Page last updated: 2024-09-03

isofloxythepin and apomorphine

isofloxythepin has been researched along with apomorphine in 2 studies

Compound Research Comparison

Studies
(isofloxythepin)
Trials
(isofloxythepin)
Recent Studies (post-2010)
(isofloxythepin)
Studies
(apomorphine)
Trials
(apomorphine)
Recent Studies (post-2010) (apomorphine)
26409,205287780

Protein Interaction Comparison

ProteinTaxonomyisofloxythepin (IC50)apomorphine (IC50)
Tryptophan 5-hydroxylase 1Rattus norvegicus (Norway rat)0.22
D(2) dopamine receptorHomo sapiens (human)0.0146
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.75
DRattus norvegicus (Norway rat)0.4744
D(3) dopamine receptorRattus norvegicus (Norway rat)0.1432
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.063
D(2) dopamine receptorBos taurus (cattle)0.3385
D(1A) dopamine receptorHomo sapiens (human)0.025
D(4) dopamine receptorHomo sapiens (human)0.025
D(1B) dopamine receptorHomo sapiens (human)0.025
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.75
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(4) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(3) dopamine receptorHomo sapiens (human)0.025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.75
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0813
E3 ubiquitin-protein ligase Mdm2Homo sapiens (human)0.205
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)1.35
DBos taurus (cattle)0.3385

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lau, YS; Runice, C1
Chlebounová, J; Dlabac, A; Metysová, J; Valchár, M1

Other Studies

2 other study(ies) available for isofloxythepin and apomorphine

ArticleYear
Prolonged inhibition of striatal dopamine receptor sites by isofloxythepin.
    European journal of pharmacology, 1985, Oct-08, Volume: 116, Issue:1-2

    Topics: Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Dibenzothiepins; Dose-Response Relationship, Drug; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1985
Induction of dopaminergic supersensitivity after a single dose of the neuroleptic isofloxythepin.
    Psychopharmacology, 1982, Volume: 76, Issue:4

    Topics: Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Dibenzothiepins; Homovanillic Acid; Humans; Hypothalamus; Male; Median Eminence; Neural Pathways; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Substantia Nigra

1982