Page last updated: 2024-09-03

isf 2405 and cadralazine

isf 2405 has been researched along with cadralazine in 7 studies

Compound Research Comparison

Studies
(isf 2405)
Trials
(isf 2405)
Recent Studies (post-2010)
(isf 2405)
Studies
(cadralazine)
Trials
(cadralazine)
Recent Studies (post-2010) (cadralazine)
910801612

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19903 (42.86)18.7374
1990's4 (57.14)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Nässberger, L1
Andersson, M; Dahlbäck, B; Englund, G; Hanson, A1
Brunel, P; Guyene, TT; Imhof, P; Lecaillon, JB; Ménard, J1
Inukai, T; Karaki, H; Mitsui, M; Nakao, K1
Hashimoto, M; Hayashi, T; Ishikawa, S; Sekine, Y; Takeyama, K; Terauchi, Y; Watari, S1
Higashio, T; Kuroda, K1
Hashimoto, M; Ishikawa, S; Kagemoto, A; Nakao, M; Negoro, T; Sekine, Y; Terauchi, Y; Watari, S1

Trials

1 trial(s) available for isf 2405 and cadralazine

ArticleYear
Influence of acetylator status on the haemodynamic effects and pharmacokinetics of cadralazine in healthy subjects.
    British journal of clinical pharmacology, 1990, Volume: 29, Issue:5

    Topics: Acetylation; Adult; Antihypertensive Agents; Blood Pressure; Forearm; Heart Rate; Hemodynamics; Humans; Male; Middle Aged; Phenotype; Pyridazines; Regional Blood Flow; Renin; Stroke Volume; Vasodilation

1990

Other Studies

6 other study(ies) available for isf 2405 and cadralazine

ArticleYear
The antihypertensive compounds hydralazine, dihydralazine and cadralazine and their metabolites inhibit myeloperoxidase activity as measured by chemiluminescence.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Antihypertensive Agents; Binding Sites; Dihydralazine; Dose-Response Relationship, Drug; Hydralazine; Luminescent Measurements; Magnetic Resonance Spectroscopy; Peroxidase; Pyridazines; Structure-Activity Relationship

1991
Inhibition of complement components C3 and C4 by cadralazine and its active metabolite.
    European journal of clinical pharmacology, 1991, Volume: 40, Issue:3

    Topics: Antihypertensive Agents; Complement C3; Complement C4; Dihydralazine; Humans; Hydralazine; Hydroxylamine; Hydroxylamines; Procainamide; Pyridazines; Vasodilator Agents

1991
Inhibitory effects of cadralazine and its metabolite, ISF-2405, on contractions and the level of cytosolic Ca2+ in vascular smooth muscle.
    European journal of pharmacology, 1990, Mar-20, Volume: 178, Issue:2

    Topics: Animals; Calcium; Cytosol; Dinoprost; Dogs; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Pyridazines; Rabbits; Vasodilator Agents; Verapamil

1990
Pharmacokinetics of an active cadralazine metabolite in plasma and blood vessels of spontaneously hypertensive rats.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:2

    Topics: Animals; Blood Pressure; Blood Vessels; Half-Life; Male; Pyridazines; Rats; Rats, Inbred SHR; Vasodilator Agents

1988
Effects of cadralazine on contractions induced by Ca2+ and norepinephrine in isolated rabbit aortic strips.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:3

    Topics: Animals; Aorta, Abdominal; Calcium; Hydralazine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Pyridazines; Rabbits

1988
Determination of ISF-2405, an active metabolite of cadralazine, in plasma and tissues by radioimmunoassay.
    Journal of pharmacobio-dynamics, 1987, Volume: 10, Issue:12

    Topics: Animals; Antibodies; Aorta; Guinea Pigs; Male; Pyridazines; Radioimmunoassay; Rats; Rats, Inbred Strains; Time Factors; Tissue Distribution

1987