isoxazoles has been researched along with baclofen in 79 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 45 (56.96) | 18.7374 |
1990's | 22 (27.85) | 18.2507 |
2000's | 9 (11.39) | 29.6817 |
2010's | 3 (3.80) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Waddington, JL | 1 |
Guidotti, A; Kurosawa, A; Naik, SR | 1 |
Agnati, L; Fuxe, K; Hökfelt, T; Johansson, O; Ljungdahl, A; Perez de la Mora, M | 1 |
Amit, Z; Robidoux, J; Smith, BR | 1 |
Ebbesson, SO; Erdö, SL; Hofmann, MH; Malz, CR; Meyer, DL | 1 |
Barolet, AW; Morris, ME | 1 |
Agmo, A; Gutiérrez, M; Guzmán, M; Pruneda, R | 1 |
Bergen, HT; Hejtmancik, JF; Pfaff, DW | 1 |
Boelen, MK; Chubb, IW; Dowton, M; Morgan, IG; Wellard, J | 1 |
Catt, KJ; Stojilković, SS; Virmani, MA | 1 |
Balcar, VJ; Dreher, B | 1 |
Michler, A | 1 |
Hicks, TP; Kaneko, T | 1 |
Agmo, A; Paredes, R; Soria, P | 1 |
Erdö, SL; Michler, A | 1 |
Karlsson, G; Olpe, HR | 1 |
Aarslew-Jensen, M; Diemer, NH; Krogsgaard-Larsen, P; Nielsen, EO; Schousboe, A | 1 |
Thalmann, RH | 2 |
Mehta, AK; Ticku, MK | 1 |
Bitran, D; Leipheimer, RE; McQuade, DB; Miller, SA; Sachs, BD | 1 |
Bond, A; Neal, H | 1 |
Alho, H; Fujimoto, M; Geffard, M; Guidotti, A; Hanbauer, I; Kataoka, Y; Kelly, GD | 1 |
Borsini, F; Giuliani, S; Meli, A | 2 |
Karobath, M; Supavilai, P | 1 |
Costa, LG; Enna, SJ; Pelley, K; Setler, P; Vaught, JL | 1 |
Gianutsos, G; Suzdak, PD | 2 |
Agmo, A; Paredes, R | 1 |
Agmo, A; Giordano, M | 1 |
Hösli, E; Hösli, L; Krogsgaard-Larsen, P | 1 |
Bristow, DR; Watling, KJ | 1 |
Chweh, AY; Swinyard, EA; Ulloque, RA | 1 |
Allan, AM; Harris, RA | 1 |
Audi, EA; Graeff, FG | 1 |
Chweh, AY; Swinyard, EA; Wolf, HH | 1 |
Lindgren, S | 1 |
Zharkovskaia, TA; Zharkovskiĭ, AM | 1 |
Gillis, RA; Hamosh, P; Hartley, B; Quest, JA; Taveira da Silva, AM | 1 |
Pelley, KA; Vaught, JL | 1 |
Borsini, F; Evangelista, S; Meli, A | 1 |
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K | 1 |
Enna, SJ; Zorn, SH | 1 |
Beart, PM; Lloyd, KG; Scatton, B | 1 |
Sawynok, J | 1 |
Meldrum, B | 1 |
Maksay, G; Ticku, MK | 1 |
Depaulis, A; Marescaux, C; Micheletti, G; Rumbach, L; Vergnes, M; Warter, JM | 1 |
Baumeister, AA; Frye, GD | 1 |
Drower, EJ; Hammond, DL | 1 |
Di Scala, G; Karli, P; Schmitt, P | 1 |
Coward, DM | 1 |
Buescher, HH; Hill, RC; Maurer, R; Roemer, D | 1 |
Clark, WG; Menon, MK; Vivonia, C | 1 |
Damgaard, I; Elster, L; Kardos, J; Krogsgaard-Larsen, P; Schousboe, A | 1 |
Liske, S; Morris, ME | 1 |
Batini, C; Billard, JM; Vigot, R | 1 |
Alger, BE; Kirov, SA; Lenz, RA; Martin, LA; Morishita, W; Pitler, TA | 1 |
Matsutani, S; Yamamoto, N | 1 |
Kulinskiĭ, VI; Mikhel'son, GV | 2 |
Eriksson, B; Magnusson, AK; Tham, R | 1 |
Agmo, A; Contreras, JL; Paredes, RG | 1 |
Ghanipoor, N; Parvini, S; Rezayat, M; Zarrindast, MR | 1 |
Broadbent, J; Harless, WE | 1 |
Parvini, S; Pirali, M; Rezayat, M; Tabarrai, E; Zarrindast, MR | 1 |
Asnis, N; Barros, HM; Gomez, R; Tannhauser, SL | 1 |
Firestone, LL; Hammond, DL; Homanics, GE; Ugarte, SD | 1 |
Allikmets, L; Matto, V; Pruus, K; Rudissaar, R; Skrebuhhova-Malmros, T | 1 |
de Almeida, OM; de Mello, FG; de Mello, MC; Gardino, PF; Hokoç, JN; Loureiro dos Santos, NE; Yamasaki, EN | 1 |
Frosini, M; Sgaragli, G; Valoti, M | 1 |
Abílio, VC; Araujo, NP; Castro, JP; Faria, RR; Frussa-Filho, R; Fukushiro, DF; Medrano, WA; Peixoto, MF; Silva, RH; Zanier-Gomes, PH | 1 |
Collingridge, GL; Isaac, JT; Lauri, SE; Maingret, F; Mulle, C; Segerstråle, M; Taira, T; Vesikansa, A | 1 |
Boehm, SL; Goldfarb, KJ; Linsenbardt, DN; Moore, EM; Serio, KM; Stepanovska, S | 1 |
Hutson, PH; McDonald, LM; Sheppard, WF; Sohal, B; Staveley, SM; Tattersall, FD | 1 |
Ang, D; De Santis, A; Pauwels, A; Scarpellini, E; Tack, J; Vanuytsel, T | 1 |
Johnston, GAR | 1 |
Alabed, S; Bergman, H; Latifeh, Y; Mohammad, HA | 1 |
3 review(s) available for isoxazoles and baclofen
Article | Year |
---|---|
Management of refractory typical GERD symptoms.
Topics: Alginates; Algorithms; Antacids; Baclofen; Chronic Disease; Esophagoscopy; Gastroesophageal Reflux; Gastrointestinal Agents; Gastroscopy; Humans; Isoxazoles; Muscle Relaxants, Central; Neurotransmitter Agents; Phosphinic Acids; Propylamines; Triazoles | 2016 |
GABA Australis, some reflections on the history of GABA receptor research in Australia.
Topics: Animals; Australia; Baclofen; Bicuculline; Cyclic AMP; Humans; Isoxazoles; Muscimol; Receptors, GABA | 2017 |
Gamma-aminobutyric acid agonists for antipsychotic-induced tardive dyskinesia.
Topics: Antipsychotic Agents; Baclofen; Dyskinesia, Drug-Induced; GABA Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Placebos; Randomized Controlled Trials as Topic; Valproic Acid | 2018 |
76 other study(ies) available for isoxazoles and baclofen
Article | Year |
---|---|
GABA-like properties of flurazepam and baclofen suggested by rotational behaviour following unilateral intranigral injection: a comparison with the GABA agonist muscimol [proceedings].
Topics: Aminobutyrates; Animals; Anti-Anxiety Agents; Baclofen; Behavior; Flurazepam; gamma-Aminobutyric Acid; Humans; Injections; Isoxazoles; Male; Oxazoles; Rats; Stereotyped Behavior; Substantia Nigra | 1977 |
Possible role of gamma aminobutyric acid (GABA) in the regulation of cAMP system in rat anterior pituitary.
Topics: Aminobutyrates; Animals; Baclofen; Cyclic AMP; Diazepam; gamma-Aminobutyric Acid; Hypothalamus; Isoniazid; Isoxazoles; Male; Nipecotic Acids; Pargyline; Picrotoxin; Pituitary Gland, Anterior; Protein Kinases; Rats; Reserpine | 1977 |
Regulation of the mesocortical dopamine neurons.
Topics: 4-Butyrolactone; Acetylcholine; Aminooxyacetic Acid; Baclofen; Cerebral Cortex; Dopamine; gamma-Aminobutyric Acid; Isoxazoles; Neurons; Pimozide; Pyrrolidinones; Sulpiride | 1977 |
GABAergic involvement in the acquisition of voluntary ethanol intake in laboratory rats.
Topics: Alcohol Drinking; Animals; Baclofen; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Isoxazoles; Male; Rats; Receptors, GABA-A | 1992 |
Changes in ligand binding to GABAA receptor sites in pacific salmon (Oncorhynchus) brain during spawning migration and "aging".
Topics: Aging; Aminobutyrates; Analgesics; Animals; Baclofen; Bicuculline; Binding, Competitive; Brain; Female; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Ligands; Male; Muscimol; Receptors, GABA-A; Salmon; Sexual Behavior, Animal | 1992 |
Changes in extracellular K+ evoked by GABA, THIP and baclofen in the guinea-pig hippocampal slice.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Electrodes; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Isoxazoles; Nipecotic Acids; Potassium; Proline; Receptors, GABA-A; Temperature | 1991 |
GABAergic drugs and conflict behavior in the rat: lack of similarities with the actions of benzodiazepines.
Topics: Alkynes; Aminocaproates; Animals; Baclofen; Behavior, Animal; Benzodiazepines; Bicuculline; Brain; Conflict, Psychological; Drug Interactions; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Nicotinic Acids; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission | 1991 |
Effects of gamma-aminobutyric acid receptor agonists and antagonist on LHRH-synthesizing neurons as detected by immunocytochemistry and in situ hybridization.
Topics: Animals; Baclofen; Bicuculline; Female; GABA-A Receptor Antagonists; Gene Expression Regulation; Gonadotropin-Releasing Hormone; Immunohistochemistry; Isoxazoles; Neurons; Nucleic Acid Hybridization; Ovariectomy; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; RNA Probes; RNA, Messenger | 1991 |
Glycinergic control of [Leu5]enkephalin levels in chicken retina.
Topics: Animals; Baclofen; Chickens; Enkephalin, Leucine; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Isoxazoles; Muscimol; Neurotransmitter Agents; Picrotoxin; Radioimmunoassay; Retina; Strychnine | 1991 |
Stimulation of luteinizing hormone release by gamma-aminobutyric acid (GABA) agonists: mediation by GABAA-type receptors and activation of chloride and voltage-sensitive calcium channels.
Topics: Amino Acid Sequence; Animals; Baclofen; Calcium Channels; Cells, Cultured; Chloride Channels; Chlorides; Female; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Isoxazoles; Luteinizing Hormone; Membrane Proteins; Molecular Sequence Data; Muscimol; Nifedipine; Pituitary Gland, Anterior; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Neurochemical correlates of gamma-aminobutyrate (GABA) inhibition in cat visual cortex.
Topics: Animals; Baclofen; Calcium; Cats; Cell Membrane; Female; GABA Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Neurons; Potassium; Pyridazines; Receptors, GABA-A; Visual Cortex | 1990 |
Involvement of GABA receptors in the regulation of neurite growth in cultured embryonic chick tectum.
Topics: Animals; Axons; Baclofen; Cells, Cultured; Chick Embryo; Culture Media; gamma-Aminobutyric Acid; Isoxazoles; Ligands; Muscimol; Receptors, GABA-A; Superior Colliculi | 1990 |
GABA(B)-related activity involved in synaptic processing of somatosensory information in S1 cortex of the anaesthetized cat.
Topics: Anesthesia; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrodes; Female; gamma-Aminobutyric Acid; Iontophoresis; Isoxazoles; Male; Muscimol; Neurons; Physical Stimulation; Somatosensory Cortex; Synapses | 1990 |
GABAergic drugs and lordosis behavior in the female rat.
Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Estradiol; Female; gamma-Aminobutyric Acid; Isoxazoles; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal; Taurine | 1989 |
Stimulation by phaclofen of inositol 1,4,5-triphosphate production in cultured neurons from chick tectum.
Topics: Animals; Baclofen; Chick Embryo; gamma-Aminobutyric Acid; Inosine Nucleotides; Inosine Triphosphate; Isoxazoles; Neurons; Receptors, GABA-A; Superior Colliculi | 1989 |
Late inhibitory postsynaptic potentials in rat prefrontal cortex may be mediated by GABAB receptors.
Topics: Animals; Baclofen; Electric Conductivity; Electric Stimulation; Evoked Potentials; Frontal Lobe; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Isoxazoles; Male; Membrane Potentials; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synapses | 1989 |
Baclofen-induced, calcium-dependent stimulation of in vivo release of D-[3H]aspartate from rat hippocampus monitored by intracerebral microdialysis.
Topics: Animals; Aspartic Acid; Baclofen; Calcium; GABA Antagonists; Hippocampus; Ischemic Attack, Transient; Isoxazoles; Male; Potassium; Rats; Rats, Inbred Strains | 1989 |
Pertussis toxin blocks a late inhibitory postsynaptic potential in hippocampal CA3 neurons.
Topics: Action Potentials; Adenylate Cyclase Toxin; Animals; Baclofen; Hippocampus; In Vitro Techniques; Isoxazoles; Neural Conduction; Neural Inhibition; Pertussis Toxin; Rats; Receptors, GABA-A; Virulence Factors, Bordetella | 1987 |
Interactions of pentobarbital and phenobarbital with GABAergic drugs against chemoconvulsants in rats.
Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Convulsants; Diazepam; Drug Interactions; Isoxazoles; Male; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Strychnine | 1988 |
Inhibition of sexual reflexes by lumbosacral injection of a GABAB agonist in the male rat.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Injections, Spinal; Isoxazoles; Lumbosacral Region; Male; Penile Erection; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal; Spinal Cord | 1988 |
Quantitative electrocortical changes in the rat induced by phencyclidine and other stimulants.
Topics: Animals; Apomorphine; Baclofen; Cerebral Cortex; Chlordiazepoxide; Chlorpromazine; Dextroamphetamine; Dioxolanes; Electroencephalography; Isoquinolines; Isoxazoles; Male; Muscimol; Phencyclidine; Rats; Rats, Inbred Strains | 1985 |
Intrinsic gamma aminobutyric acid receptors modulate the release of catecholamine from canine adrenal gland in situ.
Topics: Adrenal Medulla; Animals; Baclofen; Bicuculline; Chromaffin Granules; Dogs; Electric Stimulation; Epinephrine; Female; Hexamethonium; Hexamethonium Compounds; Histocytochemistry; Isoxazoles; Muscimol; Naloxone; Norepinephrine; Receptors, GABA-A; Splanchnic Nerves | 1986 |
Functional evidence for altered activity of GABAergic receptors following chronic desipramine treatment in rats.
Topics: Analgesics; Animals; Baclofen; Desipramine; Isoxazoles; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1986 |
Modulation of acetylcholine release from rat striatal slices by the GABA/benzodiazepine receptor complex.
Topics: Acetylcholine; Animals; Atropine; Baclofen; Benzodiazepinones; Clonazepam; Corpus Striatum; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Haloperidol; In Vitro Techniques; Isoxazoles; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
A comparison of the antinociceptive responses to the GABA-receptor agonists THIP and baclofen.
Topics: Analgesics; Animals; Baclofen; Dose-Response Relationship, Drug; Drug Tolerance; Isoxazoles; Male; Mice; Oxazoles; Postural Balance; Receptors, GABA-A | 1985 |
Parallel changes in the sensitivity of gamma-aminobutyric acid and noradrenergic receptors following chronic administration of antidepressant and GABAergic drugs. A possible role in affective disorders.
Topics: Animals; Anticonvulsants; Antidepressive Agents; Baclofen; Cerebral Cortex; Dihydroalprenolol; gamma-Aminobutyric Acid; Hippocampus; Humans; Imipramine; Isoxazoles; Kinetics; Male; Mice; Mood Disorders; Nomifensine; Receptors, Adrenergic; Receptors, GABA-A | 1985 |
GABAergic drugs and sexual behaviour in the male rat.
Topics: 4-Aminobutyrate Transaminase; Alkynes; Aminocaproates; Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal | 1985 |
GABAergic effects of reserpine following chronic treatment.
Topics: Animals; Baclofen; Binding, Competitive; Cerebral Cortex; Dihydroalprenolol; gamma-Aminobutyric Acid; Hippocampus; Imipramine; Isoxazoles; Male; Mice; Receptors, GABA-A; Reserpine | 1985 |
The locomotor-reducing effects of GABAergic drugs do not depend on the GABAA receptor.
Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Isoxazoles; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taurine | 1985 |
Autoradiographic localization of binding sites for the gamma-aminobutyric acid analogues 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol (THIP)isoguvacine and baclofen on cultured neurons of rat cerebellum and spinal cord.
Topics: Animals; Animals, Newborn; Autoradiography; Baclofen; Binding Sites; Cells, Cultured; Cerebellum; Fetus; Isonicotinic Acids; Isoxazoles; Oxazoles; Rats; Receptors, GABA-A; Spinal Cord | 1985 |
GABAB receptor-mediated enhancement of vasoactive intestinal peptide-stimulated cyclic AMP production in slices of rat cerebral cortex.
Topics: Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Bicuculline; Cerebral Cortex; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; gamma-Aminobutyric Acid; Isoxazoles; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vasoactive Intestinal Peptide | 1986 |
Effects of gamma-aminobutyric acid (GABA) receptor agonists on the neurotoxicity and anticonvulsant activity of barbiturates in mice.
Topics: Animals; Anticonvulsants; Baclofen; Barbiturates; Dose-Response Relationship, Drug; Drug Synergism; Electroshock; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Nervous System; Oxazoles; Receptors, GABA-A; Seizures | 1986 |
gamma-Aminobutyric acid agonists and antagonists alter chloride flux across brain membranes.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Animals; Baclofen; Bicuculline; Brain; Cell Membrane; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Liver; Male; Mice; Mice, Inbred DBA; Muscimol; Picrotoxin; Receptors, GABA-A; Sodium; Sulfates; Taurine; Temperature | 1986 |
GABAA receptors in the midbrain central grey mediate the antiaversive action of GABA.
Topics: Animals; Avoidance Learning; Baclofen; Electrodes, Implanted; gamma-Aminobutyric Acid; Isoxazoles; Male; Mesencephalon; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Hypnotic action of pentobarbital in mice: a possible mechanism.
Topics: Animals; Baclofen; Bicuculline; Isoxazoles; Male; Mice; Oxazoles; Pentobarbital; Receptors, GABA-A; Reflex; Sleep | 1987 |
Effects of GABAergic drugs on the GABA turnover in the substantia nigra and the corpus striatum of the rat.
Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Corpus Striatum; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1987 |
[Antiabstinent action of fenibut and baclofen on a model of abstinence induced by the benzodiazepine receptor antagonist CGS 8216 in rats receiving diazepam].
Topics: Animals; Baclofen; Behavior, Animal; Diazepam; Drug Evaluation, Preclinical; gamma-Aminobutyric Acid; Isoxazoles; Male; Pyrazoles; Rats; Receptors, GABA-A; Substance Withdrawal Syndrome; Tranquilizing Agents | 1987 |
Respiratory depressant effects of GABA alpha- and beta-receptor agonists in the cat.
Topics: Animals; Baclofen; Bicuculline; Cats; Female; Heart; Injections, Intravenous; Injections, Intraventricular; Isoxazoles; Male; Oxazoles; Receptors, GABA-A; Respiration | 1987 |
Evidence that guanosine triphosphate (GTP)-binding proteins control a synaptic response in brain: effect of pertussis toxin and GTP gamma S on the late inhibitory postsynaptic potential of hippocampal CA3 neurons.
Topics: Adenylate Cyclase Toxin; Animals; Baclofen; Brain; Electric Conductivity; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Isoxazoles; Membrane Potentials; Neural Inhibition; Neurons; Pertussis Toxin; Rats; Synapses; Thionucleotides; Time Factors; Virulence Factors, Bordetella | 1988 |
Functional responses to baclofen and 4,5,6,7-tetrahydroisoxazolo (5,4-c) pyridin-3-ol (THIP) in rats repeatedly treated with desipramine.
Topics: Analgesics; Animals; Baclofen; Behavior, Animal; Body Temperature; Desipramine; Isoxazoles; Male; Oxazoles; Rats; Rats, Inbred Strains | 1988 |
An antinociceptive profile of kojic amine: an analogue of gamma-aminobutyric acid (GABA).
Topics: Animals; Atropine; Atropine Derivatives; Baclofen; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Morphine; Motor Activity; Pain; Pyrans; Pyrones | 1987 |
Effect of GABAergic drugs in the behavioral 'despair' test in rats.
Topics: Acetates; Aminooxyacetic Acid; Animals; Baclofen; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Muscimol; Oxazoles; Picrotoxin; Rats | 1986 |
Effects of GABA-mimetic drugs on turnover of histamine in the mouse brain.
Topics: Aminooxyacetic Acid; Animals; Baclofen; Brain; Brain Chemistry; gamma-Aminobutyric Acid; Histamine; Isoxazoles; Male; Methylhistamines; Methylhistidines; Mice; Muscimol | 1986 |
The effect of mouse spinal cord transection on the antinociceptive response to the gamma-aminobutyric acid agonists THIP (4,5,6,7-tetrahydroisoxazolo [5,4-c]pyridine-3-ol) and baclofen.
Topics: Analgesics; Animals; Baclofen; Central Nervous System; Clonidine; Cordotomy; Isoxazoles; Male; Mice; Morphine; Oxazoles; Oxotremorine | 1985 |
Subchronic administration of GABAergic agonists elevates [3H]GABA binding and produces tolerance in striatal dopamine catabolism.
Topics: 3,4-Dihydroxyphenylacetic Acid; Alkynes; Aminocaproates; Aminooxyacetic Acid; Animals; Baclofen; Corpus Striatum; Dopamine; gamma-Aminobutyric Acid; Isoxazoles; Male; Pyrones; Rats; Rats, Inbred Strains; Vigabatrin | 1985 |
GABAergic mechanisms in antinociception.
Topics: Alkynes; Aminocaproates; Aminooxyacetic Acid; Analgesics; Animals; Baclofen; Bicuculline; Central Nervous System; gamma-Aminobutyric Acid; Isoxazoles; Mice; Muscimol; Pain; Rats; Stereoisomerism; Substance P; Synaptic Transmission; Vigabatrin | 1984 |
GABAergic agents as anticonvulsants in baboons with photosensitive epilepsy.
Topics: Aminocaproates; Animals; Anticonvulsants; Baclofen; Carbolines; Cerebral Cortex; Dose-Response Relationship, Drug; Epilepsies, Myoclonic; gamma-Aminobutyric Acid; Isoxazoles; Muscimol; Papio; Photic Stimulation; Receptors, Cell Surface; Receptors, GABA-A; Taurine; Vigabatrin | 1984 |
Pretreatment with GABA and modulatory ligands enhances GABA receptor binding.
Topics: Animals; Baclofen; Binding Sites; Cerebral Cortex; Drug Interactions; gamma-Aminobutyric Acid; In Vitro Techniques; Isoxazoles; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes | 1984 |
Enhancement of spike and wave discharges by GABAmimetic drugs in rats with spontaneous petit-mal-like epilepsy.
Topics: Action Potentials; Aminocaproates; Animals; Baclofen; Epilepsy, Absence; gamma-Aminobutyric Acid; Isoxazoles; Muscimol; Rats; Vigabatrin | 1984 |
Self-injurious behavior in rats produced by intranigral microinjection of GABA agonists.
Topics: Animals; Baclofen; Bicuculline; Brain; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Male; Microinjections; Muscimol; Rats; Rats, Inbred Strains; Self Mutilation; Stress, Physiological; Substantia Nigra | 1984 |
Effects of intrathecally administered THIP, baclofen and muscimol on nociceptive threshold.
Topics: Animals; Baclofen; Injections, Spinal; Isoxazoles; Male; Muscimol; Muscle Hypotonia; Nociceptors; Oxazoles; Rats; Rats, Inbred Strains; Reaction Time; Sensory Thresholds | 1984 |
Unilateral injection of GABA agonists in the superior colliculus: asymmetry to tactile stimulation.
Topics: Analgesics; Animals; Baclofen; Functional Laterality; gamma-Aminobutyric Acid; Isoxazoles; Motor Activity; Muscimol; Oxazoles; Physical Stimulation; Rats; Rats, Inbred Strains; Superior Colliculi; Touch | 1983 |
Nigral actions of GABA agonists are enhanced by chronic fluphenazine and differentiated by concomitant flurazepam.
Topics: Animals; Baclofen; Bicuculline; Female; Fluphenazine; Flurazepam; gamma-Aminobutyric Acid; Humans; Isoxazoles; Muscimol; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substantia Nigra | 1982 |
Analgesic properties of the GABA-mimetic THIP.
Topics: Analgesics; Animals; Arthritis, Experimental; Baclofen; Electric Stimulation; Isoxazoles; Macaca mulatta; Mice; Morphine; Muscimol; Oxazoles; Reaction Time | 1981 |
Interaction between phencyclidine (PCP) and GABA-ergic drugs: clinical implications.
Topics: Aminooxyacetic Acid; Anesthesia; Animals; Baclofen; Dextroamphetamine; Diazepam; Drug Interactions; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Motor Activity; Muscimol; Pain; Phencyclidine; Reflex | 1980 |
Role of GABAB receptors in intracellular Ca2+ homeostasis and possible interaction between GABAA and GABAB receptors in regulation of transmitter release in cerebellar granule neurons.
Topics: Animals; Aspartic Acid; Baclofen; Calcium; Calcium Radioisotopes; Cells, Cultured; Cerebellum; GABA Agonists; GTP-Binding Proteins; Homeostasis; Isonicotinic Acids; Isoxazoles; Mice; Neurons; Neurotransmitter Agents; Pertussis Toxin; Receptors, GABA-A; Receptors, GABA-B; Virulence Factors, Bordetella | 1994 |
Extrasynaptic effects of GABA (gamma-aminobutyric acid) agonists on myelinated axons of peripheral nerve.
Topics: Action Potentials; Animals; Axons; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Isoxazoles; Motor Neurons; Nerve Fibers, Myelinated; Peripheral Nerves; Rana catesbeiana; Ranidae; Sciatic Nerve; Spinal Nerve Roots; Synapses | 1994 |
GABA, THIP and baclofen inhibition of Purkinje cells and cerebellar nuclei neurons.
Topics: Animals; Baclofen; Cerebellar Nuclei; Dose-Response Relationship, Drug; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Neural Inhibition; Neurons; Purkinje Cells; Rats; Rats, Sprague-Dawley | 1993 |
N-ethylmaleimide blocks depolarization-induced suppression of inhibition and enhances GABA release in the rat hippocampal slice in vitro.
Topics: Analysis of Variance; Animals; Baclofen; Ethylmaleimide; Evoked Potentials; GABA Agonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isoxazoles; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA | 1997 |
Neuronal regulation of astrocyte morphology in vitro is mediated by GABAergic signaling.
Topics: Animals; Animals, Newborn; Astrocytes; Baclofen; Bicuculline; Cell Adhesion; Cells, Cultured; Coculture Techniques; GABA Agonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Isoxazoles; Muscimol; Neurons; Rats; Rats, Wistar; Signal Transduction; Sodium Channel Blockers; Tetrodotoxin; Time Factors | 1997 |
[Receptor mechanism of the neuroprotective effect of GABAergic agents].
Topics: Animals; Baclofen; Brain Ischemia; Female; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Injections, Subcutaneous; Isonipecotic Acids; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Muscimol; Neuroprotective Agents; Receptors, GABA-A; Receptors, GABA-B | 1998 |
Effects of the GABA agonists baclofen and THIP on long-term compensation in hemilabyrinthectomised rats.
Topics: Animals; Baclofen; Ear, Inner; Eye Movements; Functional Laterality; GABA Agonists; Isoxazoles; Magnetics; Nystagmus, Pathologic; Rats; Rats, Inbred Strains; Reflex, Vestibulo-Ocular | 1998 |
GABAergic drugs and sexual behaviour in the rabbit: evidence for species-specific effects.
Topics: Animals; Baclofen; Bicuculline; Copulation; Dose-Response Relationship, Drug; Escape Reaction; GABA Agents; Isoxazoles; Male; Picrotoxin; Rabbits; Rats; Sexual Behavior, Animal; Species Specificity; Structure-Activity Relationship | 1998 |
Interactions between antinociception induced by cholecystokinin antagonists and GABA agonists in the tail-flick test.
Topics: Animals; Baclofen; Benzodiazepinones; Devazepide; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; Isoxazoles; Male; Mice; Motor Activity; Pain; Pain Measurement; Phenylurea Compounds; Proglumide; Receptors, Cholecystokinin; Tail | 1998 |
Differential effects of GABA(A) and GABA(B) agonists on sensitization to the locomotor stimulant effects of ethanol in DBA/2 J mice.
Topics: Analysis of Variance; Animals; Baclofen; Central Nervous System Stimulants; Ethanol; GABA Agonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; Isoxazoles; Mice; Mice, Inbred DBA; Motor Activity; Receptors, GABA-A; Receptors, GABA-B | 1999 |
Effects of CCK antagonists on GABA mechanism-induced antinociception in the formalin test.
Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Baclofen; Dose-Response Relationship, Drug; Formaldehyde; GABA Agents; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Isoxazoles; Male; Mice; Morphine; Pain; Pain Measurement; Receptors, Cholecystokinin | 1999 |
GABA agonists differentially modify blood glucose levels of diabetic rats.
Topics: Aminooxyacetic Acid; Animals; Baclofen; Benzodiazepines; Blood Glucose; Diabetes Mellitus, Experimental; Diazepam; Dose-Response Relationship, Drug; Female; GABA Agonists; Insulin; Isoxazoles; Rats; Rats, Wistar | 1999 |
Sensory thresholds and the antinociceptive effects of GABA receptor agonists in mice lacking the beta3 subunit of the GABA(A) receptor.
Topics: Animals; Baclofen; GABA Agonists; Hot Temperature; Injections, Spinal; Injections, Subcutaneous; Isonicotinic Acids; Isoxazoles; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Nociceptors; Physical Stimulation; Protein Isoforms; Receptors, GABA-A; Sensory Thresholds; Sex Characteristics | 2000 |
Additivity and independence of neuroprotective effects of GABAA and GABAB receptor agonists in complete global cerebral ischemia.
Topics: Animals; Baclofen; Bicuculline; Brain Ischemia; Drug Interactions; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Isoxazoles; Male; Mice; Mice, Inbred CBA; Muscimol; Neuroprotective Agents; Picrotoxin | 2000 |
Involvement of GABAergic neurotransmission in the neurobiology of the apomorphine-induced aggressive behavior paradigm, a model of psychotic behavior in rats.
Topics: Aggression; Animals; Apomorphine; Baclofen; Behavior, Animal; Disease Models, Animal; GABA Agonists; Isoxazoles; Male; Neurotransmitter Agents; Psychotic Disorders; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission | 2000 |
Opposite roles of GABA and excitatory amino acids on the control of GAD expression in cultured retina cells.
Topics: Animals; Baclofen; Cells, Cultured; Chick Embryo; Cytarabine; Excitatory Amino Acid Agonists; GABA Agonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Glutamic Acid; Immunohistochemistry; Isoxazoles; Kainic Acid; Nitric Oxide; Retina | 2002 |
Changes in rectal temperature and ECoG spectral power of sensorimotor cortex elicited in conscious rabbits by i.c.v. injection of GABA, GABA(A) and GABA(B) agonists and antagonists.
Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Body Temperature Regulation; Electroencephalography; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Isoxazoles; Lateral Ventricles; Male; Muscimol; Nipecotic Acids; Preoptic Area; Rabbits; Receptors, GABA-A; Receptors, GABA-B; Rectum; Somatosensory Cortex | 2004 |
Effects of gabaergic drugs on reserpine-induced oral dyskinesia.
Topics: Analysis of Variance; Animals; Antipsychotic Agents; Baclofen; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Dyskinesia, Drug-Induced; GABA Agents; Immobility Response, Tonic; Isoxazoles; Locomotion; Male; Rats; Rats, Wistar; Reserpine | 2005 |
Endogenous activation of kainate receptors regulates glutamate release and network activity in the developing hippocampus.
Topics: Animals; Animals, Newborn; Aspartic Acid; Baclofen; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Furans; GABA Agonists; GABA Antagonists; Glutamic Acid; Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Interneurons; Isoquinolines; Isoxazoles; Membrane Potentials; Mice; Mice, Knockout; Nerve Net; Neural Inhibition; Neurons; Patch-Clamp Techniques; Picrotoxin; Probability; Receptors, Kainic Acid | 2005 |
GABAergic modulation of binge-like ethanol intake in C57BL/6J mice.
Topics: Alcoholism; Animals; Baclofen; Central Nervous System Depressants; Darkness; Dose-Response Relationship, Drug; Ethanol; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Muscimol; Postural Balance | 2007 |
Discriminative stimulus effects of tiagabine and related GABAergic drugs in rats.
Topics: Administration, Oral; Amines; Animals; Anticonvulsants; Azabicyclo Compounds; Baclofen; Benzodiazepines; Bicuculline; Brain; Cyclohexanecarboxylic Acids; Discrimination Learning; Dose-Response Relationship, Drug; GABA Agents; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; Gabapentin; gamma-Aminobutyric Acid; Generalization, Stimulus; Hypnotics and Sedatives; Injections, Intraperitoneal; Isoxazoles; Male; Nipecotic Acids; Piperazines; Pyridines; Rats; Thiophenes; Tiagabine; Zolpidem | 2008 |