isoguvacine and baclofen

isoguvacine has been researched along with baclofen in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-199010 (33.33)18.7374
1990's15 (50.00)18.2507
2000's4 (13.33)29.6817
2010's1 (3.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Drew, CA; Johnston, GA1
Gallagher, JP; Twery, MJ1
Albin, RL; Chu, DC; Penney, JB; Young, AB1
Balcar, VJ; Dreher, B1
Bickford-Wimer, PC; Hoffer, BJ; Parfitt, KD1
Ciuffi, M; Franchi-Micheli, S; Luzzi, S; Rosi, E; Zilletti, L1
Chu, DC; Penney, JB; Young, AB1
Oveissi, Y; Zarrindast, MR1
Crawford, ML; Young, JM1
Hösli, E; Hösli, L; Krogsgaard-Larsen, P1
Allan, RD; Dickenson, HW1
Allan, AM; Harris, RA1
Anderson, R; Mitchell, R1
Mitchell, R1
Demeneix, BA; Desaulles, E; Feltz, P; Loeffler, JP1
Goudreau, JL; Lookingland, KJ; Moore, KE; Wagner, EJ1
Damgaard, I; Elster, L; Kardos, J; Krogsgaard-Larsen, P; Schousboe, A1
Albin, RL; Altschuler, RA; Helfert, RH; Juiz, JM1
Hammond, DL; Washington, JD1
de Koning, HP; Jenks, BG; Leenders, HJ; Ponten, SP; Roubos, EW1
Bowery, NG; Malcangio, M; Teoh, H1
Cruijsen, PM; Dotman, CH; Jenks, BG; Roubos, EW1
Maier, SF; McGorry, M; Schwartz, B; Sisk, D; Watkins, LR; Wiertelak, EP1
Fricker, D; Le Feuvre, Y; Leresche, N1
Guan, BC; Hu, HZ; Li, ZW; Si, JQ; Zhou, XP1
Firestone, LL; Hammond, DL; Homanics, GE; Ugarte, SD1
Denda, M; Denda, S; Inomata, S; Inoue, K1
Reis, HJ; Romano-Silva, MA; Smith, TK; Vanden Berghe, P1
Gao, J; Gao, XY; Liao, ZH; Shi, Z; Wang, W; Zhong, MK; Zhou, LM; Zhu, GQ1
Chen, Q; Ding, L; Gao, R; Gao, XY; Kang, YM; Li, YH; Xiong, XQ; Zhu, GQ1

Other Studies

30 other study(ies) available for isoguvacine and baclofen

ArticleYear
Bicuculline- and baclofen-insensitive gamma-aminobutyric acid binding to rat cerebellar membranes.
    Journal of neurochemistry, 1992, Volume: 58, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Binding Sites; Calcium; Cerebellum; gamma-Aminobutyric Acid; Isonicotinic Acids; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains

1992
Somatostatin depresses GABA receptor-mediated inhibition in the rat dorsolateral septal nucleus.
    Brain research, 1990, Jun-11, Volume: 519, Issue:1-2

    Topics: Animals; Baclofen; Brain; Electric Stimulation; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Kinetics; Male; Membrane Potentials; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Somatostatin; Synapses; Time Factors

1990
Distribution and kinetics of GABAB binding sites in rat central nervous system: a quantitative autoradiographic study.
    Neuroscience, 1990, Volume: 34, Issue:2

    Topics: Animals; Autoradiography; Baclofen; Binding, Competitive; Brain; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Neurochemical correlates of gamma-aminobutyrate (GABA) inhibition in cat visual cortex.
    Life sciences, 1990, Volume: 47, Issue:15

    Topics: Animals; Baclofen; Calcium; Cats; Cell Membrane; Female; GABA Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Neurons; Potassium; Pyridazines; Receptors, GABA-A; Visual Cortex

1990
Potentiation of gamma-aminobutyric acid-mediated inhibition by isoproterenol in the cerebellar cortex: receptor specificity.
    Neuropharmacology, 1990, Volume: 29, Issue:10

    Topics: Action Potentials; Animals; Baclofen; Cerebellar Cortex; Drug Synergism; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoproterenol; Male; Neurons; Purkinje Cells; Rats; Rats, Inbred F344; Receptors, GABA-A

1990
Effect of various GABA-receptor agonists and antagonists on anaphylactic histamine release in the guinea-pig ileum.
    Agents and actions, 1987, Volume: 20, Issue:3-4

    Topics: Anaphylaxis; Animals; Baclofen; beta-Alanine; Depression, Chemical; gamma-Aminobutyric Acid; Guinea Pigs; Histamine Release; Ileum; Isonicotinic Acids; Male; Muscle, Smooth; Receptors, GABA-A; Taurine

1987
Cortical GABAB and GABAA receptors in Alzheimer's disease: a quantitative autoradiographic study.
    Neurology, 1987, Volume: 37, Issue:9

    Topics: Aged; Alzheimer Disease; Animals; Autoradiography; Baclofen; Binding, Competitive; Frontal Lobe; Humans; Isonicotinic Acids; Kinetics; Middle Aged; Rats; Receptors, GABA-A

1987
GABAA and GABAB receptor sites involvement in rat thermoregulation.
    General pharmacology, 1988, Volume: 19, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Body Temperature Regulation; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Injections, Intraventricular; Isonicotinic Acids; Male; Muscimol; Picrotoxin; Rats; Receptors, GABA-A

1988
GABAB receptor-mediated inhibition of histamine H1-receptor-induced inositol phosphate formation in slices of rat cerebral cortex.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: Animals; Baclofen; Carbachol; Cerebral Cortex; gamma-Aminobutyric Acid; Histamine; Inositol; Inositol Phosphates; Isonicotinic Acids; Kinetics; Lithium; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Histamine H1; Sugar Phosphates

1988
Autoradiographic localization of binding sites for the gamma-aminobutyric acid analogues 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol (THIP)isoguvacine and baclofen on cultured neurons of rat cerebellum and spinal cord.
    Neuroscience letters, 1985, Oct-24, Volume: 61, Issue:1-2

    Topics: Animals; Animals, Newborn; Autoradiography; Baclofen; Binding Sites; Cells, Cultured; Cerebellum; Fetus; Isonicotinic Acids; Isoxazoles; Oxazoles; Rats; Receptors, GABA-A; Spinal Cord

1985
Evidence that antagonism by delta-aminovaleric acid of GABAB receptors in the guinea-pig ileum may be due to an interaction between GABAA and GABAB receptors.
    European journal of pharmacology, 1986, Jan-14, Volume: 120, Issue:1

    Topics: Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Bicuculline; Electric Stimulation; Female; Guinea Pigs; Ileum; In Vitro Techniques; Isonicotinic Acids; Male; Muscle, Smooth; Receptors, GABA-A; Taurine

1986
gamma-Aminobutyric acid agonists and antagonists alter chloride flux across brain membranes.
    Molecular pharmacology, 1986, Volume: 29, Issue:5

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Animals; Baclofen; Bicuculline; Brain; Cell Membrane; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Liver; Male; Mice; Mice, Inbred DBA; Muscimol; Picrotoxin; Receptors, GABA-A; Sodium; Sulfates; Taurine; Temperature

1986
Biphasic effect of GABAA receptor agonists on prolactin secretion: evidence for two types of GABAA receptor complex on lactotrophes.
    European journal of pharmacology, 1986, May-13, Volume: 124, Issue:1-2

    Topics: Animals; Baclofen; Carnosine; Isonicotinic Acids; Male; Muscimol; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
Interactions of agonists and antagonists with a novel type of GABA receptor.
    Biochemical pharmacology, 1982, Aug-15, Volume: 31, Issue:16

    Topics: Animals; Baclofen; Bicuculline; Corpus Striatum; GABA Antagonists; In Vitro Techniques; Isonicotinic Acids; Kinetics; Male; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1982
Dual population of GABAA and GABAB receptors in rat pars intermedia demonstrated by release of alpha MSH caused by barium ions.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: Animals; Baclofen; Barium; Bicuculline; Female; In Vitro Techniques; Isonicotinic Acids; Male; Melanocyte-Stimulating Hormones; Pituitary Gland; Radioimmunoassay; Rats; Receptors, Cell Surface; Receptors, GABA-A; Stereoisomerism; Stimulation, Chemical

1984
GABAergic regulation of tuberoinfundibular dopaminergic neurons in the male rat.
    Brain research, 1994, Oct-03, Volume: 659, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Dopamine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Isonicotinic Acids; Male; Neurons; Osmolar Concentration; Prolactin; Pyridazines; Rats; Rats, Inbred Strains; Seizures

1994
Role of GABAB receptors in intracellular Ca2+ homeostasis and possible interaction between GABAA and GABAB receptors in regulation of transmitter release in cerebellar granule neurons.
    Journal of neuroscience research, 1994, Dec-15, Volume: 39, Issue:6

    Topics: Animals; Aspartic Acid; Baclofen; Calcium; Calcium Radioisotopes; Cells, Cultured; Cerebellum; GABA Agonists; GTP-Binding Proteins; Homeostasis; Isonicotinic Acids; Isoxazoles; Mice; Neurons; Neurotransmitter Agents; Pertussis Toxin; Receptors, GABA-A; Receptors, GABA-B; Virulence Factors, Bordetella

1994
Distribution of GABAA and GABAB binding sites in the cochlear nucleus of the guinea pig.
    Brain research, 1994, Mar-14, Volume: 639, Issue:2

    Topics: Animals; Autoradiography; Baclofen; Cerebellar Cortex; Cochlear Nucleus; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Guinea Pigs; Isonicotinic Acids; Receptors, GABA-A; Receptors, GABA-B

1994
Antagonism of L-baclofen-induced antinociception by CGP 35348 in the spinal cord of the rat.
    European journal of pharmacology, 1993, Apr-06, Volume: 234, Issue:2-3

    Topics: Analgesics; Animals; Baclofen; Dose-Response Relationship, Drug; GABA-A Receptor Antagonists; Hot Temperature; Injections, Spinal; Isonicotinic Acids; Male; Nociceptors; Organophosphorus Compounds; Pain Measurement; Pain Threshold; Postural Balance; Rats; Rats, Sprague-Dawley; Reflex; Spinal Cord

1993
Differential effects of coexisting dopamine, GABA and NPY on alpha-MSH secretion from melanotrope cells of Xenopus laevis.
    Life sciences, 1993, Volume: 52, Issue:24

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; alpha-MSH; Animals; Baclofen; Dopamine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Kinetics; Neuropeptide Y; Perfusion; Pituitary Gland; Radioimmunoassay; Xenopus laevis

1993
GABA, glutamate and substance P-like immunoreactivity release: effects of novel GABAB antagonists.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Animals; Baclofen; Benzoates; Benzylamines; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Nerve Roots; Stereoisomerism; Substance P

1996
Differential action of secreto-inhibitors on proopiomelanocortin biosynthesis in the intermediate pituitary of Xenopus laevis.
    Endocrinology, 1996, Volume: 137, Issue:11

    Topics: alpha-MSH; Analysis of Variance; Animals; Apomorphine; Baclofen; GABA Agonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; In Vitro Techniques; Isonicotinic Acids; Kinetics; Neuropeptide Y; Pituitary Gland; Pro-Opiomelanocortin; Receptors, Dopamine D2; Xenopus laevis

1996
Reversal of spinal cord non-opiate analgesia by conditioned anti-analgesia in the rat.
    Pain, 1997, Volume: 71, Issue:3

    Topics: Analgesia, Epidural; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Baclofen; Biguanides; Conditioning, Classical; Drug Evaluation, Preclinical; GABA Agonists; Isonicotinic Acids; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Spinal Cord

1997
GABAA receptor-mediated IPSCs in rat thalamic sensory nuclei: patterns of discharge and tonic modulation by GABAB autoreceptors.
    The Journal of physiology, 1997, Jul-01, Volume: 502 ( Pt 1)

    Topics: Animals; Autoreceptors; Baclofen; Cadmium; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Geniculate Bodies; Interneurons; Isonicotinic Acids; Male; Membrane Potentials; Organ Culture Techniques; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Tetrodotoxin; Thalamic Nuclei

1997
Inhibitory effect of baclofen on GABA-induced depolarization and GABA-activated current in primary sensory neurons.
    Neuroscience, 1997, Volume: 81, Issue:3

    Topics: Animals; Baclofen; Electric Conductivity; Electrophysiology; Female; GABA Agonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Male; Muscimol; Neurons, Afferent; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Time Factors

1997
Sensory thresholds and the antinociceptive effects of GABA receptor agonists in mice lacking the beta3 subunit of the GABA(A) receptor.
    Neuroscience, 2000, Volume: 95, Issue:3

    Topics: Animals; Baclofen; GABA Agonists; Hot Temperature; Injections, Spinal; Injections, Subcutaneous; Isonicotinic Acids; Isoxazoles; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Nociceptors; Physical Stimulation; Protein Isoforms; Receptors, GABA-A; Sensory Thresholds; Sex Characteristics

2000
gamma-Aminobutyric acid (A) receptor agonists accelerate cutaneous barrier recovery and prevent epidermal hyperplasia induced by barrier disruption.
    The Journal of investigative dermatology, 2002, Volume: 119, Issue:5

    Topics: Animals; Baclofen; Epidermis; GABA Agonists; GABA-A Receptor Agonists; Humidity; Hyperplasia; Isonicotinic Acids; Male; Mice; Mice, Hairless; Muscimol; Receptors, GABA-A; Wound Healing

2002
GABA-induced calcium signaling in cultured enteric neurons is reinforced by activation of cholinergic pathways.
    Neuroscience, 2006, May-12, Volume: 139, Issue:2

    Topics: Acetylcholine; Animals; Baclofen; Calcium; Calcium Channel Blockers; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Fura-2; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Hexamethonium; Isonicotinic Acids; Myenteric Plexus; Neurons; Nicotinic Antagonists; Ondansetron; Pyridoxal Phosphate; Serotonin Antagonists; Signal Transduction

2006
Regulation of cardiac sympathetic afferent reflex by GABA(A) and GABA(B) receptors in paraventricular nucleus in rats.
    The European journal of neuroscience, 2008, Volume: 27, Issue:12

    Topics: Animals; Baclofen; Bradykinin; Capsaicin; GABA Agonists; GABA Antagonists; Heart; Isonicotinic Acids; Kidney; Male; Neurons, Afferent; Organophosphorus Compounds; Paraventricular Hypothalamic Nucleus; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Reflex; Sensory System Agents; Sympathetic Nervous System; Vigabatrin

2008
GABA in Paraventricular Nucleus Regulates Adipose Afferent Reflex in Rats.
    PloS one, 2015, Volume: 10, Issue:8

    Topics: Adipose Tissue, White; Afferent Pathways; Animals; Baclofen; gamma-Aminobutyric Acid; Isonicotinic Acids; Kidney; Male; Organophosphorus Compounds; Paraventricular Hypothalamic Nucleus; Pyridazines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Vigabatrin

2015