isoproterenol has been researched along with cgp 20712a in 100 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (7.00) | 18.7374 |
1990's | 42 (42.00) | 18.2507 |
2000's | 40 (40.00) | 29.6817 |
2010's | 11 (11.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Guillaume, JL; Méjean, A; Strosberg, AD | 1 |
Majewski, H; Mian, MA; Rand, MJ | 1 |
Choi, AL; Martínez de la Escalera, G; Weiner, RI | 1 |
Esbenshade, TA; Granneman, JG; Han, C; Minneman, KP; Theroux, TL | 1 |
Brouwer, F; Hollenga, C; Zaagsma, J | 1 |
Leysen, JE; Pauwels, PJ; Van Gompel, P | 1 |
Holzer, G; Künster, A; Wessler, I | 1 |
Bowen, WP; Flint, DJ; Vernon, RG | 1 |
Cerbai, E; Masini, I; Mugelli, A | 1 |
Freissmuth, M; Nanoff, C; Schütz, W; Tuisl, E | 1 |
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
Groszmann, RJ; Kaumann, AJ | 1 |
Hollenga, C; Zaagsma, J | 1 |
Dubbin, PN; Dusting, GJ; Macdonald, PS | 1 |
Hadcock, JR; Malbon, CC | 1 |
Molenaar, P; Summers, RJ | 1 |
MacDonald, A; McKean, J | 1 |
Langer, L; Lemmer, B; Olbrich, HG; Witte, K | 1 |
Olszewski, MA; Robinson, NE; Zhang, XY | 1 |
Champigneulle, A; Elalouf, JM; Imbert-Teboul, M; Mandon, B; Siga, E | 1 |
Badran, TW; Hoey, AJ; Matthews, ML; Pegg, GG; Sillence, MN | 1 |
Charpentier, F; Rosen, MR | 1 |
Kuznetsov, V; Pak, E; Robinson, RB; Steinberg, SF | 1 |
Berry, JL; Chiu, P; Cook, SJ; Downing, SJ; Foster, RW; Small, RC | 1 |
Baude, B; Emorine, LJ; Fève, B; Krief, S; Pairault, J; Strosberg, AD; Zilberfarb, V | 1 |
Nash, MS; Osborne, NN | 1 |
Bazin, R; Charon, C; Diot-Dupuy, F; Emorine, LJ; Krief, S; Strosberg, AD | 1 |
Adachi-Akahane, S; Kitagawa, Y; Nagao, T | 1 |
Molenaar, P; Sarsero, D | 1 |
Barsh, GS; Bernstein, D; Desai, KH; Jasper, JR; Kobilka, BK; Regula, DP; Rohrer, DK; Stevens, ME | 1 |
Esbenshade, TA; Guerrero, SW; Minneman, KP; Zhong, H | 1 |
Bültmann, R; Driessen, B; Gonçalves, J; Starke, K | 1 |
Pfaffendorf, M; van Zwieten, PA; Winkler Prins, EA; Zwaveling, J | 1 |
Barker, LA; Spadari-Bratfisch, RC; Zanesco, A | 1 |
Du, F; Quaegebeur, JM; Sun, LS | 1 |
Altschuld, R; Bogdanov, KY; Cheng, H; Hohl, C; Lakatta, EG; Xiao, RP; Zhou, YY | 1 |
Altschuld, RA; Billman, GE; Castillo, LC; Hensley, J; Hohl, CM | 1 |
Bilbe, G; Kellenberger, S; Muller, K; Richener, H | 1 |
Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F | 1 |
Liu, YL; Nwosu, UC; Rice, PJ | 1 |
Doze, P; Elsinga, PH; Ensing, K; Kraan, J; Vaalburg, W; van der Mark, TW; van Waarde, A; Visser, TJ | 1 |
Herzig, S; Schröder, F | 1 |
Ajisawa, Y; Akahane, M; Andersson, KE; Hayakawa, K; Igawa, Y; Nishizawa, O; Takeda, H; Yamazaki, Y; Yoneyama, T | 1 |
Atgié, C; Berlan, M; Carpéné, C; Fontana, E; Galitzky, J; Lafontan, M | 1 |
Cerbai, E; Mugelli, A; Pino, R; Rodriguez, ML | 1 |
Guerrero, SW; Minneman, KP | 1 |
Abuin, L; Cotecchia, S; Lattion, A; Nenniger-Tosato, M | 1 |
Colucci, WS; Communal, C; Sawyer, DB; Singh, K | 1 |
Dong, E; Liang, CS; Mohan, A; Yatani, A | 1 |
Brawley, L; MacDonald, A; Shaw, AM | 1 |
Ferro, A; Gao, L; Li, J; Xu, B | 1 |
Black, JW; Prendergast, CE; Shankley, NP | 1 |
Adamson, DL; Harding, SE; Money-Kyrle, AR | 1 |
Bahouth, SW; Buffington, C; Cowan, GS; Fain, JN; Li, J; Pouncey, L | 1 |
Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S | 1 |
Heijenbrok, FJ; Mathy, MJ; Pfaffendorf, M; van Zwieten, PA | 1 |
Danilo, P; Gainullin, RZ; Moise, NS; Rosen, MR; Sosunov, EA; Steinberg, SF | 1 |
Brown, KJ; Summers, RJ | 1 |
Böhm, M; Cremers, B; Dabew, E; Maack, C; Schnabel, P; Südkamp, M; Tyroller, S | 1 |
Huang, Y; Xu, B | 1 |
Graf, EM; Harding, SE; Herzig, S; Heubach, JF; Jäger, A; Molenaar, P; Ravens, U; Schröder, F | 1 |
Chess-Williams, R; Sellers, DJ | 1 |
Bölck, B; Brixius, K; Bundkirchen, A; Mehlhorn, U; Schwinger, RH | 1 |
Karle, CA; Kathöfer, S; Kiehn, J; Schoels, W; Zhang, W; Zitron, E | 1 |
Chess-Williams, R; Chong, LK; Peachell, PT | 1 |
Brouri, F; Findji, L; Hamon, M; Hanoun, N; Le Naour, G; Lechat, P; Mediani, O; Mougenot, N | 1 |
Blaschke, M; Harding, SE; Heubach, JF; Kaumann, AJ; Ravens, U | 1 |
Black, JW; Harper, EA; Hasseldine, AR | 1 |
Chapple, CR; Chess-Williams, R; Yamanishi, T; Yasuda, K; Yoshida, K | 2 |
Chakir, K; Cheng, H; Kobilka, BK; Xiang, Y; Xiao, RP; Yang, D; Zhang, SJ | 1 |
Callebert, J; Etienne, N; Jaffré, F; Launay, JM; Maroteaux, L; Monassier, L; Nebigil, CG; Sarre, A | 1 |
Ander, AN; Drumm, JD; Duggirala, SK; Roth, DM | 1 |
Corleto, VD; Delle Fave, G; Romano, G; Severi, C; Tattoli, I | 1 |
Battaglia, F; Bonacchi, M; Casini, S; Cerbai, E; Fiorani, B; Giunti, G; Lonardo, G; Mugelli, A; Sani, G; Stefano, PL | 1 |
Caceres, VM; Krieger, MH; Moreira, MF; Santos, IN; Spadari-Bratfisch, RC; Sumitame, M | 1 |
Chandra, R; Chikaraishi, DM; Groelle, M; Portbury, AL; Ray, A; Ream, M | 1 |
Bianchetti, A; Croci, T; Di Marzo, V; Di Palo, S; Ferla, G; Guagnini, F; Matias, I; Mukenge, S; Valenti, M | 1 |
Allen, BG; Baragli, A; Boivin, B; Ethier, N; Hébert, TE; Lavoie, C; Trieu, P; Vaniotis, G; Villeneuve, LR | 1 |
Jing, Y; Shan, D; Su, Y; Wang, H; Wong, TM | 1 |
Chartier, D; Ehrlich, JR; Hébert, TE; Nattel, S; Qi, X; Yeh, YH | 1 |
Chandrasekar, B; Gu, Y; Hamid, T; Hill, BG; Luo, J; Prabhu, SD; Srivastava, S | 1 |
Galindo-Tovar, A; Kaumann, AJ | 1 |
Bang, ML; Catalucci, D; Condorelli, G | 1 |
Ali, NN; Brito-Martins, M; Harding, SE | 1 |
Boussemaere, M; Denef, C; Janssens, K; Kopka, K; Wagner, S | 1 |
Chen, P; Liu, Z; Ma, K; Yang, H; Zhang, Y; Zhou, C | 1 |
Gong, KZ; Guo, JH; Song, Y; Xia, Y; Xu, M; Zhang, P; Zhang, YY | 1 |
Bányász, T; Bárándi, L; Harmati, G; Horváth, B; Magyar, J; Nánási, PP; Szabó, G; Szénási, G; Szentandrássy, N; Szentmiklósi, JA | 1 |
Chang, AM; Jiang, XW; Sun, H; Zhang, Y | 1 |
Baker, JG; Fretwell, L; Gardiner, SM; Hill, SJ; Kemp, P; March, J | 1 |
Gao, L; Jiang, X; Li, D; Sun, H; Wang, Y; Xu, C; Yan, C | 1 |
Barnes, JL; Ghosh, PM; Ikeno, Y; Kamat, A; Katz, MS; Lu, Z; Shu, ZJ; Yeh, CK; Zhang, BX; Zhu, B | 1 |
Aflaki, M; Luo, X; Maguy, A; Nattel, S; Ordog, B; Qi, XY; Shi, Y; Tadevosyan, A; Tardif, JC; Xiao, L | 1 |
Kaumann, AJ; Newe, M; Propping, S; Ravens, U; Wirth, MP | 1 |
Amisten, S; Arányi, T; Denning, C; Dolatshad, NF; Földes, G; Harding, SE; Ketteler, R; Kodagoda, T; Kolker, L; Kriston-Vizi, J; Leja, T; Matsa, E; Mioulane, M; Schneider, MD; Vauchez, K | 1 |
Lorenz, K; Newe, M; Propping, S; Ravens, U; Wirth, MP | 1 |
Hanvey, HM; Jang, DS; Joseph, BK; McClenahan, SJ; Moore, CL; Nelson, PL; Rhee, SW | 1 |
Buonarati, OR; Catterall, WA; Chowdhury, D; Hell, JW; Hofmann, F; Lee, B; Matt, L; Nanou, E; Navedo, MF; Nieves-Cintrón, M; Nystoriak, MA; Patriarchi, T; Poomvanicha, M; Price, JL; Qian, H | 1 |
Bahn, A; Bussey, CT; Cook, RF; Cragg, PA; Fomison-Nurse, IC; Hughes, G; Lamberts, RR | 1 |
1 trial(s) available for isoproterenol and cgp 20712a
Article | Year |
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Synergism between insulin and low concentrations of isoproterenol in the stimulation of leptin release by cultured human adipose tissue.
Topics: Adipocytes; Adrenergic beta-Antagonists; Adult; Catecholamines; Dexamethasone; Drug Synergism; Female; Humans; Hyperglycemia; Imidazoles; Insulin; Isoproterenol; Leptin; Lipolysis; Male; Obesity | 2000 |
99 other study(ies) available for isoproterenol and cgp 20712a
Article | Year |
---|---|
Carazolol: a potent, selective beta 3-adrenoceptor agonist.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; CHO Cells; Cricetinae; Dithiothreitol; Lipolysis; Propanolamines; Receptors, Adrenergic, beta | 1995 |
An inhibitory effect of isoprenaline on stimulation-induced noradrenaline release from rat atria.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Electric Stimulation; Female; Heart Atria; Imidazoles; Indomethacin; Isoproterenol; Male; Norepinephrine; Phentolamine; Propanolamines; Rats; Rats, Inbred Strains | 1992 |
Beta 1-adrenergic regulation of the GT1 gonadotropin-releasing hormone (GnRH) neuronal cell lines: stimulation of GnRH release via receptors positively coupled to adenylate cyclase.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Line; Cyclic AMP; Gonadotropin-Releasing Hormone; Imidazoles; Isoproterenol; Kinetics; Mice; Mice, Transgenic; Neurons; Norepinephrine; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, LHRH | 1992 |
Coexisting beta 1- and atypical beta-adrenergic receptors cause redundant increases in cyclic AMP in human neuroblastoma cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Neuroblastoma; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured | 1992 |
Relationship between lipolysis and cyclic AMP generation mediated by atypical beta-adrenoceptors in rat adipocytes.
Topics: Adipocytes; Animals; Cattle; Cyclic AMP; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1991 |
Human beta 1- and beta 2-adrenergic receptor binding and mediated accumulation of cAMP in transfected Chinese hamster ovary cells. Profile of nebivolol and known beta-adrenergic blockers.
Topics: Adrenergic beta-Antagonists; Animals; Benzopyrans; Binding Sites; Binding, Competitive; Cell Line; Cricetinae; Cricetulus; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Models, Biological; Nebivolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Stereoisomerism; Transfection | 1991 |
Stimulation of beta 1-adrenoceptors enhances electrically evoked [3H]-acetylcholine release from rat phrenic nerve.
Topics: Acetylcholine; Adrenergic beta-Antagonists; Animals; Electric Stimulation; Female; Fenoterol; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Phentolamine; Phrenic Nerve; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Tritium | 1990 |
Characterization of the beta-adrenergic receptors of sheep adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Atenolol; Epinephrine; Imidazoles; Isoproterenol; Norepinephrine; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Sheep | 1990 |
Electrophysiological characterization of cardiac beta 2-adrenoceptors in sheep Purkinje fibers.
Topics: Action Potentials; Adrenergic beta-Antagonists; Animals; Drug Interactions; Imidazoles; Isoproterenol; Propanolamines; Purkinje Fibers; Receptors, Adrenergic, beta; Sheep | 1990 |
A different desensitization pattern of cardiac beta-adrenoceptor subtypes by prolonged in vivo infusion of isoprenaline.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Cell Membrane; Heart; Imidazoles; Infusions, Intravenous; Iodocyanopindolol; Isoproterenol; Male; Myocardium; Organ Size; Ouabain; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sarcoplasmic Reticulum; Succinate Dehydrogenase | 1989 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Catecholamines relax portal and mesenteric veins from normal and portal hypertensive rats.
Topics: Adrenergic beta-Antagonists; Animals; Buserelin; Epinephrine; Goserelin; Hypertension, Portal; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Mesenteric Veins; Muscle, Smooth, Vascular; Norepinephrine; Portal Vein; Potassium Chloride; Rats; Rats, Inbred Strains; Reference Values; Vasodilation | 1989 |
Direct evidence for the atypical nature of functional beta-adrenoceptors in rat adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Epididymis; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1989 |
Beta-adrenoceptors on endothelial cells do not influence release of relaxing factor in dog coronary arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Biological Products; Bradykinin; Coronary Vessels; Dogs; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Isoproterenol; Nitric Oxide; Propanolamines; Prostaglandin Endoperoxides, Synthetic; Receptors, Adrenergic, beta; Vasodilation | 1987 |
Down-regulation of beta-adrenergic receptors: agonist-induced reduction in receptor mRNA levels.
Topics: Adrenergic beta-Antagonists; Animals; Cell Line; Cricetinae; Cyclic AMP; DNA; Endonucleases; Imidazoles; Isoproterenol; Kinetics; Male; Nucleic Acid Hybridization; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA, Messenger; Single-Strand Specific DNA and RNA Endonucleases; Vas Deferens | 1988 |
Characterization of beta-1 and beta-2 adrenoceptors in guinea pig atrium: functional and receptor binding studies.
Topics: Animals; Electric Stimulation; Ethanolamines; Female; Guinea Pigs; Heart Atria; Heart Rate; Imidazoles; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Pindolol; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Stimulation, Chemical; Uterine Contraction; Uterus | 1987 |
Contributions of beta-adrenoceptor subtypes to responses to isoprenaline in rat isolated distal colon.
Topics: Animals; Colon; Imidazoles; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1995 |
Uncoupling of beta 1-adrenoceptors from cardiac adenylyl cyclase in cardiomyopathic and control hamsters.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cardiomyopathies; Cricetinae; Heart Ventricles; Imidazoles; Isoproterenol; Male; Membranes; Mesocricetus; Myocardium; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1 | 1993 |
Beta 2-adrenoceptor activation augments acetylcholine release from tracheal parasympathetic nerves.
Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Atropine; Electric Stimulation; Horses; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Parasympathetic Nervous System; Propanolamines; Receptors, Adrenergic, beta-2; Trachea | 1995 |
Molecular analysis of beta-adrenergic receptor subtypes in rat collecting duct: effects on cell cAMP and Ca2+ levels.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Calcium; Cyclic AMP; DNA Primers; Epinephrine; Imidazoles; Isoproterenol; Kidney Cortex; Kidney Tubules, Collecting; Male; Molecular Sequence Data; Mutagenesis; Nephrons; Norepinephrine; Pindolol; Polymerase Chain Reaction; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; RNA, Messenger | 1995 |
Cardiovascular effects of clenbuterol are beta 2-adrenoceptor-mediated in steers.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Blood Glucose; Blood Pressure; Cardiovascular Physiological Phenomena; Cardiovascular System; Cattle; Clenbuterol; Dose-Response Relationship, Drug; Heart Atria; Heart Rate; Imidazoles; Infusions, Intravenous; Isoproterenol; Male; Norepinephrine; Potassium; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1995 |
Beta-adrenergic regulation of action potentials and automaticity in young and adult canine purkinje fibers.
Topics: Action Potentials; Adrenergic beta-Antagonists; Aging; Albuterol; Animals; Cardiac Pacing, Artificial; Dogs; Imidazoles; In Vitro Techniques; Isoproterenol; Propanolamines; Purkinje Fibers; Receptors, Adrenergic, beta | 1994 |
Beta 2-adrenergic receptor actions in neonatal and adult rat ventricular myocytes.
Topics: Age Factors; Animals; Animals, Newborn; Calcium; Cells, Cultured; Cyclic AMP; Ethanolamines; Imidazoles; Isoproterenol; Male; Myocardial Contraction; Myocardium; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1995 |
Beta-adrenoceptor subtypes and the opening of plasmalemmal K(+)-channels in trachealis muscle: electrophysiological and mechanical studies in guinea-pig tissue.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Benzopyrans; Cell Membrane; Cromakalim; Electrophysiology; Female; Guinea Pigs; Heart; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Myocardium; Norepinephrine; Potassium Channels; Procaterol; Propanolamines; Pyrroles; Receptors, Adrenergic, beta; Rubidium Radioisotopes; Salmeterol Xinafoate; Trachea | 1993 |
Transcriptional modulation by n-butyric acid of beta 1-, beta 2-, and beta 3-adrenergic receptor balance in 3T3-F442A adipocytes.
Topics: 3T3 Cells; Adenylyl Cyclase Inhibitors; Adipocytes; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Animals; Base Sequence; Butyrates; Butyric Acid; DNA Primers; DNA, Complementary; Ethanolamines; Gene Expression Regulation; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Molecular Sequence Data; Oligonucleotides, Antisense; Pindolol; Polymerase Chain Reaction; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Transcription, Genetic | 1994 |
Agonist-induced effects on cyclic AMP metabolism are affected in pigment epithelial cells of the Royal College of Surgeons rat.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprostadil; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dinoprostone; Fibroblast Growth Factor 2; Imidazoles; Isoproterenol; Kinetics; Melatonin; Pigment Epithelium of Eye; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta-2; Receptors, Purinergic P1; Serotonin | 1995 |
Early alterations in the brown adipose tissue adenylate cyclase system of pre-obese Zucker rat fa/fa pups: decreased G-proteins and beta 3-adrenoceptor activities.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Animals, Suckling; Base Sequence; Female; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Imidazoles; Isoproterenol; Male; Molecular Sequence Data; Norepinephrine; Obesity; Rats; Rats, Zucker; Receptors, Adrenergic, beta; RNA, Messenger | 1995 |
Determination of beta-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective beta-antagonists.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cyclic AMP; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Membranes; Myocardium; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Tritium | 1995 |
Effects of chronic infusion of (-)-isoprenaline on rat cardiac muscarinic (M2)-cholinoceptors and beta 1- and beta 2-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Binding, Competitive; Down-Regulation; Heart Ventricles; Imidazoles; Infusion Pumps, Implantable; Isoproterenol; Male; Myocardium; N-Methylscopolamine; Pindolol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Scopolamine Derivatives | 1995 |
Targeted disruption of the mouse beta1-adrenergic receptor gene: developmental and cardiovascular effects.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Cell Membrane; Chimera; Crosses, Genetic; Death; Female; Gene Expression; Heart; Heart Rate; Heart Ventricles; Homozygote; Imidazoles; Isoproterenol; Kinetics; Lung; Male; Methoxyhydroxyphenylglycol; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Knockout; Myocardial Contraction; Myocardium; Norepinephrine; Receptors, Adrenergic, beta-1; Restriction Mapping; Stem Cells | 1996 |
Inducible expression of beta 1- and beta 2-adrenergic receptors in rat C6 glioma cells: functional interactions between closely related subtypes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Epinephrine; Gene Expression Regulation, Neoplastic; Genomic Library; Glioma; Imidazoles; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Norepinephrine; Pindolol; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Transfection; Tumor Cells, Cultured | 1996 |
Opposite modulation of noradrenaline and ATP release in guinea-pig vas deferens through prejunctional beta-adrenoceptors: evidence for the beta 2 subtype.
Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Imidazoles; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Norepinephrine; Prazosin; Propanolamines; Receptors, Adrenergic, beta-2; Suramin; Terbutaline; Vas Deferens | 1996 |
The influence of hyperthyroidism on beta-adrenoceptor-mediated relaxation of isolated small mesenteric arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Colforsin; Dose-Response Relationship, Drug; Hyperthyroidism; Imidazoles; Isoproterenol; Male; Mesenteric Arteries; Methoxamine; Muscle Contraction; Muscle Relaxation; Propanolamines; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Wistar; Thromboxane A2; Thyroxine; Vascular Resistance; Vasoconstrictor Agents | 1996 |
Sino-aortic denervation causes right atrial beta adrenoceptor down-regulation.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Down-Regulation; Heart Atria; Heart Rate; Imidazoles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Male; Muscle Denervation; Myocardium; Neurons; Norepinephrine; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Sinoatrial Node | 1997 |
Right ventricular infundibular beta-adrenoceptor complex in tetralogy of Fallot patients.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Child; Child, Preschool; Colforsin; Female; Guanosine Triphosphate; Heart Ventricles; Humans; Hypoxia; Imidazoles; In Vitro Techniques; Infant; Isoproterenol; Male; Myocardium; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sodium Fluoride; Tetralogy of Fallot | 1997 |
Localized cAMP-dependent signaling mediates beta 2-adrenergic modulation of cardiac excitation-contraction coupling.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium; Calcium Channels; Calcium Channels, L-Type; Colforsin; Cyclic AMP; Ethanolamines; Heart; Heart Ventricles; Imidazoles; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic, beta-2; Signal Transduction; Thionucleotides | 1997 |
Beta2-adrenergic receptor antagonists protect against ventricular fibrillation: in vivo and in vitro evidence for enhanced sensitivity to beta2-adrenergic stimulation in animals susceptible to sudden death.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium; Cells, Cultured; Cyclic AMP; Death, Sudden; Dogs; Ethanolamines; Exercise Test; Imidazoles; Isoproterenol; Muscle Fibers, Skeletal; Myocardial Ischemia; Myocardium; Propanolamines; Sensitivity and Specificity; Ventricular Fibrillation | 1997 |
Formoterol and isoproterenol induce c-fos gene expression in osteoblast-like cells by activating beta2-adrenergic receptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DNA, Complementary; Enzyme Activation; Ethanolamines; Formoterol Fumarate; Gene Expression; Genes, fos; Genes, Immediate-Early; Humans; Imidazoles; Isoproterenol; Osteoblasts; Propanolamines; Rats; Receptors, Adrenergic, beta-2; Tumor Cells, Cultured | 1998 |
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1998 |
Relaxation of isolated human myometrial muscle by beta2-adrenergic receptors but not beta1-adrenergic receptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Female; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Myometrium; Potassium Chloride; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1998 |
Characterisation of beta2-adrenoceptors, using the agonist [11C]formoterol and positron emission tomography.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbon Radioisotopes; Ethanolamines; Formoterol Fumarate; Imidazoles; Isoproterenol; Male; Metabolic Clearance Rate; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta-2; Tissue Distribution; Tomography, Emission-Computed | 1998 |
Effects of beta2-adrenergic stimulation on single-channel gating of rat cardiac L-type Ca2+ channels.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium Channels; Calcium Channels, L-Type; Drug Combinations; Electrophysiology; Ethanolamines; Imidazoles; Ion Channel Gating; Isoproterenol; Male; Myocardium; Propanolamines; Rats; Rats, Wistar | 1999 |
Functional and molecular biological evidence for a possible beta3-adrenoceptor in the human detrusor muscle.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colforsin; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 1999 |
Selective activation of beta3-adrenoceptors by octopamine: comparative studies in mammalian fat cells.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adult; Animals; Binding, Competitive; Biogenic Amines; Bupranolol; CHO Cells; Cricetinae; Dioxoles; Dogs; Ethanolamines; Female; Gene Expression; Guinea Pigs; Humans; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lipolysis; Male; Mammals; Mesocricetus; Norepinephrine; Octopamine; Oxygen Consumption; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Species Specificity | 1999 |
Modulation of the pacemaker current If by beta-adrenoceptor subtypes in ventricular myocytes isolated from hypertensive and normotensive rats.
Topics: Action Potentials; Adenosine; Adrenergic alpha-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Cardiomegaly; Catecholamines; GTP-Binding Protein alpha Subunits, Gi-Go; Hypertension; Imidazoles; Isoproterenol; Male; Myocardium; Norepinephrine; Patch-Clamp Techniques; Pertussis Toxin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Virulence Factors, Bordetella | 1999 |
Coupling efficiencies of beta 1- and beta 2-adrenergic receptors expressed alone or together in transfected GH3 pituitary cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Imidazoles; Iodine Radioisotopes; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Pindolol; Pituitary Gland, Anterior; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection | 1999 |
Constitutively active mutants of the beta1-adrenergic receptor.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Betaxolol; Carbazoles; Carvedilol; Cell Line; Cyclic AMP; Epinephrine; Humans; Imidazoles; Isoproterenol; Labetalol; Point Mutation; Practolol; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Timolol | 1999 |
Opposing effects of beta(1)- and beta(2)-adrenergic receptors on cardiac myocyte apoptosis : role of a pertussis toxin-sensitive G protein.
Topics: Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Apoptosis; Carbachol; Cardiotonic Agents; Cyclic AMP; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Imidazoles; Isoproterenol; Male; Muscarinic Agonists; Myocardium; Pertussis Toxin; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Second Messenger Systems; Virulence Factors, Bordetella | 1999 |
Myocardial beta-adrenoceptor down-regulation by norepinephrine is linked to reduced norepinephrine uptake activity.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Colforsin; Dobutamine; Dogs; Down-Regulation; Enzyme Activation; Guanylyl Imidodiphosphate; Heart Ventricles; Hemodynamics; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Myocardial Contraction; Norepinephrine; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Ventricular Function | 1999 |
Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Bupranolol; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Substrate Specificity; Vasodilator Agents | 2000 |
Nitric oxide-dependent vasodilatation of rabbit femoral artery by beta(2)-adrenergic stimulation or cyclic AMP elevation in vivo.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Bucladesine; Colforsin; Cyclic AMP; Enzyme Inhibitors; Femoral Artery; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Tonus; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Propanolamines; Rabbits; Vasodilation | 2000 |
Negative inotropic effects of isoprenaline on isolated left atrial assays from aged transgenic mice with cardiac over-expression of human beta(2)-adrenoceptors.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Aging; Animals; Atrial Function; Cardiotonic Agents; Dose-Response Relationship, Drug; Gene Expression Regulation; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Mice; Mice, Transgenic; Myocardial Contraction; Propanolamines; Receptors, Adrenergic, beta-2 | 2000 |
Functional evidence for a cyclic-AMP related mechanism of action of the beta(2)-adrenoceptor in human ventricular myocytes.
Topics: Adrenergic beta-Antagonists; Adult; Aged; Carbachol; Cardiotonic Agents; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Female; Heart Ventricles; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Receptors, Adrenergic, beta-2 | 2000 |
Functional assessment of beta adrenoceptor subtypes in human colonic circular and longitudinal (taenia coli) smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Colon; Female; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Terbutaline; Tetrahydronaphthalenes | 2000 |
Beta-adrenergic responses are significantly enhanced in rat carotid artery with intimal hyperplasia.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carotid Artery Injuries; Dose-Response Relationship, Drug; Drug Interactions; Electromyography; Hyperplasia; Imidazoles; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Propanolamines; Rats; Rats, Wistar | 2000 |
beta(1) and beta(2)-adrenergic receptor subtype effects in German shepherd dogs with inherited lethal ventricular arrhythmias.
Topics: Action Potentials; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Death, Sudden, Cardiac; Dog Diseases; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Microelectrodes; Myocardium; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Tachycardia, Ventricular | 2000 |
beta(1)- and beta(3)-adrenoceptor mediated smooth muscle relaxation in hypothyroid rat ileum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Hypothyroidism; Ileum; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; RNA, Messenger | 2001 |
Characterization of beta(1)-selectivity, adrenoceptor-G(s)-protein interaction and inverse agonism of nebivolol in human myocardium.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Benzopyrans; COS Cells; Ethanolamines; GTP-Binding Protein alpha Subunits, Gs; Guanylyl Imidodiphosphate; Heart; Humans; Imidazoles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Myocardial Contraction; Myocardium; Nebivolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Transfection | 2001 |
Different mechanisms mediate beta adrenoceptor stimulated vasorelaxation of coronary and femoral arteries.
Topics: Adrenergic beta-Antagonists; Animals; Arteries; Coronary Vessels; Endothelium, Vascular; Female; Femoral Artery; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; omega-N-Methylarginine; Propanolamines; Swine; Vasodilation | 2000 |
Murine ventricular L-type Ca(2+) current is enhanced by zinterol via beta(1)-adrenoceptors, and is reduced in TG4 mice overexpressing the human beta(2)-adrenoceptor.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Barium; Binding Sites; Calcium; Calcium Channels, L-Type; Electric Conductivity; Ethanolamines; GTP-Binding Protein alpha Subunits, Gi-Go; Heart Ventricles; Humans; Imidazoles; Ion Channel Gating; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Myocardium; Pertussis Toxin; Propanolamines; Protein Binding; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Virulence Factors, Bordetella | 2001 |
The effect of streptozotocin-induced diabetes on cardiac beta-adrenoceptor subtypes in the rat.
Topics: Adrenergic beta-Agonists; Animals; Binding Sites; Blood Glucose; Blood Pressure; Body Weight; Diabetes Mellitus, Experimental; Dihydroalprenolol; Heart Rate; Imidazoles; Isoproterenol; Male; Myocardium; Perfusion; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Streptozocin | 2001 |
Nebivolol, bucindolol, metoprolol and carvedilol are devoid of intrinsic sympathomimetic activity in human myocardium.
Topics: Adrenergic beta-Antagonists; Benzopyrans; Binding, Competitive; Bisoprolol; Carbazoles; Carvedilol; Ethanolamines; Female; Guanylyl Imidodiphosphate; Heart Ventricles; Humans; Imidazoles; In Vitro Techniques; Inhibitory Concentration 50; Isoproterenol; Male; Metoprolol; Middle Aged; Myocardial Contraction; Myocardium; Nebivolol; Propanolamines; Substrate Specificity; Sympathetic Nervous System; Sympathomimetics; Thermodynamics | 2001 |
Rapid component I(Kr) of the guinea-pig cardiac delayed rectifier K(+) current is inhibited by beta(1)-adrenoreceptor activation, via cAMP/protein kinase A-dependent pathways.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbazoles; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Enzyme Inhibitors; Guinea Pigs; Imidazoles; Indoles; Isoproterenol; Myocardium; Patch-Clamp Techniques; Potassium Channels, Inwardly Rectifying; Pyrroles; Xamoterol | 2002 |
Pharmacological characterisation of the beta-adrenoceptor expressed by human lung mast cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Dose-Response Relationship, Drug; Humans; Imidazoles; Isoproterenol; Lung; Mast Cells; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta | 2002 |
Toxic cardiac effects of catecholamines: role of beta-adrenoceptor downregulation.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Blood Pressure; Down-Regulation; Fibrosis; Heart Rate; Heart Ventricles; Imidazoles; Isoproterenol; Male; Muscle Contraction; Myocardial Infarction; Papillary Muscles; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 2002 |
Cardiostimulant and cardiodepressant effects through overexpressed human beta2-adrenoceptors in murine heart: regional differences and functional role of beta1-adrenoceptors.
Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Mice; Mice, Transgenic; Myocardial Contraction; Norepinephrine; Pertussis Toxin; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2003 |
Cardiac-specific overexpression of human beta2 adrenoceptors in mice exposes coupling to both Gs and Gi proteins.
Topics: Adrenergic beta-Antagonists; Animals; Atrial Function, Left; Female; Gene Expression; Genotype; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Humans; Imidazoles; Isoproterenol; Male; Mice; Mice, Transgenic; Models, Theoretical; Pertussis Toxin; Propanolamines; Receptors, Adrenergic, beta-2 | 2003 |
Role of beta-adrenoceptor subtypes in mediating relaxation of the pig bladder trigonal muscle in vitro.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Swine; Urinary Bladder | 2003 |
The third intracellular loop and the carboxyl terminus of beta2-adrenergic receptor confer spontaneous activity of the receptor.
Topics: Adrenergic beta-Antagonists; Animals; Cells, Cultured; Cyclic AMP; Imidazoles; Isoproterenol; Mice; Myocardial Contraction; Myocardium; Propanolamines; Protein Conformation; Protein Structure, Tertiary; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Signal Transduction; Subcellular Fractions | 2003 |
The functional role of beta-adrenoceptor subtypes in mediating relaxation of pig urethral smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Ethanolamines; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Swine; Urethra | 2003 |
Involvement of the serotonin 5-HT2B receptor in cardiac hypertrophy linked to sympathetic stimulation: control of interleukin-6, interleukin-1beta, and tumor necrosis factor-alpha cytokine production by ventricular fibroblasts.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Cardiomegaly; Cells, Cultured; Drug Evaluation, Preclinical; Fibroblasts; Gene Expression Regulation; Heart Ventricles; Imidazoles; Indoles; Interleukin-1; Interleukin-6; Isoproterenol; Mice; Mice, Knockout; Myocytes, Cardiac; Propanolamines; Pyridines; Quinolines; Receptor, Serotonin, 5-HT2B; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Sympathetic Nervous System; Sympathomimetics; Tumor Necrosis Factor-alpha | 2004 |
Natriuretic peptide gene expression after beta-adrenergic stimulation in adult mouse cardiac myocytes.
Topics: Adrenergic beta-Antagonists; Animals; Atrial Natriuretic Factor; Cells, Cultured; Gene Expression; Imidazoles; In Situ Nick-End Labeling; Isoproterenol; Mice; Myocytes, Cardiac; Natriuretic Peptide, Brain; Nerve Tissue Proteins; Propanolamines; RNA, Messenger | 2004 |
Beta3-adrenoceptors: relaxant function and mRNA detection in smooth muscle cells isolated from the human colon.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Colon; Gastrointestinal Motility; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Myocytes, Smooth Muscle; Propranolol; Receptors, Adrenergic, beta-3; RNA, Messenger; Tetrahydronaphthalenes | 2004 |
Pharmacological modulation of the hyperpolarization-activated current (I f) in human atrial myocytes: focus on G protein-coupled receptors.
Topics: Aged; Arrhythmias, Cardiac; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Ion Transport; Isoproterenol; Male; Membrane Potentials; Middle Aged; Myocytes, Cardiac; Patch-Clamp Techniques; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, G-Protein-Coupled; Receptors, Serotonin, 5-HT4; Serotonin | 2005 |
Evidence for two atypical conformations of beta-adrenoceptors and their interaction with Gi proteins.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Norepinephrine; Pertussis Toxin; Propanolamines; Protein Binding; Protein Conformation; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1 | 2005 |
Beta1-adrenergic receptors maintain fetal heart rate and survival.
Topics: Adrenergic beta-Antagonists; Animals; Fetal Heart; Fetal Hypoxia; Heart Rate, Fetal; Imidazoles; Isoproterenol; Mice; Mice, Inbred ICR; Mice, Knockout; Organ Culture Techniques; Oxygen; Receptors, Adrenergic, beta-1; Survival Rate; Tyrosine 3-Monooxygenase | 2006 |
Neural contractions in colonic strips from patients with diverticular disease: role of endocannabinoids and substance P.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Case-Control Studies; Colon; Diverticulum; Endocannabinoids; Female; Glycerides; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Morpholines; Muscle Contraction; Muscle, Smooth; Naphthalenes; Neurokinin-1 Receptor Antagonists; Piperidines; Polyunsaturated Alkamides; Propanolamines; Pyrazoles; Quinuclidines; Rimonabant; Substance P; Tetrodotoxin | 2006 |
Functional beta-adrenergic receptor signalling on nuclear membranes in adult rat and mouse ventricular cardiomyocytes.
Topics: Adenylyl Cyclases; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blotting, Western; Dioxoles; Ethanolamines; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Microscopy, Confocal; Myocytes, Cardiac; Nuclear Envelope; Pertussis Toxin; Propanolamines; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Signal Transduction | 2006 |
kappa-opioid receptor stimulation inhibits cardiac hypertrophy induced by beta1-adrenoceptor stimulation in the rat.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Calcium; Cardiomegaly; Cell Size; Cells, Cultured; Imidazoles; Isoproterenol; Leucine; Myocytes, Cardiac; Propanolamines; Proteins; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa | 2007 |
Adrenergic control of a constitutively active acetylcholine-regulated potassium current in canine atrial cardiomyocytes.
Topics: Acetylcholine; Action Potentials; Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Bee Venoms; Clonidine; Cyclic AMP-Dependent Protein Kinases; Dihydropyridines; Dogs; Dose-Response Relationship, Drug; Estrenes; Heart Atria; Imidazoles; Indoles; Isoproterenol; Isoquinolines; Maleimides; Myocytes, Cardiac; Patch-Clamp Techniques; Phenylephrine; Phorbol 12,13-Dibutyrate; Piperazines; Potassium Channels; Prazosin; Propanolamines; Propranolol; Protein Kinase C; Pyrrolidinones; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Sulfonamides; Type C Phospholipases | 2007 |
Downregulation of CuZn-superoxide dismutase contributes to beta-adrenergic receptor-mediated oxidative stress in the heart.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Animals; Apoptosis; Blotting, Western; Cell Line; DNA; Down-Regulation; ets-Domain Protein Elk-1; Glutathione; Imidazoles; Immunohistochemistry; Isoproterenol; Male; Myocardium; Oxidative Stress; Rats; Rats, Wistar; Receptors, Adrenergic, beta; RNA Interference; RNA, Messenger; RNA, Small Interfering; Stimulation, Chemical; Superoxide Dismutase; YY1 Transcription Factor | 2007 |
Phosphodiesterase-4 blunts inotropism and arrhythmias but not sinoatrial tachycardia of (-)-adrenaline mediated through mouse cardiac beta(1)-adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiotonic Agents; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Dose-Response Relationship, Drug; Drug Synergism; Epinephrine; Female; Heart Atria; Heart Rate; Heart Ventricles; Imidazoles; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Myocardial Contraction; Myocytes, Cardiac; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Propanolamines; Quinolones; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Rolipram; Sinoatrial Node; Tachycardia, Sinus; Tachycardia, Ventricular | 2008 |
Deciphering the beta-adrenergic response in human embryonic stem cell-derived-cardiac myocytes: closer to clinical use?
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbachol; Cell Differentiation; Cell Line; Cell Lineage; Dose-Response Relationship, Drug; Embryonic Stem Cells; Heart Failure; Humans; Imidazoles; Isoproterenol; Muscarinic Agonists; Myocardial Contraction; Myocytes, Cardiac; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Stem Cell Transplantation | 2008 |
beta(1)- and beta(2)-adrenoceptor responses in cardiomyocytes derived from human embryonic stem cells: comparison with failing and non-failing adult human heart.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Animals; Carbachol; Cell Differentiation; Cell Line; Cell Lineage; Dose-Response Relationship, Drug; Embryonic Stem Cells; Heart Failure; Humans; Imidazoles; Isoproterenol; Mice; Muscarinic Agonists; Myocardial Contraction; Myocytes, Cardiac; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Stem Cell Transplantation; Time Factors | 2008 |
Beta1-adrenoceptors in rat anterior pituitary may be constitutively active. Inverse agonism of CGP 20712A on basal 3',5'-cyclic adenosine 5'-monophosphate levels.
Topics: Adenylyl Cyclases; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Animals; Carbazoles; Carvedilol; Cell Aggregation; Cells, Cultured; Cyclic AMP; Drug Inverse Agonism; Enzyme Activation; Imidazoles; Isoproterenol; Male; Pertussis Toxin; Pituitary Gland, Anterior; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Substrate Specificity | 2008 |
Mouse embryonic stem cell-derived cardiomyocytes express functional adrenoceptors.
Topics: Animals; Cell Differentiation; Cell Line; Embryonic Stem Cells; Extracellular Signal-Regulated MAP Kinases; Gene Expression; Imidazoles; Isoproterenol; Mice; Myocytes, Cardiac; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptor, Muscarinic M2; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Tyrosine 3-Monooxygenase | 2008 |
Regulation of gap-junction protein connexin 43 by beta-adrenergic receptor stimulation in rat cardiomyocytes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Cells, Cultured; Connexin 43; Cyclic AMP-Dependent Protein Kinases; Gap Junctions; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Imidazoles; Isoproterenol; Myocytes, Cardiac; Pertussis Toxin; Propranolol; Protein Isoforms; Protein Phosphatase 2; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Signal Transduction | 2009 |
Effects of β-adrenoceptor stimulation on delayed rectifier K(+) currents in canine ventricular cardiomyocytes.
Topics: Action Potentials; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Delayed Rectifier Potassium Channels; Dogs; Heart Ventricles; Imidazoles; Isoproterenol; Kinetics; Metoprolol; Myocytes, Cardiac; Patch-Clamp Techniques; Protein Kinase Inhibitors; Receptors, Adrenergic, beta-1; Signal Transduction; Single-Cell Analysis | 2011 |
[Effects of overexpression of beta2-adrenoceptor on contraction in cardiac myocytes isolated from failure hearts of rats].
Topics: Adenoviridae; Adrenergic beta-Antagonists; Animals; Cells, Cultured; Heart Failure; Humans; Imidazoles; Isoproterenol; Male; Myocardial Contraction; Myocytes, Cardiac; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2 | 2007 |
Predicting in vivo cardiovascular properties of β-blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiovascular Agents; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Heart Rate; Humans; Imidazoles; Isoproterenol; Male; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Rats; Rats, Sprague-Dawley; Vascular Resistance; Xamoterol | 2011 |
β2-adrenoceptor transfection enhances contractile reserve of isolated rat ventricular myocytes exposed to chronic isoprenaline stimulation by improving β1-adrenoceptor responsiveness.
Topics: Adrenergic beta-Antagonists; Animals; Gene Transfer Techniques; Genetic Therapy; Heart Failure; Imidazoles; Isoproterenol; Myocardial Contraction; Myocytes, Cardiac; Primary Cell Culture; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 2012 |
Role of β-adrenergic receptors in regulation of hepatic fat accumulation during aging.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Cells, Cultured; Enzyme Activation; Fats; Hepatocytes; Imidazoles; Isoproterenol; Lipids; Liver; Male; Mice; Mice, Inbred C57BL; Propanolamines; Propranolol; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction; Time Factors | 2012 |
Exchange protein directly activated by cAMP mediates slow delayed-rectifier current remodeling by sustained β-adrenergic activation in guinea pig hearts.
Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Calcineurin; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Delayed Rectifier Potassium Channels; Egtazic Acid; Guanine Nucleotide Exchange Factors; Guinea Pigs; Hypertrophy, Left Ventricular; Imidazoles; Ion Channel Gating; Isoproterenol; Myocytes, Cardiac; NFATC Transcription Factors; Patch-Clamp Techniques; Potassium; Propanolamines; Receptors, Adrenergic, beta-1; RNA Interference; RNA, Small Interfering; Second Messenger Systems | 2014 |
Mucosa of murine detrusor impairs β2 -adrenoceptor-mediated relaxation.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Aminophenols; Animals; Colforsin; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mucous Membrane; Muscle Relaxation; Muscle, Smooth; Potassium Chloride; Sulfonamides; Urinary Bladder; Vasodilator Agents | 2015 |
Aberrant α-adrenergic hypertrophic response in cardiomyocytes from human induced pluripotent cells.
Topics: Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cell Line; Cell Size; Embryonic Stem Cells; Gene Expression; Humans; Hypertrophy; Imidazoles; Induced Pluripotent Stem Cells; Isoproterenol; Microscopy, Confocal; Myocytes, Cardiac; Phenylephrine; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction | 2014 |
β-Adrenoceptor-Mediated Relaxation of Carbachol-Pre-Contracted Mouse Detrusor.
Topics: Aminophenols; Animals; Carbachol; Cholinergic Agonists; Colforsin; Homozygote; Imidazoles; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mucous Membrane; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Sulfonamides; Urinary Bladder | 2015 |
Beta1-adrenergic receptor-mediated dilation of rat cerebral artery requires Shaker-type KV1 channels on PSD95 scaffold.
Topics: Adrenergic beta-Antagonists; Animals; Cerebral Arteries; Disks Large Homolog 4 Protein; Imidazoles; Intracellular Signaling Peptides and Proteins; Isoproterenol; Male; Membrane Proteins; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Shaker Superfamily of Potassium Channels; Vasoconstrictor Agents; Vasodilation | 2015 |
Phosphorylation of Ser1928 mediates the enhanced activity of the L-type Ca2+ channel Cav1.2 by the β2-adrenergic receptor in neurons.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium Channels, L-Type; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Female; Imidazoles; Isoproterenol; Long-Term Potentiation; Male; Mice, 129 Strain; Mice, Inbred C57BL; Mice, Transgenic; Myocytes, Cardiac; Neuronal Plasticity; Neurons; Phosphorylation; Propanolamines; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2; Serine; Signal Transduction | 2017 |
β
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Diabetes Mellitus, Type 2; Heart; Heart Rate; Imidazoles; Isolated Heart Preparation; Isoproterenol; Male; Myocardium; Rats; Rats, Zucker; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction | 2019 |