isoniazid and bm 212

isoniazid has been researched along with bm 212 in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (14.29)18.2507
2000's3 (42.86)29.6817
2010's3 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Biava, M; Deidda, D; Fioravanti, R; Maullu, C; Pompei, R; Porretta, GC1
Biava, M; Botta, M; Deidda, D; Manetti, F; Molicotti, P; Poce, G; Pompei, R; Porretta, GC; Supino, S1
Biava, M; Botta, M; De Logu, A; De Rossi, E; Manetti, F; Meleddu, R; Poce, G; Porretta, GC; Saddi, M1
Bhakta, S; Brown, AK; Castagnolo, D; Dasugari, S; Evangelopoulos, D; Maitra, A; Manetti, F; McHugh, TD; Mortazavi, PN; Petricci, E; Scalacci, N; Twist, A1
Chakraborti, AK; Dhameliya, TM; Jadhavar, PS; Pancholia, S; Shah, P; Sridevi, JP; Sriram, D; Yogeshwari, P1
Anand, A; B, S; Gokhale, R; Kumar, V; Ramesh, R; Shingare, RD; Srinivasa Reddy, D; Ummanni, R; Veeraraghavan, S; Viswanadha, S1
Biava, M; Cesare Porretta, G; Deidda, D; Manetti, F; Pompei, R; Tafi, A1

Other Studies

7 other study(ies) available for isoniazid and bm 212

ArticleYear
New pyrrole derivatives as antimycobacterial agents analogs of BM212.
    Bioorganic & medicinal chemistry letters, 1999, Oct-18, Volume: 9, Issue:20

    Topics: Antitubercular Agents; Microbial Sensitivity Tests; Mycobacterium; Piperazines; Pyrroles

1999
Antimycobacterial agents. Novel diarylpyrrole derivatives of BM212 endowed with high activity toward Mycobacterium tuberculosis and low cytotoxicity.
    Journal of medicinal chemistry, 2006, Aug-10, Volume: 49, Issue:16

    Topics: Animals; Antitubercular Agents; Chlorocebus aethiops; Microbial Sensitivity Tests; Models, Molecular; Morpholines; Mycobacterium tuberculosis; Piperazines; Pyrroles; Quantitative Structure-Activity Relationship; Vero Cells

2006
1,5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings.
    Journal of medicinal chemistry, 2008, Jun-26, Volume: 51, Issue:12

    Topics: Antitubercular Agents; Drug Resistance, Multiple, Bacterial; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Nontuberculous Mycobacteria; Piperazines; Pyrroles; Structure-Activity Relationship

2008
Design and Synthesis of 1-((1,5-Bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethylocta-2,6-dienyl)ethane-1,2-diamine (SQ109) Pyrrole Hybrid Derivatives: Discovery of Potent Antitubercul
    Journal of medicinal chemistry, 2016, Mar-24, Volume: 59, Issue:6

    Topics: Adamantane; Antitubercular Agents; Carrier Proteins; Cell Line; Cell Survival; Computational Biology; Drug Design; Drug Resistance, Multiple, Bacterial; Ethylenediamines; Humans; Microbial Sensitivity Tests; Models, Molecular; Mycobacterium; Mycobacterium tuberculosis; Pharmaceutical Preparations; Piperazines; Pyrroles; Structure-Activity Relationship

2016
Benzo[d]thiazol-2-yl(piperazin-1-yl)methanones as new anti-mycobacterial chemotypes: Design, synthesis, biological evaluation and 3D-QSAR studies.
    European journal of medicinal chemistry, 2016, Jun-30, Volume: 116

    Topics: Animals; Antitubercular Agents; Chemistry Techniques, Synthetic; Drug Design; Mice; Microbial Sensitivity Tests; Models, Molecular; Molecular Conformation; Mycobacterium tuberculosis; Piperazine; Piperazines; Quantitative Structure-Activity Relationship; RAW 264.7 Cells

2016
Repurposing of a drug scaffold: Identification of novel sila analogues of rimonabant as potent antitubercular agents.
    European journal of medicinal chemistry, 2016, Oct-21, Volume: 122

    Topics: Antitubercular Agents; Drug Repositioning; Hep G2 Cells; Humans; Microbial Sensitivity Tests; Models, Molecular; Molecular Conformation; Mycobacterium tuberculosis; Piperidines; Pyrazoles; Rimonabant; Structure-Activity Relationship

2016
Importance of the thiomorpholine introduction in new pyrrole derivatives as antimycobacterial agents analogues of BM 212.
    Bioorganic & medicinal chemistry, 2003, Feb-20, Volume: 11, Issue:4

    Topics: Anti-Bacterial Agents; Antibiotics, Antitubercular; Antifungal Agents; Antitubercular Agents; Antiviral Agents; Binding Sites; Chemical Phenomena; Chemistry, Physical; Indicators and Reagents; Isoniazid; Microbial Sensitivity Tests; Models, Molecular; Molecular Conformation; Morpholines; Mycobacterium; Piperazines; Pyrroles; Rifampin; Streptomycin; Structure-Activity Relationship

2003
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