isoproterenol and uk 68798

isoproterenol has been researched along with uk 68798 in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (27.78)18.2507
2000's6 (33.33)29.6817
2010's7 (38.89)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Refsum, H; Tande, PM; Yang, T1
Brown, AM; Cantù, F; Napolitano, C; Priori, SG; Schwartz, PJ1
Martin, CL; Mcmahon, EG; Palomo, MA1
Beatch, GN; Williams, BA1
Bril, A; Faivre, JF; Rouanet, S1
Brachmann, J; Karolyi, L; Kübler, W; Marschang, H; Schöls, W1
Khan, IA1
Blessing, WW; De Pasquale, CG; Nalivaiko, E1
Kovács, A; Szénási, G1
Abi-Gerges, N; Crijns, HJ; Heijman, J; Johnson, DM; Pollard, CE; Valentin, JP; Volders, PG1
Dai, DZ; Dai, Y; Hamed, KH; Hu, C; Yu, F1
Antoons, G; Beekman, JD; Bourgonje, VJ; de Windt, LJ; Houtman, MJ; Miedema, LF; Schoenmakers, M; Sipido, K; van der Nagel, R; van Veen, TA; Vos, MA1
Bányász, T; Hegyi, B; Horváth, B; Kistamás, K; Magyar, J; Nánási, PP; Ruzsnavszky, F; Szentandrássy, N; Váczi, K; Varró, A1
Clancy, CE; DeMarco, KR; Harvey, RD; Jeng, MT; Kurokawa, J; López-Redondo, F; Noskov, SY; Perissinotti, LL; Vorobyov, I; Wang, Y; Yang, PC1

Reviews

2 review(s) available for isoproterenol and uk 68798

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Atrial stunning: basics and clinical considerations.
    International journal of cardiology, 2003, Volume: 92, Issue:2-3

    Topics: Animals; Anti-Arrhythmia Agents; Atrial Fibrillation; Atrial Flutter; Atrial Function; Atrial Function, Left; Atrial Function, Right; Catheter Ablation; Electric Countershock; Humans; Isoproterenol; Myocardial Stunning; Phenethylamines; Sotalol; Sulfonamides; Thromboembolism; Time Factors; Verapamil

2003

Other Studies

16 other study(ies) available for isoproterenol and uk 68798

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Negative chronotropic effect of a novel class III antiarrhythmic drug, UK-68,798, devoid of beta-blocking action on isolated guinea-pig atria.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Depression, Chemical; Female; Guinea Pigs; Heart Atria; Heart Rate; In Vitro Techniques; Isoproterenol; Phenethylamines; Propranolol; Sinoatrial Node; Sulfonamides

1991
Differential response to Na+ channel blockade, beta-adrenergic stimulation, and rapid pacing in a cellular model mimicking the SCN5A and HERG defects present in the long-QT syndrome.
    Circulation research, 1996, Volume: 78, Issue:6

    Topics: Action Potentials; Animals; Cardiac Pacing, Artificial; Cation Transport Proteins; Ether-A-Go-Go Potassium Channels; Guinea Pigs; Intercellular Signaling Peptides and Proteins; Isoproterenol; Long QT Syndrome; Mexiletine; Mutation; Peptides; Phenethylamines; Potassium Channels; Potassium Channels, Voltage-Gated; Receptors, Adrenergic, beta; Sodium Channel Blockers; Sodium Channels; Sulfonamides

1996
Comparison of bidisomide, flecainide and dofetilide on action potential duration in isolated canine atria: effect of isoproterenol.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 278, Issue:1

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Dogs; Dose-Response Relationship, Drug; Flecainide; Guinea Pigs; Heart Atria; Isoproterenol; Male; Phenethylamines; Piperidines; Sulfonamides

1996
Magnesium shifts voltage dependence of activation of delayed rectifier I(K) in guinea pig ventricular myocytes.
    The American journal of physiology, 1997, Volume: 272, Issue:3 Pt 2

    Topics: Animals; Anti-Arrhythmia Agents; Cells, Cultured; Delayed Rectifier Potassium Channels; Dose-Response Relationship, Drug; Guinea Pigs; Heart; Heart Ventricles; Isoproterenol; Kinetics; Magnesium; Membrane Potentials; Patch-Clamp Techniques; Phenethylamines; Potassium Channels; Potassium Channels, Voltage-Gated; Sulfonamides

1997
Comparative effects of glibenclamide, tedisamil, dofetilide, E-4031, and BRL-32872 on protein kinase A-activated chloride current in guinea pig ventricular myocytes.
    Journal of cardiovascular pharmacology, 1998, Volume: 31, Issue:4

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Acetylcholine; Animals; Anti-Arrhythmia Agents; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Cardiotonic Agents; Chlorides; Cyclic AMP-Dependent Protein Kinases; Cyclopropanes; Glyburide; Guinea Pigs; Heart Ventricles; Hypoglycemic Agents; Ion Transport; Isoproterenol; Male; Myocardium; Patch-Clamp Techniques; Phenethylamines; Piperidines; Potassium Channels; Propranolol; Pyridines; Sulfonamides

1998
Isoproterenol specifically modulates reverse rate-dependent effects of d,l-sotalol, d-sotalol, and dofetilide.
    Journal of cardiovascular pharmacology, 2000, Volume: 35, Issue:3

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Cardiotonic Agents; Dogs; Electric Stimulation; Electrophysiology; Heart; Isomerism; Isoproterenol; Membrane Potentials; Phenethylamines; Sotalol; Sulfonamides

2000
Ventricular arrhythmias triggered by alerting stimuli in conscious rabbits pre-treated with dofetilide.
    Basic research in cardiology, 2004, Volume: 99, Issue:2

    Topics: Administration, Inhalation; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Arousal; Arrhythmias, Cardiac; Electrocardiography; Formaldehyde; Heart; Heart Ventricles; Isoproterenol; Motion; Pain; Phenethylamines; Physical Stimulation; Premedication; Propranolol; Rabbits; Stimulation, Chemical; Sulfonamides

2004
Effects of dofetilide and EGIS-7229, an antiarrhythmic agent possessing class III, IV, and IB activities, on myocardial refractoriness in hyperkalemia, hypokalemia, and during beta-adrenergic activation in the rabbit papillary muscle in vitro.
    Journal of pharmacological sciences, 2006, Volume: 100, Issue:4

    Topics: Adrenergic beta-Agonists; Animals; Anti-Arrhythmia Agents; Dose-Response Relationship, Drug; Electric Stimulation; Electrocardiography; Hyperkalemia; Hypokalemia; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Papillary Muscles; Phenethylamines; Pyridazines; Rabbits; Sulfonamides

2006
I(Ks) restricts excessive beat-to-beat variability of repolarization during beta-adrenergic receptor stimulation.
    Journal of molecular and cellular cardiology, 2010, Volume: 48, Issue:1

    Topics: Action Potentials; Aniline Compounds; Animals; Arrhythmias, Cardiac; Calcium; Cells, Cultured; Dogs; Egtazic Acid; Female; Heart Ventricles; Ion Channels; Isoproterenol; Myocytes, Cardiac; Phenethylamines; Phenyl Ethers; Potassium; Potassium Channel Blockers; Potassium Channels; Receptors, Adrenergic, beta; Sodium; Sodium-Calcium Exchanger; Sulfonamides

2010
CPU228, a derivative of dofetilide, relieves cardiac dysfunction by normalizing FKBP12.6, NADPH oxidase and protein kinase C epsilon in the myocardium.
    The Journal of pharmacy and pharmacology, 2010, Volume: 62, Issue:1

    Topics: Animals; Anti-Arrhythmia Agents; Disease Models, Animal; Dose-Response Relationship, Drug; Down-Regulation; Heart Failure; Isoproterenol; Male; NADPH Oxidases; Naphthalenes; Oxidative Stress; Phenethylamines; Phosphorylation; Protein Kinase C-epsilon; Rats; Rats, Sprague-Dawley; Sulfonamides; Tacrolimus Binding Proteins; Up-Regulation

2010
Relevance of calmodulin/CaMKII activation for arrhythmogenesis in the AV block dog.
    Heart rhythm, 2012, Volume: 9, Issue:11

    Topics: Animals; Arrhythmias, Cardiac; Atrioventricular Block; Benzylamines; Calcineurin; Calcium-Binding Proteins; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Cardiomyopathy, Hypertrophic; Cyclosporine; Disease Models, Animal; Dogs; Isoproterenol; Long QT Syndrome; Myocytes, Cardiac; Patch-Clamp Techniques; Phenethylamines; Phenotype; Phosphorylation; Random Allocation; Sulfonamides; Ventricular Remodeling

2012
Contribution of ion currents to beat-to-beat variability of action potential duration in canine ventricular myocytes.
    Pflugers Archiv : European journal of physiology, 2015, Volume: 467, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Calcium; Cardiotonic Agents; Cells, Cultured; Chromans; Dogs; Feedback, Physiological; Female; Heart Ventricles; Ion Channels; Ion Transport; Isoproterenol; Lidocaine; Male; Myocytes, Cardiac; Nisoldipine; Phenethylamines; Potassium Channel Blockers; Sulfonamides; Tetrodotoxin; Veratridine

2015
A multiscale computational modelling approach predicts mechanisms of female sex risk in the setting of arousal-induced arrhythmias.
    The Journal of physiology, 2017, 07-15, Volume: 595, Issue:14

    Topics: Adrenergic beta-Agonists; Animals; Anti-Arrhythmia Agents; Arousal; Arrhythmias, Cardiac; Estradiol; Ether-A-Go-Go Potassium Channels; Female; Guinea Pigs; Isoproterenol; Male; Models, Biological; Molecular Docking Simulation; Myocytes, Cardiac; Phenethylamines; Sex Characteristics; Sulfonamides

2017