isoproterenol has been researched along with brl 37344 in 107 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (1.87) | 18.7374 |
1990's | 66 (61.68) | 18.2507 |
2000's | 33 (30.84) | 29.6817 |
2010's | 5 (4.67) | 24.3611 |
2020's | 1 (0.93) | 2.80 |
Authors | Studies |
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Bloom, JD; Burns, MG; Claus, TH; Dolan, JA; Dutia, MD; Johnson, BD; Largis, EE; Wissner, A | 1 |
Guillaume, JL; Méjean, A; Strosberg, AD | 1 |
Akahane, M; Akahane, S; Hirabayashi, A; Miyata, H; Mukaiyama, H; Muranaka, H; Tamai, T; Tanaka, N | 1 |
Akahane, M; Akahane, S; Hirabayashi, A; Ishikawa, T; Kobayashi, J; Mukaiyama, H; Muranaka, H; Tamai, T; Tanaka, N | 1 |
Hoffmann, C; Klotz, KN; Leitz, MR; Lohse, MJ; Oberdorf-Maass, S | 1 |
Bleve, L; Colabufo, NA; Jockers, R; Milazzo, FM; Perrone, MG; Santandrea, E; Sciarroni, AF; Scilimati, A; Vitale, P | 1 |
Dauzats, M; Lafontan, M; Langin, D; Portillo, M | 1 |
Kompa, AR; Molenaar, P; Pak, HS; Roberts, SJ; Summers, RJ | 1 |
Van Liefde, I; Van Witzenburg, A; Vauquelin, G | 1 |
Belfrage, P; Ekholm, D; Lafontan, M; Langin, D; Ridderstråle, M | 1 |
Bond, RA; Vanhoutte, PM | 1 |
Canfield, P; Paraskeva, P | 1 |
Esbenshade, TA; Granneman, JG; Han, C; Minneman, KP; Theroux, TL | 1 |
Berlan, M; Bousquet-Melou, A; Galitzky, J; Montastruc, JL; Tavernier, G | 1 |
Fraeyman, N; Van de Velde, E; Van Ermen, A; Vanscheeuwijck, P | 1 |
Brouwer, F; Hollenga, C; Zaagsma, J | 2 |
Baude, B; Emorine, LJ; Fève, B; Krief, S; Pairault, J; Strosberg, AD | 1 |
MacDonald, A; McLaughlin, DP | 1 |
Lafontan, M; Langin, D; Portillo, MP; Saulnier-Blache, JS | 1 |
Chaudhry, A; Granneman, JG; Lahners, KN | 1 |
Deinum, JT; Haas, M; Hollenga, C; Zaagsma, J | 1 |
Granneman, JG | 1 |
Bast, A; Rademaker, B; van der Vliet, A | 1 |
Hollenga, C; Zaagsma, J | 1 |
Fraser, C; Giacobino, JP; Muzzin, P; Seydoux, J; Venter, JC | 1 |
Cawthorne, MA; Giacobino, JP; Klaus, S; Muzzin, P; Revelli, JP; Ricquier, D | 1 |
Cawthorne, MA; Oriowo, MA; Ruffolo, RR; Sennitt, MV; Smith, SA | 1 |
Oriowo, MA | 3 |
Croci, T; Landi, M; Manara, L | 1 |
Bronnikov, G; Mohell, N; Nedergaard, J; Unelius, L | 1 |
Casteilla, L; Giacobino, JP; Muzzin, P; Revelli, JP; Ricquier, D | 1 |
Shen, YT; Vatner, SF; Zhang, H | 1 |
Berlan, M; Bousquet-Melou, A; Galitzky, J; Lafontan, M; Montastruc, JL | 1 |
Chiyotani, A; Konno, K; Takeuchi, S; Tamaoki, J; Yamauchi, F; Yamawaki, I | 1 |
Chiba, S; Furukawa, Y; Inoue, Y; Ren, LM; Sawaki, S; Takayama, S | 1 |
Berlan, M; Carpéné, C; Galitzky, J; Lafontan, M; Portillo, M; Reverte, M | 1 |
Cawthorne, MA; Kirkham, DM; Murphy, GJ; Young, P | 1 |
Brouwer, F; de Boer, RE; Zaagsma, J | 1 |
Baude, B; Emorine, LJ; Fève, B; Krief, S; Pairault, J; Strosberg, AD; Zilberfarb, V | 1 |
Cannon, B; Dicker, A; Nedergaard, J | 1 |
el Borai, N; Ito, K; Nakano, S; Nakazawa, H; Tanaka, E; Yamakawa, A; Yamamura, M | 1 |
Arner, P; Blaak, E; Hoffstedt, J; Lönnqvist, F; Shimizu, M | 1 |
Grant, TL; Holloway, BR; Mayers, RM; Quayle, SP; Thompson, AJ | 1 |
Reverte, M; Rivas-Cabañero, L | 1 |
Feller, DR; Konkar, AA; Lezama, EJ; Miller, DD; Salazar-Bookaman, MM | 1 |
Chang, CJ; Cheng, JT; Kao, JT; Lai, CW; Lee, TL | 1 |
Houston, G; Kelly, J | 1 |
de Boer, RE; Kroezen, PA; Smit, J; Steegstra, MR; Zaagsma, J | 1 |
Dove, J; Matheny, M; Scarpace, PJ | 1 |
Collins, S; Gettys, TW; Taylor, IL; Watson, PM | 1 |
Atgié, C; Bukowiecki, LJ; D'Allaire, F | 1 |
Roberts, SJ; Summers, RJ | 1 |
Bar-Ilan, A; Geyer, O; Lazar, M; Nachman, R; Oron, Y | 1 |
Isono, K; Nagai, A; Tagaya, E; Tamaoki, J | 1 |
Borger, P; Esselink, MT; Hoekstra, Y; Kauffman, HF; Postma, DS; Vellenga, E; Zaagsma, J | 1 |
Balligand, JL; Bril, A; Gauthier, C; Khandoudi, N; Kobzik, L; Le Marec, H; Leblais, V; Trochu, JN | 1 |
de la Lande, IS; Ivar, PM; Marino, V; Parker, DA | 1 |
Gerhardt, CC; Gros, J; Issad, T; Strosberg, AD | 1 |
Ajisawa, Y; Akahane, M; Andersson, KE; Hayakawa, K; Igawa, Y; Nishizawa, O; Takeda, H; Yamazaki, Y; Yoneyama, T | 1 |
Oriowo, MA; Thulesius, O | 1 |
Atgié, C; Berlan, M; Carpéné, C; Fontana, E; Galitzky, J; Lafontan, M | 1 |
Evans, BA; Papaioannou, M; Roberts, SJ; Summers, RJ | 1 |
MacDonald, A; Watt, K | 1 |
Farias-Silva, E; Grassi-Kassisse, DM; Spadari-Bratfisch, RC; Wolf-Nunes, V | 1 |
MacAulay, L; MacDonald, A; McLean, M; Shaw, AM | 1 |
Horinouchi, T; Koike, K | 3 |
Horinouchi, T; Koike, K; Tsujitani, M | 1 |
Mahmoudian, M; Mirkhani, H; Omrani, GR; Shafiei, M | 1 |
Ajisawa, Y; Akahane, M; Igawa, Y; Komatsu, Y; Nishizawa, O; Takeda, H; Yamazaki, Y | 1 |
Carneiro, SM; Markus, RP; Scrivano, CN; Yamanouye, N | 1 |
Amusquivar, E; Cacho, J; Herrera, E | 1 |
Mills, S | 1 |
Brechet, S; Chayvialle, JA; Claustre, J; Cuber, JC; Dumoulin, V; Plaisancié, P | 1 |
Ambid, L; Atgié, C; Carpéné, C; Casteilla, L; Hanoun, N; Le Gouic, S; Marti, L; Pénicaud, L | 1 |
Nunoki, K; Sato, T; Sukegawa, J; Yamada, H; Yanagisawa, T | 1 |
Grassi-Kassisse, DM; Spadari-Bratfisch, RC; Verago, JL | 1 |
Hussein, SM; Khan, I; Oriowo, M | 1 |
Leaver, EV; Pappone, PA | 1 |
Oriowo, MA; Yousif, MH | 1 |
Bosch, RF; Eigenberger, BW; Gogel, J; Hambrock, A; Kiehn, J; Kühlkamp, V; Mewis, C; Rüb, N; Schneck, AC; Seipel, L; Zhang, W | 1 |
Horinouchi, T; Koike, K; Tanaka, Y | 1 |
Cacho, J; Crespo-Solans, MD; del Campo, S; Herrera, E; Ramos, MP | 1 |
Chapple, CR; Chess-Williams, R; Yamanishi, T; Yasuda, K; Yoshida, K | 1 |
Balligand, JL; Dessy, C; Ghisdal, P; Havaux, X; Moniotte, S; Noirhomme, P | 1 |
Chandrasekhar, B; Fatinikun, T; Kadavil, EA; Khan, I; Omu, AE; Oriowo, MA | 1 |
Badawi, JK; Bross, S; Haferkamp, A; Hatzinger, M; Michel, MS; Uecelehan, H | 1 |
Allen, BG; Baragli, A; Boivin, B; Ethier, N; Hébert, TE; Lavoie, C; Trieu, P; Vaniotis, G; Villeneuve, LR | 1 |
Frazier, EP; Michel, MC; Schneider, T | 1 |
Adamo, C; Angelone, T; Cerra, MC; Imbrogno, S; Pulerà, E; Tota, B | 1 |
Badawi, JK; Bross, S; Honeck, P; Kwon, ST; Langbein, S; Seja, T; Uecelehan, H | 1 |
Fu, L; Isobe, K; Kawakami, Y; Suzukawa, K; Takekoshi, K; Zeng, Q | 1 |
Haynes, JM | 1 |
Altan, VM; Arioglu, E; Guner, S; Ozakca, I; Ozcelikay, AT | 1 |
Angelone, T; Cerra, MC; Filice, E; Imbrogno, S; Mannarino, C; Pellegrino, D; Pulerà, E; Quintieri, AM; Recchia, A | 1 |
Arai, Y; Ikeda, Y; Masumiya, H; Nakagawa, H; Nunoki, K; Sato, T; Takemoto, J; Yanagisawa, T | 1 |
Al Zubair, K; Bexis, S; Docherty, JR | 1 |
Kurita, Y; Matsumoto, R; Mizuno, T; Mugiya, S; Otsuka, A; Ozono, S; Shinbo, H; Suzuki, T | 1 |
Calvi, P; D' Agostino, G; Maria Condino, A | 1 |
Bondareva, VM; Derkach, KV; Moyseyuk, IV; Shpakov, AO | 1 |
El-Zohairy, SN; Ezeamuzie, CI; Oriowo, MA | 1 |
Brown, JT; Church, TW; Marrion, NV | 1 |
Aitken-Buck, HM; Babakr, AA; Bunton, RW; Coffey, S; Davis, PJ; Fomison-Nurse, IC; Jones, PP; Lamberts, RR; Stiles, MK; Sugunesegran, R; van Hout, I; Williams, MJA | 1 |
107 other study(ies) available for isoproterenol and brl 37344
Article | Year |
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Disodium (R,R)-5-[2-[[2-(3-chlorophenyl)-2-hydroxyethyl]-amino] propyl]-1,3-benzodioxole-2,2-dicarboxylate (CL 316,243). A potent beta-adrenergic agonist virtually specific for beta 3 receptors. A promising antidiabetic and antiobesity agent.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Animals; Diabetes Mellitus, Type 2; Hypoglycemic Agents; Lipolysis; Male; Mice; Mice, Obese; Obesity; Substrate Specificity | 1992 |
Carazolol: a potent, selective beta 3-adrenoceptor agonist.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; CHO Cells; Cricetinae; Dithiothreitol; Lipolysis; Propanolamines; Receptors, Adrenergic, beta | 1995 |
Discovery of novel N-phenylglycine derivatives as potent and selective beta(3)-adrenoceptor agonists for the treatment of frequent urination and urinary incontinence.
Topics: Adrenergic beta-Agonists; Animals; Blood Pressure; Female; Ferrets; Glycine; Heart Rate; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Pregnancy; Pressure; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Structure-Activity Relationship; Urinary Bladder; Urinary Incontinence; Urination; Uterus | 2001 |
Relationship between stereochemistry and the beta3-adrenoceptor agonistic activity of 4'-hydroxynorephedrine derivative as an agent for treatment of frequent urination and urinary incontinence.
Topics: Administration, Oral; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Colon; Duodenum; Ethanolamines; Heart Rate; In Vitro Techniques; Injections, Intravenous; Male; Muscle Contraction; Norepinephrine; Pressure; Prodrugs; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Stereoisomerism; Structure-Activity Relationship; Tetrahydronaphthalenes; Urinary Bladder; Urinary Incontinence; Urination | 2003 |
Comparative pharmacology of human beta-adrenergic receptor subtypes--characterization of stably transfected receptors in CHO cells.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Humans; Radioligand Assay; Receptors, Adrenergic, beta; Transfection | 2004 |
Stereospecific synthesis and bio-activity of novel beta(3)-adrenoceptor agonists and inverse agonists.
Topics: Adenylyl Cyclases; Adrenergic beta-3 Receptor Agonists; Animals; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Inverse Agonism; Humans; Molecular Structure; Receptors, Adrenergic, beta-3; Stereoisomerism; Structure-Activity Relationship | 2008 |
Drop in the "atypical" beta-adrenergic response and modification of the beta/alpha 2-adrenoceptor balance in fat cells from aging rabbits.
Topics: Adipose Tissue; Adrenocorticotropic Hormone; Aging; Animals; Brimonidine Tartrate; Epinephrine; Ethanolamines; In Vitro Techniques; Isoproterenol; Lipolysis; Propanolamines; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1992 |
Localization of (-)-[125I]cyanopindolol binding in guinea-pig heart: characteristics of non-beta-adrenoceptor related binding in cardiac pacemaker and conducting regions.
Topics: Alprenolol; Animals; Ascorbic Acid; Binding Sites; Ethanolamines; Female; Guinea Pigs; Haloperidol; Heart Conduction System; Isoproterenol; Male; Myocardium; Peroxidase; Phentolamine; Pindolol; Propanolamines; Propranolol; Protein Binding; Receptors, Adrenergic, beta; Serotonin; Thiophenes; Trachea | 1992 |
Multiple beta adrenergic receptor subclasses mediate the l-isoproterenol-induced lipolytic response in rat adipocytes.
Topics: Adipose Tissue; Animals; Dose-Response Relationship, Drug; Ethanolamines; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1992 |
cAMP-dependent protein kinase activation mediated by beta 3-adrenergic receptors parallels lipolysis in rat adipocytes.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adipose Tissue; Adrenergic beta-Agonists; Animals; Cyclic AMP; Cyclic GMP; Enzyme Activation; Ethanolamines; Isoproterenol; Lipolysis; Male; Protein Kinases; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1992 |
Interaction of tertatolol at the "atypical" or beta 3-adrenoceptor in guinea-pig ileum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Electric Stimulation; Ethanolamines; Guinea Pigs; Ileum; In Vitro Techniques; Isoproterenol; Male; Methiothepin; Muscle Contraction; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Thiophenes | 1992 |
Beta-adrenoceptor agonist stimulation of acid secretion by rat stomach in vitro is mediated by 'atypical' beta-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Ethanolamines; Gastric Acid; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Stomach; Tetrahydronaphthalenes | 1992 |
Coexisting beta 1- and atypical beta-adrenergic receptors cause redundant increases in cyclic AMP in human neuroblastoma cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Neuroblastoma; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured | 1992 |
The positive chronotropic effect induced by BRL 37344 and CGP 12177, two beta-3 adrenergic agonists, does not involve cardiac beta adrenoceptors but baroreflex mechanisms.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Animals; Dogs; Ethanolamines; Heart Rate; Isoproterenol; Lipolysis; Male; Pressoreceptors; Propanolamines; Receptors, Adrenergic, beta; Reflex; Stimulation, Chemical | 1992 |
Pharmacological characterization of a beta 3-receptor agonist (BRL 37,344) and a partial agonist (CGP 12,177A) in neonatal rat liver plasma membranes.
Topics: Adenylyl Cyclase Inhibitors; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Binding, Competitive; Cell Membrane; Enzyme Activation; Ethanolamines; Humans; Isoproterenol; Liver; Propanolamines; Rats; Rats, Wistar | 1992 |
Relationship between lipolysis and cyclic AMP generation mediated by atypical beta-adrenoceptors in rat adipocytes.
Topics: Adipocytes; Animals; Cattle; Cyclic AMP; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1991 |
Inhibition by dexamethasone of beta 3-adrenergic receptor responsiveness in 3T3-F442A adipocytes. Evidence for a transcriptional mechanism.
Topics: 3T3 Cells; Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Animals; Base Sequence; Cell Membrane; Dexamethasone; Dose-Response Relationship, Drug; Ethanolamines; Isoproterenol; Kinetics; Mice; Mifepristone; Molecular Sequence Data; Oligodeoxyribonucleotides; Oligonucleotides, Antisense; Polymerase Chain Reaction; Progesterone; Propanolamines; Receptors, Adrenergic, beta; RNA; Transcription, Genetic | 1992 |
Characterization of catecholamine-mediated relaxations in rat isolated gastric fundus: evidence for an atypical beta-adrenoceptor.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Catecholamines; Ethanolamines; Gastric Fundus; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Norepinephrine; Pindolol; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Coexistence of three beta-adrenoceptor subtypes in white fat cells of various mammalian species.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cricetinae; Dogs; Ethanolamines; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lipolysis; Male; Mesocricetus; Muscle, Smooth; Pindolol; Propanolamines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Molecular cloning and expression of the rat beta 3-adrenergic receptor.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Sequence; Animals; Base Sequence; CHO Cells; Cloning, Molecular; Cricetinae; Enzyme Activation; Epinephrine; Ethanolamines; Gene Expression; Humans; Isoproterenol; Male; Molecular Sequence Data; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection | 1991 |
Differences in functional cyclic AMP compartments mediating lipolysis by isoprenaline and BRL 37344 in four adipocyte types.
Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Animals; Cattle; Cells, Cultured; Cyclic AMP; Enzyme Activation; Ethanolamines; Fatty Acids, Nonesterified; Humans; Isoproterenol; Lipolysis; Rats; Rats, Inbred Strains; Rats, Zucker; Stimulation, Chemical | 1991 |
Discrepancies in lipolytic activities induced by beta-adrenoceptor agonists in human and rat adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Aged; Alprenolol; Animals; Catecholamines; Ethanolamines; Fatty Acids, Nonesterified; Female; Glycerol; Humans; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Middle Aged; Rats; Rats, Inbred Strains; Stereoisomerism | 1990 |
Norepinephrine and BRL 37344 stimulate adenylate cyclase by different receptors in rat brown adipose tissue.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cold Temperature; Ethanolamines; Isoproterenol; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic | 1990 |
A beta adrenoceptor with atypical characteristics is involved in the relaxation of the rat small intestine.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Ethanolamines; In Vitro Techniques; Intestine, Small; Iodocyanopindolol; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Pindolol; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1990 |
Direct evidence for the atypical nature of functional beta-adrenoceptors in rat adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Epididymis; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1989 |
Discrepancies between the affinities of binding and action of the novel beta-adrenergic agonist BRL 37344 in rat brown adipose tissue.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Agonists; Animals; Binding, Competitive; Cell Membrane; Ethanolamines; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Oxygen Consumption; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reference Values | 1988 |
Control of beta 3-adrenergic receptor gene expression in brown adipocytes in culture.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Animals; Base Sequence; Cell Differentiation; Cells, Cultured; Cricetinae; Ethanolamines; Gene Expression Regulation; Half-Life; Isoproterenol; Molecular Sequence Data; Phodopus; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1995 |
The beta-adrenoceptor selectivity profile of BRL 37344 in the pithed rat.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Animals; Blood Pressure; Decerebrate State; Dose-Response Relationship, Drug; Ethanolamines; Female; Heart Rate; Isoproterenol; Oxygen Consumption; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Stereoisomerism | 1994 |
Atypical beta-adrenoceptors in the rat isolated common carotid artery.
Topics: Adrenergic beta-Agonists; Albuterol; Animals; Carotid Artery, Common; Dose-Response Relationship, Drug; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Male; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1994 |
Similar atypical beta-adrenergic receptors mediate in vitro rat adipocyte lipolysis and colonic motility inhibition.
Topics: Adipocytes; Adrenergic beta-Agonists; Alprenolol; Animals; Atrial Function; Colon; Ethanolamines; Gastrointestinal Motility; Guinea Pigs; Heart Atria; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Rats; Receptors, Adrenergic, beta; Tetrahydronaphthalenes; Trachea | 1993 |
Physiological desensitization of beta 3-adrenergic responses in brown fat cells: involvement of a postreceptor process.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Acclimatization; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cells, Cultured; Cold Temperature; Colforsin; Cricetinae; Cyclic AMP; Ethanolamines; Isoproterenol; Kinetics; Male; Mesocricetus; Norepinephrine; Oxygen Consumption; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1993 |
Expression of beta 1- and beta 3-adrenergic-receptor messages and adenylate cyclase beta-adrenergic response in bovine perirenal adipose tissue during its transformation from brown into white fat.
Topics: Adenylyl Cyclases; Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Aging; Amino Acid Sequence; Animals; Cattle; DNA Probes; Ethanolamines; Gene Expression; Isoproterenol; Molecular Sequence Data; Polymerase Chain Reaction; Receptors, Adrenergic, beta; RNA, Messenger | 1994 |
Peripheral vascular effects of beta-3 adrenergic receptor stimulation in conscious dogs.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Dogs; Ethanolamines; Female; Hemodynamics; Isoproterenol; Male; Nitric Oxide; Regional Blood Flow | 1994 |
Beta-3 adrenoceptor-mediated increase in cutaneous blood flow in the dog.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Bupranolol; Dioxoles; Dogs; Ethanolamines; Heart Rate; Isoproterenol; Male; Nitroprusside; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Regional Blood Flow; Skin | 1994 |
Atypical beta-adrenoceptor- (beta 3-adrenoceptor) mediated relaxation of canine isolated bronchial smooth muscle.
Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Bronchi; Cyclic AMP; Dogs; Ethanolamines; Female; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1993 |
Positive chronotropic and inotropic responses to BRL 37344, a beta 3-adrenoceptor agonist in isolated, blood-perfused dog atria.
Topics: Adrenergic beta-Agonists; Animals; Dogs; Dose-Response Relationship, Drug; Ethanolamines; Heart Rate; Isoproterenol; Myocardial Contraction | 1993 |
Coexistence of beta 1-, beta 2-, and beta 3-adrenoceptors in dog fat cells and their differential activation by catecholamines.
Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamines; Cell Membrane; Dogs; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Isoproterenol; Norepinephrine; Procaterol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tetrahydronaphthalenes | 1993 |
Correlation of beta 3-adrenoceptor-induced activation of cyclic AMP-dependent protein kinase with activation of lipolysis in rat white adipocytes.
Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Amino Acid Sequence; Animals; Cells, Cultured; Cyclic AMP; Enzyme Activation; Ethanolamines; Glycerol; Isoproterenol; Lipolysis; Molecular Sequence Data; Protein Kinases; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Substrate Specificity | 1993 |
The beta-adrenoceptors mediating relaxation of rat oesophageal muscularis mucosae are predominantly of the beta 3-, but also of the beta 2-subtype.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Esophagus; Ethanolamines; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1993 |
Transcriptional modulation by n-butyric acid of beta 1-, beta 2-, and beta 3-adrenergic receptor balance in 3T3-F442A adipocytes.
Topics: 3T3 Cells; Adenylyl Cyclase Inhibitors; Adipocytes; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Animals; Base Sequence; Butyrates; Butyric Acid; DNA Primers; DNA, Complementary; Ethanolamines; Gene Expression Regulation; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Molecular Sequence Data; Oligonucleotides, Antisense; Pindolol; Polymerase Chain Reaction; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Transcription, Genetic | 1994 |
Different atypical beta-adrenoceptors mediate isoprenaline-induced relaxation in vascular and non-vascular smooth muscles.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Pindolol; Rats; Receptors, Adrenergic, beta | 1995 |
Stimulation of nonshivering thermogenesis in the Syrian hamster by norepinephrine and beta-selective adrenergic agents: a phenomenon of refractoriness.
Topics: Acclimatization; Adipose Tissue, Brown; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Cold Temperature; Cricetinae; Drug Interactions; Ethanolamines; Female; Isoproterenol; Male; Mesocricetus; Norepinephrine; Oxygen Consumption; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Reproducibility of Results; Shivering | 1996 |
Regulation of heat production of brown adipocytes via typical and atypical beta-adrenoceptors in the rat.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Calorimetry; Ethanolamines; In Vitro Techniques; Isoproterenol; Male; Phenoxyacetates; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1995 |
Effects of several putative beta 3-adrenoceptor agonists on lipolysis in human omental adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Catechols; Dioxoles; Ethanolamines; Glycerol; Humans; Isoproterenol; Lipolysis; Omentum; Propanolamines; Serine | 1996 |
The acid metabolite of ZD7114 is a partial agonist of lipolysis mediated by the rat beta 3-adrenoceptor.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Dose-Response Relationship, Drug; Ethanolamines; Isoproterenol; Lipolysis; Male; Phenoxyacetates; Phenoxypropanolamines; Rats; Rats, Wistar | 1996 |
Effects of the beta 3-adrenoceptor agonist BRL 37344 on lipomobilization and plasma glucose levels in conscious fasted rabbits.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Biological Transport; Blood Glucose; Ethanolamines; Fasting; Fatty Acids, Nonesterified; Insulin; Isoproterenol; Lactic Acid; Male; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Sodium Chloride | 1996 |
Pharmacological study of atypical beta-adrenoceptors in rat esophageal smooth muscle.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Carbachol; Clenbuterol; Cyclohexane Monoterpenes; Esophagus; Ethanolamines; Female; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Phenoxyacetates; Phenoxypropanolamines; Pindolol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Serotonin Antagonists; Trachea; Tretoquinol | 1996 |
Comparison of isoproterenol with BRL37344 in activation of beta 3-adrenoceptors to inhibit the uptake of [14C]deoxy-D-glucose and translocation of glucose transporter (GLUT4) to membrane fraction in rat adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Blotting, Western; Carbon Radioisotopes; Cell Membrane; Deoxyglucose; Dose-Response Relationship, Drug; Ethanolamines; Glucose Transporter Type 4; Hypoglycemic Agents; Insulin; Isoproterenol; Male; Monosaccharide Transport Proteins; Muscle Proteins; Rats; Rats, Wistar | 1996 |
Beta 3-adrenoceptors mediating relaxation of the oesophageal tunica muscularis mucosae and distal colon in the rat: comparative pharmacology and their desensitization by BRL 37344.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dose-Response Relationship, Drug; Esophagus; Ethanolamines; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1996 |
Influence of adrenodemedullation on beta 2- and beta 3-adrenoceptors mediating relaxation of oesophageal smooth muscle of spontaneously hypertensive rats.
Topics: Adrenal Medulla; Adrenalectomy; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Esophagus; Ethanolamines; Fenoterol; Hypertension; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Propanolamines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1996 |
Effects of age on beta adrenergic subtype activation of adenylyl cyclase in brown adipose tissue.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Agonists; Age Factors; Animals; Colforsin; Dose-Response Relationship, Drug; Enzyme Activation; Ethanolamines; Gene Expression; Glucagon; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; Regression Analysis; RNA, Messenger; Sodium Fluoride | 1996 |
Beta(3)-adrenoceptors mediate smooth muscle relaxation in the rat lower oesophageal sphincter.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbachol; Esophagogastric Junction; Ethanolamines; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Nitroarginine; Potassium Channel Blockers; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1997 |
RU-486 (Mifepristone) ameliorates diabetes but does not correct deficient beta-adrenergic signalling in adipocytes from mature C57BL/6J-ob/ob mice.
Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Animals; Blood Glucose; Blotting, Northern; Blotting, Western; Colforsin; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Enzyme Activation; Ethanolamines; Glucose Transporter Type 4; GTP-Binding Protein alpha Subunits, Gs; Hormone Antagonists; Insulin; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mifepristone; Monosaccharide Transport Proteins; Muscle Proteins; Phenotype; Receptors, Adrenergic, beta; Receptors, Glucocorticoid; Signal Transduction | 1997 |
Role of beta1- and beta3-adrenoceptors in the regulation of lipolysis and thermogenesis in rat brown adipocytes.
Topics: Adipocytes; Adipose Tissue, Brown; Adrenergic alpha-Agonists; Animals; Body Temperature Regulation; Cells, Cultured; Dioxoles; Dobutamine; Epinephrine; Ethanolamines; Female; Isoproterenol; Lipolysis; Norepinephrine; Oxygen Consumption; Procaterol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1997 |
Cyclic AMP accumulation in rat soleus muscle: stimulation by beta2- but not beta3-adrenoceptors.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Catecholamines; Cyclic AMP; Ethanolamines; Indicators and Reagents; Isoproterenol; Male; Muscle, Skeletal; Osmotic Pressure; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1998 |
Beta3-adrenergic relaxation of bovine iris sphincter.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Bupranolol; Cattle; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Ethanolamines; Iris; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1998 |
Atypical adrenoceptor-mediated relaxation of canine pulmonary artery through a cAMP-dependent pathway.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cyclic AMP; Dioxoles; Dogs; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Pindolol; Propanolamines; Pulmonary Artery; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1998 |
Beta-adrenoceptor-mediated inhibition of IFN-gamma, IL-3, and GM-CSF mRNA accumulation in activated human T lymphocytes is solely mediated by the beta2-adrenoceptor subtype.
Topics: Concanavalin A; Cyclic AMP; Ethanolamines; Fenoterol; Gene Expression Regulation; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Interferon-gamma; Interleukin-3; Interleukin-4; Isoproterenol; Receptors, Adrenergic, beta-2; RNA, Messenger; T-Lymphocytes; Timolol | 1998 |
The negative inotropic effect of beta3-adrenoceptor stimulation is mediated by activation of a nitric oxide synthase pathway in human ventricle.
Topics: Adrenergic beta-Agonists; Arginine; Cyclic GMP; Ethanolamines; Female; Heart; Heart Ventricles; Humans; Isoproterenol; Kinetics; Male; Middle Aged; Myocardial Contraction; Myocardium; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Nitroarginine; Norepinephrine; omega-N-Methylarginine; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1998 |
Modulation by presynaptic beta-adrenoceptors of noradrenaline release from sympathetic nerves in human dental pulp.
Topics: Adolescent; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Adult; Albuterol; Anti-Inflammatory Agents; Corticosterone; Dental Pulp; Desipramine; Electric Stimulation; Ethanolamines; Female; Humans; Isoproterenol; Male; Norepinephrine; Propranolol; Radiopharmaceuticals; Receptors, Adrenergic, beta; Receptors, Presynaptic; Sympathetic Nervous System; Sympatholytics; Sympathomimetics; Tritium; Yohimbine | 1998 |
Stimulation of the extracellular signal-regulated kinase 1/2 pathway by human beta-3 adrenergic receptor: new pharmacological profile and mechanism of activation.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Colforsin; Cricetinae; Dioxoles; Enzyme Activation; Epinephrine; Ethanolamines; Humans; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Norepinephrine; Phentolamine; Prazosin; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction; Yohimbine | 1999 |
Functional and molecular biological evidence for a possible beta3-adrenoceptor in the human detrusor muscle.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colforsin; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 1999 |
Functional characterization of beta-adrenoceptors mediating relaxation in sheep gallbladder.
Topics: Adrenergic beta-Agonists; Animals; Ethanolamines; Female; Gallbladder; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Receptors, Adrenergic, beta; Sheep | 1999 |
Selective activation of beta3-adrenoceptors by octopamine: comparative studies in mammalian fat cells.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adult; Animals; Binding, Competitive; Biogenic Amines; Bupranolol; CHO Cells; Cricetinae; Dioxoles; Dogs; Ethanolamines; Female; Gene Expression; Guinea Pigs; Humans; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lipolysis; Male; Mammals; Mesocricetus; Norepinephrine; Octopamine; Oxygen Consumption; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Species Specificity | 1999 |
Characterization of beta-adrenoceptor mediated smooth muscle relaxation and the detection of mRNA for beta1-, beta2- and beta3-adrenoceptors in rat ileum.
Topics: Adenylate Cyclase Toxin; Animals; Colforsin; Dioxoles; Dose-Response Relationship, Drug; Ethanolamines; Ileum; Isoproterenol; Male; Muscle Relaxation; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Virulence Factors, Bordetella | 1999 |
Characterisation of the atypical beta-adrenoceptor in rabbit isolated jejunum using BRL 37344, cyanopindolol and SR 59230A.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Jejunum; Male; Pindolol; Propanolamines; Propranolol; Rabbits; Receptors, Adrenergic, beta | 1999 |
Stress-induced alteration in the lipolytic response to beta-adrenoceptor agonists in rat white adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Body Weight; Bucladesine; Eating; Epinephrine; Ethanolamines; Glycerol; Isoproterenol; Lipolysis; Male; Metoprolol; Norepinephrine; Propanolamines; Rats; Rats, Wistar; Stress, Physiological | 1999 |
Effects of propranolol and L-NAME on beta-adrenoceptor-mediated relaxation in rat carotid artery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic beta-Agonists; Animals; Carotid Artery, Common; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Phenylacetates; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Thromboxane A2; Vasoconstrictor Agents | 1999 |
Pharmacological analysis of atypical beta-adrenoceptors in the guinea pig gastric fundus using the beta(3)-adrenoceptor antagonist bupranolol.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Bupranolol; Butoxamine; Catecholamines; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3 | 1999 |
[Pharmacological analysis of atypical beta-adrenoceptors in the guinea pig gastrointestinal tissue systems].
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Digestive System; Duodenum; Epinephrine; Ethanolamines; Gastric Fundus; Guinea Pigs; Ileum; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta | 1999 |
Effects of different vasodilators on human internal mammary artery in vitro.
Topics: Ethanolamines; Female; Humans; In Vitro Techniques; Isoproterenol; Isosorbide Dinitrate; Male; Mammary Arteries; Middle Aged; Myocardial Ischemia; Nifedipine; Phenylephrine; Potassium Chloride; Propranolol; Vasoconstrictor Agents; Vasodilator Agents | 1999 |
Partial agonist activity of carteolol on atypical beta-adrenoceptors in the guinea pig duodenum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Carteolol; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Vasodilator Agents | 2000 |
Characterization of beta-adrenoceptor subtypes in the ferret urinary bladder in vitro and in vivo.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Anesthesia; Animals; Blood Pressure; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Ethanolamines; Ferrets; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pressure; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Time Factors; Urinary Bladder | 2000 |
Characterization of beta-adrenoceptors responsible for venom production in the venom gland of the snake Bothrops jararaca.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Bothrops; Crotalid Venoms; Cyclic AMP; Dioxoles; Ethanolamines; Exocrine Glands; Female; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Membranes; Metoprolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2000 |
Changes in dietary fatty acids modify the decreased lipolytic beta3-adrenergic response to hyperinsulinemia in adipocytes from pregnant and nonpregnant rats.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Dietary Fats; Epinephrine; Ethanolamines; Fatty Acids; Female; Fish Oils; Glucose Clamp Technique; Hyperinsulinism; Isoproterenol; Lipolysis; Olive Oil; Phospholipids; Plant Oils; Pregnancy; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 2000 |
Beta-adrenergic receptor subtypes mediating lipolysis in porcine adipocytes. Studies with BRL-37344, a putative beta3-adrenergic agonist.
Topics: Adenylyl Cyclases; Adipocytes; Adrenergic beta-Agonists; Animals; Cell Fractionation; Dihydroalprenolol; Ethanolamines; Intracellular Membranes; Isoproterenol; Lipolysis; Muscle, Skeletal; Receptors, Adrenergic, beta; Swine | 2000 |
Involvement of beta1- and beta2- but not beta3-adrenoceptor activation in adrenergic PYY secretion from the isolated colon.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Colon; Dobutamine; Ethanolamines; Isoproterenol; Male; Models, Animal; Organ Culture Techniques; Peptide YY; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Statistics, Nonparametric; Terbutaline; Tetrahydronaphthalenes | 2001 |
Lipolytic and antilipolytic responses of the Siberian hamster (Phodopus sungorus sungorus) white adipocytes after weight loss induced by short photoperiod exposure.
Topics: Adipocytes; Adipose Tissue; Adrenergic beta-Agonists; Adrenocorticotropic Hormone; Animals; Cricetinae; DNA; Epinephrine; Ethanolamines; Isoproterenol; Lipolysis; Male; Norepinephrine; Peptide YY; Phodopus; Photoperiod; Propanolamines; Sympathomimetics; Weight Gain; Weight Loss | 1998 |
Selectivity and potency of agonists for the three subtypes of cloned human beta-adrenoceptors expressed in Chinese hamster ovary cells.
Topics: Adrenergic beta-Agonists; Animals; Carboxylic Acids; CHO Cells; Cloning, Molecular; Cricetinae; Cyclic AMP; Dioxins; Dioxoles; Dose-Response Relationship, Drug; Ethanolamines; Humans; Isoproterenol; Molecular Structure; Protein Isoforms; Radioligand Assay; Receptors, Adrenergic, beta; Recombinant Proteins | 2000 |
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 2001 |
Metabolic markers following beta-adrenoceptor agonist infusion in footshock-stressed rats.
Topics: Adrenergic beta-Agonists; Animals; Biomarkers; Blood Glucose; Consciousness; Corticosterone; Electroshock; Ethanolamines; Foot; Glycerol; Isoproterenol; Male; Norepinephrine; Rats; Rats, Wistar; Stress, Physiological; Time Factors; Triglycerides | 2001 |
Studies on the expression and function of beta-3-adrenoceptors in the colon of rats with acetic acid-induced colitis.
Topics: Acetic Acid; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colitis, Ulcerative; Colon; Dose-Response Relationship, Drug; Ethanolamines; Female; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Peroxidase; Pindolol; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-3; RNA, Messenger | 2002 |
Beta-adrenergic potentiation of endoplasmic reticulum Ca(2+) release in brown fat cells.
Topics: Adipocytes; Adipose Tissue, Brown; Adrenergic Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium; Cells, Cultured; Endoplasmic Reticulum; Enzyme Inhibitors; Ethanolamines; Isoproterenol; Prazosin; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2; Thapsigargin | 2002 |
BRL 37344 inhibited adrenergic transmission in the rat portal vein via atypical beta-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Electric Stimulation; Ethanolamines; Female; Isoproterenol; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Portal Vein; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Sympathetic Nervous System; Synaptic Transmission | 2002 |
beta3-Adrenergic regulation of an ion channel in the heart-inhibition of the slow delayed rectifier potassium current I(Ks) in guinea pig ventricular myocytes.
Topics: Action Potentials; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Culture Techniques; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Ethanolamines; Guinea Pigs; Isoproterenol; KCNQ Potassium Channels; KCNQ1 Potassium Channel; Male; Myocytes, Cardiac; Norepinephrine; Oocytes; Potassium; Potassium Channels; Potassium Channels, Voltage-Gated; Receptors, Adrenergic, beta-3; Xenopus | 2002 |
Evidence for the primary role for 4-aminopyridine-sensitive K(v) channels in beta(3)-adrenoceptor-mediated, cyclic AMP-independent relaxations of guinea-pig gastrointestinal smooth muscles.
Topics: 4-Aminopyridine; Adrenergic Agonists; Animals; Catecholamines; Cyclic AMP; Epinephrine; Ethanolamines; Guinea Pigs; In Vitro Techniques; Ion Channel Gating; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Propanolamines; Receptors, Adrenergic, beta-3 | 2003 |
Fat accumulation in the rat during early pregnancy is modulated by enhanced insulin responsiveness.
Topics: 1-Methyl-3-isobutylxanthine; Adipocytes; Adipose Tissue; Adrenergic beta-Agonists; Animals; Blood Glucose; Colforsin; Ethanolamines; Fatty Acids, Nonesterified; Female; Gestational Age; Glucose Tolerance Test; Glycerol; Insulin; Isoproterenol; Leptin; Lipids; Lipolysis; Lumbosacral Region; Organ Size; Pregnancy; Rats; Rats, Wistar; Receptors, Adrenergic, beta-3 | 2003 |
The functional role of beta-adrenoceptor subtypes in mediating relaxation of pig urethral smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Ethanolamines; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Swine; Urethra | 2003 |
Endothelial beta3-adrenoceptors mediate vasorelaxation of human coronary microarteries through nitric oxide and endothelium-dependent hyperpolarization.
Topics: Adolescent; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Apamin; Arterioles; Bupranolol; Charybdotoxin; Child; Coronary Vessels; Endothelium, Vascular; Ethanolamines; Female; Humans; Isoproterenol; Male; Membrane Potentials; Microcirculation; Microscopy, Video; Middle Aged; Nadolol; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitroarginine; Potassium Channel Blockers; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Vasodilation | 2004 |
Evidence for the presence of beta-3-adrenoceptors mediating relaxation in the human oviduct.
Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adult; Dose-Response Relationship, Drug; Ethanolamines; Fallopian Tubes; Female; Humans; In Vitro Techniques; Isoproterenol; Middle Aged; Muscle Relaxation; Pindolol; Propranolol; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2005 |
Relaxant effects of beta-adrenergic agonists on porcine and human detrusor muscle.
Topics: Adrenergic beta-Agonists; Aged; Albuterol; Animals; Dioxoles; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Humans; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Procaterol; Propanolamines; Swine | 2005 |
Functional beta-adrenergic receptor signalling on nuclear membranes in adult rat and mouse ventricular cardiomyocytes.
Topics: Adenylyl Cyclases; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blotting, Western; Dioxoles; Ethanolamines; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Microscopy, Confocal; Myocytes, Cardiac; Nuclear Envelope; Pertussis Toxin; Propanolamines; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Signal Transduction | 2006 |
Effects of gender, age and hypertension on beta-adrenergic receptor function in rat urinary bladder.
Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Age Factors; Animals; Ethanolamines; Female; Hypertension; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Wistar; Receptors, Adrenergic, beta; Sex Factors; Urinary Bladder; Urinary Incontinence | 2006 |
Beta3-adrenoceptor in the eel (Anguilla anguilla) heart: negative inotropy and NO-cGMP-dependent mechanism.
Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Anguilla; Animals; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Depression, Chemical; Ethanolamines; GTP-Binding Proteins; Heart; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Nadolol; Nitric Oxide; Propanolamines; Receptors, Adrenergic, beta-3; Signal Transduction | 2006 |
Relaxation of human detrusor muscle by selective beta-2 and beta-3 agonists and endogenous catecholamines.
Topics: Adrenergic beta-Agonists; Aged; Catecholamines; Clenbuterol; Dose-Response Relationship, Drug; Ethanolamines; Female; Humans; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Terbutaline; Urinary Bladder | 2007 |
beta-adrenoceptor agonists downregulate adiponectin, but upregulate adiponectin receptor 2 and tumor necrosis factor-alpha expression in adipocytes.
Topics: 3T3-L1 Cells; Adenylyl Cyclases; Adipocytes; Adiponectin; Adrenergic beta-Agonists; AMP-Activated Protein Kinases; Animals; Blotting, Western; Colforsin; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Enzyme Activation; Ethanolamines; Fenoterol; Gene Expression Regulation; Isoproterenol; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Multienzyme Complexes; Protein Serine-Threonine Kinases; Receptors, Adiponectin; Receptors, Cell Surface; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonamides; Tumor Necrosis Factor-alpha; Up-Regulation | 2007 |
beta(2) and beta(3)-adrenoceptor inhibition of alpha(1)-adrenoceptor-stimulated Ca(2+) elevation in human cultured prostatic stromal cells.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Atenolol; Calcium; Cells, Cultured; Cyclic AMP; Ethanolamines; Humans; Isoproterenol; Male; Phenylephrine; Potassium Channel Blockers; Propanolamines; Propranolol; Prostate; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Stromal Cells; Xamoterol | 2007 |
Role of beta-3-adrenoceptor in catecholamine-induced relaxations in gastric fundus from control and diabetic rats.
Topics: Animals; Catecholamines; Diabetes Mellitus, Experimental; Ethanolamines; Fenoterol; Gastric Fundus; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-3; RNA, Messenger; Streptozocin | 2007 |
Beta3-adrenoceptors modulate left ventricular relaxation in the rat heart via the NO-cGMP-PKG pathway.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Ethanolamines; GTP-Binding Protein alpha Subunits, Gi-Go; Isoproterenol; Male; Nitric Oxide; Organ Culture Techniques; Rats; Rats, Wistar; Receptors, Adrenergic, beta-3; Signal Transduction; Ventricular Function, Left | 2008 |
Potentiation of potassium currents by beta-adrenoceptor agonists in human urinary bladder smooth muscle cells: a possible electrical mechanism of relaxation.
Topics: Adrenergic beta-Agonists; Apamin; Cell Line; Electrophysiology; Ethanolamines; Gene Expression Regulation; Humans; Isoproterenol; Large-Conductance Calcium-Activated Potassium Channels; Membrane Potentials; Muscle, Smooth; Patch-Clamp Techniques; Peptides; Receptors, Adrenergic, beta; Small-Conductance Calcium-Activated Potassium Channels; Urinary Bladder | 2008 |
Relaxations to beta-adrenoceptor subtype selective agonists in wild-type and NOS-3-KO mouse mesenteric arteries.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Dose-Response Relationship, Drug; Ethanolamines; Female; Formoterol Fumarate; In Vitro Techniques; Isoproterenol; Mesenteric Arteries; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Potassium Chloride; Receptors, Adrenergic, beta | 2008 |
Expression and functional role of β3 -adrenoceptors in the human ureter.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Aged; Aged, 80 and over; Albuterol; Ethanolamines; Female; Humans; Isoproterenol; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Procaterol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sympathetic Nervous System; Ureter; Urothelium | 2013 |
Involvement of β3-adrenoceptors in the inhibitory control of cholinergic activity in human bladder: Direct evidence by [(3)H]-acetylcholine release experiments in the isolated detrusor.
Topics: Acetanilides; Acetylcholine; Adrenergic beta-3 Receptor Agonists; Aminophenols; Dose-Response Relationship, Drug; Electric Stimulation; Ethanolamines; Humans; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta-3; Sulfonamides; Thiazoles; Urinary Bladder | 2015 |
[The influence of two-month treatment with bromocryptine on activity of the adenylyl cyclase signaling system in the myocardium and testes of rats with type 2 diabetes mellitus].
Topics: Adenylyl Cyclases; Administration, Oral; Animals; Blood Glucose; Bromocriptine; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Diet, High-Fat; Dioxoles; Dopamine Agonists; Drug Administration Schedule; Ethanolamines; Guanylyl Imidodiphosphate; Humans; Insulin Resistance; Isoproterenol; Male; Myocardium; Norepinephrine; Rats; Rats, Wistar; Relaxin; Signal Transduction; Streptozocin; Testis; Triglycerides | 2014 |
Cyclic Adenosine Monophosphate-Mediated Enhancement of Vascular Endothelial Growth Factor Released by Differentiated Human Monocytic Cells: The Role of Protein Kinase A.
Topics: Adrenergic Antagonists; Adrenergic beta-Agonists; Albuterol; Atenolol; Carbazoles; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Ethanolamines; Humans; Isoproterenol; Lipopolysaccharides; Macrophages; Procaterol; Pyrroles; Vascular Endothelial Growth Factor A | 2015 |
β
Topics: Adrenergic beta-Agonists; Animals; CA1 Region, Hippocampal; Cyclic AMP; Ethanolamines; Isoproterenol; Male; Membrane Potentials; Potassium Channel Blockers; Pyramidal Cells; Pyrimidines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Small-Conductance Calcium-Activated Potassium Channels; Tetrahydronaphthalenes | 2019 |
Acute interaction between human epicardial adipose tissue and human atrial myocardium induces arrhythmic susceptibility.
Topics: Adipose Tissue; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Aged; Arrhythmias, Cardiac; Ethanolamines; Female; Heart; Heart Atria; Humans; Isoproterenol; Male; Myocardial Contraction; Myocardium; Pericardium | 2020 |