isoguvacine has been researched along with gamma-aminobutyric acid in 84 studies
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 33 (39.29) | 18.7374 |
1990's | 30 (35.71) | 18.2507 |
2000's | 14 (16.67) | 29.6817 |
2010's | 7 (8.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Brehm, L; Falch, E; Frølund, B; Hansen, AB; Kristiansen, U; Krogsgaard-Larsen, P | 1 |
Ebert, B; Kehler, J; Krogsgaard-Larsen, P; Mortensen, M; Thompson, SA; Wafford, KA | 1 |
Bang-Andersen, B; Ebert, B; Frølund, B; Hansen, CP; Jensen, AA; Kristiansen, U; Krogsgaard-Larsen, P; Larsen, M; Liljefors, T; Madsen, C; Nielsen, B | 1 |
Brandsch, M; Gebauer, S; Laug, L; Schäfer, S; Thondorf, I; Voigt, V; Zebisch, K | 1 |
Balle, T; Bergmann, R; Damgaard, M; Frølund, B; Jensen, AA; Nielsen, B; Petersen, JG; Sørensen, T | 1 |
Bowery, NG; Collins, JF; Hudson, AL; Neal, MJ | 1 |
Polc, P | 1 |
Karobath, M; Lippitsch, M | 1 |
Curtis, DR; Johnston, GA; Lodge, D | 1 |
Conzelmann, U; Meyer, DK; Müller, A | 1 |
Tietz, EI; Xie, XH | 1 |
Chesler, M; Hassan, AZ; Sakatani, K | 3 |
Ching, W; Hassan, AZ; Sakatani, K | 1 |
Corbett, R; Cornfeldt, M; Dunn, RW; Fielding, S | 1 |
Hablitz, JJ; Mistry, DK | 1 |
Astier, H; Roussel, JP | 1 |
Drew, CA; Johnston, GA | 1 |
Balcar, VJ | 1 |
Gallagher, JP; Twery, MJ | 1 |
Albin, RL; Chu, DC; Penney, JB; Young, AB | 1 |
Balcar, VJ; Dreher, B | 1 |
Bickford-Wimer, PC; Hoffer, BJ; Parfitt, KD | 1 |
Ciuffi, M; Franchi-Micheli, S; Luzzi, S; Rosi, E; Zilletti, L | 1 |
Bossu, JL; Demeneix, BA; Dupont, JL; Feltz, A; Feltz, P; Taleb, O; Trouslard, J | 1 |
Brailowsky, S; Champagnat, J; Menini, C; Naquet, R; Silva-Barrat, C | 1 |
Crawford, ML; Young, JM | 1 |
Astier, H; Jourdan, J; Roussel, JP; Tapia-Arancibia, L | 1 |
Olsen, RW; Snowman, AM | 1 |
Iversen, LL; Wong, EH | 1 |
Allan, AM; Harris, RA | 1 |
Ciesielski, L; Gobaille, S; Mandel, P; Molina, V | 1 |
Kemp, JA; Marshall, GR; Woodruff, GN | 1 |
Audi, EA; Brandão, ML; Graeff, FG; Schütz, MT | 1 |
Astier, H; Roussel, JP; Tapia-Arancibia, L | 1 |
Ben-Ari, Y; Cherubini, E; Rovira, C | 1 |
Karobath, M; Supavilai, P | 1 |
Brown, DA; Scholfield, CN | 1 |
Benson, DI; Klepner, CA; Squires, RF | 1 |
Meldrum, B | 1 |
Desarmenien, M; Feltz, P; Headley, PM | 1 |
Mantegazza, P; Tammiso, R; Vicentini, L; Zambotti, F; Zonta, N | 2 |
Aaes-Jørgensen, T; Bøgesø, KP; Krogsgaard-Larsen, P; Mikkelsen, H; Schultz, B | 1 |
Falch, E; Krogsgaard-Larsen, P | 1 |
Brehm, L; Krogsgaard-Larsen, P; Schaumburg, K | 1 |
Cavagnini, F; Grandison, L; Guidotti, A; Invitti, SC; Schmid, R | 1 |
Agardh, E; Ehinger, B | 2 |
Curtis, DR; Hjeds, H; Krogsgaard-Larsen, P; Leah, JD; Peet, MJ | 1 |
Bloch, R; Bousquet, P; Feldman, J; Schwartz, J | 1 |
Snodgrass, SR; White, WF | 1 |
Goudreau, JL; Lookingland, KJ; Moore, KE; Wagner, EJ | 1 |
Barnes, EM; Calkin, PA | 1 |
de Koning, HP; Jenks, BG; Leenders, HJ; Ponten, SP; Roubos, EW | 1 |
Honmou, O; Sakatani, K; Young, W | 1 |
Darlington, CL; Hutchinson, M; Smith, PF | 1 |
Moos, FC | 1 |
Bowery, NG; Malcangio, M; Teoh, H | 1 |
Dominguez-Perrot, C; Feltz, P; Poulter, MO | 1 |
Fricker, D; Le Feuvre, Y; Leresche, N | 1 |
Guan, BC; Hu, HZ; Li, ZW; Si, JQ; Zhou, XP | 1 |
Buckingham, SD; Rauh, J; Sattelle, DB; Schnee, M | 1 |
Castel, H; Cazin, L; Le Foll, F; Louiset, E; Vaudry, H | 1 |
Bas, DE; Calamera, JC; Ritta, MN | 1 |
Ben-Ari, Y; Dzhala, V; Khalilov, I; Khazipov, R | 1 |
Barker, JL; Maric, D; Schaffner, AE; Sukhareva, M; Vautrin, J | 1 |
Buckingham, SD; Hosie, AM; Presnail, JK; Sattelle, DB | 1 |
Chub, N; O'Donovan, MJ | 1 |
Johnson, SW; Shen, KZ | 1 |
Trussell, LO; Turecek, R | 1 |
Ben-Ari, Y; Holmes, GL; Khalilov, I; Khazipov, R; Morozova, E; Tyzio, R | 1 |
Doepner, RF; Geigerseder, C; Krieger, A; Mayerhofer, A; Thalhammer, A | 1 |
Holmes, GL; Isaev, D; Isaeva, E; Khazipov, R | 1 |
Reis, HJ; Romano-Silva, MA; Smith, TK; Vanden Berghe, P | 1 |
Ennis, M; Hayar, A | 1 |
Ben-Ari, Y; Holmes, GL; Khazipov, R; Tyzio, R | 1 |
Aniksztejn, L; Becq, H; Ben-Ari, Y; Bulteau, C; Cossart, R; Crepel, V; Delalande, O; Dorfmüller, G; Dulac, O; Epsztein, J; Fohlen, M; Jorquera, I; Khalilov, I; Khazipov, R; Milh, M; Minlebaev, M; Mukhtarov, M; Nardou, R; Oliver, V; Represa, A; Rheims, S; Tyzio, R; Zilberter, Y | 1 |
Arisi, I; Brandi, R; Capsoni, S; Cattaneo, A; Cherubini, E; D'Onofrio, M; Franzot, J; Lagostena, L; Rosato-Siri, M | 1 |
Kaila, K; Ruusuvuori, E; Viitanen, T; Voipio, J | 1 |
Brame, LS; Cao, A; Fang, YT; Fung, KM; Humphreys, MR; Kropp, BP; Lin, HK; Shih, PT; Wu, W; Yang, Q | 1 |
Chen, Q; Ding, L; Gao, R; Gao, XY; Kang, YM; Li, YH; Xiong, XQ; Zhu, GQ | 1 |
Allain, AE; Branchereau, P; Cattaert, D; Delpy, A; Martin, E; Meyrand, P | 1 |
4 review(s) available for isoguvacine and gamma-aminobutyric acid
Article | Year |
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GABA-agonists as anti-epileptic agents.
Topics: Animals; Anticonvulsants; Barbiturates; Benzodiazepines; Disease Models, Animal; Epilepsy; Etomidate; gamma-Aminobutyric Acid; Hydroxybutyrates; Isonicotinic Acids; Mice; Muscimol; Rats; Receptors, Cell Surface; Receptors, GABA-A; Sodium Oxybate | 1981 |
THIP, isoguvacine, isoguvacine oxide, and related GABA agonists.
Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; Humans; Isonicotinic Acids; Isoxazoles; Oxazoles; Pipecolic Acids; Receptors, Cell Surface; Receptors, GABA-A; Tissue Distribution | 1981 |
GABA agonists. Development and interactions with the GABA receptor complex.
Topics: Amino Acids; Animals; Benzodiazepines; Brain Chemistry; Cats; Chemical Phenomena; Chemistry; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Mice; Models, Structural; Muscimol; Receptors, Cell Surface; Receptors, GABA-A; Structure-Activity Relationship | 1981 |
Muscimol, a psychoactive constituent of Amanita muscaria, as a medicinal chemical model structure.
Topics: Agaricales; Amanita; Animals; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Magnetic Resonance Spectroscopy; Models, Chemical; Models, Structural; Molecular Conformation; Muscimol; Nipecotic Acids; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Stereoisomerism | 1981 |
80 other study(ies) available for isoguvacine and gamma-aminobutyric acid
Article | Year |
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Partial GABAA receptor agonists. Synthesis and in vitro pharmacology of a series of nonannulated analogs of 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol.
Topics: Animals; Cells, Cultured; Cerebral Cortex; GABA-A Receptor Agonists; Isoxazoles; Magnetic Resonance Spectroscopy; Mice; Neurons; Rats; Rats, Sprague-Dawley | 1995 |
Bioisosteric determinants for subtype selectivity of ligands for heteromeric GABA(A) receptors.
Topics: Animals; GABA Agonists; GABA Antagonists; Humans; Inhibitory Concentration 50; Ligands; Oocytes; Protein Subunits; Receptors, GABA-A; Transfection; Xenopus | 2001 |
5-Substituted imidazole-4-acetic acid analogues: synthesis, modeling, and pharmacological characterization of a series of novel gamma-aminobutyric acid(C) receptor agonists.
Topics: Animals; Brain; Cell Line; GABA Agonists; GABA-A Receptor Agonists; Humans; Imidazoles; In Vitro Techniques; Ligands; Membrane Potentials; Models, Molecular; Mutation; Oocytes; Patch-Clamp Techniques; Protein Structure, Tertiary; Protein Subunits; Radioligand Assay; Rats; Receptors, GABA; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship | 2007 |
Three-dimensional quantitative structure-activity relationship analyses of substrates of the human proton-coupled amino acid transporter 1 (hPAT1).
Topics: Amino Acid Transport Systems; Caco-2 Cells; Endocytosis; Humans; Kinetics; Models, Chemical; Models, Molecular; Molecular Conformation; Quantitative Structure-Activity Relationship; Substrate Specificity; Symporters | 2011 |
Synthesis and pharmacological evaluation of 6-aminonicotinic acid analogues as novel GABA(A) receptor agonists.
Topics: Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Humans; Ligands; Models, Molecular; Molecular Structure; Niacin; Receptors, GABA-A; Structure-Activity Relationship | 2014 |
Isoguvacine, isonipecotic acid, muscimol and N-methyl isoguvacine on the GABA receptor in rat sympathetic ganglia.
Topics: Animals; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Ganglia, Autonomic; Isonicotinic Acids; Isonipecotic Acids; Membrane Potentials; Muscimol; Rats; Receptors, Neurotransmitter; Structure-Activity Relationship | 1978 |
Effects of GABA-mimetic agents on the cat spinal cord.
Topics: Animals; Bicuculline; Cats; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Ibotenic Acid; Isonicotinic Acids; Isoxazoles; Male; Muscimol; Neurons, Afferent; Spinal Cord | 1979 |
THIP and isoguvacine are partial agonists of GABA-stimulated benzodiazepine receptor binding.
Topics: Animals; Benzodiazepines; Cerebral Cortex; Drug Synergism; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Muscimol; Oxazoles; Rats; Receptors, Drug | 1979 |
Does uptake limit the actions of GABA agonists in vivo? Experiments with muscimol, isoguvacine and THIP in cat spinal cord.
Topics: Aminobutyrates; Animals; Biological Transport; Cats; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Muscimol; Neurons; Nipecotic Acids; Oxazoles; Spinal Cord | 1978 |
Effects of GABA receptor stimulation on the release of [3H]GABA from slices of rat neostriatum.
Topics: Animals; Convulsants; Corpus Striatum; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sodium Channels; Tetrodotoxin | 1992 |
Reduction in potency of selective gamma-aminobutyric acidA agonists and diazepam in CA1 region of in vitro hippocampal slices from chronic flurazepam-treated rats.
Topics: Animals; Diazepam; Evoked Potentials; Flurazepam; gamma-Aminobutyric Acid; Hippocampus; Isonicotinic Acids; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1992 |
GABA-sensitivity of dorsal column axons: an in vitro comparison between adult and neonatal rat spinal cords.
Topics: Action Potentials; Aging; Animals; Animals, Newborn; Axons; gamma-Aminobutyric Acid; Isonicotinic Acids; Neural Conduction; Rats; Receptors, GABA-A; Spinal Cord | 1991 |
Age-dependent extrasynaptic modulation of axonal conduction by exogenous and endogenous GABA in the rat optic nerve.
Topics: Action Potentials; Age Factors; Animals; Animals, Newborn; Axons; Cells, Cultured; gamma-Aminobutyric Acid; Isonicotinic Acids; Neural Conduction; Nipecotic Acids; Optic Nerve; Proline; Rats; Receptors, GABA-A; Synapses | 1991 |
GABAmimetic agents display anxiolytic-like effects in the social interaction and elevated plus maze procedures.
Topics: Aminooxyacetic Acid; Animals; Anti-Anxiety Agents; Conflict, Psychological; Diazepam; Exploratory Behavior; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Muscimol; Rats; Rats, Inbred Strains; Social Behavior; Valproic Acid | 1991 |
Activation of subconductance states by gamma-aminobutyric acid and its analogs in chick cerebral neurons.
Topics: Analgesics; Animals; Cells, Cultured; Cerebral Cortex; Chick Embryo; Chlorides; Electric Conductivity; gamma-Aminobutyric Acid; Ion Channel Gating; Ion Channels; Isonicotinic Acids; Isoxazoles; Muscimol; Neurons | 1990 |
Involvement of dihydropyridine-sensitive calcium channels in the GABAA potentiation of TRH-induced TSH release.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Drug Synergism; GABA Antagonists; gamma-Aminobutyric Acid; GTP-Binding Proteins; In Vitro Techniques; Isonicotinic Acids; Male; Nifedipine; omega-Conotoxins; Peptides, Cyclic; Pertussis Toxin; Pituitary Gland; Pyridazines; Rats; Rats, Inbred Strains; Thyrotropin; Thyrotropin-Releasing Hormone; Virulence Factors, Bordetella | 1990 |
Bicuculline- and baclofen-insensitive gamma-aminobutyric acid binding to rat cerebellar membranes.
Topics: Animals; Baclofen; Bicuculline; Binding Sites; Calcium; Cerebellum; gamma-Aminobutyric Acid; Isonicotinic Acids; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains | 1992 |
GABAA receptors modulate axonal conduction in dorsal columns of neonatal rat spinal cord.
Topics: Action Potentials; Animals; Animals, Newborn; Axons; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Male; Neural Conduction; Osmolar Concentration; Reaction Time; Receptors, GABA-A; Spinal Cord | 1991 |
Presence of a highly efficient "binding" to bacterial contamination can distort data from binding studies.
Topics: Animals; Cats; Cerebral Cortex; GABA Antagonists; gamma-Aminobutyric Acid; Gram-Positive Bacteria; Isonicotinic Acids; Muscimol; Nipecotic Acids; Proline; Pyridazines; Radioligand Assay; Receptors, GABA-A; Tritium | 1990 |
Somatostatin depresses GABA receptor-mediated inhibition in the rat dorsolateral septal nucleus.
Topics: Animals; Baclofen; Brain; Electric Stimulation; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Kinetics; Male; Membrane Potentials; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Somatostatin; Synapses; Time Factors | 1990 |
Distribution and kinetics of GABAB binding sites in rat central nervous system: a quantitative autoradiographic study.
Topics: Animals; Autoradiography; Baclofen; Binding, Competitive; Brain; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Neurochemical correlates of gamma-aminobutyrate (GABA) inhibition in cat visual cortex.
Topics: Animals; Baclofen; Calcium; Cats; Cell Membrane; Female; GABA Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Neurons; Potassium; Pyridazines; Receptors, GABA-A; Visual Cortex | 1990 |
Potentiation of gamma-aminobutyric acid-mediated inhibition by isoproterenol in the cerebellar cortex: receptor specificity.
Topics: Action Potentials; Animals; Baclofen; Cerebellar Cortex; Drug Synergism; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoproterenol; Male; Neurons; Purkinje Cells; Rats; Rats, Inbred F344; Receptors, GABA-A | 1990 |
Effect of various GABA-receptor agonists and antagonists on anaphylactic histamine release in the guinea-pig ileum.
Topics: Anaphylaxis; Animals; Baclofen; beta-Alanine; Depression, Chemical; gamma-Aminobutyric Acid; Guinea Pigs; Histamine Release; Ileum; Isonicotinic Acids; Male; Muscle, Smooth; Receptors, GABA-A; Taurine | 1987 |
Spontaneous and GABA-evoked chloride channels on pituitary intermediate lobe cells and their internal Ca requirements.
Topics: Animals; Calcium; Cells, Cultured; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Ions; Isonicotinic Acids; Membrane Potentials; Pituitary Gland; Receptors, GABA-A | 1987 |
Relationship between tolerance to GABAA agonist and bursting properties in neocortical neurons during GABA-withdrawal syndrome.
Topics: Animals; Cerebral Cortex; Drug Tolerance; Electrophysiology; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Male; Neurons; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome | 1989 |
GABAB receptor-mediated inhibition of histamine H1-receptor-induced inositol phosphate formation in slices of rat cerebral cortex.
Topics: Animals; Baclofen; Carbachol; Cerebral Cortex; gamma-Aminobutyric Acid; Histamine; Inositol; Inositol Phosphates; Isonicotinic Acids; Kinetics; Lithium; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Histamine H1; Sugar Phosphates | 1988 |
Effect of norfloxacin, a new quinolone, on GABA modulation of TRH-induced TSH release from perifused rat pituitaries.
Topics: Animals; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Norfloxacin; Perfusion; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thyrotropin; Thyrotropin-Releasing Hormone | 1988 |
Avermectin B1a modulation of gamma-aminobutyric acid/benzodiazepine receptor binding in mammalian brain.
Topics: Animals; Bicuculline; Brain; Cattle; Cell Membrane; Cerebral Cortex; Etazolate; gamma-Aminobutyric Acid; Isonicotinic Acids; Ivermectin; Lactones; Muscimol; Pentobarbital; Rats; Receptors, GABA-A | 1985 |
Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.
Topics: Androstanes; Animals; Azasteroids; Bicuculline; Cell Membrane; Cerebral Cortex; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isonicotinic Acids; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, GABA-A; Taurine | 1985 |
gamma-Aminobutyric acid agonists and antagonists alter chloride flux across brain membranes.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Animals; Baclofen; Bicuculline; Brain; Cell Membrane; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Liver; Male; Mice; Mice, Inbred DBA; Muscimol; Picrotoxin; Receptors, GABA-A; Sodium; Sulfates; Taurine; Temperature | 1986 |
Effects of the potentiation of the GABAergic neurotransmission in the olfactory bulbs on mouse-killing behavior.
Topics: Aggression; Aminocaproates; Animals; Brain Chemistry; Drug Synergism; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Motor Activity; Muscimol; Nipecotic Acids; Olfactory Bulb; Proline; Rats; Rats, Inbred Strains; Synaptic Transmission; Valproic Acid; Vigabatrin | 1986 |
Quantitative evaluation of the potencies of GABA-receptor agonists and antagonists using the rat hippocampal slice preparation.
Topics: Action Potentials; Animals; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isonicotinic Acids; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1986 |
Modulation of the brain aversive system by GABAergic and serotonergic mechanisms.
Topics: Animals; Avoidance Learning; Benzodiazepines; Cerebral Ventricles; Chlordiazepoxide; Drug Interactions; gamma-Aminobutyric Acid; Isonicotinic Acids; Midazolam; Muscimol; Pentobarbital; Periaqueductal Gray; Rats; Receptors, GABA-A; Serotonin | 1986 |
Evidence for a dual effect of gamma-aminobutyric acid on thyrotropin (TSH)-releasing hormone-induced TSH release from perifused rat pituitaries.
Topics: Animals; Bicuculline; Dose-Response Relationship, Drug; Drug Synergism; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Male; Muscimol; Perfusion; Picrotoxin; Pituitary Gland; Pyridazines; Rats; Rats, Inbred Strains; Thyrotropin; Thyrotropin-Releasing Hormone | 1987 |
Somatic and dendritic actions of gamma-aminobutyric acid agonists and uptake blockers in the hippocampus in vivo.
Topics: Acetylcholine; Action Potentials; Animals; Dendrites; gamma-Aminobutyric Acid; Hippocampus; Isonicotinic Acids; Isoxazoles; Male; Muscimol; Rats; Synaptic Transmission | 1984 |
The effect of temperature and chloride ions on the stimulation of [3H]flunitrazepam binding by the muscimol analogues THIP and piperidine-4-sulfonic acid.
Topics: Animals; Anti-Anxiety Agents; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Oxazoles; Piperidines; Rats; Stimulation, Chemical; Temperature; Tritium | 1980 |
Inhibition of GABA uptake potentiates the conductance increase produced by GABA-mimetic compounds on single neurones in isolated olfactory cortex slices of the guinea-pig.
Topics: Animals; Central Nervous System; Cerebral Cortex; Electric Stimulation; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Isonicotinic Acids; Muscimol; Neural Conduction; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Olfactory Pathways; Proline; Sodium; Taurine | 1984 |
Multiple benzodiazepine receptor complexes: some benzodiazepine recognition sites are coupled to GABA receptors and ionophores.
Topics: Animals; Anions; Benzodiazepines; Bicuculline; Brain; Buffers; Flunitrazepam; gamma-Aminobutyric Acid; Haplorhini; Hot Temperature; Ionophores; Isonicotinic Acids; Isoxazoles; Macromolecular Substances; Papio; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter | 1980 |
Does glial uptake affect GABA responses? AN intracellular study on rat dorsal root ganglion neurones in vitro.
Topics: Animals; beta-Alanine; gamma-Aminobutyric Acid; Ganglia, Spinal; In Vitro Techniques; Isonicotinic Acids; Membrane Potentials; Muscimol; Neuroglia; Neurons; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1980 |
Effects of some GABA-mimetic drugs on the antinociceptive activity of morphine and beta-endorphin in rats.
Topics: Analgesics; Animals; beta-Endorphin; Bicuculline; Drug Interactions; Endorphins; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Morphine; Muscimol; Nicotinic Acids; Nipecotic Acids; Rats | 1981 |
gamma-Aminobutyric acid- and benzodiazepine-binding sites in human anterior pituitary tissue.
Topics: Adult; Aged; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Humans; Isonicotinic Acids; Isoxazoles; Middle Aged; Muscimol; Pituitary Gland, Anterior; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A | 1982 |
(3H)-muscimol, (3H)-nipecotic acid and (3H)-isoguvacine as autoradiographic markers for GABA neurotransmission.
Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; Goldfish; Guinea Pigs; Isonicotinic Acids; Muscimol; Neuroglia; Neurons; Nipecotic Acids; Oxazoles; Rabbits; Receptors, Cell Surface; Receptors, GABA-A; Retina; Synaptic Transmission | 1982 |
Glycine antagonists structurally related to muscimol, THIP, or isoguvacine.
Topics: Animals; Cats; gamma-Aminobutyric Acid; Glycine; Interneurons; Isonicotinic Acids; Isoxazoles; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Glycine; Spinal Cord; Structure-Activity Relationship | 1982 |
Pharmacological analysis of the central cardiovascular effects of four GABA analogues.
Topics: Animals; Atropine; Bicuculline; Blood Pressure; Brain; GABA Antagonists; gamma-Aminobutyric Acid; Heart Rate; Isonicotinic Acids; Isoxazoles; Kainic Acid; Muscimol; Pyrones; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Retinal GABA neuron labelling with [3H]isoguvacine in different species.
Topics: Animals; Autoradiography; Cell Count; Chickens; gamma-Aminobutyric Acid; Goldfish; Guinea Pigs; Humans; Isonicotinic Acids; Neurons; Rabbits; Rats; Retina; Retinal Ganglion Cells; Tritium | 1983 |
Isoguvacine binding, uptake, and release: relation to the GABA system.
Topics: 3-O-Methylglucose; Animals; Binding Sites; Biological Transport; Brain; Carbon Radioisotopes; gamma-Aminobutyric Acid; Isonicotinic Acids; Kinetics; Methylglucosides; Rats; Synaptosomes; Tritium | 1983 |
The effect of GABAergic agents on opiate analgesia.
Topics: Animals; Drug Interactions; Endorphins; gamma-Aminobutyric Acid; Injections, Intraventricular; Isonicotinic Acids; Male; Morphine; Muscimol; Narcotics; Nicotinic Acids; Nipecotic Acids; Pain; Rats; Reaction Time; Time Factors | 1980 |
GABAergic regulation of tuberoinfundibular dopaminergic neurons in the male rat.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Dopamine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Isonicotinic Acids; Male; Neurons; Osmolar Concentration; Prolactin; Pyridazines; Rats; Rats, Inbred Strains; Seizures | 1994 |
Effects of GABA on axonal conduction and extracellular potassium activity in the neonatal rat optic nerve.
Topics: Action Potentials; Animals; Animals, Newborn; Axons; Extracellular Space; gamma-Aminobutyric Acid; Isonicotinic Acids; Neural Conduction; Optic Nerve; Potassium; Rats; Receptors, GABA-A | 1994 |
gamma-Aminobutyric acid-A (GABAA) agonists down-regulate GABAA/benzodiazepine receptor polypeptides from the surface of chick cortical neurons.
Topics: Androstanes; Animals; Azasteroids; Blotting, Western; Cells, Cultured; Cerebral Cortex; Chick Embryo; Down-Regulation; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Molecular Weight; Neurons; Receptors, GABA-A | 1994 |
Differential effects of coexisting dopamine, GABA and NPY on alpha-MSH secretion from melanotrope cells of Xenopus laevis.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; alpha-MSH; Animals; Baclofen; Dopamine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Kinetics; Neuropeptide Y; Perfusion; Pituitary Gland; Radioimmunoassay; Xenopus laevis | 1993 |
GABA and potassium effects on corticospinal and primary afferent tracts of neonatal rat spinal dorsal columns.
Topics: Afferent Pathways; Animals; Animals, Newborn; gamma-Aminobutyric Acid; Isonicotinic Acids; Neural Conduction; Potassium; Pyramidal Tracts; Rats; Rats, Inbred Strains; Spinal Cord | 1993 |
Further evidence on the contribution of GABAA receptors to the GABA-mediated inhibition of medial vestibular nucleus neurones in vitro.
Topics: Action Potentials; Animals; Brain Stem; Dose-Response Relationship, Drug; GABA Agonists; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Isonicotinic Acids; Neurons; Receptors, GABA-A; Time Factors; Vestibular Nuclei | 1995 |
GABA-induced facilitation of the periodic bursting activity of oxytocin neurones in suckled rats.
Topics: Animals; Animals, Suckling; Electrophysiology; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Microinjections; Neurons; Osmotic Pressure; Oxytocin; Paraventricular Hypothalamic Nucleus; Periodicity; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Supraoptic Nucleus | 1995 |
GABA, glutamate and substance P-like immunoreactivity release: effects of novel GABAB antagonists.
Topics: Animals; Baclofen; Benzoates; Benzylamines; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Nerve Roots; Stereoisomerism; Substance P | 1996 |
Recombinant GABAA receptor desensitization: the role of the gamma 2 subunit and its physiological significance.
Topics: Cells, Cultured; Computer Simulation; Electrophysiology; GABA Agonists; gamma-Aminobutyric Acid; Humans; Isonicotinic Acids; Kidney; Kinetics; Membrane Potentials; Patch-Clamp Techniques; Protein Binding; Receptors, GABA-A; Recombinant Proteins; Synaptic Transmission; Taurine; Transfection | 1996 |
GABAA receptor-mediated IPSCs in rat thalamic sensory nuclei: patterns of discharge and tonic modulation by GABAB autoreceptors.
Topics: Animals; Autoreceptors; Baclofen; Cadmium; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Geniculate Bodies; Interneurons; Isonicotinic Acids; Male; Membrane Potentials; Organ Culture Techniques; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Tetrodotoxin; Thalamic Nuclei | 1997 |
Inhibitory effect of baclofen on GABA-induced depolarization and GABA-activated current in primary sensory neurons.
Topics: Animals; Baclofen; Electric Conductivity; Electrophysiology; Female; GABA Agonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Muscimol; Neurons, Afferent; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Time Factors | 1997 |
Pharmacology of skeletal muscle GABA-gated chloride channels in the cockroach Periplaneta americana.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Flunitrazepam; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Isonicotinic Acids; Male; Motor Neurons; Muscle, Skeletal; Periplaneta; Picrotoxin; Receptors, GABA; Sesterterpenes | 1997 |
Multiple modulatory effects of the neuroactive steroid pregnanolone on GABAA receptor in frog pituitary melanotrophs.
Topics: Action Potentials; Animals; Cells, Cultured; Evoked Potentials; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Membrane Potentials; Patch-Clamp Techniques; Pituitary Gland; Pregnanolone; Protein Conformation; Rana ridibunda; Receptors, GABA-A | 1997 |
Occurrence of GABA and GABA receptors in human spermatozoa.
Topics: Bicuculline; Cell Membrane; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Isonicotinic Acids; Male; Muscimol; Receptors, GABA; Semen; Sperm Motility; Spermatozoa; Tritium | 1998 |
Dual role of GABA in the neonatal rat hippocampus.
Topics: Animals; Animals, Newborn; Bicuculline; Diazepam; Electrophysiology; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isonicotinic Acids; Nerve Net; Rats; Rats, Wistar | 1999 |
Surface-accessible GABA supports tonic and quantal synaptic transmission.
Topics: Adsorption; Animals; Cells, Cultured; Chloride Channels; Electrophysiology; Exocytosis; Female; Flow Cytometry; GABA Agonists; gamma-Aminobutyric Acid; Gangliosides; Isonicotinic Acids; Liposomes; Membrane Potentials; Membrane Proteins; Neurons; Pregnancy; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptic Transmission | 2000 |
Alternative splicing of a Drosophila GABA receptor subunit gene identifies determinants of agonist potency.
Topics: Alternative Splicing; Amino Acid Sequence; Animals; Drosophila melanogaster; Drosophila Proteins; Embryo, Nonmammalian; Exons; Female; GABA Agonists; gamma-Aminobutyric Acid; Gene Library; Genetic Variation; In Vitro Techniques; Isonicotinic Acids; Isonipecotic Acids; Membrane Potentials; Molecular Sequence Data; Muscimol; Oocytes; Patch-Clamp Techniques; Protein Subunits; Receptors, GABA-A; Recombinant Proteins; Sulfonic Acids; Xenopus laevis | 2001 |
Post-episode depression of GABAergic transmission in spinal neurons of the chick embryo.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Anterior Horn Cells; Bicuculline; Chick Embryo; Chloride Channels; Chlorides; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gramicidin; Ion Transport; Isonicotinic Acids; Membrane Potentials; Nerve Tissue Proteins; Patch-Clamp Techniques; Periodicity; Receptors, GABA-A; Refractory Period, Electrophysiological; Spinal Cord; Synaptic Transmission; Tetrodotoxin | 2001 |
Potentiation of GABA(A) receptor agonists by GABA uptake inhibitors in the rat ventral midbrain.
Topics: Animals; Carrier Proteins; Drug Synergism; Electrophysiology; GABA Agonists; GABA Plasma Membrane Transport Proteins; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Mesencephalon; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Organic Anion Transporters; Oximes; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sodium; Suprachiasmatic Nucleus | 2001 |
Reciprocal developmental regulation of presynaptic ionotropic receptors.
Topics: Animals; Brain Stem; Evoked Potentials; GABA Agonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Ion Channel Gating; Isonicotinic Acids; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Receptors, Glycine; Receptors, Presynaptic; Synaptic Transmission | 2002 |
Developmental changes in GABAergic actions and seizure susceptibility in the rat hippocampus.
Topics: Aging; Animals; Animals, Newborn; Bicuculline; Disease Susceptibility; Excitatory Postsynaptic Potentials; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isonicotinic Acids; Male; Membrane Potentials; Neural Inhibition; Patch-Clamp Techniques; Potassium; Pyramidal Cells; Rats; Seizures; Time Factors | 2004 |
Stimulation of TM3 Leydig cell proliferation via GABA(A) receptors: a new role for testicular GABA.
Topics: Animals; Animals, Newborn; Carrier Proteins; Cell Division; Cell Line; Enzyme Activation; GABA Agonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Isoenzymes; Isonicotinic Acids; Leydig Cells; Male; Membrane Proteins; Membrane Transport Proteins; Mice; Mice, Inbred BALB C; Proliferating Cell Nuclear Antigen; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, GABA-A; Testis | 2004 |
Anticonvulsant action of GABA in the high potassium-low magnesium model of ictogenesis in the neonatal rat hippocampus in vivo and in vitro.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Bicuculline; Disease Models, Animal; Drug Interactions; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isonicotinic Acids; Lipoproteins; Magnesium; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium; Pyridazines; Rats; Seizures | 2005 |
GABA-induced calcium signaling in cultured enteric neurons is reinforced by activation of cholinergic pathways.
Topics: Acetylcholine; Animals; Baclofen; Calcium; Calcium Channel Blockers; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Fura-2; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Hexamethonium; Isonicotinic Acids; Myenteric Plexus; Neurons; Nicotinic Antagonists; Ondansetron; Pyridoxal Phosphate; Serotonin Antagonists; Signal Transduction | 2006 |
Endogenous GABA and glutamate finely tune the bursting of olfactory bulb external tufted cells.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Animals, Newborn; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Neurons; Olfactory Bulb; Pyridazines; Rats; Rats, Sprague-Dawley; Valine | 2007 |
Timing of the developmental switch in GABA(A) mediated signaling from excitation to inhibition in CA3 rat hippocampus using gramicidin perforated patch and extracellular recordings.
Topics: Action Potentials; Age Factors; Animals; Animals, Newborn; Bicuculline; Calcium Channels; Electrophysiology; Excitatory Postsynaptic Potentials; Female; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gramicidin; Hippocampus; Inhibitory Postsynaptic Potentials; Isonicotinic Acids; Male; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-A | 2007 |
Inhibitory actions of the gamma-aminobutyric acid in pediatric Sturge-Weber syndrome.
Topics: Action Potentials; Bumetanide; Cerebral Cortex; Diazepam; Epilepsy; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Infant; Isonicotinic Acids; Membrane Potentials; Neural Inhibition; Neurons; Receptors, GABA-A; Receptors, Glutamate; Sodium Potassium Chloride Symporter Inhibitors; Solute Carrier Family 12, Member 2; Sturge-Weber Syndrome | 2009 |
In the adult hippocampus, chronic nerve growth factor deprivation shifts GABAergic signaling from the hyperpolarizing to the depolarizing direction.
Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antibodies, Neutralizing; Biophysics; Bumetanide; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Hippocampus; In Vitro Techniques; Ion Channel Gating; Isonicotinic Acids; K Cl- Cotransporters; Mice; Mice, Transgenic; Nerve Growth Factor; Neurons; Patch-Clamp Techniques; Pyridazines; Quinoxalines; Receptors, Nicotinic; RNA, Messenger; Sodium Potassium Chloride Symporter Inhibitors; Symporters | 2010 |
The K+-Cl cotransporter KCC2 promotes GABAergic excitation in the mature rat hippocampus.
Topics: Animals; Anticonvulsants; Barium; Bicarbonates; CA1 Region, Hippocampal; Carbonic Anhydrase Inhibitors; Chlorides; Diuretics; Electric Stimulation; Electrophysiology; Epilepsy; Furosemide; GABA Agonists; gamma-Aminobutyric Acid; Hippocampus; Hydrogen-Ion Concentration; Isonicotinic Acids; K Cl- Cotransporters; Microelectrodes; Potassium; Pyramidal Cells; Rats; Receptors, GABA-A; Spectrometry, Fluorescence; Symporters | 2010 |
Linking γ-aminobutyric acid A receptor to epidermal growth factor receptor pathways activation in human prostate cancer.
Topics: Autocrine Communication; Cell Line, Tumor; Cell Proliferation; ErbB Receptors; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gefitinib; Gene Expression Regulation, Neoplastic; Humans; Isonicotinic Acids; Male; Paracrine Communication; Phosphorylation; Picrotoxin; Prostate; Prostatic Neoplasms; Protein Kinase Inhibitors; Quinazolines; Receptors, GABA-A; Signal Transduction; src-Family Kinases | 2014 |
GABA in Paraventricular Nucleus Regulates Adipose Afferent Reflex in Rats.
Topics: Adipose Tissue, White; Afferent Pathways; Animals; Baclofen; gamma-Aminobutyric Acid; Isonicotinic Acids; Kidney; Male; Organophosphorus Compounds; Paraventricular Hypothalamic Nucleus; Pyridazines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Vigabatrin | 2015 |
Depolarizing GABA/glycine synaptic events switch from excitation to inhibition during frequency increases.
Topics: Animals; Chlorides; Embryo, Mammalian; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glycine; Isonicotinic Acids; Mice; Microscopy, Fluorescence; Motor Neurons; Patch-Clamp Techniques; Spinal Cord | 2016 |