isoproterenol and labetalol

isoproterenol has been researched along with labetalol in 60 studies

Research

Studies (60)

TimeframeStudies, this research(%)All Research%
pre-199035 (58.33)18.7374
1990's13 (21.67)18.2507
2000's6 (10.00)29.6817
2010's6 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chen, M; Fang, H; Liu, Z; Shi, Q; Tong, W; Vijay, V1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Bellman, K; Knegtel, RM; Settimo, L1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Jones, LH; Nadanaciva, S; Rana, P; Will, Y1
Prichard, BN; Richards, DA; Tuckman, J1
Brittain, RT; Levy, GP1
Boakes, AJ; Knight, EJ; Prichard, BN; Richards, DA; Tuckman, J1
Cohn, JN; Mehta, J1
Dobbs, RJ; Prichard, BN; Richards, DA1
Hashimoto, K; Hashimoto, T; Iizuka, H; Imai, S; Matsuda, H; Tsukada, T1
Carey, B; Whalley, ET2
Drew, GM; Hilditch, A; Levy, GP1
Murray, A; Rawlins, MD; Sanders, GL1
Nencini, P1
Leopold, IH; Murray, DL1
Prichard, BN; Richards, DA1
Doggrell, SA1
Mills, RG; Roberts, MS; Shen, JJ; Wanwimolruk, S1
Latini, R; Mennini, T; Riva, E1
Kato, T; Kinjo, N; Moromizato, H; Noguchi, K; Sakanashi, M1
Hicks, PR; Rankin, AP1
Lathers, CM; Levin, RM; Spivey, WH; Tumer, N1
den Boer, MO; Sassen, LM; Saxena, PR; van der Giessen, WJ; Verdouw, PD1
Colindres, RE; Cubeddu, LX; Fuenmayor, N; Powell, JR; Varin, F; Villagra, VG2
Blasucci, DJ; Chodosh, S; Tuck, J1
Drummer, OH; Louis, WJ; Tung, LH1
Cleroux, J; Giannattasio, C; Grassi, G; Mancia, G; Seravalle, G; Zanchetti, A1
Carr, ME; Cubeddu, LX; Fuenmayor, NJ1
Palkama, A; Raij, K; Uusitalo, H; Uusitalo, R1
Honda, K; Miyata-Osawa, A; Nakagawa, C; Shiono, K; Takenaka, T1
Bompart, F; Graham, BR; Liu, JB; Prichard, BN; Tomlinson, B1
Matsumura, Y; Morimoto, S1
Lucchesi, BR; Lynch, JJ; Montgomery, DG1
Hurwitz, MD; Kallenbach, JM; Pincus, PS1
Doggrell, SA; Hughes, EW1
Berlin, E; Gjöres, JE; Thulesius, O1
Giorgetti, F; Re, L; Rossini, L1
Re, L; Rossini, L1
Abiko, Y; Ichihara, K; Kameda, H; Monma, Y; Okuoka, Y; Tanabe, T1
D'Ascenzo, G; Gennari, C; Maioli, E; Nami, R; Nardi, PL; Pizzuti, M1
Hlede, M; Morandin, F; Pessina, AC; Rossi, GP; Semplicini, A1
Elliott, HL; McLean, K; Meredith, PA; Reid, JL; Sumner, DJ1
Endo, J; Ohshika, H; Takemura, H; Tanaka, M1
Germond, C; Kallenbach, J; Lewis, M; Muller, F; Steyn, J; Zaltzman, M; Zwi, S1
Abassi, ZA; Cuda, G; Golomb, E; Keiser, HR; Panchal, VR; Stylianou, M; Trachewsky, D1
Conti, A; Forlani, A; Monopoli, A; Ongini, E1
Guy, S; McDermott, BJ; Riddell, JG; Shanks, RG; Tham, TC1
Kemp, GJ; Odoom, JE; Radda, GK1
Chen, IJ; Chen, SJ; Cheng, CJ; Chiu, CC; Huang, YC; Lin, YT; Wu, BN1
Abuin, L; Cotecchia, S; Lattion, A; Nenniger-Tosato, M1
Chen, IJ; Chiang, LC; Chiu, CC; Liang, JC; Lin, YT; Tsai, CH; Wu, JR; Yeh, JL1
Accinni, R; Bonacina, E; Brenna, S; Pinelli, A; Tomasoni, L; Trivulzio, S1
Acharya, M; Lau-Cam, CA1

Reviews

2 review(s) available for isoproterenol and labetalol

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
A review of the animal pharmacology of labetalol, a combined alpha- and beta-adrenoceptor-blocking drug.
    British journal of clinical pharmacology, 1976, Volume: 3, Issue:4 Suppl 3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Autonomic Fibers, Preganglionic; Desoxycorticosterone; Dogs; Electric Stimulation; Ethanolamines; Guinea Pigs; Hemodynamics; Hypertension; Hypertension, Renal; In Vitro Techniques; Isoproterenol; Labetalol; Male; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Phentolamine; Phenylephrine; Propranolol; Rabbits; Rats

1976

Trials

8 trial(s) available for isoproterenol and labetalol

ArticleYear
Hemodynamic effects of labetalol, an alpha and beta adrenergic blocking agent, in hypertensive subjects.
    Circulation, 1977, Volume: 55, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Amyl Nitrite; Blood Pressure; Cardiac Output; Clinical Trials as Topic; Dose-Response Relationship, Drug; Ethanolamines; Heart Rate; Hemodynamics; Humans; Hypertension; Isoproterenol; Labetalol; Male; Middle Aged; Phenylephrine; Physical Exertion; Renin; Valsalva Maneuver; Vascular Resistance

1977
Concurrent antagonism of isoproterenol and norepinephrine after labetalol.
    Clinical pharmacology and therapeutics, 1978, Volume: 23, Issue:3

    Topics: Adult; Blood Pressure; Dose-Response Relationship, Drug; Ethanolamines; Heart Rate; Humans; Isoproterenol; Labetalol; Male; Norepinephrine

1978
Mechanism of the vasodilatory effect of carvedilol in normal volunteers: a comparison with labetalol.
    Journal of cardiovascular pharmacology, 1987, Volume: 10 Suppl 11

    Topics: Adrenergic beta-Antagonists; Angiotensin II; Blood Pressure; Carbazoles; Carvedilol; Half-Life; Heart Rate; Humans; Isoproterenol; Labetalol; Phenylephrine; Propanolamines; Random Allocation; Vasodilation

1987
The effects of dilevalol, metoprolol, and placebo on ventilatory function in asthmatics.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 2

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Aged; Asthma; Female; Forced Expiratory Volume; Hemodynamics; Humans; Isoproterenol; Labetalol; Male; Metoprolol; Middle Aged; Respiratory Function Tests

1988
Beta blockade by oral propranolol and labetalol.
    Clinical pharmacology and therapeutics, 1985, Volume: 37, Issue:3

    Topics: Administration, Oral; Adrenergic beta-Antagonists; Adult; Blood Pressure; Double-Blind Method; Ethanolamines; Heart Rate; Humans; Injections, Intravenous; Isometric Contraction; Isoproterenol; Labetalol; Male; Propranolol; Random Allocation

1985
Vasodilating mechanism and response to physiological pressor stimuli of acute doses of carvedilol compared with labetalol, propranolol and hydralazine.
    Drugs, 1988, Volume: 36 Suppl 6

    Topics: Adrenergic beta-Antagonists; Adult; Angiotensin II; Antihypertensive Agents; Blood Pressure; Carbazoles; Carvedilol; Cold Temperature; Double-Blind Method; Exercise; Heart Rate; Hemodynamics; Humans; Hydralazine; Isoproterenol; Labetalol; Male; Middle Aged; Phenylephrine; Posture; Propanolamines; Propranolol; Vasodilator Agents

1988
Clinical pharmacology of carvedilol in normal volunteers.
    Clinical pharmacology and therapeutics, 1987, Volume: 41, Issue:1

    Topics: Adult; Angiotensin II; Blood Pressure; Carbazoles; Carvedilol; Dose-Response Relationship, Drug; Heart Rate; Humans; Isoproterenol; Kinetics; Labetalol; Male; Phenylephrine; Propanolamines; Random Allocation; Receptors, Adrenergic

1987
The dose dependency of the alpha- and beta-adrenoceptor antagonist activity of carvedilol in man.
    British journal of clinical pharmacology, 1995, Volume: 40, Issue:1

    Topics: Administration, Oral; Adrenergic beta-Antagonists; Adult; Blood Pressure; Carbazoles; Carvedilol; Double-Blind Method; Exercise; Heart Rate; Humans; Isoproterenol; Labetalol; Male; Phenylephrine; Propanolamines; Vasodilator Agents

1995

Other Studies

50 other study(ies) available for isoproterenol and labetalol

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
FDA-approved drug labeling for the study of drug-induced liver injury.
    Drug discovery today, 2011, Volume: 16, Issue:15-16

    Topics: Animals; Benchmarking; Biomarkers, Pharmacological; Chemical and Drug Induced Liver Injury; Drug Design; Drug Labeling; Drug-Related Side Effects and Adverse Reactions; Humans; Pharmaceutical Preparations; Reproducibility of Results; United States; United States Food and Drug Administration

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
    Pharmaceutical research, 2014, Volume: 31, Issue:4

    Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation

2014
Development of a cell viability assay to assess drug metabolite structure-toxicity relationships.
    Bioorganic & medicinal chemistry letters, 2016, 08-15, Volume: 26, Issue:16

    Topics: Adenosine Triphosphate; Benzbromarone; Cell Line; Cell Survival; Chromans; Cytochrome P-450 CYP2C9; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Humans; Pharmaceutical Preparations; Thiazolidinediones; Troglitazone

2016
Assessment of alpha- and beta-adrenoceptor blocking actions of labetalol.
    British journal of clinical pharmacology, 1976, Volume: 3, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Blood Pressure; Dose-Response Relationship, Drug; Ethanolamines; Heart Rate; Humans; Isoproterenol; Labetalol; Male; Phenylephrine

1976
Pharmacological basis for antihypertensive effects of intravenous labetalol.
    British heart journal, 1977, Volume: 39, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adult; Antihypertensive Agents; Blood Pressure; Depression, Chemical; Dose-Response Relationship, Drug; Ethanolamines; Heart Rate; Humans; Isoproterenol; Labetalol; Male; Phenylephrine; Physical Exertion

1977
Adrenoceptor blockade of the circulatory responses to intravenous isoproterenol.
    Clinical pharmacology and therapeutics, 1978, Volume: 24, Issue:3

    Topics: Adrenergic beta-Antagonists; Adult; Blood Pressure; Cardiac Output; Heart Rate; Hemodynamics; Humans; Isoproterenol; Labetalol; Male; Myocardial Contraction; Phentolamine; Propranolol; Stroke Volume; Time Factors

1978
Hypotensive and vascular effects of labetalol in the normotensive rat and dog.
    Japanese heart journal, 1978, Volume: 19, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Flow Velocity; Blood Pressure; Dogs; Ethanolamines; Female; Femoral Artery; Heart Rate; Isoproterenol; Kidney; Labetalol; Male; Phentolamine; Propranolol; Rats; Regional Blood Flow; Vasomotor System

1978
Beta-adrenoceptor agonist activity of labetolol on the isolated uterus of the rat.
    British journal of pharmacology, 1979, Volume: 67, Issue:1

    Topics: Acetylcholine; Adrenergic beta-Agonists; Animals; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Labetalol; Rats; Uterine Contraction; Uterus

1979
Labetalol possesses beta-adrenoceptor agonist action on the rat isolated uterus.
    The Journal of pharmacy and pharmacology, 1979, Volume: 31, Issue:11

    Topics: Adrenergic beta-Agonists; Animals; Estrus; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Labetalol; Pregnancy; Propranolol; Rats; Uterine Contraction

1979
The relationships between the cardiovascular effects, alpha- and beta-adrenoceptor blocking actions and plasma concentration of labetalol in doca hypertensive rats.
    Clinical and experimental hypertension, 1979, Volume: 1, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Depression, Chemical; Desoxycorticosterone; Dose-Response Relationship, Drug; Ethanolamines; Heart Rate; Hypertension; Isoproterenol; Labetalol; Male; Phenylephrine; Rats

1979
Interdose control of beta-blockade and arterial blood pressure during chronic oral labetalol treatment.
    British journal of clinical pharmacology, 1979, Volume: 8, Issue:Suppl 2

    Topics: Adrenergic beta-Antagonists; Adult; Blood Pressure; Drug Administration Schedule; Ethanolamines; Heart Rate; Humans; Hypertension; Isoproterenol; Labetalol; Male; Time Factors

1979
The influence of calcium on the antilipolytic action of propranolol, timolol, labetalol, verapamil, procaine, and papaverine in rat adipocytes.
    Pharmacological research communications, 1979, Volume: 11, Issue:9

    Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adrenocorticotropic Hormone; Animals; Calcium; In Vitro Techniques; Isoproterenol; Labetalol; Lipolysis; Male; Papaverine; Procaine; Propranolol; Rats; Timolol; Vasodilator Agents; Verapamil

1979
Ocular hypotensive action of labetalol.
    American journal of ophthalmology, 1979, Volume: 88, Issue:3 Pt 1

    Topics: Animals; Ethanolamines; Female; Intraocular Pressure; Isoproterenol; Labetalol; Norepinephrine; p-Hydroxyamphetamine; Phenoxybenzamine; Pupil; Rabbits; Sympathectomy; Timolol

1979
The effects of labetalol and dilevalol on isolated cardiovascular preparations of the guinea-pig and rat.
    The Journal of pharmacy and pharmacology, 1992, Volume: 44, Issue:12

    Topics: Animals; Guinea Pigs; Isoproterenol; Labetalol; Male; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Rats, Wistar

1992
Response to beta-blockers in maternal and fetal rat hearts in vitro.
    Life sciences, 1991, Volume: 48, Issue:18

    Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Female; Heart; Heart Rate; Isoproterenol; Labetalol; Metoprolol; Pregnancy; Pregnancy, Animal; Propranolol; Rats; Rats, Inbred Strains

1991
The alpha- and beta-adrenoceptor blocking activities of labetalol and its RR-SR (50:50) stereoisomers.
    British journal of pharmacology, 1991, Volume: 104, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Cerebral Cortex; Dose-Response Relationship, Drug; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Labetalol; Male; Myocardium; Phenylephrine; Prazosin; Propranolol; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Stereoisomerism

1991
Comparative effects of arotinolol, labetalol and propranolol on regional myocardial dysfunction induced by flow-limiting coronary stenosis in anesthetized dogs.
    Japanese journal of pharmacology, 1990, Volume: 53, Issue:3

    Topics: Adrenergic beta-Antagonists; Anesthesia; Animals; Blood Pressure; Cardiomyopathies; Coronary Vessels; Dogs; Female; Heart Rate; Hemodynamics; Isoproterenol; Labetalol; Male; Myocardial Contraction; Phenylephrine; Propanolamines; Propranolol

1990
Massive adrenaline doses in labetalol overdose.
    Anaesthesia and intensive care, 1991, Volume: 19, Issue:3

    Topics: Adult; Dobutamine; Dopamine; Drug Overdose; Epinephrine; Female; Humans; Isoproterenol; Labetalol

1991
The effect of dilevalol on cardiac autonomic neural discharge, plasma catecholamines, and myocardial beta receptor density associated with coronary occlusion.
    Journal of clinical pharmacology, 1990, Volume: 30, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Autonomic Nervous System; Blood Pressure; Catecholamines; Cats; Coronary Vessels; Electrophysiology; Epinephrine; Heart Rate; Isoproterenol; Labetalol; Myocardium; Neurons; Norepinephrine; Phenylephrine; Receptors, Adrenergic, beta

1990
Effects of dilevalol in the anesthetized pig with a partially occluded coronary artery.
    Cardiovascular drugs and therapy, 1990, Volume: 4, Issue:6

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthesia; Animals; Chloralose; Coronary Circulation; Coronary Disease; Heart; Hemodynamics; Isoproterenol; Labetalol; Myocardial Contraction; Myocardial Reperfusion; Swine

1990
Actions of dilevalol on adrenoceptors.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 2

    Topics: Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Decerebrate State; Dose-Response Relationship, Drug; Guinea Pigs; Heart Rate; In Vitro Techniques; Isoproterenol; Labetalol; Muscle, Smooth; Phenylephrine; Receptors, Adrenergic; Trachea; Vasodilator Agents

1988
Effects of dilevalol on forearm circulation in essential hypertension.
    The American journal of cardiology, 1989, Jun-05, Volume: 63, Issue:19

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Female; Forearm; Hemodynamics; Humans; Hypertension; Infusions, Intra-Arterial; Isoproterenol; Labetalol; Male; Middle Aged; Propranolol; Regional Blood Flow

1989
Comparison of the effects of adrenergic agonists and alpha-, beta 1-, beta 2-antagonists on the intraocular pressure and adenylate cyclase activity in the ciliary processes of the rabbit.
    Acta ophthalmologica, 1985, Volume: 63, Issue:1

    Topics: Acebutolol; Adenylyl Cyclases; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Ciliary Body; Intraocular Pressure; Isoproterenol; Labetalol; Metoprolol; Rats; Timolol; Water

1985
Autonomic and antihypertensive activity of oral amosulalol (YM-09538), a combined alpha- and beta-adrenoceptor blocking agent in conscious rats.
    Japanese journal of pharmacology, 1985, Volume: 38, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Autonomic Nervous System; Blood Pressure; Ethanolamines; Heart Rate; Isoproterenol; Labetalol; Male; Phenylephrine; Prazosin; Propranolol; Rats; Rats, Inbred SHR; Rats, Inbred Strains

1985
Effects of labetalol on renin release from rat kidney cortical slices.
    Journal of pharmacobio-dynamics, 1986, Volume: 9, Issue:11

    Topics: Animals; In Vitro Techniques; Isoproterenol; Kidney Cortex; Labetalol; Male; Norepinephrine; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Renin

1986
Cardiac electrophysiologic actions of SCH 19927 (Dilevalol), the R,R-isomer of labetalol.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:3

    Topics: Animals; Atrioventricular Node; Blood Pressure; Dogs; Electrophysiology; Heart; Heart Rate; Isomerism; Isoproterenol; Labetalol; Male

1986
Massive propranolol overdose.
    The American journal of medicine, 1986, Volume: 81, Issue:6

    Topics: Acebutolol; Adult; Dose-Response Relationship, Drug; Female; Humans; Isoproterenol; Labetalol; Suicide, Attempted

1986
Comparison of the effects of labetalol and SCH 19927, the R1R isomer of labetalol, on the rat isolated right ventricle and aorta.
    Journal of autonomic pharmacology, 1985, Volume: 5, Issue:4

    Topics: Animals; Aorta; Cocaine; Dioxanes; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Idazoxan; In Vitro Techniques; Isoproterenol; Labetalol; Male; Myocardial Contraction; Norepinephrine; Phenylephrine; Rats; Rats, Inbred Strains; Serotonin; Stereoisomerism; Vasoconstriction

1985
Alpha- and beta-adrenoceptor blockade by labetalol in human isolated arteries and veins.
    British journal of clinical pharmacology, 1980, Volume: 9, Issue:6

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arteries; Ethanolamines; Guinea Pigs; Humans; In Vitro Techniques; Isoproterenol; Labetalol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Rats; Veins

1980
[Cholinergic antagonism by beta-blockers. I. Spectrum of interactions].
    Bollettino della Societa italiana di biologia sperimentale, 1980, May-15, Volume: 56, Issue:9

    Topics: Abdominal Muscles; Acetylcholine; Adrenergic beta-Antagonists; Animals; Guinea Pigs; Heart; Ileum; Isoproterenol; Labetalol; Male; Metoprolol; Pindolol; Practolol; Propranolol; Receptors, Cholinergic; Sotalol

1980
[Cholinergic antagonism by beta-blockers. II. Sequence of interactions and final steady state effects].
    Bollettino della Societa italiana di biologia sperimentale, 1980, May-15, Volume: 56, Issue:9

    Topics: Acetylcholine; Adrenergic beta-Antagonists; Animals; Drug Interactions; Guinea Pigs; Heart; Isoproterenol; Labetalol; Male; Metoprolol; Practolol; Propranolol; Receptors, Cholinergic; Time Factors

1980
[Effects of labetalol on the circulatory system (author's transl)].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1980, Volume: 76, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Cardiovascular System; Carotid Sinus; Dogs; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Guinea Pigs; Hemodynamics; In Vitro Techniques; Isoproterenol; Labetalol; Male; Norepinephrine; Rabbits; Rana catesbeiana; Rats; Reflex; Vasodilator Agents

1980
[Exogenous adrenergic stimulation by intravenous infusions of isoproterenol and blood levels of cyclic AMP before and after beta-blocking in humans].
    Bollettino della Societa italiana di cardiologia, 1980, Volume: 25, Issue:7

    Topics: Adrenergic beta-Antagonists; Adult; Cyclic AMP; Cyclic GMP; Ethanolamines; Female; Humans; Hypertension; Isoproterenol; Labetalol; Male; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sympathetic Nervous System

1980
Alpha-adrenoceptor blockade by labetalol during long-term dosing.
    Clinical pharmacology and therapeutics, 1983, Volume: 33, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Dose-Response Relationship, Drug; Ethanolamines; Female; Heart Rate; Humans; Hypertension; Isoproterenol; Labetalol; Male; Middle Aged; Phenylephrine

1983
Comparison of medroxalol and labetalol, drugs with combined alpha- and beta-adrenoceptor antagonist properties.
    British journal of clinical pharmacology, 1984, Volume: 17, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Blood Pressure; Depression, Chemical; Double-Blind Method; Drug Evaluation; Ethanolamines; Heart Rate; Humans; Isoproterenol; Labetalol; Male; Norepinephrine; Phenylephrine; Posture

1984
Potentiation of isoproterenol-induced salivation by labetalol.
    Japanese journal of pharmacology, 1982, Volume: 32, Issue:4

    Topics: Amylases; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Epinephrine; Ethanolamines; Hydroxydopamines; In Vitro Techniques; Isoproterenol; Labetalol; Male; Oxidopamine; Parotid Gland; Potassium; Rats; Rats, Inbred Strains; Reserpine; Salivation

1982
Survival following massive overdose of adrenergic blocking agents (acebutolol and labetalol).
    European heart journal, 1983, Volume: 4, Issue:5

    Topics: Acebutolol; Adult; Atropine; Blood Pressure; Dopamine; Ethanolamines; Female; Heart Rate; Hemodynamics; Humans; Isoproterenol; Labetalol; Suicide, Attempted; Trimipramine

1983
Angiotensin II maintains, but does not mediate, isoproterenol-induced cardiac hypertrophy in rats.
    The American journal of physiology, 1994, Volume: 267, Issue:4 Pt 2

    Topics: Actins; Angiotensin II; Animals; Base Sequence; Biphenyl Compounds; Blood Pressure; Captopril; Cardiomegaly; DNA; DNA Primers; Dose-Response Relationship, Drug; Gene Expression; Genes, fos; Heart; Hydralazine; Hydroxyproline; Imidazoles; Isoproterenol; Labetalol; Losartan; Male; Methyldopa; Molecular Sequence Data; Myocardium; Myosins; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; RNA; RNA, Messenger; Tetrazoles; Transcription, Genetic

1994
Beta 1 and beta 2 adrenoceptors are involved in mediating vasodilation in the human coronary artery.
    Pharmacological research, 1993, Volume: 27, Issue:3

    Topics: Adult; Binding, Competitive; Coronary Vessels; Dinoprost; Female; Humans; In Vitro Techniques; Iodine Radioisotopes; Isoproterenol; Kinetics; Labetalol; Male; Pindolol; Receptors, Adrenergic, beta; Vasodilation

1993
The regulation of total creatine content in a myoblast cell line.
    Molecular and cellular biochemistry, 1996, May-24, Volume: 158, Issue:2

    Topics: Animals; Atenolol; Bucladesine; Butoxamine; Cell Line; Clenbuterol; Creatine; Energy Metabolism; Insulin; Insulin-Like Growth Factor I; Isoproterenol; Labetalol; Methoxamine; Mice; Muscle, Skeletal; Norepinephrine; Phentolamine; Propranolol; Sodium; Triiodothyronine

1996
Eugenodilol: a third-generation beta-adrenoceptor blocker, derived from eugenol, with alpha-adrenoceptor blocking and beta2-adrenoceptor agonist-associated vasorelaxant activities.
    Journal of cardiovascular pharmacology, 1999, Volume: 34, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Anesthesia; Animals; Aorta, Thoracic; Bradycardia; Dose-Response Relationship, Drug; Drug Interactions; Eugenol; Female; Guinea Pigs; Hypotension; In Vitro Techniques; Isoproterenol; Labetalol; Male; Muscle Contraction; Phenylephrine; Radioligand Assay; Rats; Rats, Wistar; Time Factors; Trachea; Vasodilator Agents

1999
Constitutively active mutants of the beta1-adrenergic receptor.
    FEBS letters, 1999, Sep-03, Volume: 457, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Betaxolol; Carbazoles; Carvedilol; Cell Line; Cyclic AMP; Epinephrine; Humans; Imidazoles; Isoproterenol; Labetalol; Point Mutation; Practolol; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Timolol

1999
Pharmacological effects of an aldehyde type alpha/beta-adrenoceptor blocking agent with vasodilating properties.
    General pharmacology, 2000, Volume: 34, Issue:6

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Aorta; Atenolol; Benzaldehydes; Blood Pressure; Cardiovascular Agents; Depression, Chemical; Dose-Response Relationship, Drug; Guinea Pigs; Heart Atria; Heart Rate; Isoproterenol; Labetalol; Mecamylamine; Models, Animal; Muscle, Smooth, Vascular; Myocardial Contraction; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Regression Analysis; Stimulation, Chemical; Vasodilator Agents

2000
Isoproterenol-induced myocardial infarction in rabbits. Protection by propranolol or labetalol: a proposed non-invasive procedure.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2004, Volume: 23, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Electrocardiography; Isoproterenol; Labetalol; Lipid Peroxides; Male; Myocardial Infarction; Myocardium; Partial Thromboplastin Time; Propranolol; Rabbits; Vitamin E

2004
Attenuating action of taurine and labetalol on cardiovascular alterations by pyridoxal-isoproterenol, a vitamin-drug interaction with cardiopathologic significance.
    Advances in experimental medicine and biology, 2009, Volume: 643

    Topics: Animals; Antihypertensive Agents; Cardiovascular System; Drug Interactions; Electrocardiography; Isoproterenol; Labetalol; Male; Mice; Pyridoxal; Taurine

2009