dawley

1993
N-ethylmaleimide blocks depolarization-induced suppression of inhibition and enhances GABA release in the rat hippocampal slice in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Feb-01, Volume: 17, Issue:3

    Topics: Analysis of Variance; Animals; Baclofen; Ethylmaleimide; Evoked Potentials; GABA Agonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isoxazoles; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA

1997
Neuronal regulation of astrocyte morphology in vitro is mediated by GABAergic signaling.
    Glia, 1997, Volume: 20, Issue:1

    Topics: Animals; Animals, Newborn; Astrocytes; Baclofen; Bicuculline; Cell Adhesion; Cells, Cultured; Coculture Techniques; GABA Agonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Isoxazoles; Muscimol; Neurons; Rats; Rats, Wistar; Signal Transduction; Sodium Channel Blockers; Tetrodotoxin; Time Factors

1997
[Receptor mechanism of the neuroprotective effect of GABAergic agents].
    Biulleten' eksperimental'noi biologii i meditsiny, 1998, Volume: 125, Issue:2

    Topics: Animals; Baclofen; Brain Ischemia; Female; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Injections, Subcutaneous; Isonipecotic Acids; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Muscimol; Neuroprotective Agents; Receptors, GABA-A; Receptors, GABA-B

1998
Effects of the GABA agonists baclofen and THIP on long-term compensation in hemilabyrinthectomised rats.
    Brain research, 1998, Jun-08, Volume: 795, Issue:1-2

    Topics: Animals; Baclofen; Ear, Inner; Eye Movements; Functional Laterality; GABA Agonists; Isoxazoles; Magnetics; Nystagmus, Pathologic; Rats; Rats, Inbred Strains; Reflex, Vestibulo-Ocular

1998
GABAergic drugs and sexual behaviour in the rabbit: evidence for species-specific effects.
    Journal of psychopharmacology (Oxford, England), 1998, Volume: 12, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Copulation; Dose-Response Relationship, Drug; Escape Reaction; GABA Agents; Isoxazoles; Male; Picrotoxin; Rabbits; Rats; Sexual Behavior, Animal; Species Specificity; Structure-Activity Relationship

1998
Interactions between antinociception induced by cholecystokinin antagonists and GABA agonists in the tail-flick test.
    Pharmacology & toxicology, 1998, Volume: 83, Issue:4

    Topics: Animals; Baclofen; Benzodiazepinones; Devazepide; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; Isoxazoles; Male; Mice; Motor Activity; Pain; Pain Measurement; Phenylurea Compounds; Proglumide; Receptors, Cholecystokinin; Tail

1998
Differential effects of GABA(A) and GABA(B) agonists on sensitization to the locomotor stimulant effects of ethanol in DBA/2 J mice.
    Psychopharmacology, 1999, Volume: 141, Issue:2

    Topics: Analysis of Variance; Animals; Baclofen; Central Nervous System Stimulants; Ethanol; GABA Agonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; Isoxazoles; Mice; Mice, Inbred DBA; Motor Activity; Receptors, GABA-A; Receptors, GABA-B

1999
Effects of CCK antagonists on GABA mechanism-induced antinociception in the formalin test.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1999, Volume: 9, Issue:1-2

    Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Baclofen; Dose-Response Relationship, Drug; Formaldehyde; GABA Agents; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Isoxazoles; Male; Mice; Morphine; Pain; Pain Measurement; Receptors, Cholecystokinin

1999
GABA agonists differentially modify blood glucose levels of diabetic rats.
    Japanese journal of pharmacology, 1999, Volume: 80, Issue:4

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Benzodiazepines; Blood Glucose; Diabetes Mellitus, Experimental; Diazepam; Dose-Response Relationship, Drug; Female; GABA Agonists; Insulin; Isoxazoles; Rats; Rats, Wistar

1999
Sensory thresholds and the antinociceptive effects of GABA receptor agonists in mice lacking the beta3 subunit of the GABA(A) receptor.
    Neuroscience, 2000, Volume: 95, Issue:3

    Topics: Animals; Baclofen; GABA Agonists; Hot Temperature; Injections, Spinal; Injections, Subcutaneous; Isonicotinic Acids; Isoxazoles; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Nociceptors; Physical Stimulation; Protein Isoforms; Receptors, GABA-A; Sensory Thresholds; Sex Characteristics

2000
Additivity and independence of neuroprotective effects of GABAA and GABAB receptor agonists in complete global cerebral ischemia.
    Bulletin of experimental biology and medicine, 2000, Volume: 130, Issue:8

    Topics: Animals; Baclofen; Bicuculline; Brain Ischemia; Drug Interactions; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Isoxazoles; Male; Mice; Mice, Inbred CBA; Muscimol; Neuroprotective Agents; Picrotoxin

2000
Involvement of GABAergic neurotransmission in the neurobiology of the apomorphine-induced aggressive behavior paradigm, a model of psychotic behavior in rats.
    Methods and findings in experimental and clinical pharmacology, 2000, Volume: 22, Issue:8

    Topics: Aggression; Animals; Apomorphine; Baclofen; Behavior, Animal; Disease Models, Animal; GABA Agonists; Isoxazoles; Male; Neurotransmitter Agents; Psychotic Disorders; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission

2000
Opposite roles of GABA and excitatory amino acids on the control of GAD expression in cultured retina cells.
    Brain research, 2002, Jan-18, Volume: 925, Issue:1

    Topics: Animals; Baclofen; Cells, Cultured; Chick Embryo; Cytarabine; Excitatory Amino Acid Agonists; GABA Agonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Glutamic Acid; Immunohistochemistry; Isoxazoles; Kainic Acid; Nitric Oxide; Retina

2002
Changes in rectal temperature and ECoG spectral power of sensorimotor cortex elicited in conscious rabbits by i.c.v. injection of GABA, GABA(A) and GABA(B) agonists and antagonists.
    British journal of pharmacology, 2004, Volume: 141, Issue:1

    Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Body Temperature Regulation; Electroencephalography; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Isoxazoles; Lateral Ventricles; Male; Muscimol; Nipecotic Acids; Preoptic Area; Rabbits; Receptors, GABA-A; Receptors, GABA-B; Rectum; Somatosensory Cortex

2004
Effects of gabaergic drugs on reserpine-induced oral dyskinesia.
    Behavioural brain research, 2005, May-07, Volume: 160, Issue:1

    Topics: Analysis of Variance; Animals; Antipsychotic Agents; Baclofen; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Dyskinesia, Drug-Induced; GABA Agents; Immobility Response, Tonic; Isoxazoles; Locomotion; Male; Rats; Rats, Wistar; Reserpine

2005
Endogenous activation of kainate receptors regulates glutamate release and network activity in the developing hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, May-04, Volume: 25, Issue:18

    Topics: Animals; Animals, Newborn; Aspartic Acid; Baclofen; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Furans; GABA Agonists; GABA Antagonists; Glutamic Acid; Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Interneurons; Isoquinolines; Isoxazoles; Membrane Potentials; Mice; Mice, Knockout; Nerve Net; Neural Inhibition; Neurons; Patch-Clamp Techniques; Picrotoxin; Probability; Receptors, Kainic Acid

2005
GABAergic modulation of binge-like ethanol intake in C57BL/6J mice.
    Pharmacology, biochemistry, and behavior, 2007, Volume: 88, Issue:1

    Topics: Alcoholism; Animals; Baclofen; Central Nervous System Depressants; Darkness; Dose-Response Relationship, Drug; Ethanol; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Muscimol; Postural Balance

2007
Discriminative stimulus effects of tiagabine and related GABAergic drugs in rats.
    Psychopharmacology, 2008, Volume: 197, Issue:4

    Topics: Administration, Oral; Amines; Animals; Anticonvulsants; Azabicyclo Compounds; Baclofen; Benzodiazepines; Bicuculline; Brain; Cyclohexanecarboxylic Acids; Discrimination Learning; Dose-Response Relationship, Drug; GABA Agents; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; Gabapentin; gamma-Aminobutyric Acid; Generalization, Stimulus; Hypnotics and Sedatives; Injections, Intraperitoneal; Isoxazoles; Male; Nipecotic Acids; Piperazines; Pyridines; Rats; Thiophenes; Tiagabine; Zolpidem

2008