isoproterenol and xamoterol

isoproterenol has been researched along with xamoterol in 34 studies

Research

Studies (34)

TimeframeStudies, this research(%)All Research%
pre-199013 (38.24)18.7374
1990's14 (41.18)18.2507
2000's5 (14.71)29.6817
2010's1 (2.94)24.3611
2020's1 (2.94)2.80

Authors

AuthorsStudies
Barlow, JJ; Main, BG; Snow, HM1
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Hasebe, N; Honda, H; Obara, A; Onodera, S; Yahara, O; Yamashita, H1
Nagao, T; Narita, H; Watanabe, H; Yabana, H1
Kjaerulf-Jensen, H; Korsgaard, N; Lindeberg, H; Vigholt-Sørensen, E1
Barnett, DB; Lu, XY1
Katayama, K; Kohno, M; Kumada, T; Kusukawa, R; Matsuzaki, M; Miura, T; Ozaki, M; Toma, Y; Yonezawa, F1
Limas, C; Limas, CJ1
Boomsma, F; Brodde, OE; Daul, A; Man in 't Veld, AJ; Michel, MC; Michel-Reher, M; Schlieper, P1
Böhm, M; Erdmann, E; Mittmann, C; Schwinger, RH1
Ehrendorfer, S; Fischer, G; Grohs, JG; Raberger, G; Schneider, W1
Barnett, DB; Haworth, D; Kowalski, MT; Lu, X; Thomson, DS1
Burkard, WP; Eigenmann, R; Goodman, M; Holck, M; Märki, HP; Melmon, KL; Osterrieder, W1
Apperley, GH; Drew, GM; Gurden, JM1
Abrahamsson, T1
Hadfield, SE; Slee, SJ; Snow, HM1
Charlier, AA; Hanet, C; Marlow, HF; Pouleur, H; Rousseau, MF1
Malta, E; Mian, MA; Raper, C1
Nielsen-Kudsk, F; Vigholt Sørensen, E1
Cavero, I; Hicks, PE; Langer, SZ; Lefevre-Borg, F; Manoury, P1
Hattori, Y; Kanno, M; Nakao, Y; Sakuma, I1
Bobik, A; Jennings, G; Oddie, C; Restall, R1
Carlier, J; el Allaf, D1
Kawai, C; Kihara, Y; Lee, JD; Nakamura, Y; Ohyagi, A; Sasayama, S1
Arnold, IR; Barnett, DB; Mistry, R1
Fischmeister, R; Jurevicius, J; Skeberdis, VA1
Brodde, OE; Fuchs, B; Gorf, A; Jakubetz, J; Poller, U; Pönicke, K; Radke, J; Schmuck, S1
Brodde, OE; Daul, AE; Karl, I; Mennicke, K; Philipp, T; Schäfers, RF1
Karle, CA; Kathöfer, S; Kiehn, J; Schoels, W; Zhang, W; Zitron, E1
Steinle, JJ1
Haynes, JM1
Baker, JG; Fretwell, L; Gardiner, SM; Hill, SJ; Kemp, P; March, J1
Ali, A; Emran, TB; Imran, M; Ismail, ISB; Latif, Z; Muhammad, N; Saeed, L; Safi, SZ; Shah, H; Subramaniyan, V1

Reviews

1 review(s) available for isoproterenol and xamoterol

ArticleYear
Old and new inotropic drugs.
    Resuscitation, 1984, Volume: 11, Issue:3-4

    Topics: Adrenergic beta-Agonists; Aminopyridines; Amrinone; Cardiac Glycosides; Cardiotonic Agents; Catecholamines; Glucagon; Hemodynamics; Humans; Imidazoles; Isoproterenol; Myocardial Contraction; Practolol; Prenalterol; Propanolamines; Stimulation, Chemical; Xamoterol

1984

Trials

2 trial(s) available for isoproterenol and xamoterol

ArticleYear
Cardiac effects of beta-adrenoceptor antagonists with intrinsic sympathomimetic activity in humans: beta1- and/or beta2-adrenoceptor mediated?
    Journal of cardiovascular pharmacology, 1999, Volume: 33, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Blood Pressure; Cardiovascular Physiological Phenomena; Celiprolol; Cross-Over Studies; Diastole; Heart; Heart Rate; Humans; Isoproterenol; Male; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Single-Blind Method; Sympathomimetics; Terbutaline; Time Factors; Xamoterol

1999
Ketotifen and cardiovascular effects of xamoterol following single and chronic dosing in healthy volunteers.
    British journal of clinical pharmacology, 1999, Volume: 47, Issue:1

    Topics: Adrenergic beta-Agonists; Adult; Anti-Allergic Agents; Dose-Response Relationship, Drug; Double-Blind Method; Drug Interactions; Electrocardiography; Hemodynamics; Humans; Isoproterenol; Ketotifen; Male; Placebos; Reproducibility of Results; Tachycardia; Xamoterol

1999

Other Studies

31 other study(ies) available for isoproterenol and xamoterol

ArticleYear
Beta-adrenoceptor stimulant properties of amidoalkylamino-substituted 1-aryl-2-ethanols and 1-(aryloxy)-2-propanols.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Dogs; Ethanolamines; Heart Rate; Propanolamines; Receptors, Adrenergic, beta; Structure-Activity Relationship

1981
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Effect of xamoterol in Shy-Drager syndrome.
    Circulation, 1992, Volume: 85, Issue:2

    Topics: Adrenergic beta-Agonists; Aged; Blood Pressure; Blood Pressure Monitors; Circadian Rhythm; Heart Rate; Humans; Isoproterenol; Male; Middle Aged; Monitoring, Physiologic; Norepinephrine; Osmolar Concentration; Posture; Propanolamines; Shy-Drager Syndrome; Xamoterol

1992
Selective and full beta 1-adrenoceptor agonist action of a catechol derivative of denopamine (T-0509) in the guinea-pig cardiac muscle and trachea: comparison with denopamine, xamoterol and isoprenaline.
    British journal of pharmacology, 1992, Volume: 106, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Bisoprolol; Ethanolamines; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Papillary Muscles; Propanolamines; Trachea; Xamoterol

1992
Myocardial ultrastructure in the isolated rabbit heart exposed to dopamine, dobutamine, isoprenaline, G-strofanthin, xamoterol and hypoxia.
    Pharmacology & toxicology, 1992, Volume: 71, Issue:4

    Topics: Adrenergic Agonists; Animals; Cell Hypoxia; Dobutamine; Dopamine; Female; Isoproterenol; Male; Mitochondria, Heart; Myocardial Contraction; Myocardium; Oxygen Consumption; Rabbits; Stimulation, Chemical; Strophanthins; Xamoterol

1992
Cardiac beta-adrenoceptor regulation and the effects of partial agonism.
    The American journal of cardiology, 1991, May-06, Volume: 67, Issue:12

    Topics: Adrenergic beta-Agonists; Animals; Down-Regulation; Heart; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Xamoterol

1991
Effects of the partial beta 1-adrenergic agonist, xamoterol, on hemodynamics and regional myocardial function during acute coronary occlusion in dogs.
    Journal of cardiovascular pharmacology, 1990, Volume: 15, Issue:2

    Topics: Acute Disease; Adrenergic beta-Antagonists; Anesthesia; Animals; Coronary Disease; Dogs; Heart; Hemodynamics; Isoproterenol; Myocardial Contraction; Propanolamines; Xamoterol

1990
Effects of xamoterol on the reversible cycling of cardiac beta-adrenoceptors.
    Journal of cardiovascular pharmacology, 1990, Volume: 16, Issue:6

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell-Free System; Colchicine; Cytochalasin B; Heart; Heart Failure; Heparin; Isoproterenol; Myocardium; Propanolamines; Protein Kinases; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Xamoterol

1990
Agonist-induced desensitization of beta-adrenoceptor function in humans. Subtype-selective reduction in beta 1- or beta 2-adrenoceptor-mediated physiological effects by xamoterol or procaterol.
    Circulation, 1990, Volume: 81, Issue:3

    Topics: Adrenergic beta-Agonists; Adult; Blood Pressure; Ethanolamines; Exercise Test; Heart Rate; Humans; Isoproterenol; Lymphocytes; Male; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Tachyphylaxis; Time Factors; Xamoterol

1990
Effects of xamoterol on inotropic and lusitropic properties of the human myocardium and on adenylate cyclase activity.
    American heart journal, 1990, Volume: 120, Issue:6 Pt 1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Dose-Response Relationship, Drug; Heart Atria; Heart Failure; Humans; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Xamoterol

1990
Haemodynamic and metabolic effects of xamoterol in exercising dogs.
    European journal of pharmacology, 1990, Feb-20, Volume: 177, Issue:1-2

    Topics: Animals; Blood Glucose; Cardiac Output; Dogs; Dose-Response Relationship, Drug; Female; Glucose; Heart Rate; Hemodynamics; Isoproterenol; Lactates; Male; Physical Conditioning, Animal; Propanolamines; Pyruvates; Vascular Resistance; Xamoterol

1990
Comparison of the effects of xamoterol and isoprenaline on rat cardiac beta-adrenoceptors: studies of function and regulation.
    British journal of pharmacology, 1990, Volume: 99, Issue:1

    Topics: Animals; Down-Regulation; Female; Heart; Heart Rate; In Vitro Techniques; Iodine Radioisotopes; Isoproterenol; Male; Pindolol; Propanolamines; Rats; Receptors, Adrenergic, beta; Xamoterol

1990
In vitro pharmacological properties of a series of isoprenaline derivatives.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:8

    Topics: Animals; Aorta, Thoracic; Binding, Competitive; Catecholamines; Dihydroalprenolol; Dobutamine; Dogs; Electrophysiology; Female; Guinea Pigs; In Vitro Techniques; Isomerism; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Myocardial Contraction; Papillary Muscles; Potassium; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Xamoterol

1989
A comparison of the properties of prenalterol and corwin at beta 1- and beta 2-adrenoreceptors in vitro.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Cats; Dogs; Guinea Pigs; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Prenalterol; Propanolamines; Receptors, Adrenergic, beta; Xamoterol

1989
Characterization of the beta 1-adrenoceptor stimulatory effects of the partial beta 1-agonists acebutolol, xamoterol, H142/08 and H201/70.
    European journal of pharmacology, 1989, May-02, Volume: 164, Issue:1

    Topics: Acebutolol; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Female; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Propanolamines; Rats; Renin; Uterine Contraction; Xamoterol

1989
The cardiovascular pharmacology of xamoterol, cicloprolol, prenalterol and pindolol in the anaesthetised dog.
    British journal of clinical pharmacology, 1989, Volume: 28 Suppl 1

    Topics: Adrenergic beta-Agonists; Anesthesia; Animals; Dogs; Dose-Response Relationship, Drug; Hemodynamics; Hindlimb; Isoproterenol; Pindolol; Prenalterol; Propanolamines; Regional Blood Flow; Reserpine; Xamoterol

1989
Left ventricular sensitivity to beta-adrenoceptor-stimulating drugs in patients with ischemic heart disease and varying degrees of ventricular dysfunction.
    Circulation research, 1987, Volume: 61, Issue:4 Pt 2

    Topics: Aged; Coronary Disease; Dose-Response Relationship, Drug; Female; Heart; Heart Diseases; Heart Ventricles; Humans; Isoproterenol; Male; Middle Aged; Propanolamines; Receptors, Adrenergic, beta; Sympathomimetics; Xamoterol

1987
The in vitro pharmacology of xamoterol (ICI 118,587).
    British journal of pharmacology, 1985, Volume: 85, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cats; Female; Fenoterol; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Male; Muscle, Smooth; Norepinephrine; Pindolol; Propanolamines; Rats; Refractory Period, Electrophysiological; Species Specificity; Uterine Contraction; Xamoterol

1985
Single and combined myocardial pharmacodynamics of xamoterol, isoprenaline and g-strophanthin in the isolated rabbit heart.
    European journal of pharmacology, 1986, Jun-24, Volume: 125, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Coronary Circulation; Drug Interactions; Female; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Ouabain; Oxygen Consumption; Propanolamines; Rabbits; Xamoterol

1986
Comparative analysis of beta-1 adrenoceptor agonist and antagonist potency and selectivity of cicloprolol, xamoterol and pindolol.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Betaxolol; Blood Pressure; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Pindolol; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta; Trachea; Xamoterol

1987
Pharmacological analysis of the cardiac actions of xamoterol, a beta adrenoceptor antagonist with partial agonistic activity, in guinea pig heart: evidence for involvement of adenylate cyclase system in its cardiac stimulant actions.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Adenosine; Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbachol; Cyclic AMP; Dose-Response Relationship, Drug; Female; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Rate; Iodocyanopindolol; Isoproterenol; Male; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Xamoterol

1987
Cardioselectivity, kinetics, hemodynamics, and metabolic effects of xamoterol.
    Clinical pharmacology and therapeutics, 1984, Volume: 35, Issue:5

    Topics: Adrenergic beta-Agonists; Adult; Blood Pressure; Female; Heart Rate; Humans; Isoproterenol; Kinetics; Male; Physical Exertion; Propanolamines; Xamoterol

1984
Effect of ICI 118,587 on left ventricular function during graded treadmill exercise in conscious dogs.
    The American journal of cardiology, 1984, Nov-01, Volume: 54, Issue:8

    Topics: Adrenergic beta-Agonists; Animals; Dogs; Heart; Heart Rate; Isoproterenol; Myocardial Contraction; Physical Exertion; Propanolamines; Propranolol; Xamoterol

1984
Subtype selective regulation of coupling of rat cardiac beta adrenoceptors to adenylate cyclase.
    European journal of pharmacology, 1993, May-15, Volume: 245, Issue:3

    Topics: Adenylyl Cyclases; Animals; Binding Sites; Down-Regulation; Humans; Infusions, Intravenous; Isoproterenol; Male; Myocardium; Rats; Receptors, Adrenergic, beta; Xamoterol

1993
Pharmacological characterization of the receptors involved in the beta-adrenoceptor-mediated stimulation of the L-type Ca2+ current in frog ventricular myocytes.
    British journal of pharmacology, 1997, Volume: 121, Issue:7

    Topics: Albuterol; Animals; Calcium Channels; Calcium Channels, L-Type; Dobutamine; Dose-Response Relationship, Drug; In Vitro Techniques; Isoproterenol; Myocardium; Propanolamines; Rana esculenta; Receptors, Adrenergic, beta; Xamoterol

1997
Rapid component I(Kr) of the guinea-pig cardiac delayed rectifier K(+) current is inhibited by beta(1)-adrenoreceptor activation, via cAMP/protein kinase A-dependent pathways.
    Cardiovascular research, 2002, Feb-01, Volume: 53, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbazoles; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Enzyme Inhibitors; Guinea Pigs; Imidazoles; Indoles; Isoproterenol; Myocardium; Patch-Clamp Techniques; Potassium Channels, Inwardly Rectifying; Pyrroles; Xamoterol

2002
Sympathetic neurotransmission modulates expression of inflammatory markers in the rat retina.
    Experimental eye research, 2007, Volume: 84, Issue:1

    Topics: Adrenergic beta-Agonists; Animals; Cells, Cultured; Dinoprostone; Endothelium, Vascular; Female; Gene Expression Regulation; Inflammation Mediators; Isoproterenol; Nitric Oxide Synthase Type II; Rats; Rats, Sprague-Dawley; Receptors, Prostaglandin E; Retina; Retinal Vessels; RNA, Messenger; Sympathetic Nervous System; Synaptic Transmission; Xamoterol

2007
beta(2) and beta(3)-adrenoceptor inhibition of alpha(1)-adrenoceptor-stimulated Ca(2+) elevation in human cultured prostatic stromal cells.
    European journal of pharmacology, 2007, Sep-10, Volume: 570, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Atenolol; Calcium; Cells, Cultured; Cyclic AMP; Ethanolamines; Humans; Isoproterenol; Male; Phenylephrine; Potassium Channel Blockers; Propanolamines; Propranolol; Prostate; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Stromal Cells; Xamoterol

2007
Predicting in vivo cardiovascular properties of β-blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2011, Volume: 25, Issue:12

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiovascular Agents; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Heart Rate; Humans; Imidazoles; Isoproterenol; Male; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Rats; Rats, Sprague-Dawley; Vascular Resistance; Xamoterol

2011
Mechanisms of β-adrenergic receptors agonists in mediating pro and anti-apoptotic pathways in hyperglycemic Müller cells.
    Molecular biology reports, 2022, Volume: 49, Issue:10

    Topics: Adrenergic beta-Agonists; Brain-Derived Neurotrophic Factor; Caspase 3; Caspase 8; Cyclic AMP Response Element-Binding Protein; Cytochromes c; Ependymoglial Cells; Glucose; Humans; Isoproterenol; Propranolol; Reactive Oxygen Species; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Salmeterol Xinafoate; Xamoterol

2022