Page last updated: 2024-08-23

isothiuronium and clobenpropit

isothiuronium has been researched along with clobenpropit in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Jansen, FP; Leurs, R; Maeyama, K; Mochizuki, T; Timmerman, H; Windhorst, AD; Yamatodani, A1
Fujii, Y; Hossen, MA; Kamei, C; Kayasuga, R; Sugimoto, Y1
Fujii, Y; Harada, C; Harusawa, S; Hirai, T; Kamei, C; Kurihara, T1
Bräuner-Osborne, H; Dawit, S; Du, Y; Hansen, KB; Kurtkaya, NL; Kurtkaya, S; Kvist, T; Le, P; Lewis, I; Mullasseril, P; Murphy, TJ; Ogden, KK; Orr, AG; Qui, M; Snyder, JP; Traynelis, SF; Vance, KM; Vellano, KM; Yuan, H1

Other Studies

4 other study(ies) available for isothiuronium and clobenpropit

ArticleYear
Brain penetration of the histamine H3 receptor antagonists thioperamide and clobenpropit in rat and mouse, determined with ex vivo [125I]iodophenpropit binding.
    Brain research, 1996, Dec-16, Volume: 743, Issue:1-2

    Topics: Animals; Brain; Cerebral Cortex; Corpus Striatum; Histamine Antagonists; Imidazoles; Iodine Radioisotopes; Isothiuronium; Male; Mice; Mice, Inbred BALB C; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Thiourea

1996
Histamine H3 receptors regulate vascular permeability changes in the skin of mast cell-deficient mice.
    International immunopharmacology, 2003, Volume: 3, Issue:12

    Topics: Animals; Capillary Permeability; Chlorpheniramine; Diphenhydramine; Evans Blue; Female; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Injections, Intradermal; Injections, Intravenous; Isothiuronium; Mast Cells; Mice; Mice, Mutant Strains; Piperidines; Receptors, Histamine H3; Skin; Thiourea; Tryptophan

2003
Intracerebroventricular administration of histamine H3 receptor antagonists decreases seizures in rat models of epilepsia.
    Methods and findings in experimental and clinical pharmacology, 2004, Volume: 26, Issue:4

    Topics: Amygdala; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Electroencephalography; Electroshock; Epilepsy, Tonic-Clonic; Histamine Agonists; Histamine Antagonists; Imidazoles; Injections, Intraventricular; Isothiuronium; Kindling, Neurologic; Lateral Ventricles; Male; Methylhistamines; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Seizures; Thiourea

2004
Implementation of a fluorescence-based screening assay identifies histamine H3 receptor antagonists clobenpropit and iodophenpropit as subunit-selective N-methyl-D-aspartate receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 333, Issue:3

    Topics: Aniline Compounds; Animals; Cell Line; Cricetinae; Drug Evaluation, Preclinical; Electrophysiology; Excitatory Amino Acid Antagonists; Fluorescent Dyes; Histamine H3 Antagonists; Humans; Imidazoles; Isothiuronium; Microscopy, Fluorescence; Oocytes; Patch-Clamp Techniques; Piperidines; Radioligand Assay; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Thiourea; Xanthenes; Xenopus laevis

2010