isoproterenol has been researched along with cgp 12177 in 197 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 52 (26.40) | 18.7374 |
| 1990's | 100 (50.76) | 18.2507 |
| 2000's | 40 (20.30) | 29.6817 |
| 2010's | 4 (2.03) | 24.3611 |
| 2020's | 1 (0.51) | 2.80 |
| Authors | Studies |
|---|---|
| Guillaume, JL; Méjean, A; Strosberg, AD | 1 |
| Arch, JR; Henson, SM; Kaumann, AJ; Kelly, J; Molenaar, P; Sarsero, D | 1 |
| Charlton, SJ; Dickson, CJ; Duca, JS; Fairhurst, RA; Hornak, V; McKay, DJ; Pearlstein, RA; Reilly, J; Sandham, DA; Shaw, D; Sykes, DA; Velez-Vega, C | 1 |
| Dauzats, M; Lafontan, M; Langin, D; Portillo, M | 1 |
| Van Liefde, I; Van Witzenburg, A; Vauquelin, G | 2 |
| Johansson, LH; Persson, H; Rosengren, E | 1 |
| Morin, D; Sapena, R; Tillement, JP; Urien, S; Zini, R | 1 |
| Kaneko, M; Kawashima, Y; Matsuda, H; Sakagoshi, N; Sawa, Y; Watanabe, Y; Yoshida, H | 1 |
| Litthauer, D; Oelofsen, W; van de Venter, M | 1 |
| Horackova, M; Wilkinson, M | 1 |
| Berlan, M; Bousquet-Melou, A; Galitzky, J; Montastruc, JL; Tavernier, G | 1 |
| Fraeyman, N; Van de Velde, E; Van Ermen, A; Vanscheeuwijck, P | 1 |
| Baude, B; Emorine, LJ; Fève, B; Krief, S; Pairault, J; Strosberg, AD | 1 |
| Behlke, J; Boehmer, FD; Engstroem, U; Grosse, R; Hollenberg, M; Kuehn, H; Langen, P; Wallukat, G | 1 |
| Moon, TW; Perry, SF; Reid, SD | 1 |
| Duman, RS; Fishman, PH; Nussbaum, E | 1 |
| Matheny, M; Scarpace, PJ | 1 |
| Collins, P; Johnson, A; O'Donnell, L; Owens, D; Tomkin, GH | 1 |
| Bouanani, N; Corsin, A; Crozatier, B; Gilson, N | 1 |
| Lafontan, M; Langin, D; Portillo, MP; Saulnier-Blache, JS | 1 |
| Leysen, JE; Pauwels, PJ; Van Gompel, P | 1 |
| Couraud, PO; Durieu-Trautmann, O; Foignant-Chaverot, N; Gounon, P; Perdomo, J; Strosberg, AD | 1 |
| Limas, C; Limas, CJ | 2 |
| Endoh, M; Ishihata, A; Norota, I; Satoh, H; Shibasaki, T | 1 |
| Olson, MF; Pon, DJ; Schimmer, BP; Tsao, J | 1 |
| Böhm, M; Erdmann, E; Schwinger, RH | 1 |
| Eliasson, EL; Johansson, LH; Persson, H; Rosengren, E | 1 |
| Gierschik, P; Jakobs, KH; Müller, U; Reithmann, C; Werdan, K | 1 |
| Hirsch, DJ; Morgunov, NS | 1 |
| Baldi, G; Bertora, P; Bevilacqua, M; Chebat, E; Norbiato, G; Vago, T | 1 |
| Johansen, O; Mjøs, OD; Sager, G | 1 |
| Bouscarel, B; Cortinovis, C; Mayer, D; Murat, JC; Paris, H | 1 |
| Creese, I; Riva, MA | 1 |
| Abrass, IB; Allen, JM; Palmiter, RD | 1 |
| Feldman, RD | 1 |
| Iwasaki, T; Kawamoto, H; Matsumori, Y; Ohyanagi, M; Shibata, R | 1 |
| Korichneva, IL; Krasnikova, TL; Radiukhin, VA | 1 |
| Cardone, F; Cignarelli, M; Corso, M; De Pergola, G; Di Paolo, S; Garruti, G; Giorgino, R; Nardelli, G | 1 |
| Labouesse, J; Pianet, I; Teissié, J; Volker, TT | 1 |
| Hui, KK; Yu, JL | 1 |
| Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
| Kim, D; Margolis, TI; Marsh, JD | 1 |
| Choi, AH; Lee, PW | 1 |
| Aarbakke, J; Bang, BE; Pedersen, M; Sager, G | 1 |
| Reithmann, C; Werdan, K | 1 |
| Porzig, H; Reuter, H | 1 |
| Wilkinson, DA; Wilkinson, M | 1 |
| Brinkmann, M; Brodde, OE; Wang, XL | 1 |
| De Blasi, A; Fratelli, M; Insel, PA; Lipartiti, M; Motulsky, HJ | 1 |
| Cotecchia, S; De Blasi, A; Fratelli, M; Lipartiti, M | 1 |
| Anakwe, OO; Moger, WH; Murphy, PR | 1 |
| Hertel, C; Portenier, M; Staehelin, M | 1 |
| Feldman, RD; Motulsky, HJ; Thede-Reynolds, KR | 1 |
| Molinoff, PB; Reynolds, EE | 1 |
| Cervantes-Olivier, P; Delavier-Klutchko, C; Desmandril, M; Durieu-Trautmann, O; Kaveri, S; Strosberg, AD | 1 |
| Hiramatsu, Y; Nezu, E; Yoneyama, T; Yoshimura, K | 1 |
| Agli, B; Giudicelli, Y; Lacasa, D | 1 |
| Lang, PH; Lemmer, B | 1 |
| Coulter, SJ; Hertel, C; Perkins, JP | 1 |
| Levin, BE; Sullivan, AC | 1 |
| Giudicelli, Y; Leneveu, MC; Pecquery, R | 1 |
| Cunningham, EM; DeBlasi, A; Insel, PA; Motulsky, HJ | 1 |
| Algeri, S; Costantini, C; Cotecchia, S; De Blasi, A; Fratelli, M; Lipartiti, M; Sacchetti, G | 1 |
| Watson-Wright, WM; Wilkinson, M | 1 |
| Fishman, PH; Kassis, S; Olasmaa, M; Sullivan, M | 1 |
| Arinze, IJ; Graham, SM; Kawai, Y; Yoshioka, H | 1 |
| De Blasi, A; Fratelli, M; Lipartiti, M; Wielosz, M | 1 |
| Marsh, JD; Roberts, DJ | 1 |
| Lang, CH; McDonough, KH; Shepherd, RE | 1 |
| Box, RJ; Staehelin, M | 1 |
| Gjerde, I; Jacobsen, S; Refsnes, M; Sandnes, D | 1 |
| Harden, TK; Perkins, JP; Toews, ML; Waldo, GL | 1 |
| Hertel, C; Perkins, JP | 1 |
| Clementi, F; Sher, E | 1 |
| Hertel, C; Müller, P; Portenier, M; Staehelin, M | 2 |
| Montandon, JB; Porzig, H | 1 |
| Baer, M; Chanton, C; Porzig, H | 1 |
| Hertel, C; Staehelin, M | 1 |
| Delavier-Klutchko, C; Hoebeke, J; Strosberg, AD | 1 |
| Hertel, C; Perkins, JP; Staehelin, M | 1 |
| Simons, P; Staehelin, M | 1 |
| Horinouchi, T; Koike, K; Takayanagi, I | 1 |
| Langer, L; Lemmer, B; Olbrich, HG; Witte, K | 1 |
| Bouloumie, A; Galitzky, J; Lafontan, M; Langin, D; Remaury, A; Tavernier, G; Valet, P | 1 |
| Bono, M; Calls, J; Cases, A; Esforzado, N; Gaya, J; Jimenez, W; Revert, L; Rivera, F | 1 |
| Bellanger, AC; Buhler, JM; de Rouffignac, C; Dublineau, I; Elalouf, JM; Tessiot, C | 1 |
| Brodde, OE; Elsinga, PH; Vaalburg, W; Van Waarde, A; Visser, GM | 1 |
| Arner, P; Enocksson, S; Lönnqvist, F; Nordenström, J; Shimizu, M | 1 |
| Benovic, JL; Frielle, T; Ledeen, RW; Saito, M | 1 |
| Begin-Heick, N; Ghorbani, M; Himms-Hagen, J; Kates, AL; Triandafillou, J | 1 |
| Carlsson, B; Drvota, V; Häggblad, J; Sylvén, C; Wei, H | 1 |
| Oriowo, MA | 1 |
| Horinouchi, T; Koike, K; Muramatsu, M; Ohki, S; Takayanagi, I | 1 |
| Nunnally, MH; Parker, EM; Perkins, JP; Ross, EM; Swigart, P | 1 |
| Battarbee, HD; O'Donnell, JM; Zavecz, JH | 1 |
| Bronnikov, G; Mohell, N; Nedergaard, J; Unelius, L | 1 |
| Hirsch, DJ; Morgunov, NS; You, YD | 1 |
| Brunello, N; Perez, J; Racagni, G; Rovescalli, AC; Steardo, L; Vitali, S | 1 |
| Sanghani, MP; Scarpace, PJ | 1 |
| Berlan, M; Bousquet-Melou, A; Galitzky, J; Lafontan, M; Montastruc, JL | 1 |
| Change, HT; Chen, CF; Liao, JF | 1 |
| Baumgold, J; Curran, P; Fishman, PH; Zhou, XM | 1 |
| Chaudhry, A; Granneman, JG | 1 |
| Laurent, S; Nicolas, P; Perret, GY; Vassy, R; Yin, Y | 1 |
| Armour, JA; Boudreau, G; Cardinal, R; Watson-Wright, WM; Wilkinson, M | 1 |
| Berlan, M; Carpéné, C; Galitzky, J; Lafontan, M; Portillo, M; Reverte, M | 1 |
| Fujii, N; Homma, S; Ikegami, H; Miyazaki, H | 1 |
| Van Ermen, A; Van Liefde, I; Vauquelin, G | 1 |
| Morin, D; Sapena, R; Tillement, JP; Zini, R | 1 |
| Cowburn, RF; Fowler, CJ; O'Neill, C; Ravid, R; Vestling, M; Winblad, B | 1 |
| Adachi-Akahane, S; Kitagawa, Y; Nagao, T | 1 |
| Cannon, B; Dicker, A; Nedergaard, J | 1 |
| el Borai, N; Ito, K; Nakano, S; Nakazawa, H; Tanaka, E; Yamakawa, A; Yamamura, M | 1 |
| Arner, P; Blaak, E; Hoffstedt, J; Lönnqvist, F; Shimizu, M | 1 |
| el Hadri, K; Fève, B; Pairault, J | 1 |
| Reverte, M; Rivas-Cabañero, L | 1 |
| Barber, R; Carsrud, ND; Clark, RB; Dickey, BF; Knoll, BJ; Millman, EE; Moore, RH; Morrison, KJ; Trial, J; Tuvim, M | 1 |
| Arner, P; Hellström, L; Langin, D; Reynisdottir, S; Rössner, S | 1 |
| Arner, P; Blaak, EE; Gafvels, ME; Lonnqvist, F; Shimizu, M | 1 |
| Chen, CM; Ko, FN; Lin, CH; Teng, CM; Yang, CM | 1 |
| Barbe, P; Berlan, M; Galitzky, J; Hainer, V; Kunesova, M; Lafontan, M; Stich, V | 1 |
| Scarpace, PJ | 1 |
| Baamonde, C; Dierssen, M; Flórez, J; García-Calatayud, S; Lumbreras, MA; Vallina, IF | 1 |
| Chen, J; Fu, D; Javitch, JA; Liapakis, G | 1 |
| Garnier, V; Sapena, R; Tillement, JP; Zini, R | 1 |
| Arner, P; Large, V; Lönnqvist, F; Reynisdottir, S; Thörne, A; Van Harmelen, V; Wennlund, A | 1 |
| Barbe, P; Berlan, M; Crampes, F; De Glisezinski, I; Galitzky, J; Lafontan, M; Riviere, D; Senard, JM; Thalamas, C | 1 |
| Garnier, V; Morin, D; Tillement, JP; Zini, R | 1 |
| Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F | 1 |
| Lisá, V; Myslivecek, J; Trojan, S; Tucek, S | 1 |
| Honjyo, H; Kogure, A; Kondo, M; Sakane, N; Umekawa, T; Yoshida, T | 1 |
| Gerhardt, CC; Gros, J; Issad, T; Strosberg, AD | 1 |
| Bergström, D; Fowler, CJ; Jacobsson, SO | 1 |
| Ajisawa, Y; Akahane, M; Andersson, KE; Hayakawa, K; Igawa, Y; Nishizawa, O; Takeda, H; Yamazaki, Y; Yoneyama, T | 1 |
| Fowler, CJ; Sjöberg, E; Vedin, V | 1 |
| Dai, W; Hall, HS; Knoll, BJ; Moore, RH; Rosenfeld, JL | 1 |
| Adli, H; Bazin, R; Perret, GY | 1 |
| Garnier, V; Tillement, JP; Zini, R | 1 |
| Crema, F; de Ponti, F; Frigo, G; Gibelli, G; Modini, C | 1 |
| Faundez, V; Kelly, RB; Marullo, S | 1 |
| Gao, BB; Han, QD | 1 |
| Fontenot, HJ; Kennedy, RH; Wang, SN; Zhou, W | 1 |
| Farias-Silva, E; Grassi-Kassisse, DM; Spadari-Bratfisch, RC; Wolf-Nunes, V | 1 |
| Grace, AA; Kaumann, AJ; Lowe, MD | 1 |
| Berdeaux, A; Bévérelli, F; Gauthier, C; Le Marec, H; Leblais, V; Rautureau, Y; Trochu, JN | 1 |
| Brown, D; Freestone, NS; Heubach, JF; Kaumann, AJ; Ravens, U; Wettwer, E | 1 |
| Horinouchi, T; Koike, K | 3 |
| Horinouchi, T; Koike, K; Tsujitani, M | 1 |
| Coussin, F; Macrez, N; Mironneau, J; Morel, JL; Viard, P | 1 |
| Kalavantavanich, K; Schramm, CM | 1 |
| Asano, A; Fushiki, T; Kawada, T; Kayahashi, S; Kimura, K; Mizukami, J; Morimatsu, M; Saito, M; Sasaki, N; Yoshida, T | 1 |
| Koike, K; Yamamoto, Y | 1 |
| Ito, M; Nakagawa, M; Saikawa, T; Takahashi, N; Teshima, Y; Yasunaga, S; Yonemochi, H | 1 |
| Brawley, L; MacDonald, A; Shaw, AM | 1 |
| Baamonde, C; Dierssen, M; Flórez, J; García-Calatayud, S; Lumbreras, MA; Martínez-Cué, C; Vallina, IF | 1 |
| Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S | 1 |
| McLean, AJ; Milligan, G | 1 |
| Ajisawa, Y; Akahane, M; Igawa, Y; Komatsu, Y; Nishizawa, O; Takeda, H; Yamazaki, Y | 1 |
| Amusquivar, E; Cacho, J; Herrera, E | 1 |
| Ansonoff, MA; Etgen, AM | 1 |
| Bourin, MC; Crozatier, B; Germack, R; León-Velarde, F; Mohammadi, K; Richalet, JP | 1 |
| Engelhardt, S; Hein, L; Kaumann, AJ; Lohse, M; Molenaar, P | 1 |
| Ambid, L; Atgié, C; Carpéné, C; Casteilla, L; Hanoun, N; Le Gouic, S; Marti, L; Pénicaud, L | 1 |
| Han, S; Kim, JS; Kim, KT; Namgung, U; Suh, BC | 1 |
| Danner, I; Escande, D; Gauthier, C | 1 |
| Ikeda, T; Izawa, T; Komabayashi, T; Suda, K | 1 |
| Bergersen, H; Brennesvik, EO; Brørs, O; Jebens, E; Jensen, J; Oseland, H | 1 |
| Frontera, M; Gianotti, M; Justo, R; Oliver, J; Pujol, E; Roca, P; Rodriguez-Cuenca, S | 1 |
| Horinouchi, T; Koike, K; Tanaka, Y | 1 |
| Colledge, WH; Grace, AA; Joseph, SS; Kaumann, AJ; Lynham, JA; Molenaar, P | 1 |
| Horinouchi, T; Koike, K; Matsushita, M; Tanaka, Y; Tsuru, H | 1 |
| Colledge, WH; Grace, AA; Joseph, SS; Kaumann, AJ; Lynham, JA | 1 |
| Colledge, WH; Joseph, SS; Kaumann, AJ | 1 |
| Kinsella, BT; O'Meara, SJ | 1 |
| Desfontis, JC; Gogny, M; Holopherne, D; Le Coz, O; Mallem, Y; Reculeau, O | 1 |
| Caceres, VM; Krieger, MH; Moreira, MF; Santos, IN; Spadari-Bratfisch, RC; Sumitame, M | 1 |
| Carter, AA; Hill, SJ | 1 |
| Badawi, JK; Bross, S; Haferkamp, A; Hatzinger, M; Michel, MS; Uecelehan, H | 1 |
| Frazier, EP; Michel, MC; Schneider, T | 1 |
| Baranowska, U; Godlewski, G; Malinowska, B; Schlicker, E | 1 |
| Maruyama, T; Matsui, T; Miyata, K; Nagase, I; Sasamata, M; Sato, S; Takasu, T; Uchida, H; Ukai, M; Yamaguchi, O | 1 |
| Kaumann, A; Molenaar, P; Semmler, AB | 1 |
| Advenier, C; Bardou, M; Breuiller-Fouché, M; Cecchi, R; Croci, T; Descamps, L; Fradin, Y; Germain, G; Guagnini, F; Leroy, MJ; Marini, P; Pascal, M; Rouget, C; Viviani, N | 1 |
| Koike, K; Matsushita, M; Tanaka, Y | 1 |
| Badawi, JK; Bross, S; Honeck, P; Kwon, ST; Langbein, S; Seja, T; Uecelehan, H | 1 |
| Galindo-Tovar, A; Kaumann, AJ; Vargas, ML | 1 |
| dos Santos, IN; Spadari-Bratfisch, RC | 1 |
| Alewijnse, AE; Michel, MC; Vrydag, W | 1 |
| Anisuzzaman, AS; Ikeda, T; Itoh, H; Koshiji, T; Muramatsu, I; Nishimune, A; Sasaki, M; Uwada, J; Yoshiki, H | 1 |
| Abdelkrim, MA; Chatagnon, G; Desfontis, JC; Gogny, M; Mallem, MY; Noireaud, J | 1 |
| Gendvilienė, V; Jurevičius, J; Skeberdis, VA; Treinys, R; Zablockaitė, D | 1 |
| Iiboshi, Y; Kasuya, Y; Obara, K; Shigematsu, M; Takahasi, H; Tanaka, Y; Yoshioka, K | 1 |
1 review(s) available for isoproterenol and cgp 12177
| Article | Year |
|---|---|
Receptor-specific mechanisms of desensitization of beta-adrenergic receptor function.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Catecholamines; Cell Line; Concanavalin A; Cyclic AMP; Enzyme Activation; Erythrocytes; Guanosine Triphosphate; Isoproterenol; Kinetics; Models, Biological; Phosphorylation; Propanolamines; Rana catesbeiana; Rana pipiens; Receptors, Adrenergic, beta | 1984 |
196 other study(ies) available for isoproterenol and cgp 12177
| Article | Year |
|---|---|
Carazolol: a potent, selective beta 3-adrenoceptor agonist.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; CHO Cells; Cricetinae; Dithiothreitol; Lipolysis; Propanolamines; Receptors, Adrenergic, beta | 1995 |
Effects of (-)-RO363 at human atrial beta-adrenoceptor subtypes, the human cloned beta 3-adrenoceptor and rodent intestinal beta 3-adrenoceptors.
Topics: Adenylyl Cyclases; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Aged; Animals; Autoradiography; Catechols; CHO Cells; Colon; Cricetinae; Dose-Response Relationship, Drug; Female; Guinea Pigs; Humans; Male; Middle Aged; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1997 |
Uncoupling the Structure-Activity Relationships of β2 Adrenergic Receptor Ligands from Membrane Binding.
Topics: Binding Sites; Cell Membrane; Dose-Response Relationship, Drug; Humans; Ligands; Models, Molecular; Molecular Structure; Receptors, Adrenergic, beta-2; Structure-Activity Relationship | 2016 |
Drop in the "atypical" beta-adrenergic response and modification of the beta/alpha 2-adrenoceptor balance in fat cells from aging rabbits.
Topics: Adipose Tissue; Adrenocorticotropic Hormone; Aging; Animals; Brimonidine Tartrate; Epinephrine; Ethanolamines; In Vitro Techniques; Isoproterenol; Lipolysis; Propanolamines; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1992 |
Multiple beta adrenergic receptor subclasses mediate the l-isoproterenol-induced lipolytic response in rat adipocytes.
Topics: Adipose Tissue; Animals; Dose-Response Relationship, Drug; Ethanolamines; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1992 |
The role of Mg2+ on the formation of the ternary complex between agonist, beta-adrenoceptor, and GS-protein and an interpretation of high and low affinity binding of beta-adrenoceptor agonists.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; GTP-Binding Proteins; Guinea Pigs; Isoproterenol; Lung; Magnesium; Male; Propanolamines; Receptors, Adrenergic, beta | 1992 |
Labelling of rat brain beta-adrenoceptors: (3H)CGP-12177 or (125I)iodocyanopindolol?
Topics: Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Hippocampus; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Male; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Serotonin; Tritium | 1992 |
Alterations in the beta-adrenergic receptor system after hypothermic ischemia in hearts with preischemic beta-receptor desensitization.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Cell Membrane; Heart Ventricles; Hypothermia; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Perfusion; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Tritium | 1992 |
The effect of high concentrations of alpha 2-adrenoceptor antagonists on the lipolytic responsiveness of isolated human adipocytes.
Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Dioxanes; Female; Humans; Idazoxan; Isoproterenol; Lipolysis; Norepinephrine; Propanolamines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1992 |
Characterization of cell-surface beta-adrenergic ([3H]CGP-12177) binding in adult rat ventricular myocytes: lack of regulation by beta-agonists at physiological concentrations.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Down-Regulation; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Myocardium; Norepinephrine; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley | 1992 |
The positive chronotropic effect induced by BRL 37344 and CGP 12177, two beta-3 adrenergic agonists, does not involve cardiac beta adrenoceptors but baroreflex mechanisms.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Animals; Dogs; Ethanolamines; Heart Rate; Isoproterenol; Lipolysis; Male; Pressoreceptors; Propanolamines; Receptors, Adrenergic, beta; Reflex; Stimulation, Chemical | 1992 |
Pharmacological characterization of a beta 3-receptor agonist (BRL 37,344) and a partial agonist (CGP 12,177A) in neonatal rat liver plasma membranes.
Topics: Adenylyl Cyclase Inhibitors; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Binding, Competitive; Cell Membrane; Enzyme Activation; Ethanolamines; Humans; Isoproterenol; Liver; Propanolamines; Rats; Rats, Wistar | 1992 |
Inhibition by dexamethasone of beta 3-adrenergic receptor responsiveness in 3T3-F442A adipocytes. Evidence for a transcriptional mechanism.
Topics: 3T3 Cells; Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Animals; Base Sequence; Cell Membrane; Dexamethasone; Dose-Response Relationship, Drug; Ethanolamines; Isoproterenol; Kinetics; Mice; Mifepristone; Molecular Sequence Data; Oligodeoxyribonucleotides; Oligonucleotides, Antisense; Polymerase Chain Reaction; Progesterone; Propanolamines; Receptors, Adrenergic, beta; RNA; Transcription, Genetic | 1992 |
Modulation of the beta-adrenergic-response in cultured rat heart cells. II. Mammary-derived growth inhibitor (MDGI) blocks induction of beta-adrenergic supersensitivity. Dissociation from lipid-binding activity of MDGI.
Topics: Amino Acid Sequence; Animals; Arachidonic Acid; Arachidonic Acids; Binding, Competitive; Carrier Proteins; Dose-Response Relationship, Drug; Fatty Acid Binding Protein 3; Fatty Acid-Binding Protein 7; Fatty Acid-Binding Proteins; Growth Inhibitors; Heart; Isoproterenol; Lactates; Molecular Sequence Data; Neoplasm Proteins; Nerve Tissue Proteins; Peptides; Propanolamines; Prostaglandins D; Rats; Receptors, Adrenergic, beta | 1991 |
Characterization of beta-adrenoreceptors of rainbow trout (Oncorhynchus mykiss) erythrocytes.
Topics: Animals; Binding, Competitive; Cell Compartmentation; Dihydroalprenolol; Erythrocytes; Female; Hydrogen-Ion Concentration; Isoproterenol; Male; Propanolamines; Receptors, Adrenergic, beta; Trout | 1991 |
Characterization and regulation of beta 1-adrenergic receptors in a human neuroepithelioma cell line.
Topics: Adrenergic beta-Antagonists; Binding, Competitive; Cell Membrane; Cyclic AMP; DNA Probes; Down-Regulation; Epinephrine; Humans; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Neuroectodermal Tumors, Primitive, Peripheral; Norepinephrine; Nucleic Acid Hybridization; Pindolol; Propanolamines; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured | 1991 |
Adenylate cyclase agonist properties of CGP-12177A in brown fat: evidence for atypical beta-adrenergic receptors.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cell Membrane; Enzyme Activation; Female; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Myocardium; Propanolamines; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta | 1991 |
Beta-adrenergic effects on cellular cholesterologenesis and low density lipoprotein metabolism.
Topics: Adrenergic beta-Antagonists; Cholesterol; Humans; In Vitro Techniques; Isoproterenol; Leukocytes, Mononuclear; Lipoproteins, LDL; Lymphocytes; Propanolamines; Receptors, LDL; Reference Values | 1991 |
Beta-adrenoceptors and adenylate cyclase activity in hypertrophied and failing rabbit left ventricle.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cardiomegaly; Colforsin; Cyclic AMP; Female; GTP-Binding Proteins; Heart Arrest; Isoproterenol; Male; Nucleotidases; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Sodium Fluoride | 1991 |
Coexistence of three beta-adrenoceptor subtypes in white fat cells of various mammalian species.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cricetinae; Dogs; Ethanolamines; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lipolysis; Male; Mesocricetus; Muscle, Smooth; Pindolol; Propanolamines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Human beta 1- and beta 2-adrenergic receptor binding and mediated accumulation of cAMP in transfected Chinese hamster ovary cells. Profile of nebivolol and known beta-adrenergic blockers.
Topics: Adrenergic beta-Antagonists; Animals; Benzopyrans; Binding Sites; Binding, Competitive; Cell Line; Cricetinae; Cricetulus; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Models, Biological; Nebivolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Stereoisomerism; Transfection | 1991 |
Immortalization of brain capillary endothelial cells with maintenance of structural characteristics of the blood-brain barrier endothelium.
Topics: Adrenergic beta-Antagonists; Animals; Antigens, Polyomavirus Transforming; Biomarkers; Blood-Brain Barrier; Capillaries; Cattle; Cell Division; Cell Line, Transformed; Cells, Cultured; Cerebrovascular Circulation; Culture Techniques; Cyclic AMP; Endothelins; Endothelium, Vascular; Fibroblast Growth Factor 2; Intercellular Junctions; Isoproterenol; Microscopy, Electron; Plasmids; Propanolamines; Radioimmunoassay; Receptors, Adrenergic, beta; Simian virus 40; Transfection | 1991 |
Effects of xamoterol on the reversible cycling of cardiac beta-adrenoceptors.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell-Free System; Colchicine; Cytochalasin B; Heart; Heart Failure; Heparin; Isoproterenol; Myocardium; Propanolamines; Protein Kinases; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Xamoterol | 1990 |
Different mechanisms involved in the positive inotropic effects of benzimidazole derivative UD-CG 115 BS (pimobendan) and its demethylated metabolite UD-CG 212 Cl in canine ventricular myocardium.
Topics: Animals; Carbachol; Cardiotonic Agents; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Propanolamines; Pyridazines; Vasodilator Agents | 1991 |
Regulation of adenylyl cyclase activity by beta-adrenergic agonists in a desensitization-resistant mutant cell line.
Topics: Adenylyl Cyclases; Adrenal Cortex Neoplasms; Adrenocorticotropic Hormone; Animals; Gene Expression; Iodocyanopindolol; Isoproterenol; Mice; Mutation; Pindolol; Plasmids; Propanolamines; Receptors, Adrenergic, beta; Sodium Fluoride; Transfection; Tumor Cells, Cultured | 1991 |
Evidence against spare or uncoupled beta-adrenoceptors in the human heart.
Topics: Adrenergic beta-Antagonists; Adult; Binding Sites; Cell Membrane; Electric Stimulation; Female; Heart; Humans; Isoproterenol; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta | 1990 |
An analysis of the beta 2-adrenoceptor selectivity in three series of beta-adrenoceptor agonists.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Catechols; Enzyme Activation; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Kinetics; Male; Nordefrin; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Resorcinols; Terbutaline | 1990 |
Pseudomonas exotoxin A prevents beta-adrenoceptor-induced upregulation of Gi protein alpha-subunits and adenylyl cyclase desensitization in rat heart muscle cells.
Topics: Adenosine Diphosphate Ribose; Adenylyl Cyclases; ADP Ribose Transferases; Adrenergic beta-Antagonists; Animals; Bacterial Toxins; Cells, Cultured; Colforsin; Exotoxins; GTP-Binding Proteins; Heart; Isoproterenol; Kinetics; Macromolecular Substances; Muscle, Smooth; Myocardium; NAD; Norepinephrine; Propanolamines; Pseudomonas aeruginosa Exotoxin A; Rats; Receptors, Adrenergic, beta; Virulence Factors | 1990 |
Adenylate cyclase uncoupled beta-adrenergic receptors in salamander proximal tubules.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Ambystoma; Animals; Cyclic AMP; In Vitro Techniques; Isoproterenol; Kidney Tubules, Proximal; Kinetics; Perfusion; Phenylephrine; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta | 1990 |
Respiratory-burst stimulants desensitize beta-2 adrenoceptors on human polymorphonuclear leukocytes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenergic beta-Antagonists; Binding, Competitive; Granulomatous Disease, Chronic; Humans; In Vitro Techniques; Isoproterenol; Isoquinolines; Kinetics; Neutrophils; Piperazines; Propanolamines; Protein Kinase C; Receptors, Adrenergic, beta; Superoxides | 1990 |
Effects of insulin on mononuclear leukocyte beta-adrenoceptor density and adenylate cyclase coupling.
Topics: Adenylyl Cyclases; Adult; Cyclic AMP; Humans; In Vitro Techniques; Insulin; Isoproterenol; Kinetics; Neutrophils; Propanolamines; Receptors, Adrenergic, beta | 1990 |
Study of beta-adrenoceptors and beta-adrenergic responsiveness in cultured "preneoplastic-like" and neoplastic rat hepatocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Antagonists; Albuterol; Animals; Atenolol; Binding, Competitive; Cells, Cultured; Cyclic AMP; Epinephrine; Isoproterenol; Kinetics; Liver Neoplasms, Experimental; Norepinephrine; Precancerous Conditions; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta | 1985 |
Comparison of two putatively selective radioligands for labeling central nervous system beta-adrenergic receptors: inadequacy of [3H]dihydroalprenolol.
Topics: Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Kinetics; Male; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin | 1989 |
Beta 2-adrenergic receptor regulation after transfection into a cell line deficient in the cAMP-dependent protein kinase.
Topics: Adenylyl Cyclases; Animals; Cell Compartmentation; Cell Line; Cell Membrane; Endocytosis; Gene Expression Regulation; Isoproterenol; Mice; Polyribosomes; Propanolamines; Protein Biosynthesis; Protein Kinases; Receptors, Adrenergic, beta; RNA, Messenger; Transfection | 1989 |
Beta-adrenergic desensitization reduces the sensitivity of adenylate cyclase for magnesium in permeabilized lymphocytes.
Topics: Adenylyl Cyclases; Adolescent; Adrenergic beta-Agonists; Adult; Humans; Isoproterenol; Lymphocytes; Magnesium; Propanolamines; Protein Kinases; Receptors, Adrenergic, beta | 1989 |
Intracellular distribution of cardiac beta-adrenoceptors in SHR and WKY.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Aging; Animals; Heart; Hypertension; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta | 1989 |
[Dependence of kinetic constants of intact human lymphocyte beta2-adrenoreceptors on the nature of the radioligands used].
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Ethylmaleimide; Humans; Isoproterenol; Kinetics; Lymphocytes; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Temperature | 1989 |
Influence of lactate on isoproterenol-induced lipolysis and beta-adrenoceptors distribution in human fat cells.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adult; Cell Membrane; Cells, Cultured; Humans; Isoproterenol; Lactates; Lipolysis; Middle Aged; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Serotonin Antagonists | 1989 |
Signal transduction by membrane receptors in viable electropermeabilized cells: isoproterenol-stimulated cyclic AMP synthesis in C6 glioma cells.
Topics: Adenosine Triphosphate; Adrenergic beta-Antagonists; Animals; Cell Line; Cell Membrane; Cell Membrane Permeability; Cell Nucleus; Cyclic AMP; Electric Stimulation; Glioma; Guanosine Triphosphate; Isoproterenol; Kinetics; Propanolamines; Receptors, Adrenergic, beta; Signal Transduction | 1989 |
Effects of calcium channel blockers and ketotifen on beta 2 adrenergic receptor regulation in intact human lymphocytes.
Topics: Adrenergic beta-Antagonists; Calcium Channel Blockers; Cyclic AMP; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Ketotifen; Lymphocytes; Propanolamines; Radioimmunoassay; Receptors, Adrenergic, beta | 1989 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Mechanism of diminished contractile response to catecholamines during acidosis.
Topics: Acidosis; Animals; Catecholamines; Cells, Cultured; Chick Embryo; Hydrogen-Ion Concentration; Isoproterenol; Myocardial Contraction; Myocardium; Propanolamines; Receptors, Adrenergic, beta | 1988 |
Does the beta-adrenergic receptor function as a reovirus receptor?
Topics: Adenylyl Cyclases; Animals; Cell Line; Humans; Isoproterenol; L Cells; Mammalian orthoreovirus 3; Mice; Propanolamines; Receptors, Adrenergic, beta; Receptors, Virus; Reoviridae | 1988 |
The human promyelocytic leukemia cell (HL-60 cell) beta-adrenergic receptor.
Topics: Cyclic AMP; Humans; Isoproterenol; Leukemia, Myeloid, Acute; Propanolamines; Receptors, Adrenergic, beta; Tumor Cells, Cultured | 1988 |
Homologous vs. heterologous desensitization of the adenylate cyclase system in heart cells.
Topics: Adenylyl Cyclases; Alprostadil; Animals; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Isoproterenol; Myocardium; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta | 1988 |
Regulation by 8-Br-cAMP of beta-adrenoceptors in cultured myocardial cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Antagonists; Animals; Cells, Cultured; Cyclic AMP; Heart; Isoproterenol; Kinetics; Myocardium; Propanolamines; Rats; Receptors, Adrenergic, beta | 1985 |
Beta-adrenergic [( 3H]CGP-12177) binding to brain slices and single intact pineal glands.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain; Cerebral Cortex; Cricetinae; In Vitro Techniques; Isoproterenol; Kinetics; Male; Mesocricetus; Phentolamine; Pineal Gland; Propanolamines; Rats; Rats, Inbred Strains; Timolol | 1985 |
Selective labelling of beta 1-adrenoceptors in rabbit lung membranes by (-)[3H]bisoprolol.
Topics: Adrenergic beta-Antagonists; Animals; Bisoprolol; Female; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Kinetics; Ligands; Lung; Male; Propanolamines; Rabbits; Radioligand Assay; Receptors, Adrenergic, beta | 1985 |
Agonist-induced redistribution of beta-adrenergic receptors on intact human mononuclear leukocytes: redistributed receptors are nonfunctional.
Topics: Adrenergic beta-Antagonists; Adult; Cyclic AMP; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Leukocytes; Ligands; Male; Propanolamines; Receptors, Adrenergic, beta | 1985 |
Agonist-induced beta-adrenergic receptor internalization on intact human mononuclear leukocytes: effect of temperature of mononuclear leukocyte separation.
Topics: Adrenergic beta-Agonists; Cell Separation; Humans; Isoproterenol; Leukocytes; Male; Propanolamines; Receptors, Adrenergic, beta; Temperature; Tritium | 1986 |
Characterization of beta-adrenergic binding sites on rodent Leydig cells.
Topics: Adrenergic beta-Antagonists; Androgens; Animals; Binding, Competitive; Cell Separation; Cells, Cultured; Colforsin; Isoproterenol; Kinetics; Leydig Cells; Luteinizing Hormone; Male; Mice; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1985 |
Evidence for the appearance of an uncoupled form of the beta-adrenergic receptor distinct from the internalized receptor.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cells, Cultured; Dose-Response Relationship, Drug; Glioma; Isoproterenol; Propanolamines; Receptor Aggregation; Receptors, Adrenergic, beta; Time Factors | 1986 |
Temperature-dependent binding of hydrophilic beta-adrenergic receptor ligands to intact human lymphocytes.
Topics: Adolescent; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Binding, Competitive; Cell Membrane; Humans; In Vitro Techniques; Isoproterenol; Ligands; Lymphocytes; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Temperature | 1986 |
Down regulation of beta adrenergic receptors in S49 lymphoma cells induced by atypical agonists.
Topics: Adrenergic beta-Agonists; Animals; Binding Sites; Celiprolol; Cell Division; Cell Line; Isoproterenol; Kinetics; Lymphoma; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Time Factors | 1986 |
The beta 2-adrenergic receptors of human epidermoid carcinoma cells bear two different types of oligosaccharides which influence expression on the cell surface.
Topics: Adrenergic beta-Antagonists; Binding Sites; Carcinoma, Squamous Cell; Cell Line; Cell Membrane; Chromatography, Affinity; Cyclic AMP; Glycosylation; Humans; Isoproterenol; Monensin; Oligosaccharides; Propanolamines; Receptors, Adrenergic, beta; Tunicamycin | 1988 |
Augmentation and inhibition of beta-adrenergic agonists-stimulated tissue cyclic AMP accumulation by alpha-adrenergic agonists in rat parotid gland.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Calcium; Cyclic AMP; In Vitro Techniques; Isoproterenol; Male; Methoxamine; Parotid Gland; Phenylephrine; Propanolamines; Rats; Rats, Inbred Strains | 1987 |
Direct assessment of beta-adrenergic receptors in intact rat adipocytes by binding of [3H]CGP 12177. Evidence for agonist high-affinity binding complex and for beta 1 and beta 2 receptor subtypes.
Topics: Adipose Tissue; Animals; Chemical Phenomena; Chemistry; Epinephrine; Isoproterenol; Molecular Conformation; Norepinephrine; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Temperature | 1985 |
Evidence for two specific affinity states of 3H-antagonist binding to cardiac beta-adrenergic receptors and influence of Gpp(NH)p.
Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Myocardium; Propanolamines; Rats; Receptors, Adrenergic, beta | 1985 |
A comparison of catecholamine-induced internalization of beta-adrenergic receptors and receptor-mediated endocytosis of epidermal growth factor in human astrocytoma cells. Inhibition by phenylarsine oxide.
Topics: Adenosine Triphosphate; Arsenicals; Astrocytoma; Catecholamines; Cell Line; Dithiothreitol; Endocytosis; Epidermal Growth Factor; Humans; Iodocyanopindolol; Isoproterenol; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1985 |
Beta-1 receptor is the predominant beta-adrenoreceptor on rat brown adipose tissue.
Topics: Adipose Tissue, Brown; Animals; Binding, Competitive; In Vitro Techniques; Isoproterenol; Kinetics; Male; Norepinephrine; Oxygen Consumption; Propanolamines; Rats; Receptors, Adrenergic, beta; Tritium | 1986 |
Estradiol treatment decreases the lipolytic responses of hamster white adipocytes through a reduction in the activity of the adenylate cyclase catalytic subunit.
Topics: Adenylyl Cyclase Inhibitors; Adipose Tissue; Adrenocorticotropic Hormone; Animals; Clonidine; Cricetinae; Cyclic AMP; Epinephrine; Estradiol; Glycerol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Lipolysis; Male; Mesocricetus; Propanolamines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Theophylline | 1986 |
Desensitization and redistribution of beta-adrenergic receptors on human mononuclear leukocytes.
Topics: Adolescent; Adult; Binding, Competitive; Cyclic AMP; Drug Tolerance; Female; Humans; Iodocyanopindolol; Isoproterenol; Leukocytes; Male; Monocytes; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1986 |
Stress induced desensitization of lymphocyte beta-adrenoceptors in young and aged rats.
Topics: Age Factors; Animals; Corticosterone; Dihydroalprenolol; Isoproterenol; Lymphocytes; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological | 1986 |
The muscle slice--a new preparation for the characterization of beta-adrenergic binding in fast- and slow-twitch skeletal muscle.
Topics: Animals; Binding, Competitive; Hot Temperature; In Vitro Techniques; Isoproterenol; Male; Mice; Muscles; Organ Specificity; Propanolamines; Receptors, Adrenergic, beta; Species Specificity | 1986 |
Desensitization of the beta-adrenergic receptor-coupled adenylate cyclase in cultured mammalian cells. Receptor sequestration versus receptor function.
Topics: Adenylyl Cyclases; Animals; Arsenicals; Cell Line; Concanavalin A; Dose-Response Relationship, Drug; Humans; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Time Factors | 1986 |
Beta-adrenergic receptors in guinea-pig liver plasma membranes and thermal lability of [3H]dihydroalprenolol binding sites.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Guinea Pigs; Hot Temperature; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Virulence Factors, Bordetella | 1986 |
Regulation of beta adrenergic receptors on rat mononuclear leukocytes by stress: receptor redistribution and down-regulation are altered with aging.
Topics: Aging; Animals; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Male; Monocytes; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological; Time Factors | 1987 |
Adenylate cyclase regulation in intact cultured myocardial cells.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cell Membrane; Cells, Cultured; Chick Embryo; Cyclic AMP; Heart Ventricles; Homeostasis; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Propanolamines; Receptors, Adrenergic, beta | 1987 |
Myocardial adrenergic responsiveness after lethal and nonlethal doses of endotoxin.
Topics: Adenosine Triphosphate; Animals; Binding, Competitive; Cyclic AMP; Endotoxins; Epinephrine; Heart Conduction System; Isoproterenol; Lethal Dose 50; Male; Myocardium; Norepinephrine; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sympathetic Nervous System | 1987 |
Bromoacetylalprenololmenthane binding to beta-receptors modulates the rate of hormone-induced internalization but not desensitization in S49 cells.
Topics: Alprenolol; Cell Line; Cell Membrane; Cyclic AMP; Isoproterenol; Kinetics; Lymphoma; Propanolamines; Receptors, Adrenergic, beta | 1987 |
Down-regulation of surface beta-adrenoceptors on intact human mononuclear leukocytes. Time-course and isoproterenol concentration dependence.
Topics: Adenylyl Cyclases; Adolescent; Adult; Dose-Response Relationship, Drug; Female; Humans; Iodocyanopindolol; Isoproterenol; Leukocytes; Male; Middle Aged; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Time Factors | 1987 |
Rapid recovery of cardiac beta-adrenergic receptors after isoproterenol-induced "down"-regulation.
Topics: Adenosine Triphosphate; Animals; Colchicine; Cyclic AMP; Cytoplasm; Dihydroalprenolol; Drug Tolerance; Isoproterenol; Male; Monensin; Myocardium; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1984 |
Relationship between an altered membrane form and a low affinity form of the beta-adrenergic receptor occurring during catecholamine-induced desensitization. Evidence for receptor internalization.
Topics: Astrocytoma; Cell Line; Centrifugation, Density Gradient; Concanavalin A; Humans; Isoproterenol; Methylmannosides; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Time Factors | 1984 |
Agonist-induced internalization of the beta adrenergic receptor in a smooth muscle cell line.
Topics: Animals; Cell Line; Dose-Response Relationship, Drug; Isoproterenol; Kinetics; Muscle, Smooth; Phenylephrine; Propanolamines; Receptors, Adrenergic, beta | 1984 |
Some unique properties of CGP-12177.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cyclic AMP; Digitonin; Dihydroalprenolol; Glioma; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Stereoisomerism | 1984 |
Changes in beta-adrenoceptor binding properties and receptor-cyclase coupling during in vitro maturation of rat reticulocytes.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Cells, Cultured; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Reticulocytes | 1984 |
Properties of beta-adrenoceptor sites in metabolizing and nonmetabolizing rat reticulocytes and in resealed reticulocyte ghosts.
Topics: Adrenergic beta-Antagonists; Animals; Cell Membrane; Cold Temperature; Cytosol; Dihydroalprenolol; Energy Metabolism; Female; Isoproterenol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reticulocytes; Timolol | 1981 |
Reappearance of beta-adrenergic receptors after isoproterenol treatment in intact C6-cells.
Topics: Adrenergic beta-Antagonists; Animals; Cations; Cell Line; Cycloheximide; Glioma; Isoproterenol; Kinetics; Lysosomes; Propanolamines; Rats; Receptors, Adrenergic, beta; Temperature | 1983 |
Determination of the desensitization of beta-adrenergic receptors by [3H]CGP-12177.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Binding Sites; Binding, Competitive; Cell Line; Cell Membrane; Centrifugation, Density Gradient; Dihydroalprenolol; Glioma; Humans; Isoproterenol; Propanolamines; Receptors, Adrenergic, beta | 1983 |
The human carcinoma cell line A431 possesses large numbers of functional beta-adrenergic receptors.
Topics: Adrenergic beta-Antagonists; Binding, Competitive; Carcinoma, Squamous Cell; Cell Line; Dihydroalprenolol; Humans; Isoproterenol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 1984 |
Evidence for intravesicular beta-adrenergic receptors in membrane fractions from desensitized cells: binding of the hydrophilic ligand CGP-12177 only in the presence of alamethicin.
Topics: Alamethicin; Animals; Anti-Bacterial Agents; Cells, Cultured; Centrifugation, Density Gradient; Glioma; Isoproterenol; Pindolol; Propanolamines; Rats; Receptors, Adrenergic, beta | 1983 |
Rapid and reversible disappearance of beta-adrenergic cell surface receptors.
Topics: Animals; Cell Line; Endocytosis; Glioma; Isoproterenol; Lymphoma; Propanolamines; Receptors, Adrenergic, beta; Time Factors | 1982 |
Signal transduction pathway involved in beta 3-adrenoceptor-mediated relaxation in guinea pig taenia caecum.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Butoxamine; Cecum; Culture Techniques; Cyclic AMP; Guinea Pigs; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction | 1995 |
Uncoupling of beta 1-adrenoceptors from cardiac adenylyl cyclase in cardiomyopathic and control hamsters.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cardiomyopathies; Cricetinae; Heart Ventricles; Imidazoles; Isoproterenol; Male; Membranes; Mesocricetus; Myocardium; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1 | 1993 |
Molecular mechanisms underlying regional variations of catecholamine-induced lipolysis in rat adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Base Sequence; Brimonidine Tartrate; Bucladesine; Catecholamines; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Dioxanes; DNA Primers; Epididymis; Gene Expression; Idazoxan; Isoproterenol; Lipase; Lipolysis; Male; Molecular Sequence Data; Organ Specificity; Polymerase Chain Reaction; Propanolamines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; RNA, Messenger; Skin | 1995 |
Reversible decrease of surface beta 2-adrenoceptor number and response in lymphocytes of patients with pheochromocytoma.
Topics: Adrenal Gland Neoplasms; Adrenergic beta-Antagonists; Adult; Aged; Case-Control Studies; Catecholamines; Down-Regulation; Female; Humans; Isoproterenol; Lymphocytes; Male; Middle Aged; Pheochromocytoma; Propanolamines; Radioimmunoassay; Radioligand Assay; Receptors, Adrenergic, beta-2 | 1995 |
Predominant expression of beta 1-adrenergic receptor in the thick ascending limb of rat kidney. Absolute mRNA quantitation by reverse transcription and polymerase chain reaction.
Topics: Adrenergic beta-Antagonists; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA; Gene Expression; Isoproterenol; Kidney Cortex; Kidney Medulla; Molecular Sequence Data; Mutagenesis, Site-Directed; Nephrons; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; RNA-Directed DNA Polymerase; RNA, Messenger; Transcription, Genetic | 1993 |
Myocardial and pulmonary uptake of S-1'-[18F]fluorocarazolol in intact rats reflects radioligand binding to beta-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Carbazoles; Chlorpromazine; Fluorine Radioisotopes; Isoproterenol; Lung; Male; Myocardium; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Tomography, Emission-Computed | 1995 |
Demonstration of an in vivo functional beta 3-adrenoceptor in man.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adult; Analysis of Variance; Animals; Body Temperature Regulation; Cells, Cultured; Dobutamine; Female; Humans; Isoproterenol; Kinetics; Lipolysis; Male; Mammals; Metoprolol; Microdialysis; Middle Aged; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reference Values; Regional Blood Flow; Terbutaline; Time Factors | 1995 |
Modulation by GM1 ganglioside of beta 1-adrenergic receptor-induced cyclic AMP formation in Sf9 cells.
Topics: Adenosine Monophosphate; Adrenergic beta-Antagonists; Animals; Baculoviridae; Cell Line; G(M1) Ganglioside; Humans; Insecta; Isoproterenol; Propanolamines; Receptors, Adrenergic, beta; Transfection | 1995 |
Apparent lack of beta 3-adrenoceptors and of insulin regulation of glucose transport in brown adipose tissue of guinea pigs.
Topics: Acclimatization; Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic alpha-Agonists; Animals; Body Temperature Regulation; Cell Membrane; Dioxoles; Epinephrine; Ethanolamines; Female; Glucose Transporter Type 4; Guinea Pigs; Insulin; Isoproterenol; Monosaccharide Transport Proteins; Muscle Proteins; Norepinephrine; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Temperature; Time Factors | 1995 |
Beta-adrenergic receptor function in cultured AT-1 cardiomyocytes.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Calcium; Cell Line; Cyclic AMP; Cytosol; Heart; Heart Neoplasms; Isoproterenol; Kinetics; Mice; Mice, Transgenic; Myocardial Contraction; Myocardium; Potassium; Propanolamines; Receptors, Adrenergic, beta; Time Factors; Tumor Cells, Cultured | 1995 |
Atypical beta-adrenoceptors in the rat isolated common carotid artery.
Topics: Adrenergic beta-Agonists; Albuterol; Animals; Carotid Artery, Common; Dose-Response Relationship, Drug; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Male; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1994 |
Involvement of beta 3-adrenoceptor in the relaxation response in guinea pig taenia caecum.
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Binding, Competitive; Butoxamine; Cecum; Dose-Response Relationship, Drug; Epinephrine; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Microsomes; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta | 1994 |
Carboxyl-terminal domains in the avian beta 1-adrenergic receptor that regulate agonist-promoted endocytosis.
Topics: Animals; Endocytosis; Iodocyanopindolol; Isoproterenol; Mice; Peptide Fragments; Pindolol; Propanolamines; Receptors, Adrenergic, beta-1; Turkeys | 1995 |
Cardiac beta-adrenoceptor-effector coupling in portal vein-stenosed rats.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Constriction; Cyclic AMP; Heart; Hypertension; Isoproterenol; Male; Myocardial Contraction; Portal Vein; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1995 |
Physiological desensitization of beta 3-adrenergic responses in brown fat cells: involvement of a postreceptor process.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Acclimatization; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cells, Cultured; Cold Temperature; Colforsin; Cricetinae; Cyclic AMP; Ethanolamines; Isoproterenol; Kinetics; Male; Mesocricetus; Norepinephrine; Oxygen Consumption; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1993 |
Response of mouse proximal straight tubule and medullary thick ascending limb to beta-agonist.
Topics: Adrenergic beta-Antagonists; Animals; Electrophysiology; Furosemide; In Vitro Techniques; Isoproterenol; Kidney Medulla; Kidney Tubules; Kidney Tubules, Proximal; Kinetics; Membrane Potentials; Mice; Perfusion; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta | 1993 |
Heterologous sensitization of adenylate cyclase activity by serotonin in the rat cerebral cortex.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Colforsin; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Male; Phorbol 12,13-Dibutyrate; Propanolamines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Somatostatin; Tetradecanoylphorbol Acetate; Vasoactive Intestinal Peptide | 1993 |
Atypical beta-adrenergic receptors in rat liver: evidence for transient expression during aging.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Aging; Animals; Isoproterenol; Liver; Male; Propanolamines; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta | 1994 |
Beta-3 adrenoceptor-mediated increase in cutaneous blood flow in the dog.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Bupranolol; Dioxoles; Dogs; Ethanolamines; Heart Rate; Isoproterenol; Male; Nitroprusside; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Regional Blood Flow; Skin | 1994 |
Characterization of agonist-induced internalization and down-regulation of beta-adrenergic receptors in isolated rat lung and heart preparations.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Cycloheximide; Down-Regulation; Endocytosis; Heart; Hypertonic Solutions; Iodocyanopindolol; Isoproterenol; Lung; Male; Myocardium; Organ Specificity; Pindolol; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Sucrose; Terbutaline | 1993 |
Modulation of adenylylcyclase by protein kinase C in human neurotumor SK-N-MC cells: evidence that the alpha isozyme mediates both potentiation and desensitization.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Alkaloids; Aluminum Compounds; Animals; Brain; Cell Line; Cell Membrane; Cholera Toxin; Colforsin; Cyclic AMP; Dopamine; Drug Synergism; Fluorides; GTP-Binding Proteins; Humans; Isoenzymes; Isoproterenol; Kinetics; Manganese; Neuroblastoma; Neuropeptide Y; Propanolamines; Protein Kinase C; Rats; Sphingosine; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1994 |
Influence of cell type upon the desensitization of the beta 3-adrenergic receptor.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; CHO Cells; Cricetinae; Humans; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Sodium Fluoride | 1994 |
Antagonism between T3 and amiodarone on the contractility and the density of beta-adrenoceptors of chicken cardiac myocytes.
Topics: Adrenergic beta-Antagonists; Amiodarone; Animals; Calcium; Chick Embryo; Heart; Iodocyanopindolol; Isoproterenol; Myocardial Contraction; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Triiodothyronine | 1994 |
Minimal modification of canine ventricular myocyte cell surface beta adrenoceptors despite desensitisation of ventricular function during exogenous beta adrenoceptor challenge.
Topics: Animals; Cell Membrane; Cells, Cultured; Dogs; Epinephrine; Female; Isoproterenol; Male; Myocardial Contraction; Myocardium; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Stimulation, Chemical; Time Factors | 1994 |
Isoproterenol and selective agonists stimulate similar atypical beta-adrenoceptors in rat adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Animals; Isoproterenol; Lipolysis; Male; Propanolamines; Rats; Rats, Sprague-Dawley | 1993 |
Coexistence of beta 1-, beta 2-, and beta 3-adrenoceptors in dog fat cells and their differential activation by catecholamines.
Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamines; Cell Membrane; Dogs; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Isoproterenol; Norepinephrine; Procaterol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tetrahydronaphthalenes | 1993 |
Dynamic exercise induces translocation of beta-adrenergic receptors in human lymphocytes.
Topics: Adrenergic beta-Antagonists; Adult; Cell Membrane; Cyclic AMP; Exercise; Exercise Test; Humans; Isoproterenol; Lymphocytes; Propanolamines; Propranolol; Radioimmunoassay; Receptors, Adrenergic, beta | 1993 |
No functional atypical beta-adrenergic receptors in human omental adipocytes.
Topics: Adipose Tissue; Dose-Response Relationship, Drug; Humans; Isoproterenol; Lipolysis; Omentum; Propanolamines; Receptors, Adrenergic, beta | 1994 |
Isoproterenol interacts differently with beta-adrenoceptors in astrocytes and neurons isolated from the adult rat brain.
Topics: Animals; Astrocytes; Binding, Competitive; Cerebral Cortex; Guanylyl Imidodiphosphate; Isoproterenol; Neurons; Propanolamines; Protein Conformation; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1994 |
Disrupted beta 1-adrenoceptor-G protein coupling in the temporal cortex of patients with Alzheimer's disease.
Topics: Aged; Alzheimer Disease; Binding, Competitive; Female; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Isoproterenol; Male; Middle Aged; Propanolamines; Protein Binding; Receptors, Adrenergic, beta; Signal Transduction; Synaptic Membranes; Temporal Lobe | 1993 |
Determination of beta-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective beta-antagonists.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cyclic AMP; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Membranes; Myocardium; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Tritium | 1995 |
Stimulation of nonshivering thermogenesis in the Syrian hamster by norepinephrine and beta-selective adrenergic agents: a phenomenon of refractoriness.
Topics: Acclimatization; Adipose Tissue, Brown; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Cold Temperature; Cricetinae; Drug Interactions; Ethanolamines; Female; Isoproterenol; Male; Mesocricetus; Norepinephrine; Oxygen Consumption; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Reproducibility of Results; Shivering | 1996 |
Regulation of heat production of brown adipocytes via typical and atypical beta-adrenoceptors in the rat.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Calorimetry; Ethanolamines; In Vitro Techniques; Isoproterenol; Male; Phenoxyacetates; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1995 |
Effects of several putative beta 3-adrenoceptor agonists on lipolysis in human omental adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Catechols; Dioxoles; Ethanolamines; Glycerol; Humans; Isoproterenol; Lipolysis; Omentum; Propanolamines; Serine | 1996 |
Triiodothyronine regulates beta 3-adrenoceptor expression in 3T3-F442A differentiating adipocytes.
Topics: 3T3 Cells; Adenylyl Cyclases; Adipocytes; Adrenergic beta-Antagonists; Animals; Base Sequence; Cell Differentiation; Cell Nucleus; Colforsin; Dactinomycin; DNA Primers; Gene Expression; Glycerolphosphate Dehydrogenase; Guanosine 5'-O-(3-Thiotriphosphate); Isoproterenol; Kinetics; Mice; Molecular Sequence Data; Propanolamines; Protein Biosynthesis; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Recombinant Proteins; RNA, Messenger; Transcription, Genetic; Transfection; Triiodothyronine | 1996 |
Effects of the beta 3-adrenoceptor agonist BRL 37344 on lipomobilization and plasma glucose levels in conscious fasted rabbits.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Biological Transport; Blood Glucose; Ethanolamines; Fasting; Fatty Acids, Nonesterified; Insulin; Isoproterenol; Lactic Acid; Male; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Sodium Chloride | 1996 |
Repetitive endocytosis and recycling of the beta 2-adrenergic receptor during agonist-induced steady state redistribution.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Antibodies, Monoclonal; Endocytosis; Flow Cytometry; Humans; Isoproterenol; Kidney; Kinetics; Models, Theoretical; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-2; Recombinant Proteins; Time Factors; Transfection | 1996 |
Regulation of lipolysis in fat cells of obese women during long-term hypocaloric diet.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipocytes; Adrenergic beta-Agonists; Adult; Brimonidine Tartrate; Bucladesine; Catecholamines; Colforsin; Dobutamine; Energy Intake; Female; Food Deprivation; Glucose; Humans; Insulin; Insulin Resistance; Isoproterenol; Lipolysis; Middle Aged; Obesity; Propanolamines; Quinoxalines; Terbutaline; Time Factors | 1996 |
Agonist and antagonist properties of beta 3-adrenoceptors in human omental and mouse 3T3-L1 adipocytes.
Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Humans; Isoproterenol; Lipolysis; Mice; Omentum; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Yohimbine | 1996 |
Pharmacological characteristics of BDTI, a new isoquinoline-derived beta 2-adrenoceptor agonist, in canine trachea and rat heart.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Atenolol; Carbachol; Cells, Cultured; Dogs; Dose-Response Relationship, Drug; Female; Heart; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Myocardium; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Trachea; Tretoquinol | 1996 |
In vivo increase in beta-adrenergic lipolytic response in subcutaneous adipose tissue of obese subjects submitted to a hypocaloric diet.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adult; Diet, Reducing; Dobutamine; Energy Intake; Female; Glycerol; Humans; Isoproterenol; Kinetics; Lipolysis; Male; Middle Aged; Obesity; Propanolamines; Receptors, Adrenergic, beta | 1997 |
Thermoregulation with age: role of beta-adrenergic signal transduction.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Body Temperature; Carrier Proteins; Cold Temperature; Gene Expression; Guanosine Diphosphate; Ion Channels; Isoproterenol; Membrane Proteins; Mitochondria; Mitochondrial Proteins; Oxygen Consumption; Propanolamines; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Uncoupling Protein 1 | 1997 |
Alterations of central noradrenergic transmission in Ts65Dn mouse, a model for Down syndrome.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Animals; Brain; Cell Membrane; Cerebellum; Cerebral Cortex; Chromosome Mapping; Chromosomes, Human, Pair 21; Colforsin; Cyclic AMP; Down Syndrome; Hippocampus; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Mice; Mice, Neurologic Mutants; Norepinephrine; Organ Specificity; Propanolamines; Receptors, Adrenergic, beta; Reference Values; Signal Transduction | 1997 |
Constitutive activation of the beta2 adrenergic receptor alters the orientation of its sixth membrane-spanning segment.
Topics: Adrenergic beta-Agonists; Binding Sites; Binding, Competitive; Cell Membrane; Cysteine; Ethyl Methanesulfonate; Humans; Indicators and Reagents; Isoproterenol; Ligands; Propanolamines; Protein Conformation; Receptors, Adrenergic, beta-2 | 1997 |
A match between binding to beta-adrenoceptors and stimulation of adenylyl cyclase parameters of (-)isoproterenol and salbutamol on rat brain.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Albuterol; Animals; Brain; Cerebellum; Cerebral Cortex; Cyclic AMP; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Male; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Synaptosomes | 1997 |
Noradrenaline-induced lipolysis in isolated mesenteric, omental and subcutaneous adipocytes from obese subjects.
Topics: Adipocytes; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adult; Dobutamine; Dose-Response Relationship, Drug; Female; Humans; Isoproterenol; Lipolysis; Male; Mesentery; Middle Aged; Norepinephrine; Obesity; Omentum; Propanolamines; Terbutaline; Yohimbine | 1997 |
Simulated microgravity increases beta-adrenergic lipolysis in human adipose tissue.
Topics: Adipocytes; Adipose Tissue; Adrenergic beta-Agonists; Adult; Bucladesine; Dobutamine; Epinephrine; Glycerol; Head-Down Tilt; Humans; Isoproterenol; Lipolysis; Male; Microdialysis; Propanolamines; Receptors, Adrenergic, beta; Terbutaline; Weightlessness | 1998 |
Evidence for the stabilisation of the high-affinity state of beta-adrenoceptors by an endogenous factor in rat brain.
Topics: Animals; Brain; Cholic Acids; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Male; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Synaptosomes; Temperature | 1998 |
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1998 |
Heterologous regulation of muscarinic and beta-adrenergic receptors in rat cardiomyocytes in culture.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; Bucladesine; Carbachol; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Inhibitors; Female; Indoles; Isoproterenol; Isoquinolines; Kinetics; Male; Maleimides; Muscarinic Agonists; Myocardium; N-Methylscopolamine; Propanolamines; Protein Kinase C; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Sulfonamides; Thionucleotides; Tritium | 1998 |
Trp64Arg mutation of beta3-adrenoceptor gene deteriorates lipolysis induced by beta3-adrenoceptor agonist in human omental adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adult; Amino Acid Sequence; Female; Humans; Isoproterenol; Lipolysis; Middle Aged; Mutation; Omentum; Propanolamines; Receptors, Adrenergic, beta; Sulfonamides | 1999 |
Stimulation of the extracellular signal-regulated kinase 1/2 pathway by human beta-3 adrenergic receptor: new pharmacological profile and mechanism of activation.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Colforsin; Cricetinae; Dioxoles; Enzyme Activation; Epinephrine; Ethanolamines; Humans; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Norepinephrine; Phentolamine; Prazosin; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction; Yohimbine | 1999 |
The effect of hydrogen peroxide upon beta-adrenoceptor density and function in C6 rat glioma cells.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Cell Death; Colforsin; Culture Media, Serum-Free; Cyclic AMP; Glioma; GTP-Binding Protein alpha Subunits, Gs; Hydrogen Peroxide; Isoproterenol; L-Lactate Dehydrogenase; Propanolamines; Rats; Receptors, Adrenergic, beta; Tumor Cells, Cultured | 1999 |
Functional and molecular biological evidence for a possible beta3-adrenoceptor in the human detrusor muscle.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colforsin; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 1999 |
Evidence for cooperative binding of (-)Isoproterenol to rat brain beta1-adrenergic receptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Allosteric Site; Animals; Blood Platelets; Brain; Cell Membrane; Diamide; Dithiothreitol; Edetic Acid; Humans; Isoproterenol; Lysergic Acid Diethylamide; Magnesium; Molecular Weight; Propanolamines; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, beta-1; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1999 |
Specific changes in beta2-adrenoceptor trafficking kinetics and intracellular sorting during downregulation.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Biological Transport; Cell Line; Down-Regulation; Endocytosis; Humans; Isoproterenol; Kinetics; Propanolamines; Protease Inhibitors; Radioligand Assay; Receptors, Adrenergic, beta-2; Sensitivity and Specificity; Time Factors; Tritium | 1999 |
Interaction of amiodarone and triiodothyronine on the expression of beta-adrenoceptors in brown adipose tissue of rat.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amiodarone; Animals; Anti-Arrhythmia Agents; Drug Interactions; Gene Expression; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Isoproterenol; Male; Propanolamines; Proteins; Rats; Rats, Wistar; Receptors, Adrenergic, beta; RNA, Messenger; Triiodothyronine | 1999 |
A GppNHp-insensitivity factor modulates the activation of beta-adrenoceptor-coupled Gs protein in rat cortex and cerebellum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Astrocytes; Cerebellum; Cerebral Cortex; Cholic Acids; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Kinetics; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Synaptosomes | 1999 |
Atypical beta-adrenoceptors mediating relaxation in the human colon: functional evidence for beta3-rather than beta4-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colon; Ethanolamines; Female; Humans; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes | 1999 |
Beta 2-adrenergic receptor endocytic pathway is controlled by a saturable mechanism distinct from that of transferrin receptor.
Topics: 3,3'-Diaminobenzidine; Adrenergic beta-Agonists; Arrestin; Cell Line; Centrifugation, Density Gradient; Endocytosis; Humans; Iodocyanopindolol; Isoproterenol; Microscopy, Fluorescence; Phosphorylation; Propanolamines; Propranolol; Protein Processing, Post-Translational; Receptors, Adrenergic, beta-2; Receptors, Transferrin; Recombinant Fusion Proteins; Temperature; Transfection | 1999 |
No functional beta 3-adrenergic receptors expressed in rat skeletal muscle cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Cells, Cultured; Cyclic AMP; Isoproterenol; Muscle, Skeletal; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1998 |
Propofol-induced alterations in myocardial beta-adrenoceptor binding and responsiveness.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Anesthetics, Intravenous; Animals; Cell Membrane; Heart; Heart Ventricles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardium; Propanolamines; Propofol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1999 |
Stress-induced alteration in the lipolytic response to beta-adrenoceptor agonists in rat white adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Body Weight; Bucladesine; Eating; Epinephrine; Ethanolamines; Glycerol; Isoproterenol; Lipolysis; Male; Metoprolol; Norepinephrine; Propanolamines; Rats; Rats, Wistar; Stress, Physiological | 1999 |
Blockade of putative beta4- and beta1-adrenoceptors by carvedilol in ferret myocardium.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbazoles; Carvedilol; Dose-Response Relationship, Drug; Ferrets; Heart Atria; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Propanolamines; Receptors, Adrenergic, beta; Sinoatrial Node | 1999 |
Beta 3-adrenoceptor stimulation induces vasorelaxation mediated essentially by endothelium-derived nitric oxide in rat thoracic aorta.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Cyclic GMP; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Nadolol; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Phenylephrine; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes; Vasoconstriction; Vasodilation | 1999 |
Beta4-adrenoceptors are more effective than beta1-adrenoceptors in mediating arrhythmic Ca2+ transients in mouse ventricular myocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Mice; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Time Factors | 1999 |
Pharmacological analysis of atypical beta-adrenoceptors in the guinea pig gastric fundus using the beta(3)-adrenoceptor antagonist bupranolol.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Bupranolol; Butoxamine; Catecholamines; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3 | 1999 |
[Pharmacological analysis of atypical beta-adrenoceptors in the guinea pig gastrointestinal tissue systems].
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Digestive System; Duodenum; Epinephrine; Ethanolamines; Gastric Fundus; Guinea Pigs; Ileum; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta | 1999 |
Beta-3 adrenergic stimulation of L-type Ca(2+) channels in rat portal vein myocytes.
Topics: 1-Propanol; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Barium; Calcium Channels, L-Type; Cells, Cultured; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; Isoproterenol; Isoquinolines; Membrane Potentials; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Portal Vein; Propanolamines; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Sulfonamides | 2000 |
Dexamethasone potentiates high-affinity beta-agonist binding and g(s)alpha protein expression in airway smooth muscle.
Topics: Adrenergic beta-Agonists; Animals; Blotting, Western; Cattle; Dexamethasone; Glucocorticoids; GTP-Binding Protein alpha Subunits, Gs; Isoproterenol; Ligands; Membrane Proteins; Muscle, Smooth; Propanolamines; Radioligand Assay; Trachea; Tritium | 2000 |
Mutated human beta3-adrenergic receptor (Trp64Arg) lowers the response to beta3-adrenergic agonists in transfected 3T3-L1 preadipocytes.
Topics: 3T3 Cells; Adenylyl Cyclases; Adipocytes; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Animals; Cyclic AMP; Dioxoles; Epinephrine; Humans; Isoproterenol; Kinetics; Mice; Mutagenesis, Site-Directed; Norepinephrine; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Recombinant Proteins; Sulfonamides; Transfection | 2000 |
The effects of beta-adrenoceptor agonists on KCl-induced rhythmic contraction in the ureter of guinea pig.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Calcium Channels, L-Type; Dose-Response Relationship, Drug; Guinea Pigs; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Periodicity; Potassium Chloride; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Ureter | 2000 |
Rapid electrical stimulation of contraction reduces the density of beta-adrenergic receptors and responsiveness of cultured neonatal rat cardiomyocytes. Possible involvement of microtubule disassembly secondary to mechanical stress.
Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antineoplastic Agents, Phytogenic; Cells, Cultured; Colforsin; Diacetyl; Dihydroalprenolol; Down-Regulation; Electric Stimulation; Enzyme Inhibitors; Heart Failure; Isoproterenol; Microtubules; Muscle Fibers, Skeletal; Myocardial Contraction; Myocardium; Pacemaker, Artificial; Paclitaxel; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stress, Mechanical; Tritium; Vasodilator Agents | 2000 |
Role of endothelium/nitric oxide in atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Norepinephrine; Oxadiazoles; Phenoxyacetates; Phenoxypropanolamines; Phenylacetates; Pindolol; Propanolamines; Propranolol; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Vasodilation | 2000 |
Short-term effects of postnatal manipulation on central beta-adrenoceptor transmission.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenocorticotropic Hormone; Animals; Animals, Suckling; Cerebellum; Cerebral Cortex; Colforsin; Corticosterone; Cyclic AMP; Emotions; Female; Handling, Psychological; Hippocampus; Isoproterenol; Male; Norepinephrine; Pregnancy; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Restraint, Physical; Signal Transduction; Stress, Physiological; Tritium | 1999 |
Functional assessment of beta adrenoceptor subtypes in human colonic circular and longitudinal (taenia coli) smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Colon; Female; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Terbutaline; Tetrahydronaphthalenes | 2000 |
Ligand regulation of green fluorescent protein-tagged forms of the human beta(1)- and beta(2)-adrenoceptors; comparisons with the unmodified receptors.
Topics: Betaxolol; Binding, Competitive; Cell Line; Dihydroalprenolol; Endocytosis; Green Fluorescent Proteins; Humans; Isoproterenol; Kinetics; Ligands; Luminescent Proteins; Microscopy, Confocal; Oligopeptides; Peptides; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Tritium | 2000 |
Partial agonist activity of carteolol on atypical beta-adrenoceptors in the guinea pig duodenum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Carteolol; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Vasodilator Agents | 2000 |
Characterization of beta-adrenoceptor subtypes in the ferret urinary bladder in vitro and in vivo.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Anesthesia; Animals; Blood Pressure; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Ethanolamines; Ferrets; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pressure; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Time Factors; Urinary Bladder | 2000 |
Changes in dietary fatty acids modify the decreased lipolytic beta3-adrenergic response to hyperinsulinemia in adipocytes from pregnant and nonpregnant rats.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Dietary Fats; Epinephrine; Ethanolamines; Fatty Acids; Female; Fish Oils; Glucose Clamp Technique; Hyperinsulinism; Isoproterenol; Lipolysis; Olive Oil; Phospholipids; Plant Oils; Pregnancy; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 2000 |
Evidence that oestradiol attenuates beta-adrenoceptor function in the hypothalamus of female rats by altering receptor phosphorylation and sequestration.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Centrifugation, Density Gradient; Cyclic AMP; Enzyme Activation; Estradiol; Female; GTP-Binding Proteins; Hypothalamus; Isoproterenol; Phosphoprotein Phosphatases; Phosphorylation; Preoptic Area; Propanolamines; Protamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 2000 |
Differential alterations in cardiac adrenergic signaling in chronic hypoxia or norepinephrine infusion.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Cholera Toxin; Chronic Disease; Colforsin; GTP-Binding Proteins; Guanosine Triphosphate; Heart Rate; Heart Ventricles; Hypertrophy, Left Ventricular; Hypertrophy, Right Ventricular; Hypoxia; Isoproterenol; Male; Myocardium; Norepinephrine; Pertussis Toxin; Propanolamines; Protein Kinase C; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Signal Transduction; Sodium Fluoride; Sympathomimetics; Tritium; Virulence Factors, Bordetella; Weight Gain | 2001 |
Abolition of (-)-CGP 12177-evoked cardiostimulation in double beta1/beta2-adrenoceptor knockout mice. Obligatory role of beta1-adrenoceptors for putative beta4-adrenoceptor pharmacology.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Binding, Competitive; Bucladesine; Dose-Response Relationship, Drug; Female; Genotype; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Membranes; Mice; Mice, Knockout; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sinoatrial Node; Tritium | 2001 |
Lipolytic and antilipolytic responses of the Siberian hamster (Phodopus sungorus sungorus) white adipocytes after weight loss induced by short photoperiod exposure.
Topics: Adipocytes; Adipose Tissue; Adrenergic beta-Agonists; Adrenocorticotropic Hormone; Animals; Cricetinae; DNA; Epinephrine; Ethanolamines; Isoproterenol; Lipolysis; Male; Norepinephrine; Peptide YY; Phodopus; Photoperiod; Propanolamines; Sympathomimetics; Weight Gain; Weight Loss | 1998 |
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 2001 |
Selective inhibition of beta(2)-adrenergic receptor-mediated cAMP generation by activation of the P2Y(2) receptor in mouse pineal gland tumor cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine Diphosphate; Adenosine Triphosphate; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Bombesin; Calcium; Cyclic AMP; Extracellular Space; Isoproterenol; Mice; Pertussis Toxin; Phosphodiesterase Inhibitors; Pinealoma; Propanolamines; Receptors, Adrenergic, beta-2; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Signal Transduction; Thionucleotides; Tritium; Tumor Cells, Cultured; Uridine Triphosphate; Virulence Factors, Bordetella | 2001 |
Beta(3)-adrenoceptors control Cl(-) conductance in rabbit nasal epithelium.
Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Amiloride; Animals; Chlorides; Isoproterenol; Membrane Potentials; Nasal Mucosa; Propanolamines; Rabbits; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes | 2001 |
Beta-adrenergic receptors and adenylate cyclase activity in the parotid acinar cells from acute streptozotocin-induced diabetic rats.
Topics: Adenylyl Cyclases; Amylases; Animals; Diabetes Mellitus, Experimental; Enzyme Activation; Isoproterenol; Male; Norepinephrine; Parotid Gland; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Streptozocin | 2000 |
Quantitative determination of cell surface beta-adrenoceptors in different rat skeletal muscles.
Topics: Adrenergic beta-Agonists; Animals; In Vitro Techniques; Isoproterenol; Kinetics; Male; Muscle Contraction; Muscle Fibers, Fast-Twitch; Muscle Fibers, Slow-Twitch; Muscle, Skeletal; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Cell Surface; Stimulation, Chemical | 2002 |
Sex-dependent thermogenesis, differences in mitochondrial morphology and function, and adrenergic response in brown adipose tissue.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Weight; Bucladesine; Calorimetry, Indirect; Colforsin; DNA; Female; Isoproterenol; Light; Lipolysis; Male; Mitochondria; Norepinephrine; Organ Size; Oxygen Consumption; Propanolamines; Rats; Rats, Wistar; Respiratory Mechanics; Sex Characteristics; Thermogenesis; Triglycerides | 2002 |
Evidence for the primary role for 4-aminopyridine-sensitive K(v) channels in beta(3)-adrenoceptor-mediated, cyclic AMP-independent relaxations of guinea-pig gastrointestinal smooth muscles.
Topics: 4-Aminopyridine; Adrenergic Agonists; Animals; Catecholamines; Cyclic AMP; Epinephrine; Ethanolamines; Guinea Pigs; In Vitro Techniques; Ion Channel Gating; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Propanolamines; Receptors, Adrenergic, beta-3 | 2003 |
Intrinsic sympathomimetic activity of (-)-pindolol mediated through a (-)-propranolol-resistant site of the beta1-adrenoceptor in human atrium and recombinant receptors.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Animals; Binding Sites; CHO Cells; Cricetinae; Cyclic AMP; Drug Interactions; Drug Resistance; Female; Heart; Heart Atria; Humans; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Norepinephrine; omega-N-Methylarginine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Recombinant Proteins; Stereoisomerism; Sympathomimetics | 2003 |
Characterization of beta 3-adrenoceptor-mediated relaxation in rat abdominal aorta smooth muscle.
Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Animals; Aorta, Abdominal; Dose-Response Relationship, Drug; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth, Vascular; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-3; Vasoconstriction; Vasodilation | 2003 |
Markedly reduced effects of (-)-isoprenaline but not of (-)-CGP12177 and unchanged affinity of beta-blockers at Gly389-beta1-adrenoceptors compared to Arg389-beta1-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Arginine; Cricetinae; Dose-Response Relationship, Drug; Glycine; Humans; Isoproterenol; Polymorphism, Genetic; Propanolamines; Protein Binding; Receptors, Adrenergic, beta-1 | 2004 |
Aspartate138 is required for the high-affinity ligand binding site but not for the low-affinity binding site of the beta1-adrenoceptor.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aspartic Acid; Binding Sites; Bupranolol; CHO Cells; Cricetinae; Cricetulus; Drug Interactions; Isoproterenol; Ligands; Propanolamines; Receptors, Adrenergic, beta-1 | 2004 |
The effect of the farnesyl protein transferase inhibitor SCH66336 on isoprenylation and signalling by the prostacyclin receptor.
Topics: Adrenergic beta-Agonists; Alkyl and Aryl Transferases; Amino Acid Motifs; Animals; Calcium Signaling; Carrier Proteins; Cell Line; Cell Line, Tumor; Cyclic AMP; Dose-Response Relationship, Drug; Endocytosis; Epoprostenol; Farnesyltranstransferase; Heat-Shock Proteins; HSP40 Heat-Shock Proteins; Humans; Iloprost; Isoproterenol; Kidney; Leukemia, Erythroblastic, Acute; Mice; Mutagenesis, Site-Directed; Organophosphorus Compounds; Piperidines; Proline; Propanolamines; Protein Prenylation; Protein Processing, Post-Translational; Proto-Oncogene Proteins p21(ras); Pyridines; Receptors, Adrenergic, beta-2; Receptors, Epoprostenol; Receptors, Thromboxane A2, Prostaglandin H2; Recombinant Fusion Proteins; Signal Transduction; Transfection | 2005 |
Beta-adrenoceptor-mediated vascular relaxation in spontaneously hypertensive rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Tetrahydronaphthalenes | 2005 |
Evidence for two atypical conformations of beta-adrenoceptors and their interaction with Gi proteins.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Norepinephrine; Pertussis Toxin; Propanolamines; Protein Binding; Protein Conformation; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1 | 2005 |
Characterization of isoprenaline- and salmeterol-stimulated interactions between beta2-adrenoceptors and beta-arrestin 2 using beta-galactosidase complementation in C2C12 cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Arrestins; beta-Arrestin 2; beta-Arrestins; beta-Galactosidase; Cell Line; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Genetic Complementation Test; Humans; Isoproterenol; Mutation; Propanolamines; Propranolol; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Salmeterol Xinafoate; Transfection | 2005 |
Relaxant effects of beta-adrenergic agonists on porcine and human detrusor muscle.
Topics: Adrenergic beta-Agonists; Aged; Albuterol; Animals; Dioxoles; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Humans; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Procaterol; Propanolamines; Swine | 2005 |
Effects of gender, age and hypertension on beta-adrenergic receptor function in rat urinary bladder.
Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Age Factors; Animals; Ethanolamines; Female; Hypertension; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Wistar; Receptors, Adrenergic, beta; Sex Factors; Urinary Bladder; Urinary Incontinence | 2006 |
Recruitment of functionally active heart beta2-adrenoceptors in the initial phase of endotoxic shock in pithed rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiovascular Physiological Phenomena; Fenoterol; Heart Rate; Isoproterenol; Lipopolysaccharides; Male; Myocardium; Prenalterol; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Shock, Septic; Tachycardia | 2006 |
Effect of (R)-2-(2-aminothiazol-4-yl)-4'-{2-[(2-hydroxy-2-phenylethyl)amino]ethyl} acetanilide (YM178), a novel selective beta3-adrenoceptor agonist, on bladder function.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Animals; Carbachol; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Humans; Isoproterenol; Muscle Contraction; Propanolamines; Thiazoles; Urinary Bladder | 2007 |
The effects of both noradrenaline and CGP12177, mediated through human beta1 -adrenoceptors, are reduced by PDE3 in human atrium but PDE4 in CHO cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adrenergic beta-Agonists; Aged; Animals; Atrial Appendage; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Drug Synergism; Female; Humans; Isometric Contraction; Isoproterenol; Male; Middle Aged; Norepinephrine; Phosphodiesterase Inhibitors; Propanolamines; Quinolones; Receptors, Adrenergic, beta-1; Rolipram; Signal Transduction | 2007 |
In vitro and in vivo pharmacological characterization of ethyl-4-[trans-4-[((2S)-2-hydroxy-3-[4-hydroxy-3[(methylsulfonyl)amino]-phenoxy]propyl) amino]cyclohexyl]benzoate hydrochloride (SAR150640), a new potent and selective human beta3-adrenoceptor agoni
Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Benzoates; Binding, Competitive; Cell Line; Cell Line, Tumor; Cells, Cultured; Cyclic AMP; Female; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Isoproterenol; Macaca fascicularis; Molecular Structure; Myometrium; Obstetric Labor, Premature; Oxytocin; Pregnancy; Propanolamines; Receptors, Adrenergic, beta-3; Sulfonamides; Tocolytic Agents; Transfection; Uterine Contraction; Vasotocin | 2007 |
Studies on the mechanisms underlying beta-adrenoceptor-mediated relaxation of rat abdominal aorta.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Abdominal; Cyclic AMP; In Vitro Techniques; Isoproterenol; Large-Conductance Calcium-Activated Potassium Channels; Male; Muscle Relaxation; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 2006 |
Relaxation of human detrusor muscle by selective beta-2 and beta-3 agonists and endogenous catecholamines.
Topics: Adrenergic beta-Agonists; Aged; Catecholamines; Clenbuterol; Dose-Response Relationship, Drug; Ethanolamines; Female; Humans; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Terbutaline; Urinary Bladder | 2007 |
Phosphodiesterases PDE3 and PDE4 jointly control the inotropic effects but not chronotropic effects of (-)-CGP12177 despite PDE4-evoked sinoatrial bradycardia in rat atrium.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Animals; Arrhythmia, Sinus; Atrial Function, Left; Atrial Function, Right; Bradycardia; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Drug Partial Agonism; Female; Heart Atria; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Propanolamines; Quinolones; Rats; Rats, Sprague-Dawley; Rolipram; Stimulation, Chemical; Tachycardia | 2009 |
Adrenoceptors and adaptive mechanisms in the heart during stress.
Topics: Adaptation, Physiological; Adrenergic beta-Agonists; Adult; Animals; Epinephrine; Female; Heart; Homeostasis; Humans; Isoproterenol; Male; Myocytes, Cardiac; Norepinephrine; Propanolamines; Protein Isoforms; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction; Stress, Psychological | 2008 |
Do gene polymorphisms alone or in combination affect the function of human beta3-adrenoceptors?
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Binding, Competitive; Biphenyl Compounds; Cell Line; Cyclic AMP; Humans; Isoproterenol; Mutagenesis, Site-Directed; Norepinephrine; Phenethylamines; Polymorphism, Single Nucleotide; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-3; Thiazoles; Transfection | 2009 |
Regional quantification of muscarinic acetylcholine receptors and β-adrenoceptors in human airways.
Topics: Aged; Carbachol; Female; Humans; In Vitro Techniques; Isoproterenol; Ligands; Lung; Male; Middle Aged; Muscle Contraction; N-Methylscopolamine; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic | 2012 |
Autoantibodies against cardiac β(1)-adrenoceptor do not affect the low-affinity state β(1)-adrenoceptor-mediated inotropy in rat cardiomyocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Animals; Autoantibodies; Bisoprolol; Isoproterenol; Male; Myocardial Contraction; Myocytes, Cardiac; Phosphodiesterase Inhibitors; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1 | 2012 |
β₃-Adrenergic regulation of L-type Ca²⁺ current and force of contraction in human ventricle.
Topics: Adolescent; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adult; Aged; Aged, 80 and over; Aminophenols; Biomechanical Phenomena; Calcium Channels, L-Type; Calcium Signaling; Female; Heart Ventricles; Humans; Isoproterenol; Male; Membrane Potentials; Middle Aged; Myocardial Contraction; Nitric Oxide Synthase; Patch-Clamp Techniques; Phosphoric Diester Hydrolases; Propanolamines; Receptors, Adrenergic, beta-3; Sulfonamides; Young Adult | 2014 |
Pharmacological properties of β-adrenoceptors mediating rat superior mesenteric artery relaxation and the effects of chemical sympathetic denervation.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Isoproterenol; Male; Mesenteric Artery, Superior; Muscle Relaxation; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Sympathectomy, Chemical | 2020 |