Page last updated: 2024-08-17

isatin and 5-bromoisatin

isatin has been researched along with 5-bromoisatin in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (37.50)29.6817
2010's5 (62.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chibale, K; Chiyanzu, I; Gut, J; Hansell, E; McKerrow, JH; Rosenthal, PJ1
Benkendorff, K; Bremner, JB; Locke, JM; Pyne, SG; Ranson, M; Vine, KL1
Danks, MK; Edwards, CC; Hatfield, MJ; Hyatt, JL; Moak, T; Potter, PM; Tsurkan, L; Wadkins, RM; Wierdl, M1
Fassihi, A; Mohammadpour, M; Sabet, R; Sadeghi, A1
Boardman, P; Choi, K; Griffin, JH; Jin, X; Khosla, C; Klöck, C; Lanza, G; Madrid, PB; Raimundo, BC; Spencer, A1
Dung, do TM; Dung, PT; Han, BW; Han, SB; Huong, TL; Kang, JS; Kim, KR; Kim, Y; Nam, NH; Oanh, DT; Park, SH; Quyen, D; Thao, le T; Yun, J1
Guo, Q; Han, K; Liu, F; Liu, W; Song, B; Teng, Y; Wang, P; Yang, Y; Yao, Q; Yu, P; Zhou, Y1
Fan, ZC; Gao, ML; Han, KL; Liu, H; Sun, H; Teng, YO; Wang, J; Yu, P; Zhang, YM; Zhao, HY; Zhou, Y1

Other Studies

8 other study(ies) available for isatin and 5-bromoisatin

ArticleYear
Synthesis and evaluation of isatins and thiosemicarbazone derivatives against cruzain, falcipain-2 and rhodesain.
    Bioorganic & medicinal chemistry letters, 2003, Oct-20, Volume: 13, Issue:20

    Topics: Drug Evaluation, Preclinical; Isatin; Magnetic Resonance Spectroscopy; Protease Inhibitors; Spectrometry, Mass, Fast Atom Bombardment; Thiosemicarbazones

2003
In vitro cytotoxicity evaluation of some substituted isatin derivatives.
    Bioorganic & medicinal chemistry, 2007, Jan-15, Volume: 15, Issue:2

    Topics: Animals; Antineoplastic Agents; Apoptosis; Caspase 3; Caspase 7; Cell Line, Tumor; Cell Survival; Cyclin-Dependent Kinase 2; Enzyme Activators; Enzyme Inhibitors; Humans; Indicators and Reagents; Isatin; Magnetic Resonance Spectroscopy; Mice; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship

2007
Selective inhibition of carboxylesterases by isatins, indole-2,3-diones.
    Journal of medicinal chemistry, 2007, Apr-19, Volume: 50, Issue:8

    Topics: Acetylcholinesterase; Butyrylcholinesterase; Carboxylic Ester Hydrolases; Cholinesterase Inhibitors; Humans; Hydrophobic and Hydrophilic Interactions; Isatin; Models, Molecular; Quantitative Structure-Activity Relationship

2007
QSAR study of isatin analogues as in vitro anti-cancer agents.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Drug Design; Humans; Isatin; Linear Models; Models, Biological; Molecular Structure; Quantitative Structure-Activity Relationship

2010
Acylideneoxoindoles: a new class of reversible inhibitors of human transglutaminase 2.
    Bioorganic & medicinal chemistry letters, 2011, May-01, Volume: 21, Issue:9

    Topics: Enzyme Activation; Enzyme Inhibitors; GTP-Binding Proteins; Humans; Indoles; Inhibitory Concentration 50; Protein Glutamine gamma Glutamyltransferase 2; Structure-Activity Relationship; Transglutaminases

2011
Novel isatin-based hydroxamic acids as histone deacetylase inhibitors and antitumor agents.
    European journal of medicinal chemistry, 2013, Volume: 70

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Humans; Hydroxamic Acids; Isatin; Molecular Structure; Protein Tyrosine Phosphatase, Non-Receptor Type 1; Structure-Activity Relationship

2013
Design, synthesis and in vitro cytotoxicity evaluation of 5-(2-carboxyethenyl)isatin derivatives as anticancer agents.
    Bioorganic & medicinal chemistry letters, 2014, Jan-15, Volume: 24, Issue:2

    Topics: Antineoplastic Agents; Apoptosis; Cytotoxins; Drug Design; Drug Screening Assays, Antitumor; Hep G2 Cells; HT29 Cells; Humans; K562 Cells

2014
Synthesis and anti-cancer activity evaluation of 5-(2-carboxyethenyl)-isatin derivatives.
    European journal of medicinal chemistry, 2016, Apr-13, Volume: 112

    Topics: Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Drug Screening Assays, Antitumor; Humans; Isatin; Jurkat Cells; Leukemia, T-Cell; Membrane Potential, Mitochondrial; Mitochondria; Neoplasms

2016