isoproterenol has been researched along with cyanopindolol in 65 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 14 (21.54) | 18.7374 |
1990's | 36 (55.38) | 18.2507 |
2000's | 14 (21.54) | 29.6817 |
2010's | 1 (1.54) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Charlton, SJ; Dickson, CJ; Duca, JS; Fairhurst, RA; Hornak, V; McKay, DJ; Pearlstein, RA; Reilly, J; Sandham, DA; Shaw, D; Sykes, DA; Velez-Vega, C | 1 |
Kompa, AR; Molenaar, P; Pak, HS; Roberts, SJ; Summers, RJ | 1 |
Tran, VT | 1 |
Liggett, SB | 1 |
Houslay, MD; Milligan, G; Strassheim, D | 1 |
Esbenshade, TA; Granneman, JG; Han, C; Minneman, KP; Theroux, TL | 1 |
Emmerich, B; Göhly, U; Haen, E; Hallek, M; Kamp, T; Remien, J | 1 |
MacDonald, A; McLaughlin, DP | 1 |
Lafontan, M; Langin, D; Portillo, MP; Saulnier-Blache, JS | 1 |
Carpéné, C; Dauzats, M; Lafontan, M; Larrouy, D; Quideau, N; Saulnier-Blache, JS | 1 |
Borst, SE; Conolly, ME; Hui, KK | 1 |
Caron, MG; Hausdorff, WP; Hnatowich, M; Lefkowitz, RJ; O'Dowd, BF | 1 |
Hintze, TH; Homcy, CJ; Nejima, J; Susanni, EE; Uemura, N; Vatner, DE; Vatner, SF | 1 |
Korichneva, IL; Krasnikova, TL; Radiukhin, VA | 1 |
Cardone, F; Cignarelli, M; Corso, M; De Pergola, G; Di Paolo, S; Garruti, G; Giorgino, R; Nardelli, G | 1 |
Grogan, DM; Hatjis, CG; Koritnik, DR | 1 |
Grogan, DM; Hatjis, CG | 1 |
Chung, MK; Gulick, T; Lange, LG; Pieper, SJ; Schreiner, GF | 1 |
Crews, A; Hatjis, CG | 1 |
Göthert, M; Hillenbrand, K; Schlicker, E | 1 |
Malta, E; Molenaar, P | 1 |
Gagne, B; Labrie, F; Lavoie, M; Poyet, P | 1 |
Levitzki, A; Marbach, I; Shiloach, J | 1 |
Engel, G; Göthert, M; Hillenbrand, K; Hoyer, D; Schlicker, E | 1 |
Crooke, ST; Heckman, GD; Nambi, P; Schmidt, DB; Stassen, FL; Whitman, MH | 1 |
Molenaar, P; Summers, RJ | 1 |
Blankesteijn, WM; de Pont, JJ; Graafsma, SJ; Thien, T; Willems, PH | 1 |
Bejarano, P; Green, SA; Hall, IP; Liggett, SB; Turki, J | 1 |
Hirsch, DJ; Morgunov, NS; You, YD | 1 |
Kompa, AR; Molenaar, P; Russell, FD; Summers, RJ | 1 |
Chiyotani, A; Konno, K; Takeuchi, S; Tamaoki, J; Yamauchi, F; Yamawaki, I | 1 |
Dombrowski, MP; Gauvin, JM; Hayashi, RH; Hurd, WW | 1 |
Clark, CJ; Connell, JM; Milligan, G | 1 |
Molenaar, P; Sarsero, D | 1 |
Molenaar, P; Roberts, SJ; Russell, FD; Summers, RJ | 1 |
Oriowo, MA | 1 |
Esbenshade, TA; Guerrero, SW; Minneman, KP; Zhong, H | 1 |
Cui, Y; Iwase, M; Kalthof, B; Sato, N; Shen, YT; Uechi, M; Vatner, DE; Vatner, SF | 1 |
Abraini, JH; Kriem, B; Rostain, JC | 1 |
Bouanani, NE; Crozatier, B; Su, JB; Xiong, L | 1 |
Gabilondo, AM; Krasel, C; Lohse, MJ | 1 |
Díaz-Laviada, I; Guillén, A; Haro, A; Nieto, JL | 1 |
Björntorp, P; Edén, S; Liu, X; Yang, S | 1 |
Houston, G; Kelly, J | 1 |
Cohen-Tannoudji, J; Coudouel, N; Lécrivain, JL; Legrand, C; Maltier, JP; Robin, MT | 1 |
Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F | 1 |
Isono, K; Nagai, A; Tagaya, E; Tamaoki, J | 1 |
Dhalla, NS; Elimban, V; Persad, S; Siddiqui, F | 1 |
Baranski, TJ; Bourne, HR; Iiri, T; Lichtarge, O; Meng, EC; Nissenson, RA; Sheikh, SP; Vilardarga, JP | 1 |
Guerrero, SW; Minneman, KP | 1 |
MacDonald, A; Watt, K | 1 |
Brawley, L; MacDonald, A; Shaw, AM | 2 |
Brink, CB; Neubig, RR; Wade, SM | 1 |
Evans, BA; Hutchinson, DS; Summers, RJ | 1 |
Engelhardt, S; Hein, L; Kaumann, AJ; Lohse, M; Molenaar, P | 1 |
Green, SA; Liggett, SB; Rathz, DA; Schuster, AJ | 1 |
Hussein, SM; Khan, I; Oriowo, M | 1 |
Barakat, H; Christian, B; Davis, J; Hickner, R; McConnaughey, MM; Privette, J; Sheets, KA | 1 |
Ishii, K; Karikomi, Y; Kubota, Y; Nakahara, T; Sakamoto, K | 1 |
Brown, MJ; O'Shaughnessy, KM; Sandilands, A; Yeo, G | 1 |
Chandrasekhar, B; Fatinikun, T; Kadavil, EA; Khan, I; Omu, AE; Oriowo, MA | 1 |
Desfontis, JC; Gogny, M; Holopherne, D; Le Coz, O; Mallem, Y; Reculeau, O | 1 |
Clark, RB; Dai, W; Friedman, J; Godines, V; Knoll, BJ; Millman, EE; Moore, RH; Tran, TM; Vaughan, DJ | 1 |
Amour, J; Birenbaum, A; Heymes, C; Loyer, X; Michelet, P; Riou, B | 1 |
1 trial(s) available for isoproterenol and cyanopindolol
Article | Year |
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Differences in beta-adrenergic receptor densities in omental and subcutaneous adipose tissue from obese African American and Caucasian women.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adult; Black or African American; Cell Membrane; Female; Humans; Immunoblotting; Isoproterenol; Kinetics; Lipolysis; Obesity, Morbid; Omentum; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; White People | 2004 |
64 other study(ies) available for isoproterenol and cyanopindolol
Article | Year |
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Uncoupling the Structure-Activity Relationships of β2 Adrenergic Receptor Ligands from Membrane Binding.
Topics: Binding Sites; Cell Membrane; Dose-Response Relationship, Drug; Humans; Ligands; Models, Molecular; Molecular Structure; Receptors, Adrenergic, beta-2; Structure-Activity Relationship | 2016 |
Localization of (-)-[125I]cyanopindolol binding in guinea-pig heart: characteristics of non-beta-adrenoceptor related binding in cardiac pacemaker and conducting regions.
Topics: Alprenolol; Animals; Ascorbic Acid; Binding Sites; Ethanolamines; Female; Guinea Pigs; Haloperidol; Heart Conduction System; Isoproterenol; Male; Myocardium; Peroxidase; Phentolamine; Pindolol; Propanolamines; Propranolol; Protein Binding; Receptors, Adrenergic, beta; Serotonin; Thiophenes; Trachea | 1992 |
Human retinal pigment epithelial cells possess beta 2-adrenergic receptors.
Topics: Adenylyl Cyclases; Betaxolol; Cells, Cultured; Cyclic AMP; Epinephrine; Humans; Isoproterenol; Norepinephrine; Pigment Epithelium of Eye; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1992 |
Functional properties of the rat and human beta 3-adrenergic receptors: differential agonist activation of recombinant receptors in Chinese hamster ovary cells.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Enzyme Activation; Humans; Isoproterenol; Pindolol; Rats; Receptors, Adrenergic, beta; Recombinant Proteins | 1992 |
Regulation of cardiac adenylate cyclase activity in rodent models of obesity.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Binding, Competitive; Disease Models, Animal; GTP-Binding Proteins; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Membranes; Mice; Mice, Obese; Myocardium; Obesity; Pindolol; Rats; Rats, Zucker; Receptors, Adrenergic, beta; Stimulation, Chemical | 1992 |
Coexisting beta 1- and atypical beta-adrenergic receptors cause redundant increases in cyclic AMP in human neuroblastoma cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Neuroblastoma; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured | 1992 |
Reduced responsiveness of adenylate cyclase to forskolin in human lymphoma cells.
Topics: Adenylyl Cyclase Inhibitors; Aged; B-Lymphocytes; Binding Sites; Cholera Toxin; Colforsin; Cyclic AMP; Female; Humans; Isoproterenol; Lymphoma, Non-Hodgkin; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Signal Transduction; Tumor Cells, Cultured | 1991 |
Characterization of catecholamine-mediated relaxations in rat isolated gastric fundus: evidence for an atypical beta-adrenoceptor.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Catecholamines; Ethanolamines; Gastric Fundus; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Norepinephrine; Pindolol; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Coexistence of three beta-adrenoceptor subtypes in white fat cells of various mammalian species.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cricetinae; Dogs; Ethanolamines; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lipolysis; Male; Mesocricetus; Muscle, Smooth; Pindolol; Propanolamines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Photoperiodic control of adipocyte alpha 2-adrenoceptors in Syrian hamsters: role of testosterone.
Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brain; Brimonidine Tartrate; Cricetinae; Dioxanes; Idazoxan; Isoproterenol; Kidney; Light; Lipolysis; Male; Mesocricetus; Periodicity; Pindolol; Quinoxalines; Receptors, Adrenergic, alpha; Testosterone | 1990 |
Beta-adrenergic receptors on human lymphocytes: comparison of down-regulation in vivo and in vitro.
Topics: Adrenergic beta-Antagonists; Down-Regulation; Humans; Isoproterenol; Lymphocytes; Pindolol; Receptors, Adrenergic, beta; Terbutaline; Time Factors | 1990 |
A mutation of the beta 2-adrenergic receptor impairs agonist activation of adenylyl cyclase without affecting high affinity agonist binding. Distinct molecular determinants of the receptor are involved in physical coupling to and functional activation of
Topics: Adenylyl Cyclases; Amino Acid Sequence; Cell Compartmentation; DNA Mutational Analysis; Endocytosis; Enzyme Activation; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Isoproterenol; Macromolecular Substances; Molecular Sequence Data; Mutation; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Structure-Activity Relationship | 1990 |
Chronic norepinephrine elicits desensitization by uncoupling the beta-receptor.
Topics: Adenylyl Cyclases; Animals; Colforsin; Dogs; Drug Tolerance; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Heart Ventricles; Hemodynamics; Isoproterenol; Norepinephrine; Organ Size; Pindolol; Receptors, Adrenergic, beta; Sodium Fluoride; Sodium-Potassium-Exchanging ATPase; Ventricular Function | 1989 |
[Dependence of kinetic constants of intact human lymphocyte beta2-adrenoreceptors on the nature of the radioligands used].
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Ethylmaleimide; Humans; Isoproterenol; Kinetics; Lymphocytes; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Temperature | 1989 |
Influence of lactate on isoproterenol-induced lipolysis and beta-adrenoceptors distribution in human fat cells.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adult; Cell Membrane; Cells, Cultured; Humans; Isoproterenol; Lactates; Lipolysis; Middle Aged; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Serotonin Antagonists | 1989 |
Treatment of oophorectomized guinea pigs with intrauterine 17 beta-estradiol pellets may modulate myometrial beta-adrenergic receptor binding properties.
Topics: Adrenergic beta-Antagonists; Animals; Estradiol; Female; Guanosine Triphosphate; Guinea Pigs; Isoproterenol; Myometrium; Ovariectomy; Pindolol; Progesterone; Receptors, Adrenergic, beta | 1989 |
Pregnancy-induced changes in the interaction of guinea pig myometrial beta-adrenergic receptors with l-isoproterenol.
Topics: Adrenergic beta-Antagonists; Animals; Female; Guanosine Triphosphate; Guinea Pigs; Isoproterenol; Myometrium; Pindolol; Pregnancy; Pregnancy, Animal; Receptors, Adrenergic, beta | 1989 |
Immune cytokine inhibition of beta-adrenergic agonist stimulated cyclic AMP generation in cardiac myocytes.
Topics: Animals; Animals, Newborn; Biological Products; Cells, Cultured; Culture Media; Cyclic AMP; Cytokines; Isoproterenol; Lymphocyte Activation; Lymphocytes; Macrophages; Myocardium; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Spleen | 1988 |
Regulation of guinea pig myometrial beta-adrenoreceptors by guanosine triphosphate and magnesium ion.
Topics: Animals; Female; Guanosine Triphosphate; Guinea Pigs; Iodine Radioisotopes; Isoproterenol; Magnesium; Myometrium; Pindolol; Pregnancy; Propranolol; Radioimmunoassay; Receptors, Adrenergic, beta | 1988 |
Cyanopindolol is a highly potent and selective antagonist at the presynaptic serotonin autoreceptor in the rat brain cortex.
Topics: Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Isoproterenol; Male; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Stereoisomerism | 1985 |
Analysis of agonist dissociation constants as assessed by functional antagonism in guinea pig left atria.
Topics: Adenosine; Adrenergic beta-Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Benzofurans; Carbachol; Catechols; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Myocardial Contraction; Nifedipine; Pindolol; Propanolamines | 1986 |
Characteristics of the beta-adrenergic receptor in the rat ventral prostate using [125I]cyanopindolol.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Chemical Precipitation; Epinephrine; Isoproterenol; Male; Norepinephrine; Pindolol; Polyethylene Glycols; Prostate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1986 |
Gi affects the agonist-binding properties of beta-adrenoceptors in the presence of Gs.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Catalysis; Cholera Toxin; Erythrocyte Membrane; GTP-Binding Proteins; Isoproterenol; Lymphoma; Pertussis Toxin; Pindolol; Receptors, Adrenergic, beta; Turkeys; Virulence Factors, Bordetella | 1988 |
Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites.
Topics: Animals; Cerebral Cortex; In Vitro Techniques; Isoproterenol; Ketanserin; Kinetics; Male; Pindolol; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Subcellular Fractions; Swine | 1986 |
Induction of functional beta-adrenergic receptors in rat aortic smooth muscle cells by sodium butyrate.
Topics: Adenylyl Cyclases; Animals; Butyrates; Butyric Acid; Cell Membrane; Cells, Cultured; Isoproterenol; Kinetics; Muscle, Smooth, Vascular; Pindolol; Rats; Receptors, Adrenergic, beta | 1986 |
Characterization of beta-1 and beta-2 adrenoceptors in guinea pig atrium: functional and receptor binding studies.
Topics: Animals; Electric Stimulation; Ethanolamines; Female; Guinea Pigs; Heart Atria; Heart Rate; Imidazoles; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Pindolol; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Stimulation, Chemical; Uterine Contraction; Uterus | 1987 |
Forskolin-stimulated adenylyl cyclase activity is decreased but beta 2-adrenoceptor function is unchanged in primary hypertension.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Adult; Binding, Competitive; Cell Membrane; Colforsin; Female; Hemodynamics; Humans; Hypertension; Isoproterenol; Leukocytes, Mononuclear; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Sex Factors | 1993 |
Influence of beta 2-adrenergic receptor genotypes on signal transduction in human airway smooth muscle cells.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Down-Regulation; Genotype; Humans; Isoproterenol; Muscle, Smooth; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta-2; Second Messenger Systems; Signal Transduction; Trachea | 1995 |
Response of mouse proximal straight tubule and medullary thick ascending limb to beta-agonist.
Topics: Adrenergic beta-Antagonists; Animals; Electrophysiology; Furosemide; In Vitro Techniques; Isoproterenol; Kidney Medulla; Kidney Tubules; Kidney Tubules, Proximal; Kinetics; Membrane Potentials; Mice; Perfusion; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta | 1993 |
Regulation of beta-adrenoceptors in the guinea-pig sinoatrial node.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Catechols; Chromatography, High Pressure Liquid; Densitometry; Down-Regulation; Drug Interactions; Female; Guinea Pigs; Heart Atria; Isoproterenol; Male; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Sinoatrial Node | 1994 |
Atypical beta-adrenoceptor- (beta 3-adrenoceptor) mediated relaxation of canine isolated bronchial smooth muscle.
Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Bronchi; Cyclic AMP; Dogs; Ethanolamines; Female; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1993 |
Cocaine selectively inhibits beta-adrenergic receptor binding in pregnant human myometrium.
Topics: Adrenergic beta-Antagonists; Binding, Competitive; Cocaine; Dihydroergotoxine; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Isoproterenol; Least-Squares Analysis; Molecular Structure; Myometrium; Pindolol; Pregnancy; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1993 |
Guanine nucleotide regulatory protein alterations in young Milan hypertensive strain rats.
Topics: Adenylyl Cyclases; Alprostadil; Amino Acid Sequence; Animals; Cell Membrane; Cells, Cultured; Colforsin; GTP-Binding Proteins; Hypertension; Immune Sera; Isoproterenol; Molecular Sequence Data; Muscle, Smooth, Vascular; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Signal Transduction | 1994 |
Effects of chronic infusion of (-)-isoprenaline on rat cardiac muscarinic (M2)-cholinoceptors and beta 1- and beta 2-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Binding, Competitive; Down-Regulation; Heart Ventricles; Imidazoles; Infusion Pumps, Implantable; Isoproterenol; Male; Myocardium; N-Methylscopolamine; Pindolol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Scopolamine Derivatives | 1995 |
Characterization and localization of atypical beta-adrenoceptors in rat ileum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Female; Ileum; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1995 |
Different atypical beta-adrenoceptors mediate isoprenaline-induced relaxation in vascular and non-vascular smooth muscles.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Pindolol; Rats; Receptors, Adrenergic, beta | 1995 |
Inducible expression of beta 1- and beta 2-adrenergic receptors in rat C6 glioma cells: functional interactions between closely related subtypes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Epinephrine; Gene Expression Regulation, Neoplastic; Genomic Library; Glioma; Imidazoles; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Norepinephrine; Pindolol; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Transfection; Tumor Cells, Cultured | 1996 |
Identification and functional role of beta-adrenergic receptor subtypes in primate and rodent: in vivo versus isolated myocytes.
Topics: Adrenergic beta-Antagonists; Animals; Betaxolol; Blood Pressure; Cells, Cultured; Coronary Vessels; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardium; Papio; Pindolol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Vascular Resistance; Ventricular Function, Left; Ventricular Function, Right | 1996 |
Role of 5-HT1b receptor in the pressure-induced behavioral and neurochemical disorders in rats.
Topics: Adrenergic beta-Agonists; Animals; Atmospheric Pressure; Behavior, Animal; Brain Chemistry; Calibration; Dopamine; Electrochemistry; Electrodes; High Pressure Neurological Syndrome; Isoproterenol; Male; Motor Activity; Neostriatum; Pindolol; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1996 |
Propranolol therapy in experimental heart failure in rabbits improves cardiac response to catecholamines without beta-adrenoceptor up-regulation.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Cardiac Output, Low; Catecholamines; Female; Heart; Heart Function Tests; Heart Rate; Hemodynamics; Isoproterenol; Male; Myocardium; Norepinephrine; Pindolol; Propranolol; Rabbits; Receptors, Adrenergic, beta; Up-Regulation; Ventricular Function | 1995 |
Mutations of Tyr326 in the beta 2-adrenoceptor disrupt multiple receptor functions.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alanine; Animals; Cell Membrane; CHO Cells; Cloning, Molecular; Cricetinae; Gene Expression; Humans; Iodine Radioisotopes; Isoproterenol; Mutagenesis, Site-Directed; Mutation; Phenylalanine; Pindolol; Protein Binding; Radioligand Assay; Receptors, Adrenergic, beta-2; Transfection; Tyrosine | 1996 |
Effect of endurance physical training on rat liver adenylyl cyclase system.
Topics: Adaptation, Physiological; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Colforsin; Enzyme Activation; Fluorides; Glucagon; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Liver; Male; Manganese; Physical Conditioning, Animal; Physical Endurance; Pindolol; Random Allocation; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1996 |
Growth hormone treatment of hypophysectomized rats increases catecholamine-induced lipolysis and the number of beta-adrenergic receptors in adipocytes: no differences in the effects of growth hormone on different fat depots.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Female; Growth Hormone; Hypophysectomy; Iodine Radioisotopes; Isoproterenol; Lipolysis; Male; Norepinephrine; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1996 |
Beta 3-adrenoceptors mediating relaxation of the oesophageal tunica muscularis mucosae and distal colon in the rat: comparative pharmacology and their desensitization by BRL 37344.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dose-Response Relationship, Drug; Esophagus; Ethanolamines; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1996 |
Molecular mechanisms of adenylyl cyclase desensitization in pregnant rat myometrium following in vivo administration of the beta-adrenergic agonist, isoproterenol.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Drug Tolerance; Female; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Myometrium; Pindolol; Pregnancy; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; RNA, Messenger | 1998 |
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1998 |
Atypical adrenoceptor-mediated relaxation of canine pulmonary artery through a cAMP-dependent pathway.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cyclic AMP; Dioxoles; Dogs; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Pindolol; Propanolamines; Pulmonary Artery; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1998 |
Alterations in cardiac membrane beta-adrenoceptors and adenylyl cyclase due to hypochlorous acid.
Topics: Adenosine Diphosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Ascorbic Acid; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hypochlorous Acid; Immunoblotting; Isoproterenol; Lipid Peroxidation; Methionine; Myocardium; Pertussis Toxin; Pindolol; Propane; Rats; Receptors, Adrenergic; Sodium Fluoride; Virulence Factors, Bordetella | 1999 |
Similar structures and shared switch mechanisms of the beta2-adrenoceptor and the parathyroid hormone receptor. Zn(II) bridges between helices III and VI block activation.
Topics: Animals; Binding, Competitive; Evolution, Molecular; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Histidine; Humans; Isoproterenol; Models, Molecular; Mutation; Pindolol; Protein Engineering; Protein Structure, Secondary; Receptors, Adrenergic, beta-2; Receptors, Parathyroid Hormone; Rod Opsins; Secretin; Sequence Alignment; Signal Transduction; Zinc | 1999 |
Coupling efficiencies of beta 1- and beta 2-adrenergic receptors expressed alone or together in transfected GH3 pituitary cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Imidazoles; Iodine Radioisotopes; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Pindolol; Pituitary Gland, Anterior; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection | 1999 |
Characterisation of the atypical beta-adrenoceptor in rabbit isolated jejunum using BRL 37344, cyanopindolol and SR 59230A.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Jejunum; Male; Pindolol; Propanolamines; Propranolol; Rabbits; Receptors, Adrenergic, beta | 1999 |
Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Bupranolol; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Substrate Specificity; Vasodilator Agents | 2000 |
Role of endothelium/nitric oxide in atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Norepinephrine; Oxadiazoles; Phenoxyacetates; Phenoxypropanolamines; Phenylacetates; Pindolol; Propanolamines; Propranolol; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Vasodilation | 2000 |
Agonist-directed trafficking of porcine alpha(2A)-adrenergic receptor signaling in Chinese hamster ovary cells: l-isoproterenol selectively activates G(s).
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Binding Sites; Brimonidine Tartrate; CHO Cells; Cricetinae; Drug Interactions; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Isoproterenol; Kinetics; Oxymetazoline; Pindolol; Protein Binding; Quinoxalines; Receptors, Adrenergic, alpha-2; Serotonin Antagonists; Signal Transduction; Swine; Yohimbine | 2000 |
beta(1)-Adrenoceptors compensate for beta(3)-adrenoceptors in ileum from beta(3)-adrenoceptor knock-out mice.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Genotype; Ileum; In Vitro Techniques; Isoproterenol; Mice; Mice, Knockout; Muscle Relaxation; Muscle, Smooth; Pindolol; Propranolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2001 |
Abolition of (-)-CGP 12177-evoked cardiostimulation in double beta1/beta2-adrenoceptor knockout mice. Obligatory role of beta1-adrenoceptors for putative beta4-adrenoceptor pharmacology.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Binding, Competitive; Bucladesine; Dose-Response Relationship, Drug; Female; Genotype; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Membranes; Mice; Mice, Knockout; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sinoatrial Node; Tritium | 2001 |
The Ile164 beta(2)-adrenoceptor polymorphism alters salmeterol exosite binding and conventional agonist coupling to G(s).
Topics: Adrenergic beta-Agonists; Albuterol; Amino Acid Substitution; Animals; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Genotype; Humans; Iodine Radioisotopes; Isoproterenol; Metaproterenol; Pindolol; Polymorphism, Genetic; Radioligand Assay; Receptors, Adrenergic, beta-2; Salmeterol Xinafoate; Terbutaline | 2001 |
Studies on the expression and function of beta-3-adrenoceptors in the colon of rats with acetic acid-induced colitis.
Topics: Acetic Acid; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colitis, Ulcerative; Colon; Dose-Response Relationship, Drug; Ethanolamines; Female; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Peroxidase; Pindolol; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-3; RNA, Messenger | 2002 |
Characterization of mexiletine as an antagonist of beta-adrenoceptor in Chinese hamster ovary cells expressing cloned human beta-adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Drug Interactions; Female; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lidocaine; Mexiletine; Pindolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection | 2004 |
Functional responses of human beta1 adrenoceptors with defined haplotypes for the common 389R>G and 49S>G polymorphisms.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cells, Cultured; Cyclic AMP; DNA, Complementary; Down-Regulation; Genotype; Haplotypes; Humans; Iodine Radioisotopes; Isoproterenol; Kidney; Ligands; Pindolol; Polymorphism, Genetic; Receptors, Adrenergic, beta-1 | 2004 |
Evidence for the presence of beta-3-adrenoceptors mediating relaxation in the human oviduct.
Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adult; Dose-Response Relationship, Drug; Ethanolamines; Fallopian Tubes; Female; Humans; In Vitro Techniques; Isoproterenol; Middle Aged; Muscle Relaxation; Pindolol; Propranolol; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2005 |
Beta-adrenoceptor-mediated vascular relaxation in spontaneously hypertensive rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Tetrahydronaphthalenes | 2005 |
Role of the G protein-coupled receptor kinase site serine cluster in beta2-adrenergic receptor internalization, desensitization, and beta-arrestin translocation.
Topics: Adenylyl Cyclases; Alanine; Arrestins; Aspartic Acid; beta-Arrestin 1; beta-Arrestin 2; beta-Arrestins; Binding Sites; Blotting, Western; Cell Line; Cell Membrane; Cyclic AMP-Dependent Protein Kinases; DNA, Complementary; Epinephrine; G-Protein-Coupled Receptor Kinase 1; Green Fluorescent Proteins; Humans; Isoproterenol; Kinetics; Mutation; Phosphorylation; Pindolol; Protein Structure, Tertiary; Protein Transport; Receptors, Adrenergic, beta-2; Serine; Time Factors; Transfection | 2006 |
Preservation of the positive lusitropic effect of beta-adrenoceptors stimulation in diabetic cardiomyopathy.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathies; Colforsin; Diabetes Complications; Diabetes Mellitus, Experimental; Echocardiography; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Papillary Muscles; Phentolamine; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 2008 |