isoproterenol has been researched along with thiazoles in 48 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 15 (31.25) | 18.7374 |
1990's | 11 (22.92) | 18.2507 |
2000's | 15 (31.25) | 29.6817 |
2010's | 4 (8.33) | 24.3611 |
2020's | 3 (6.25) | 2.80 |
Authors | Studies |
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Brundin, J; Stjärne, L | 1 |
Strosberg, AM | 1 |
Guellaen, G; Hanoune, J; Lacombe, ML; Strosberg, AD; Vauquelin, G | 1 |
Waldeck, B | 1 |
Daly, JW; Skolnick, P; Stalvey, LP | 1 |
Jolly, SR; Lech, JJ; Menahan, LA | 1 |
Buckley, HT; Harrison, DC; Strosberg, AM | 1 |
Kiyoto, S; Matsuo, M; Satake, N; Shibata, S; Zhou, Q | 1 |
Ballabeni, V; Barocelli, E; Chiavarini, M; Impicciatore, M; Mingiardi, MR; Morini, G; Ronchini, F | 1 |
Endoh, M; Hirano, K; Norota, I; Satoh, H | 1 |
Sheng, BH; Yang, XM; Zhao, DH | 1 |
Gray, WD; Rauh, CE | 1 |
Berkoz, B; Edwards, JA; Fried, JH; Halpern, O; Lewis, GS; Miller, LM; Roszkowski, AP; Strosberg, AM | 1 |
Lockwood, RH; Lum, BK | 1 |
Ancla, M; de Brux, J; Laborit, H; Pavlovitchova, H | 1 |
Bachmann, W; Häring, HU; Kirsch, DM | 1 |
Ayala, GA; Banerjee, P; Bowser, EN; Hargis, GK; Kukreja, SC; Williams, GA | 1 |
Ahrén, B; Lundquist, I | 1 |
Inoue, T; Satoh, M; Tomozawa, Y | 1 |
Bleasdale, JE; Jacob, CS; Sizer, KM; Smith, CL; Swanson, ML | 2 |
Heard, SO; Perkins, M; Toth, I | 1 |
Barnes, PJ; Giembycz, MA; Kelly, JJ | 1 |
Forest, C; Franckhauser-Vogel, S; Glorian, M; Robin, D; Robin, P | 1 |
Asano, M; Hazama, H; Imuta, H; Iwasawa, K; Kawakami, Y; Morita, T; Nakajima, T; Nakamura, F; Okuda, Y; Omata, M; Oonuma, H; Suzuki, J; Suzuki, S | 1 |
Bretscher, A; Cao, TT; Deacon, HW; Reczek, D; von Zastrow, M | 1 |
Fukamachi, H; Higa, T; Shindo, K; Suzuki, H; Takei, M; Ueno, A | 1 |
Alves-Guerra, MC; Bouillaud, F; Cassard-Doulcier, AM; del Mar Gonzalez-Barroso, M; Gelly, C; Pecqueur, C; Ricquier, D; Sanchis, D | 1 |
Aizawa, Y; Hasebe, N; Kawabe, J; Kikuchi, K; Takehara, N | 1 |
Furuse, Y; Hisatome, I; Ogino, K; Sasaki, N; Shimoyama, M | 1 |
Hashimoto, K; Hori, M; Imahashi, K; Kusuoka, H; Nishimura, T; Terakawa, T; Yoshioka, J | 1 |
Gaidarov, I; Keen, JH; Santini, F | 1 |
Gotoda, T; Harada, K; Iizuka, Y; Ishibashi, S; Kimura, S; Ohashi, K; Okazaki, H; Osuga, J; Shimano, H; Shionoiri, F; Tamura, Y; Tomita, S; Yahagi, N; Yamada, N | 1 |
Antoine, B; Beale, EG; Chauvet, G; Forest, C; Quette, J; Tordjman, J | 1 |
Adamson, PB; Foreman, RD; Schwartz, PJ; Shibano, T; Vanoli, E | 1 |
Becq, F; Norez, C; Robert, R | 1 |
Comini, M; Menozzi, A; Morini, G; Poli, E; Pozzoli, C | 1 |
Prasad, SV; Rockman, HA; Volovyk, ZM; Wolf, MJ | 1 |
Maruyama, T; Matsui, T; Miyata, K; Nagase, I; Sasamata, M; Sato, S; Takasu, T; Uchida, H; Ukai, M; Yamaguchi, O | 1 |
Amit, O; Chigaev, A; Sklar, LA; Waller, A | 1 |
Alewijnse, AE; Michel, MC; Vrydag, W | 1 |
Andersson, KE; Bouchelouche, K; Bouchelouche, P; Korstanje, C; Nordling, J; Svalø, J | 1 |
Calvi, P; D' Agostino, G; Maria Condino, A | 1 |
Alexandre, EC; Antunes, E; Claudino, MA; Costa, FF; da Silva, FH; de Nucci, G; Fertrin, KY; Franco-Penteado, CF; Leiria, LO; Mónica, FZ; Renno, A | 1 |
De Wachter, S; Eastham, J; Gillespie, J; Persyn, S; Wyndaele, JJ | 1 |
Su, G; Su, X; You, H | 1 |
Berezina, TP; Evlakhov, VI; Poyassov, IZ | 1 |
Beyhoff, N; Blumrich, A; Foryst-Ludwig, A; Goeritzer, M; Grune, J; Jaeger, C; Kasch, J; Kintscher, U; Klopfleisch, R; Luettges, K; Müller, OJ; Ritter, D; Smeir, E; Thiele, A | 1 |
48 other study(ies) available for isoproterenol and thiazoles
Article | Year |
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Beta2-adrenoceptors facilitating noradrenaline secretion from human vasoconstrictor nerves.
Topics: Adrenergic beta-Antagonists; Adult; Aged; Albuterol; Arteries; Electric Stimulation; Female; Humans; Isoproterenol; Male; Middle Aged; Norepinephrine; Omentum; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic; Secretory Rate; Terbutaline; Thiazoles; Vasomotor System; Veins | 1976 |
The cardiovascular pharmacology and hemodynamic activity of tazolol, a selective myocardial beta-stimulant.
Topics: Adrenergic beta-Agonists; Amphetamine; Animals; Blood Pressure; Dogs; Drug Interactions; Female; Heart Rate; Hemodynamics; Isoproterenol; Male; Myocardial Contraction; Propanolamines; Propranolol; Reserpine; Thiazoles; Time Factors | 1976 |
Tazolol (1-isopropylamino-3-(2-thiazoloxy)-2-propanol) as a beta-adrenergic blocker.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Carcinoma, Hepatocellular; Female; In Vitro Techniques; Isoproterenol; Liver; Liver Neoplasms; Myocardium; Propanolamines; Rats; Stimulation, Chemical; Thiazoles | 1976 |
Analysis of the beta-receptor mediated effect on slow-contracting skeletal muscle in vitro.
Topics: Adrenergic beta-Antagonists; Animals; Dopamine; Electric Stimulation; Epinephrine; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Norepinephrine; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reserpine; Terbutaline; Thiazoles; Tyramine | 1977 |
Blockade of central beta-adrenergic receptors by tazolol (1-isopropylamino-3-(2-thiazoloxy)-2-propanol).
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Cerebral Cortex; Cyclic AMP; Isoproterenol; Male; Propanolamines; Purkinje Cells; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Thiazoles | 1977 |
Comparison of isoproterenol, salbutamol and tazolol as lipolytic agents with isolated rodent adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Albuterol; Animals; In Vitro Techniques; Isoproterenol; Lipid Metabolism; Male; Mice; Propanolamines; Rats; Thiazoles | 1978 |
Circulatory effects of tazolol in experimental myocardial infarction.
Topics: Adrenergic beta-Agonists; Animals; Blood Pressure; Cardiac Output; Dogs; Drug Evaluation; Heart Rate; Hemodynamics; Infusions, Parenteral; Isoproterenol; Propanolamines; Shock, Cardiogenic; Thiazoles; Time Factors; Vascular Resistance | 1975 |
Mode of relaxing action of FK336, a new antianginal agent, in rabbit aorta.
Topics: Acetylcholine; Animals; Aorta; Calcium; Guanylate Cyclase; In Vitro Techniques; Inosine Monophosphate; Isoproterenol; Male; Muscle Relaxation; Nitroglycerin; Norepinephrine; Potassium Chloride; Rabbits; Thiazoles; Vasodilator Agents | 1992 |
Pharmacological properties of new 1,2-benzisothiazolyloxypropanolamines on cardiac and tracheal beta-receptors.
Topics: Adrenergic beta-Antagonists; Animals; Carbachol; Heart; Heart Atria; Isoproterenol; Male; Molecular Structure; Myocardium; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Structure-Activity Relationship; Thiazoles; Trachea | 1992 |
Effects of a new 1,3-thiazole derivative ZSY-39 on force of contraction and cyclic AMP content in canine ventricular muscle.
Topics: Animals; Carbachol; Cardiotonic Agents; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Female; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Phosphodiesterase Inhibitors; Pyridines; Thiazoles | 1990 |
[Effects of thioproline on isolated guinea pig papillary muscles].
Topics: Animals; Anti-Arrhythmia Agents; Calcium Chloride; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Papillary Muscles; Thiazoles; Thiazolidines; Verapamil | 1986 |
The anticonvulsant action of the carbonic anhydrase inhibitor methazolamide: possible involvement of a noradrenergic mechanism.
Topics: Animals; Anticonvulsants; Benserazide; Body Temperature; Carbonic Anhydrase Inhibitors; Dihydroxyphenylalanine; Dopamine beta-Hydroxylase; Dose-Response Relationship, Drug; Electroshock; Ethanolamines; Isoproterenol; Levobunolol; Male; Methazolamide; Mice; Motor Activity; Norepinephrine; Phenoxybenzamine; Phentolamine; Phenytoin; Practolol; Propranolol; Rats; Reserpine; Serotonin; Thiazoles; Thiourea; Tolazoline | 1974 |
Selective -adrenergic myocardial stimulant.
Topics: Acetanilides; Adrenergic beta-Agonists; Amino Alcohols; Amphetamine; Animals; Blood Pressure; Dogs; Female; Heart; Heart Rate; Isoproterenol; Male; Muscle Contraction; Propylamines; Propylene Glycols; Stimulation, Chemical; Thiazoles | 1972 |
Effects of adrenergic agonists and antagonists on potassium metabolism.
Topics: Albuterol; Animals; Blood Glucose; Blood Pressure; Butoxamine; Cats; Epinephrine; Ethanolamines; Heart Rate; Hyperkalemia; Isoproterenol; Norepinephrine; Pancreas; Phenethylamines; Phenoxybenzamine; Phenylephrine; Potassium; Potassium Chloride; Practolol; Propanolamines; Propranolol; Propylamines; Sotalol; Sulfonamides; Sympatholytics; Sympathomimetics; Thiazoles; Time Factors; Toluene | 1974 |
[Effect of 2-amino-(isothioureyl methylene)-4-thiazole dihydrochloride (Agr 307) on biochemical, electrocardiographic and histological modifications of the rat myocardium caused by isoproterenol].
Topics: Animals; Electrocardiography; Heart; Isoproterenol; Monoamine Oxidase Inhibitors; Myocardium; Rats; Thiazoles; Thiourea | 1970 |
Ciglitazone reverses cAMP-induced post-insulin receptor resistance in rat adipocytes in vitro.
Topics: 3-O-Methylglucose; Adipose Tissue; Animals; Biological Transport; Cyclic AMP; Insulin; Insulin Resistance; Isoproterenol; Male; Methylglucosides; Rats; Receptor, Insulin; Thiazoles; Thiazolidinediones | 1984 |
Characterization of the beta-adrenergic receptor mediating secretion of parathyroid hormone.
Topics: Adrenergic beta-Agonists; Animals; Cattle; Dose-Response Relationship, Drug; Humans; Isoproterenol; Parathyroid Hormone; Practolol; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, beta; Terbutaline; Thiazoles; Time Factors | 1980 |
Effects of selective and non-selective beta-adrenergic agents on insulin secretion in vivo.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Butoxamine; Carbachol; Dose-Response Relationship, Drug; Female; Glucose; Insulin; Insulin Secretion; Isoproterenol; Metoprolol; Mice; Propanolamines; Propranolol; Terbutaline; Thiazoles | 1981 |
Expression of type I interleukin-1 receptor mRNA and its regulation in cultured astrocytes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Astrocytes; Blotting, Northern; Bucladesine; Cells, Cultured; Coloring Agents; Cyclic AMP-Dependent Protein Kinases; Cycloheximide; Humans; Interleukin-1; Isoproterenol; Propranolol; Protein Synthesis Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Interleukin-1; Recombinant Proteins; RNA, Messenger; Stimulation, Chemical; Tetrazolium Salts; Thiazoles | 1995 |
Pioglitazone promotes insulin-induced activation of phosphoinositide 3-kinase in 3T3-L1 adipocytes by inhibiting a negative control mechanism.
Topics: 1-Phosphatidylinositol 4-Kinase; 3',5'-Cyclic-AMP Phosphodiesterases; 3T3 Cells; Adipocytes; Animals; Cell Differentiation; Cyclic AMP; Enzyme Activation; Hypoglycemic Agents; Immunosorbent Techniques; Insulin; Insulin-Like Growth Factor I; Isoproterenol; Kinetics; Male; Mice; Mice, Inbred C57BL; Phosphotransferases (Alcohol Group Acceptor); Phosphotyrosine; Pioglitazone; Thiazoles; Thiazolidinediones; Tyrosine | 1994 |
The role of platelet-activating factor in lipopolysaccharide-induced myocardial depression in guinea pigs.
Topics: Animals; Azepines; Depression, Chemical; Drug Interactions; Escherichia coli; Female; Guinea Pigs; Isoproterenol; Lipopolysaccharides; Male; Myocardial Contraction; Phenylephrine; Platelet Activating Factor; Platelet Membrane Glycoproteins; Quinolinium Compounds; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Thiazoles; Time Factors; Triazoles | 1995 |
Pioglitazone promotes insulin-induced activation of phosphoinositide 3-kinase in 3T3-L1 adipocytes by inhibiting a negative control mechanism.
Topics: 3T3 Cells; Adipocytes; Animals; Cell Differentiation; Cyclic AMP; Insulin; Insulin-Like Growth Factor I; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Phosphatidylinositol 3-Kinases; Phosphotransferases (Alcohol Group Acceptor); Pioglitazone; Precipitin Tests; Thiazoles; Thiazolidinediones | 1994 |
Phosphodiesterase 4 in macrophages: relationship between cAMP accumulation, suppression of cAMP hydrolysis and inhibition of [3H]R-(-)-rolipram binding by selective inhibitors.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Binding Sites; Brain; Chromatography, Ion Exchange; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Guinea Pigs; Isoenzymes; Isoproterenol; Kinetics; Macrophages, Peritoneal; Male; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pyrrolidinones; Quinazolines; Rats; Regression Analysis; Rolipram; Stereoisomerism; Thiazoles; Tritium | 1996 |
Glucocorticoids repress induction by thiazolidinediones, fibrates, and fatty acids of phosphoenolpyruvate carboxykinase gene expression in adipocytes.
Topics: 3T3 Cells; Adipocytes; Adrenergic beta-Agonists; Animals; Clofibrate; Dexamethasone; Enzyme Induction; Fatty Acids; Gene Expression Regulation, Enzymologic; Genes; Glucocorticoids; Hypoglycemic Agents; Isoproterenol; Male; Mice; Phosphoenolpyruvate Carboxykinase (GTP); Protein Biosynthesis; Proteins; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Regulatory Sequences, Nucleic Acid; RNA, Messenger; Rosiglitazone; Thiazoles; Thiazolidinediones; Trans-Activators; Transcription Factors | 1998 |
Troglitazone inhibits voltage-dependent calcium currents in guinea pig cardiac myocytes.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, T-Type; Cardiotonic Agents; Chromans; Cyclic AMP; Electric Conductivity; Guinea Pigs; Hypoglycemic Agents; Isoproterenol; Kinetics; Myocardium; Nifedipine; Thiazoles; Thiazolidinediones; Troglitazone; Verapamil | 1999 |
A kinase-regulated PDZ-domain interaction controls endocytic sorting of the beta2-adrenergic receptor.
Topics: Actins; Adrenergic beta-Agonists; Binding Sites; Biotinylation; Bridged Bicyclo Compounds, Heterocyclic; Carrier Proteins; Cell Line; Endocytosis; Endosomes; Humans; Isoproterenol; Lysosomes; Molecular Sequence Data; Phosphoproteins; Receptor Protein-Tyrosine Kinases; Receptors, Adrenergic, beta-2; Recombinant Proteins; Serine; Sodium-Hydrogen Exchangers; Thiazoles; Thiazolidines | 1999 |
The effects of S1319, a novel marine sponge-derived beta2-adrenoceptor agonist, on IgE-mediated activation of human cultured mast cells.
Topics: Adrenergic beta-Agonists; Albuterol; Benzothiazoles; Cells, Cultured; Chymases; Cross-Linking Reagents; Cyclic AMP; Ethanolamines; Formoterol Fumarate; Humans; Immunoglobulin E; Inositol 1,4,5-Trisphosphate; Isoproterenol; Mast Cells; Mitogen-Activated Protein Kinase 1; Phosphorylation; Serine Endopeptidases; Thiazoles; Tryptases; Tumor Necrosis Factor-alpha | 2000 |
Transcriptional activation of the human ucp1 gene in a rodent cell line. Synergism of retinoids, isoproterenol, and thiazolidinedione is mediated by a multipartite response element.
Topics: Adipocytes; Animals; Base Sequence; Carrier Proteins; Cell Line; COS Cells; DNA; Drug Synergism; Enhancer Elements, Genetic; Genes, Reporter; Humans; Ion Channels; Isoproterenol; Membrane Proteins; Mice; Mitochondrial Proteins; Molecular Sequence Data; Mutagenesis, Site-Directed; Rats; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Response Elements; Retinoids; Sequence Homology, Nucleic Acid; Thiazoles; Thiazolidinediones; Transcription Factors; Transcriptional Activation; Transfection; Uncoupling Protein 1 | 2000 |
Glucose modifies the cross-talk between insulin and the beta-adrenergic signalling system in vascular smooth muscle cells.
Topics: Animals; Cells, Cultured; Chromans; Glucose; Insulin; Insulin Receptor Substrate Proteins; Insulin Resistance; Isoproterenol; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Phosphatidylinositol 3-Kinases; Phosphoproteins; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Thiazoles; Thiazolidinediones; Troglitazone | 2000 |
Ca(2+)-sensitizing effect is involved in the positive inotropic effect of troglitazone.
Topics: Animals; Calcium; Calcium Channels, L-Type; Cardiotonic Agents; Chromans; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Heart Ventricles; Isoproterenol; Male; Patch-Clamp Techniques; Rats; Rats, Wistar; Ryanodine; Sarcoplasmic Reticulum; Thapsigargin; Thiazoles; Thiazolidinediones; Troglitazone; Ventricular Pressure | 2001 |
Troglitazone enhances glucose uptake induced by alpha-adrenoceptor stimulation via phosphatidylinositol 3-kinase in rat heart.
Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Androstadienes; Animals; Catecholamines; Chromans; Glucose; Heart; Hemodynamics; Humans; In Vitro Techniques; Insulin; Isoproterenol; Male; Myocardium; Phentolamine; Phenylephrine; Phosphates; Phosphatidylinositol 3-Kinases; Phosphocreatine; Phosphodiesterase Inhibitors; Phosphoinositide-3 Kinase Inhibitors; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Sugar Phosphates; Thiazoles; Thiazolidinediones; Time Factors; Troglitazone; Wortmannin | 2001 |
G protein-coupled receptor/arrestin3 modulation of the endocytic machinery.
Topics: Adrenergic beta-Agonists; Animals; Arrestins; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chlorocebus aethiops; Coated Pits, Cell-Membrane; COS Cells; Endocytosis; GTP-Binding Proteins; Humans; Image Processing, Computer-Assisted; Isoproterenol; Receptor, Muscarinic M1; Receptors, Adrenergic, beta-2; Receptors, Cell Surface; Receptors, Muscarinic; Recombinant Fusion Proteins; Thiazoles; Thiazolidines | 2002 |
Lipolysis in the absence of hormone-sensitive lipase: evidence for a common mechanism regulating distinct lipases.
Topics: Adipocytes; Animals; Cell Differentiation; Chromans; Cyclic AMP-Dependent Protein Kinases; Embryo, Mammalian; Enzyme Inhibitors; Hydrolysis; Isoproterenol; Isoquinolines; Lipase; Lipolysis; Mice; Mice, Knockout; Sterol Esterase; Sulfonamides; Thiazoles; Thiazolidinediones; Tissue Extracts; Triglycerides; Troglitazone; Tumor Necrosis Factor-alpha | 2002 |
Thiazolidinediones block fatty acid release by inducing glyceroneogenesis in fat cells.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Cells, Cultured; Cyclic AMP; Enzyme Activation; Esterification; Fatty Acids; Female; Gene Expression; Glycerol; Glycerol Kinase; Homeostasis; Hypoglycemic Agents; Isoproterenol; Lipid Metabolism; Lipolysis; Phosphoenolpyruvate Carboxykinase (GTP); Pioglitazone; Pyruvic Acid; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Rosiglitazone; Thiazoles; Thiazolidinediones; Transcription Factors; Viscera | 2003 |
Combined sodium and calcium channel blockade in prevention of lethal arrhythmias.
Topics: Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Calcium Channel Blockers; Death, Sudden, Cardiac; Depression, Chemical; Dogs; Drug Synergism; Drug Therapy, Combination; Heart Rate; Isoproterenol; Myocardial Infarction; Physical Conditioning, Animal; Propranolol; Sodium Channel Blockers; Thiazoles; Ventricular Fibrillation | 2003 |
Disruption of CFTR chloride channel alters mechanical properties and cAMP-dependent Cl- transport of mouse aortic smooth muscle cells.
Topics: Adrenergic beta-Agonists; Angiotensin II; Animals; Aorta, Thoracic; Benzoates; Cells, Cultured; Chlorides; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Genistein; Glyburide; In Vitro Techniques; Isoproterenol; Mice; Mice, Inbred CFTR; Muscle, Smooth, Vascular; ortho-Aminobenzoates; Quinolizines; Serotonin; Thiazoles; Thiazolidines; Vasoactive Intestinal Peptide; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2005 |
Benzisothiazoles and beta-adrenoceptors: synthesis and pharmacological investigation of novel propanolamine and oxypropanolamine derivatives in isolated rat tissues.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Synergism; Heart Atria; Ileum; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myocardial Contraction; Propanolamines; Propranolol; Rats; Thiazoles | 2005 |
Agonist-stimulated beta-adrenergic receptor internalization requires dynamic cytoskeletal actin turnover.
Topics: Actin Cytoskeleton; Actin Depolymerizing Factors; Actins; Adrenergic beta-Agonists; Bridged Bicyclo Compounds, Heterocyclic; Cell Culture Techniques; Endocytosis; Humans; Isoproterenol; Kidney; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Thiazoles; Thiazolidines | 2006 |
Effect of (R)-2-(2-aminothiazol-4-yl)-4'-{2-[(2-hydroxy-2-phenylethyl)amino]ethyl} acetanilide (YM178), a novel selective beta3-adrenoceptor agonist, on bladder function.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Animals; Carbachol; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Humans; Isoproterenol; Muscle Contraction; Propanolamines; Thiazoles; Urinary Bladder | 2007 |
Galphas-coupled receptor signaling actively down-regulates alpha4beta1-integrin affinity: a possible mechanism for cell de-adhesion.
Topics: Adrenergic beta-Agonists; Cell Adhesion; Chemokine CXCL12; Down-Regulation; Histamine Agonists; Humans; Integrin alpha4beta1; Isoproterenol; Leukocytes, Mononuclear; Oligopeptides; Phenylurea Compounds; Protein Binding; Protein Conformation; Receptor Cross-Talk; Receptors, Adrenergic, beta-2; Receptors, CXCR4; Receptors, Histamine H2; Recombinant Proteins; Signal Transduction; Thiazoles; U937 Cells | 2008 |
Do gene polymorphisms alone or in combination affect the function of human beta3-adrenoceptors?
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Binding, Competitive; Biphenyl Compounds; Cell Line; Cyclic AMP; Humans; Isoproterenol; Mutagenesis, Site-Directed; Norepinephrine; Phenethylamines; Polymorphism, Single Nucleotide; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-3; Thiazoles; Transfection | 2009 |
The novel β3-adrenoceptor agonist mirabegron reduces carbachol-induced contractile activity in detrusor tissue from patients with bladder outflow obstruction with or without detrusor overactivity.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Aged; Aged, 80 and over; Carbachol; Humans; In Vitro Techniques; Inhibitory Concentration 50; Isoproterenol; Male; Middle Aged; Muscle Contraction; Thiazoles; Urinary Bladder; Urinary Bladder Neck Obstruction; Urinary Bladder, Overactive | 2013 |
Involvement of β3-adrenoceptors in the inhibitory control of cholinergic activity in human bladder: Direct evidence by [(3)H]-acetylcholine release experiments in the isolated detrusor.
Topics: Acetanilides; Acetylcholine; Adrenergic beta-3 Receptor Agonists; Aminophenols; Dose-Response Relationship, Drug; Electric Stimulation; Ethanolamines; Humans; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta-3; Sulfonamides; Thiazoles; Urinary Bladder | 2015 |
Urinary Bladder Dysfunction in Transgenic Sickle Cell Disease Mice.
Topics: Acetanilides; Adenosine Triphosphate; Anemia, Sickle Cell; Animals; Atropine; Calcium Chloride; Carbachol; Disease Models, Animal; Diuresis; Electric Stimulation; Hemoglobin, Sickle; Humans; Isoproterenol; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle Contraction; Muscle, Smooth; Phenylephrine; Potassium Chloride; Thiazoles; Urethra; Urinary Bladder | 2015 |
The actions of isoprenaline and mirabegron in the isolated whole rat and guinea pig bladder.
Topics: Acetanilides; Animals; Arecoline; Carbachol; Female; Guinea Pigs; In Vitro Techniques; Isoproterenol; Muscarinic Agonists; Muscle Contraction; Rats, Sprague-Dawley; Thiazoles; Urinary Bladder | 2016 |
Novel thiazole-pyrazolone hybrids as potent ACE inhibitors and their cardioprotective effect on isoproterenol-induced myocardial infarction.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Apoptosis; Apoptosis Regulatory Proteins; Cytokines; Disease Models, Animal; Drug Design; Inflammation Mediators; Isoproterenol; Male; Mitochondria, Heart; Myocardial Infarction; Myocytes, Cardiac; Oxidative Stress; Pyrazolones; Rats, Sprague-Dawley; Thiazoles | 2020 |
Role of β
Topics: Acetanilides; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Capillary Permeability; Disease Models, Animal; Isoproterenol; Lung; Nebivolol; Propranolol; Pulmonary Circulation; Pulmonary Embolism; Rabbits; Receptors, Adrenergic, beta; Thiazoles; Vascular Resistance | 2020 |
Liver X Receptor Agonist AZ876 Induces Beneficial Endogenous Cardiac Lipid Reprogramming and Protects Against Isoproterenol-Induced Cardiac Damage.
Topics: Aniline Compounds; Animals; Cellular Reprogramming; Disease Models, Animal; Fatty Acids; Fibrosis; Heart Diseases; Isoproterenol; Liver X Receptors; Male; Mice; Mice, 129 Strain; Myocardium; Thiazoles | 2021 |