isoxazoles has been researched along with 1,2-benzisoxazole in 14 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 2 (14.29) | 29.6817 |
| 2010's | 12 (85.71) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Lemma-Gray, P; Liu, XC | 1 |
| Buckheit, RW; Cullen, MD; Cushman, M; De Clercq, E; Deng, BL; Fanwick, PE; Hartman, TL; Pannecouque, C; Zhou, Z | 1 |
| Keeling, S; Mason, C; Moses, JE; Ritson, DJ; Sharma, P; Spiteri, C; Zhang, F | 1 |
| Keeling, S; Macdonald, SJ; Moses, JE; Sharma, P; Spiteri, C; Zhang, F | 1 |
| Driver, TG; Pan, M; Stokes, BJ; Urnezis, LK; Vogel, CV | 1 |
| Deadman, J; Jones, ED; Le, G; Smith, JA | 1 |
| Endo, T; Kanda, T; Nakamura, H; Sakuma, S; Yamakawa, T; Yamasaki, S | 1 |
| Uto, Y | 3 |
| Gowda, DC; Shantharam, CS; Sridhara, MB; Suhas, R; Suyoga Vardhan, DM | 1 |
| Dubrovskiy, AV; Jain, P; Larock, RC; Lushington, GH; Porubsky, P; Santini, C; Shi, F | 1 |
| Ellman, JA; Otley, KD | 1 |
| Anusha, S; Ashwini, N; Bender, A; Fuchs, JE; Garg, M; Kanojia, D; Koeffler, HP; Madan, V; Mohan, CD; Rakesh, KS; Rangappa, KS; Rangappa, S; Swaroop, TR | 1 |
2 review(s) available for isoxazoles and 1,2-benzisoxazole
| Article | Year |
|---|---|
1,2-Benzisoxazole compounds: a patent review (2009 - 2014).
Topics: Animals; Anticonvulsants; Antipsychotic Agents; Drug Design; Humans; Isoxazoles; Patents as Topic; Protein Kinase Inhibitors | 2015 |
1, 2-Benzisoxazole: A Privileged Structure with a Potential for Polypharmacology.
Topics: Central Nervous System Agents; Central Nervous System Diseases; Humans; Isoxazoles; Molecular Structure; Polypharmacology | 2016 |
12 other study(ies) available for isoxazoles and 1,2-benzisoxazole
| Article | Year |
|---|---|
Biocatalysis of isomerization of 1,2-benzisoxazole by bovine serum albumin in an organic solvent.
Topics: Acetonitriles; Binding Sites; Catalysis; Isoxazoles; Kinetics; Serum Albumin, Bovine; Solvents; Stereoisomerism; Water | 2001 |
Synthesis and anti-HIV activity of new alkenyldiarylmethane (ADAM) non-nucleoside reverse transcriptase inhibitors (NNRTIs) incorporating benzoxazolone and benzisoxazole rings.
Topics: Animals; Anti-HIV Agents; Benzoxazoles; Cell Line; Crystallography, X-Ray; Drug Design; HIV-1; HIV-2; Humans; In Vitro Techniques; Isoxazoles; Methane; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Protein Conformation; Rats; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 2006 |
An efficient entry to 1,2-benzisoxazoles via 1,3-dipolar cycloaddition of in situ generated nitrile oxides and benzyne.
Topics: Benzene Derivatives; Cyclization; Isoxazoles; Molecular Structure; Nitriles; ortho-Aminobenzoates; Oxides | 2010 |
An improved synthesis of 1,2-benzisoxazoles: TBAF mediated 1,3-dipolar cycloaddition of nitrile oxides and benzyne.
Topics: Benzene Derivatives; Catalysis; Cyclization; Isoxazoles; Nitriles; Oxides | 2010 |
Intramolecular Fe(II)-catalyzed N-O or N-N bond formation from aryl azides.
Topics: Azides; Bromides; Catalysis; Combinatorial Chemistry Techniques; Ferrous Compounds; Indazoles; Isoxazoles; Molecular Structure; Pyrazoles | 2010 |
Microwave-promoted synthesis of 3-amino-substituted 1,2-benzisoxazoles.
Topics: Amines; Anticonvulsants; Antipsychotic Agents; Benzoxazoles; Isoxazoles; Microwaves; Oxazoles; Time Factors | 2010 |
Biological evaluation of novel benzisoxazole derivatives as PPARĪ“ agonists.
Topics: Animals; Cell Differentiation; Cell Line; Cells, Cultured; Cerebral Cortex; Humans; Isoxazoles; Oligodendroglia; PPAR delta; Rats; Rats, Wistar | 2011 |
Benzisoxazole analogs as glycogen synthase activators, a patent evaluation (WO2011057956).
Topics: Animals; Diabetes Mellitus, Type 2; Drug Design; Enzyme Activation; Enzyme Activators; Glycogen Synthase; Humans; Hypoglycemic Agents; Isoxazoles; Molecular Structure; Patents as Topic; Structure-Activity Relationship | 2012 |
Inhibition of protein glycation by urea and thiourea derivatives of glycine/proline conjugated benzisoxazole analogue - synthesis and structure-activity studies.
Topics: Animals; Cattle; Dose-Response Relationship, Drug; Glycine; Isoxazoles; Molecular Structure; Proline; Serum Albumin, Bovine; Structure-Activity Relationship; Urea | 2013 |
Solution-phase synthesis of a diverse library of benzisoxazoles utilizing the [3 + 2] cycloaddition of in situ-generated nitrile oxides and arynes.
Topics: Benzene Derivatives; Catalysis; Combinatorial Chemistry Techniques; Cycloaddition Reaction; Isoxazoles; Nitriles; Oxides; Palladium; Small Molecule Libraries | 2013 |
A Lewis Acid Catalyzed annulation to 2,1-benzisoxazoles.
Topics: Catalysis; Cyclization; Isoxazoles; Lewis Acids; Molecular Structure; Nitroso Compounds | 2014 |
Synthesis of 1,2-benzisoxazole tethered 1,2,3-triazoles that exhibit anticancer activity in acute myeloid leukemia cell lines by inhibiting histone deacetylases, and inducing p21 and tubulin acetylation.
Topics: Acetylation; Animals; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Cyclin D; Cyclin-Dependent Kinase Inhibitor p21; G1 Phase Cell Cycle Checkpoints; Histone Deacetylase Inhibitors; Histone Deacetylases; Histones; Humans; Isoxazoles; Leukemia, Myeloid, Acute; Mice; Mice, Inbred C57BL; Triazoles; Tubulin | 2015 |